Page last updated: 2024-09-02

sr 95531 and n-methylaspartate

sr 95531 has been researched along with n-methylaspartate in 19 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(n-methylaspartate)
Trials
(n-methylaspartate)
Recent Studies (post-2010) (n-methylaspartate)
610020910,408591,902

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)n-methylaspartate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)5.175

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (5.26)18.2507
2000's6 (31.58)29.6817
2010's12 (63.16)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chuang, DM; Yu, O1
Bourguignon, JP; Gérard, A; Lebrethon, MC; Parent, AS1
Balthazart, J; Cornil, CA; Motte, P; Seutin, V1
Bensen, AL; Bromberg, DA; Overstreet Wadiche, L; Westbrook, GL1
Lachamp, PM; Liu, SJ; Liu, Y1
Blankenship, AG; Copenhagen, DR; Edwards, RH; Feller, MB; Ford, KJ; Johnson, J; Seal, RP1
Bannai, H; Inoue, T; Launey, T; Lévi, S; Mikoshiba, K; Racine, V; Schweizer, C; Sibarita, JB; Triller, A1
Martin, LJ; Orser, BA; Paulsen, O; Salter, MW; Vargas-Caballero, M1
Dergacheva, O; Jameson, H; Lovett-Barr, MR; Mendelowitz, D; Wang, X1
Gire, DH; Pandipati, S; Schoppa, NE1
Li, WC; Roberts, A; Soffe, SR1
Felmy, F; Grothe, B; Meyer, EM; Porres, CP1
Kalinina, NI; Kurchavyĭ, GG; Veselkin, NP1
Caspary, DM; Llano, DA; Turner, J1
Kawabe, K; Kawabe, T; Sapru, HN1
Chu, CP; Liu, H; Qiu, DL; Sun, L; Zhao, GY; Zhao, SN1
Chitravanshi, VC; Kawabe, K; Sapru, HN1
Aimone, JB; Dieni, CV; Kuo, CT; Overstreet-Wadiche, L; Panichi, R; Wadiche, JI1
Chen, L; Huang, M; Jiang, B; Li, S; Li, Y; Wang, L; Wang, X; Yang, Y; Zhang, X1

Other Studies

19 other study(ies) available for sr 95531 and n-methylaspartate

ArticleYear
Long-term GABA treatment elicits supersensitivity of quisqualate-preferring metabotropic glutamate receptor in cultured rat cerebellar neurons.
    Journal of neurochemistry, 1993, Volume: 61, Issue:2

    Topics: Animals; Baclofen; Carbachol; Cells, Cultured; Cerebellum; Drug Tolerance; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kainic Acid; N-Methylaspartate; Neurons; Potassium Chloride; Pyridazines; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glutamate

1993
Factors accounting for perinatal occurrence of pulsatile gonadotropin-releasing hormone secretion in vitro in rats.
    Biology of reproduction, 2005, Volume: 72, Issue:1

    Topics: Animals; Dinoprostone; Embryo, Mammalian; Feedback, Physiological; Female; GABA Antagonists; Glutamates; Gonadotropin-Releasing Hormone; In Vitro Techniques; Labor, Obstetric; Male; N-Methylaspartate; Oxytocin; Pregnancy; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate

2005
Electrophysiological and neurochemical characterization of neurons of the medial preoptic area in Japanese quail (Coturnix japonica).
    Brain research, 2004, Dec-17, Volume: 1029, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Aromatase; Coturnix; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Isonicotinic Acids; Kainic Acid; Male; N-Methylaspartate; Neurons; Norepinephrine; Preoptic Area; Pyridazines; Sympathomimetics

2004
GABAergic signaling to newborn neurons in dentate gyrus.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Age Factors; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Blotting, Northern; Cells, Cultured; Dentate Gyrus; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Flow Cytometry; Fluorescent Antibody Technique; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Green Fluorescent Proteins; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; N-Methylaspartate; Neural Inhibition; Neurons; Parvalbumins; Patch-Clamp Techniques; Pro-Opiomelanocortin; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Signal Transduction; Synapses; Synaptic Transmission; Zolpidem

