sr 95531 has been researched along with isoxazoles in 20 studies
| Studies (sr 95531) | Trials (sr 95531) | Recent Studies (post-2010) (sr 95531) | Studies (isoxazoles) | Trials (isoxazoles) | Recent Studies (post-2010) (isoxazoles) |
|---|---|---|---|---|---|
| 610 | 0 | 209 | 8,633 | 900 | 3,337 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 5 (25.00) | 18.2507 |
| 2000's | 8 (40.00) | 29.6817 |
| 2010's | 7 (35.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Andre, JM; Boulanger, T; Durant, F; Hoffmann, R; Rognan, D; Vercauteren, DP; Wermuth, CG | 1 |
| Heinricher, MM; Kaplan, HJ | 1 |
| Catt, KJ; Stojilković, SS; Virmani, MA | 1 |
| Balcar, VJ; Dreher, B | 1 |
| Dzubay, JA; Jones, MV; Sahara, Y; Westbrook, GL | 1 |
| Maksay, G; McKernan, R | 1 |
| Ebert, B; Fjalland, B; Hansen, SL; Kristiansen, U | 1 |
| Jonas, P; Jones, MV; Sahara, Y; Westbrook, GL | 1 |
| Frølund, B; Jørgensen, AT; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Tagmose, L | 1 |
| Babich, M; Branda, EM; Elfline, GS; Quock, RM | 1 |
| Ebert, B; Frølund, B; Jensen, LS; Kehler, J; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Storustovu, SI | 1 |
| Park, JB; Skalska, S; Son, S; Stern, JE | 1 |
| Amar, M; Baux, G; Fossier, P; Le Roux, N; Moreau, A | 1 |
| Dretchen, KL; Gillis, RA; Herman, MA; Sahibzada, N; Vicini, S | 1 |
| Branco, T; Chadderton, P; Duguid, I; Häusser, M; London, M | 1 |
| Caspary, DM; Duque, D; Malmierca, MS | 1 |
| Corbin, JG; Huntsman, MM; Martin, BS | 1 |
| Gangadharan, G; Hwang, EM; Lee, B; Lee, S; Paydar, A; Shin, HS | 1 |
| Finn, DA; Helms, M; Jensen, J; Kaplan, JS; Nipper, MA; Richardson, BD; Rossi, DJ | 1 |
| Browning, KN; McMenamin, CA; Travagli, RA | 1 |
20 other study(ies) available for sr 95531 and isoxazoles
| Article | Year |
|---|---|
Structure and molecular modeling of GABAA receptor antagonists.
Topics: Alkaloids; Androstanes; Azasteroids; Azepines; Bicuculline; Crystallization; Dibenzazepines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Isoxazoles; Lactones; Models, Molecular; Molecular Conformation; Molecular Structure; Piperidines; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship; Tubocurarine; X-Ray Diffraction | 1992 |
GABA-mediated inhibition in rostral ventromedial medulla: role in nociceptive modulation in the lightly anesthetized rat.
Topics: Analgesics; Anesthesia; Animals; Bicuculline; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Medulla Oblongata; Microinjections; Nociceptors; Pyridazines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Receptors, Glycine; Receptors, Neurotransmitter | 1991 |
Stimulation of luteinizing hormone release by gamma-aminobutyric acid (GABA) agonists: mediation by GABAA-type receptors and activation of chloride and voltage-sensitive calcium channels.
Topics: Amino Acid Sequence; Animals; Baclofen; Calcium Channels; Cells, Cultured; Chloride Channels; Chlorides; Female; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Isoxazoles; Luteinizing Hormone; Membrane Proteins; Molecular Sequence Data; Muscimol; Nifedipine; Pituitary Gland, Anterior; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex | 1990 |
Defining affinity with the GABAA receptor.
Topics: Animals; Animals, Newborn; beta-Alanine; Cells, Cultured; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Hippocampus; Isoxazoles; Ligands; Muscimol; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Receptors, GABA-A | 1998 |
Entropy as the predominant driving force of binding to human recombinant alpha(x)beta(3)gamma(2) GABA(A) receptors.
Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Entropy; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; L Cells; Membranes; Mice; Muscimol; Piperidines; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Temperature; Tritium | 2001 |
Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Cerebral Cortex; Electrophysiology; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Receptors, GABA-A; Xenopus laevis | 2001 |
Microscopic kinetics and energetics distinguish GABA(A) receptor agonists from antagonists.
Topics: Animals; Brain; Diffusion; Electrophysiology; Energy Metabolism; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Inhibitory Concentration 50; Isoxazoles; Kinetics; Muscimol; Phosphinic Acids; Protein Binding; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2001 |
Design and synthesis of a new series of 4-alkylated 3-isoxazolol GABA A antagonists.
