sr 95531 has been researched along with pentobarbital in 12 studies
Studies (sr 95531) | Trials (sr 95531) | Recent Studies (post-2010) (sr 95531) | Studies (pentobarbital) | Trials (pentobarbital) | Recent Studies (post-2010) (pentobarbital) |
---|---|---|---|---|---|
610 | 0 | 209 | 10,272 | 175 | 439 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (41.67) | 18.2507 |
2000's | 4 (33.33) | 29.6817 |
2010's | 3 (25.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ho, IK; Kimura, T; Miyaoka, T; Saunders, PA | 1 |
Bormann, J; Feigenspan, A | 1 |
Lukasiewicz, PD; Maple, BR; Werblin, FS | 1 |
Cestari, IN; Uchida, I; Yang, J | 1 |
Bracamontes, J; Steinbach, JH; Ueno, S; Weiss, DS; Zorumski, C | 1 |
Dreyfus, H; Jellali, A; Pattnaik, B; Picaud, S; Sahel, J | 1 |
Mathers, DA; Puil, E; Ran, I | 1 |
Czajkowski, C; Mercado, J | 1 |
Czajkowski, C; Sharkey, LM | 1 |
Czajkowski, C; Venkatachalan, SP | 1 |
Barg, S; Birnir, B; Jin, Y; Jin, Z; Korol, SV | 1 |
Chesnoy-Marchais, D | 1 |
12 other study(ies) available for sr 95531 and pentobarbital
Article | Year |
---|---|
Effects of pentobarbital tolerance and dependence on convulsant and GABAA receptor antagonist binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Convulsants; GABA Antagonists; Male; Pentobarbital; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Substance-Related Disorders | 1992 |
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction | 1994 |
A novel GABA receptor on bipolar cell terminals in the tiger salamander retina.
Topics: Animals; Bicuculline; Chlorides; Crotonates; Electrophysiology; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Urodela | 1994 |
The differential antagonism by bicuculline and SR95531 of pentobarbitone-induced currents in cultured hippocampal neurons.
Topics: Anesthetics, General; Anesthetics, Intravenous; Animals; Bicuculline; Binding Sites; Cells, Cultured; Chloride Channels; Chlorides; Etomidate; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Models, Molecular; Neurons; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A | 1996 |
Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor.
Topics: Allosteric Regulation; Allosteric Site; Amino Acid Sequence; Animals; Bicuculline; Binding Sites; Binding, Competitive; Cell Line; Coturnix; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Transport; Models, Chemical; Molecular Sequence Data; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pentobarbital; Point Mutation; Pregnanediones; Pregnanolone; Protein Binding; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship | 1997 |
GABAC receptors are localized with microtubule-associated protein 1B in mammalian cone photoreceptors.
Topics: Animals; Cell Separation; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C3H; Microtubule-Associated Proteins; Patch-Clamp Techniques; Pentobarbital; Phosphinic Acids; Pyridazines; Pyridines; Receptors, GABA; Retina; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells | 2000 |
Pentobarbital induces thalamic oscillations in brain slices, modulated by GABA and glycine receptors.
Topics: Animals; Basal Ganglia; Electric Stimulation; Extracellular Space; Fourier Analysis; GABA Antagonists; Glycine Agents; Hypnotics and Sedatives; In Vitro Techniques; Nerve Net; Organophosphorus Compounds; Pentobarbital; Pyridazines; Rats; Receptors, GABA; Receptors, Glycine; Strychnine; Thalamus | 2004 |
Gamma-aminobutyric acid (GABA) and pentobarbital induce different conformational rearrangements in the GABA A receptor alpha1 and beta2 pre-M1 regions.
Topics: Amino Acid Substitution; Animals; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Pentobarbital; Protein Structure, Tertiary; Pyridazines; Rats; Receptors, GABA-A; Xenopus laevis | 2008 |
Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.
Topics: Animals; Benzodiazepines; Binding Sites; Cysteine; Dose-Response Relationship, Drug; Electrophysiology; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Inhibitory Concentration 50; Ligands; Microinjections; Muscimol; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A; Xenopus | 2008 |
Structural link between γ-aminobutyric acid type A (GABAA) receptor agonist binding site and inner β-sheet governs channel activation and allosteric drug modulation.
Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Benzodiazepines; Binding Sites; Drug Design; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Molecular Sequence Data; Oocytes; Pentobarbital; Protein Structure, Secondary; Pyridazines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis | 2012 |
In intact islets interstitial GABA activates GABA(A) receptors that generate tonic currents in α-cells.
Topics: Animals; gamma-Aminobutyric Acid; Gene Expression Regulation; Glucagon-Secreting Cells; Ion Channel Gating; Pentobarbital; Protein Subunits; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2013 |
Persistent GABAA/C responses to gabazine, taurine and beta-alanine in rat hypoglossal motoneurons.
Topics: Animals; beta-Alanine; Bicuculline; Brain Stem; Central Nervous System Agents; Chlorine; GABA Agents; Hypoglossal Nerve; Midazolam; Motor Neurons; Neuroprotective Agents; Patch-Clamp Techniques; Pentobarbital; Phosphinic Acids; Pregnanolone; Pyridazines; Pyridines; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Strychnine; Taurine; Tissue Culture Techniques | 2016 |