2005
Glutamatergic modulation of cerebellar interneuron activity is mediated by an enhancement of GABA release and requires protein kinase A/RIM1alpha signaling.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Jan-14, Volume: 29, Issue:2

    Topics: Action Potentials; Animals; Animals, Newborn; Cerebellum; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; GTP-Binding Proteins; In Vitro Techniques; Interneurons; Long-Term Potentiation; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methylaspartate; Patch-Clamp Techniques; Pyridazines; Signal Transduction; Synaptic Potentials

2009
Synaptic and extrasynaptic factors governing glutamatergic retinal waves.
    Neuron, 2009, Apr-30, Volume: 62, Issue:2

    Topics: Amino Acid Transport Systems, Acidic; Animals; Animals, Newborn; Aspartic Acid; Calcium; Dihydro-beta-Erythroidine; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; In Vitro Techniques; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Biological; N-Methylaspartate; Neural Inhibition; Nicotinic Antagonists; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Retinal Ganglion Cells; Synapses; Synaptic Transmission; Time Factors; Valine; Vesicular Glutamate Transport Protein 1

2009
Activity-dependent tuning of inhibitory neurotransmission based on GABAAR diffusion dynamics.
    Neuron, 2009, Jun-11, Volume: 62, Issue:5

    Topics: Animals; Animals, Newborn; Biotinylation; Calcineurin; Calcium; Carrier Proteins; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Hippocampus; Inhibitory Postsynaptic Potentials; Long-Term Synaptic Depression; Membrane Proteins; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Protein Transport; Pyridazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA-A; Signal Transduction; Synapsins; Tissue Culture Techniques

2009
alpha5 Subunit-containing GABA(A) receptors mediate a slowly decaying inhibitory synaptic current in CA1 pyramidal neurons following Schaffer collateral activation.
    Neuropharmacology, 2010, Volume: 58, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; CA1 Region, Hippocampal; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Imidazoles; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Knockout; N-Methylaspartate; Neural Inhibition; Neural Pathways; Pyramidal Cells; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Zolpidem

2010
The lateral paragigantocellular nucleus modulates parasympathetic cardiac neurons: a mechanism for rapid eye movement sleep-dependent changes in heart rate.
    Journal of neurophysiology, 2010, Volume: 104, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Biophysics; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Heart; Heart Rate; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Medulla Oblongata; N-Methylaspartate; Neurons; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Sleep, REM; Time Factors; Vagus Nerve; Valine

2010
Adrenergic receptor-mediated disinhibition of mitral cells triggers long-term enhancement of synchronized oscillations in the olfactory bulb.
    Journal of neurophysiology, 2010, Volume: 104, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Agonists; Animals; Animals, Newborn; Bicuculline; Biological Clocks; Biophysical Phenomena; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; N-Methylaspartate; Neurons; Norepinephrine; Olfactory Bulb; Pyridazines; Quinoxalines; Rats; Receptors, Adrenergic; Valine

2010
Specific brainstem neurons switch each other into pacemaker mode to drive movement by activating NMDA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Dec-08, Volume: 30, Issue:49

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Biological Clocks; Brain Stem; Cadmium Chloride; Dihydro-beta-Erythroidine; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Glycyrrhetinic Acid; Humans; In Vitro Techniques; Larva; Models, Biological; Movement; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Periodicity; Pyridazines; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Swimming; Xenopus

2010
NMDA currents modulate the synaptic input-output functions of neurons in the dorsal nucleus of the lateral lemniscus in Mongolian gerbils.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Mar-23, Volume: 31, Issue:12

    Topics: Action Potentials; Animals; Brain Stem; Calcium; Calcium Channels; Calcium Signaling; Electrophysiological Phenomena; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; gamma-Aminobutyric Acid; Gerbillinae; In Vitro Techniques; Male; Membranes; N-Methylaspartate; Neurons; Pyridazines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