Topics: Alkylation; Animals; Binding Sites; Drug Design; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; Humans; Isoxazoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Pyridazines; Receptors, GABA; Receptors, GABA-A; Structure-Activity Relationship | 2003 |
Antagonism by NOS inhibition of the behavioral effects of benzodiazepine and GABAA receptor agonists in the mouse elevated plus-maze.
Topics: Animals; Anxiety; Behavior, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; GABA Agonists; GABA-A Receptor Agonists; Injections, Intraventricular; Isoxazoles; Male; Mice; Nitric Oxide Synthase; Nitroarginine; Pyrazoles; Pyridazines | 2004 |
4-aryl-5-(4-piperidyl)-3-isoxazolol GABAA antagonists: synthesis, pharmacology, and structure-activity relationships.
Topics: Animals; Female; GABA-A Receptor Antagonists; Humans; In Vitro Techniques; Isoxazoles; Models, Molecular; Molecular Conformation; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Structure-Activity Relationship; Xenopus | 2007 |
Dual GABAA receptor-mediated inhibition in rat presympathetic paraventricular nucleus neurons.
Topics: Animals; Bicuculline; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Isoxazoles; Male; Medulla Oblongata; Neural Inhibition; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Synapses | 2007 |
Impaired GABAergic transmission disrupts normal homeostatic plasticity in rat cortical networks.
Topics: Animals; Cerebral Cortex; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Homeostasis; Isoxazoles; Long-Term Potentiation; Models, Neurological; Neural Inhibition; Neuronal Plasticity; Organ Culture Techniques; Pyramidal Cells; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission | 2008 |
Tonic GABAA receptor conductance in medial subnucleus of the tractus solitarius neurons is inhibited by activation of μ-opioid receptors.
Topics: Analgesics, Opioid; Animals; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Opioid, mu; Sodium Channel Blockers; Solitary Nucleus; Tetrodotoxin | 2012 |
Tonic inhibition enhances fidelity of sensory information transmission in the cerebellar cortex.
Topics: Action Potentials; Afferent Pathways; Animals; Animals, Newborn; Cerebellar Cortex; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Functional Laterality; GABA Agonists; GABA Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Isoxazoles; Ketamine; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Physical Stimulation; Pyridazines; Rats; Rats, Sprague-Dawley; Sensation; Vibrissae | 2012 |
Modulation of stimulus-specific adaptation by GABA(A) receptor activation or blockade in the medial geniculate body of the anaesthetized rat.
Topics: Acoustic Stimulation; Adaptation, Physiological; Anesthesia, General; Animals; GABA Antagonists; GABA-A Receptor Agonists; GABAergic Neurons; Geniculate Bodies; Isoxazoles; Male; Pyridazines; Rats; Rats, Inbred F344; Receptors, GABA-A | 2014 |
Deficient tonic GABAergic conductance and synaptic balance in the fragile X syndrome amygdala.
Topics: Amygdala; Animals; Excitatory Postsynaptic Potentials; Feedback, Physiological; Fragile X Mental Retardation Protein; Fragile X Syndrome; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABAergic Neurons; Inhibitory Postsynaptic Potentials; Isoxazoles; Mice; Phthalazines; Protein Subunits; Pyridazines; Receptors, GABA-A; Synapses; Triazoles | 2014 |
Extrasynaptic GABAA receptors in mediodorsal thalamic nucleus modulate fear extinction learning.
Topics: Animals; Extinction, Psychological; Fear; Integrases; Isoxazoles; Male; Mediodorsal Thalamic Nucleus; Mice; Mice, Knockout; Pyridazines; Receptors, GABA-A; Synapses; Transfection | 2014 |
Pharmacologically Counteracting a Phenotypic Difference in Cerebellar GABAA Receptor Response to Alcohol Prevents Excessive Alcohol Consumption in a High Alcohol-Consuming Rodent Genotype.
Topics: Alcohol Drinking; Analysis of Variance; Animals; Animals, Newborn; Cerebellum; Dose-Response Relationship, Drug; Ethanol; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Genotype; In Vitro Techniques; Isoxazoles; Kynurenic Acid; Locomotion; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Patch-Clamp Techniques; Pyridazines; Receptors, GABA-A; Species Specificity; Sucrose | 2016 |
Perinatal high fat diet increases inhibition of dorsal motor nucleus of the vagus neurons regulating gastric functions.
Topics: Animals; Bicuculline; Brain Stem; Diet, High-Fat; GABA Agonists; GABA Antagonists; Gastrointestinal Motility; Isoxazoles; Male; Neural Inhibition; Neurons; Pyridazines; Rats, Sprague-Dawley; Vagus Nerve | 2018 |