Page last updated: 2024-09-02

sr 95531 and pentobarbital

sr 95531 has been researched along with pentobarbital in 12 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(pentobarbital)
Trials
(pentobarbital)
Recent Studies (post-2010) (pentobarbital)
610020910,272175439

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (41.67)18.2507
2000's4 (33.33)29.6817
2010's3 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ho, IK; Kimura, T; Miyaoka, T; Saunders, PA1
Bormann, J; Feigenspan, A1
Lukasiewicz, PD; Maple, BR; Werblin, FS1
Cestari, IN; Uchida, I; Yang, J1
Bracamontes, J; Steinbach, JH; Ueno, S; Weiss, DS; Zorumski, C1
Dreyfus, H; Jellali, A; Pattnaik, B; Picaud, S; Sahel, J1
Mathers, DA; Puil, E; Ran, I1
Czajkowski, C; Mercado, J1
Czajkowski, C; Sharkey, LM1
Czajkowski, C; Venkatachalan, SP1
Barg, S; Birnir, B; Jin, Y; Jin, Z; Korol, SV1
Chesnoy-Marchais, D1

Other Studies

12 other study(ies) available for sr 95531 and pentobarbital

ArticleYear
Effects of pentobarbital tolerance and dependence on convulsant and GABAA receptor antagonist binding.
    Life sciences, 1992, Volume: 50, Issue:22

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Convulsants; GABA Antagonists; Male; Pentobarbital; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Substance-Related Disorders

1992
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction

1994
A novel GABA receptor on bipolar cell terminals in the tiger salamander retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:3 Pt 1

    Topics: Animals; Bicuculline; Chlorides; Crotonates; Electrophysiology; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Urodela

1994
The differential antagonism by bicuculline and SR95531 of pentobarbitone-induced currents in cultured hippocampal neurons.
    European journal of pharmacology, 1996, Jun-20, Volume: 307, Issue:1

    Topics: Anesthetics, General; Anesthetics, Intravenous; Animals; Bicuculline; Binding Sites; Cells, Cultured; Chloride Channels; Chlorides; Etomidate; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Models, Molecular; Neurons; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A

1996
Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: Allosteric Regulation; Allosteric Site; Amino Acid Sequence; Animals; Bicuculline; Binding Sites; Binding, Competitive; Cell Line; Coturnix; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Transport; Models, Chemical; Molecular Sequence Data; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pentobarbital; Point Mutation; Pregnanediones; Pregnanolone; Protein Binding; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship

1997
GABAC receptors are localized with microtubule-associated protein 1B in mammalian cone photoreceptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Sep-15, Volume: 20, Issue:18

    Topics: Animals; Cell Separation; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C3H; Microtubule-Associated Proteins; Patch-Clamp Techniques; Pentobarbital; Phosphinic Acids; Pyridazines; Pyridines; Receptors, GABA; Retina; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells

2000
Pentobarbital induces thalamic oscillations in brain slices, modulated by GABA and glycine receptors.
    Neuropharmacology, 2004, Volume: 47, Issue:7

    Topics: Animals; Basal Ganglia; Electric Stimulation; Extracellular Space; Fourier Analysis; GABA Antagonists; Glycine Agents; Hypnotics and Sedatives; In Vitro Techniques; Nerve Net; Organophosphorus Compounds; Pentobarbital; Pyridazines; Rats; Receptors, GABA; Receptors, Glycine; Strychnine; Thalamus

2004
Gamma-aminobutyric acid (GABA) and pentobarbital induce different conformational rearrangements in the GABA A receptor alpha1 and beta2 pre-M1 regions.
    The Journal of biological chemistry, 2008, May-30, Volume: 283, Issue:22

    Topics: Amino Acid Substitution; Animals; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Pentobarbital; Protein Structure, Tertiary; Pyridazines; Rats; Receptors, GABA-A; Xenopus laevis

2008
Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.
    Molecular pharmacology, 2008, Volume: 74, Issue:1

    Topics: Animals; Benzodiazepines; Binding Sites; Cysteine; Dose-Response Relationship, Drug; Electrophysiology; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Inhibitory Concentration 50; Ligands; Microinjections; Muscimol; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A; Xenopus

2008
Structural link between γ-aminobutyric acid type A (GABAA) receptor agonist binding site and inner β-sheet governs channel activation and allosteric drug modulation.
    The Journal of biological chemistry, 2012, Feb-24, Volume: 287, Issue:9

    Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Benzodiazepines; Binding Sites; Drug Design; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Molecular Sequence Data; Oocytes; Pentobarbital; Protein Structure, Secondary; Pyridazines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2012
In intact islets interstitial GABA activates GABA(A) receptors that generate tonic currents in α-cells.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: Animals; gamma-Aminobutyric Acid; Gene Expression Regulation; Glucagon-Secreting Cells; Ion Channel Gating; Pentobarbital; Protein Subunits; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2013
Persistent GABAA/C responses to gabazine, taurine and beta-alanine in rat hypoglossal motoneurons.
    Neuroscience, 2016, 08-25, Volume: 330

    Topics: Animals; beta-Alanine; Bicuculline; Brain Stem; Central Nervous System Agents; Chlorine; GABA Agents; Hypoglossal Nerve; Midazolam; Motor Neurons; Neuroprotective Agents; Patch-Clamp Techniques; Pentobarbital; Phosphinic Acids; Pregnanolone; Pyridazines; Pyridines; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Strychnine; Taurine; Tissue Culture Techniques

2016