2011
[Inhibitory regulation of glutamate receptors in the frog motoneuron].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2012, Volume: 98, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Evoked Potentials; Excitatory Amino Acids; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Kainic Acid; Microelectrodes; Motor Neurons; N-Methylaspartate; Organ Culture Techniques; Poisons; Pyridazines; Rana ridibunda; Receptors, Ionotropic Glutamate; Spinal Cord; Strychnine

2012
Diminished cortical inhibition in an aging mouse model of chronic tinnitus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Nov-14, Volume: 32, Issue:46

    Topics: Acoustic Stimulation; Aging; Animals; Auditory Cortex; Auditory Threshold; Cerebral Cortex; Chronic Disease; Disease Models, Animal; Evoked Potentials, Auditory, Brain Stem; Flavoproteins; GABA Antagonists; gamma-Aminobutyric Acid; Hearing Loss, Noise-Induced; Male; Mice; Mice, Inbred CBA; N-Methylaspartate; Neural Inhibition; Pyridazines; Receptors, GABA-A; Reflex, Startle; Tinnitus

2012
Tonic γ-aminobutyric acid-ergic activity in the hypothalamic arcuate nucleus is attenuated in the spontaneously hypertensive rat.
    Hypertension (Dallas, Tex. : 1979), 2013, Volume: 62, Issue:2

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Arterial Pressure; Baroreflex; Denervation; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Heart Rate; Hypertension; Male; N-Methylaspartate; Neuropeptide Y; Pyridazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY

2013
N-methyl-d-aspartate inhibits cerebellar Purkinje cell activity via the excitation of molecular layer interneurons under in vivo conditions in mice.
    Brain research, 2014, Apr-29, Volume: 1560

    Topics: Action Potentials; Anesthetics, Intravenous; Animals; Biotin; Cell Membrane; Cerebellum; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; GABA-A Receptor Antagonists; Interneurons; Mice, Inbred ICR; Microelectrodes; N-Methylaspartate; Purkinje Cells; Pyridazines; Receptors, N-Methyl-D-Aspartate; Tissue Culture Techniques; Urethane

2014
GABA and glycine receptors in the nucleus ambiguus mediate tachycardia elicited by chemical stimulation of the hypothalamic arcuate nucleus.
    American journal of physiology. Heart and circulatory physiology, 2015, Jul-01, Volume: 309, Issue:1

    Topics: Animals; Arcuate Nucleus of Hypothalamus; GABA Antagonists; GABA-A Receptor Agonists; Glycine Agents; Heart; Male; Medulla Oblongata; Microinjections; Muscimol; N-Methylaspartate; Pyridazines; Rats, Wistar; Receptors, GABA-A; Receptors, Glycine; Stimulation, Chemical; Strychnine; Tachycardia

2015
Low excitatory innervation balances high intrinsic excitability of immature dentate neurons.
    Nature communications, 2016, Apr-20, Volume: 7

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Dentate Gyrus; Electric Stimulation; Entorhinal Cortex; Excitatory Postsynaptic Potentials; Female; Gene Expression; Integrases; Male; Mice; Mice, Transgenic; Microtomy; N-Methylaspartate; Nestin; Neural Inhibition; Neural Stem Cells; Neurogenesis; Neuronal Plasticity; Neurons; Patch-Clamp Techniques; Pyridazines; Synapses; Tamoxifen; Tissue Culture Techniques

2016
Inhibition of Cdk5 rejuvenates inhibitory circuits and restores experience-dependent plasticity in adult visual cortex.
    Neuropharmacology, 2018, Volume: 128

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cyclin-Dependent Kinase 5; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; N-Methylaspartate; Neuronal Plasticity; Neurons; Phosphopyruvate Hydratase; Piperidines; Pyridazines; Sensory Deprivation; Visual Cortex; Visual Pathways

2018