Page last updated: 2024-09-02

sr 95531 and isoguvacine

sr 95531 has been researched along with isoguvacine in 16 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(isoguvacine)
Trials
(isoguvacine)
Recent Studies (post-2010) (isoguvacine)
6100209178030

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (43.75)18.2507
2000's6 (37.50)29.6817
2010's3 (18.75)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Astier, H; Roussel, JP1
Balcar, VJ1
Feltz, P; Zhang, ZW1
Balcar, VJ; Dreher, B1
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ1
Hammond, DL; McGowan, MK1
Ashworth-Preece, M; Jarrott, B; Krstew, E; Lawrence, AJ1
Ebert, B; Fjalland, B; Hansen, SL; Kristiansen, U1
Balthazart, J; Cornil, CA; Motte, P; Seutin, V1
Holmes, GL; Isaev, D; Isaeva, E; Khazipov, R1
Ennis, M; Hayar, A1
Gao, J; Gao, XY; Liao, ZH; Shi, Z; Wang, W; Zhong, MK; Zhou, LM; Zhu, GQ1
Garcia-Rill, E; Ye, M1
Arisi, I; Brandi, R; Capsoni, S; Cattaneo, A; Cherubini, E; D'Onofrio, M; Franzot, J; Lagostena, L; Rosato-Siri, M1
Cai, L; Ji, F; Lu, W; Ma, TF; Ren, SQ; Tian, T; Zhang, N; Zhao, XL1
Chen, Q; Ding, L; Gao, R; Gao, XY; Kang, YM; Li, YH; Xiong, XQ; Zhu, GQ1

Other Studies

16 other study(ies) available for sr 95531 and isoguvacine

ArticleYear
Involvement of dihydropyridine-sensitive calcium channels in the GABAA potentiation of TRH-induced TSH release.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; GTP-Binding Proteins; In Vitro Techniques; Isonicotinic Acids; Male; Nifedipine; omega-Conotoxins; Peptides, Cyclic; Pertussis Toxin; Pituitary Gland; Pyridazines; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella

1990
Presence of a highly efficient "binding" to bacterial contamination can distort data from binding studies.
    Neurochemical research, 1990, Volume: 15, Issue:12

    Topics: Animals; Cats; Cerebral Cortex; GABA Antagonists; gamma-Aminobutyric Acid; Gram-Positive Bacteria; Isonicotinic Acids; Muscimol; Nipecotic Acids; Proline; Pyridazines; Radioligand Assay; Receptors, GABA-A; Tritium

1990
Bicuculline blocks nicotinic acetylcholine response in isolated intermediate lobe cells of the pig.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; GABA Antagonists; In Vitro Techniques; Isonicotinic Acids; Membrane Potentials; Pyridazines; Receptors, Nicotinic; Solutions; Swine

1991
Neurochemical correlates of gamma-aminobutyrate (GABA) inhibition in cat visual cortex.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Baclofen; Calcium; Cats; Cell Membrane; Female; GABA Antagonists; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Neurons; Potassium; Pyridazines; Receptors, GABA-A; Visual Cortex

1990
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
    Brain research, 1994, Oct-03, Volume: 659, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1994
Antinociception produced by microinjection of L-glutamate into the ventromedial medulla of the rat: mediation by spinal GABAA receptors.
    Brain research, 1993, Aug-20, Volume: 620, Issue:1

    Topics: Animals; Behavior, Animal; Bicuculline; Diazepam; GABA Antagonists; Glutamates; Glutamic Acid; Injections, Spinal; Isonicotinic Acids; Male; Medulla Oblongata; Microinjections; Nociceptors; Pyridazines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, GABA; Skin Temperature; Spinal Cord

1993
Functional GABAA receptors on rat vagal afferent neurones.
    British journal of pharmacology, 1997, Volume: 120, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Autoradiography; Bicuculline; Brain Stem; Denervation; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Image Processing, Computer-Assisted; In Vitro Techniques; Isonicotinic Acids; Male; Neurons, Afferent; Nodose Ganglion; Presynaptic Terminals; Pyridazines; Rats; Rats, Inbred WKY; Receptors, GABA-A; Vagus Nerve

1997
Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
    British journal of pharmacology, 2001, Volume: 133, Issue:4

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Cerebral Cortex; Electrophysiology; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Receptors, GABA-A; Xenopus laevis

2001
Electrophysiological and neurochemical characterization of neurons of the medial preoptic area in Japanese quail (Coturnix japonica).
    Brain research, 2004, Dec-17, Volume: 1029, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Aromatase; Coturnix; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Isonicotinic Acids; Kainic Acid; Male; N-Methylaspartate; Neurons; Norepinephrine; Preoptic Area; Pyridazines; Sympathomimetics

2004
Anticonvulsant action of GABA in the high potassium-low magnesium model of ictogenesis in the neonatal rat hippocampus in vivo and in vitro.
    Journal of neurophysiology, 2005, Volume: 94, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Bicuculline; Disease Models, Animal; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Lipoproteins; Magnesium; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Pyridazines; Rats; Seizures

2005
Endogenous GABA and glutamate finely tune the bursting of olfactory bulb external tufted cells.
    Journal of neurophysiology, 2007, Volume: 98, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Neurons; Olfactory Bulb; Pyridazines; Rats; Rats, Sprague-Dawley; Valine

2007
Regulation of cardiac sympathetic afferent reflex by GABA(A) and GABA(B) receptors in paraventricular nucleus in rats.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Baclofen; Bradykinin; Capsaicin; GABA Agonists; GABA Antagonists; Heart; Isonicotinic Acids; Kidney; Male; Neurons, Afferent; Organophosphorus Compounds; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Reflex; Sensory System Agents; Sympathetic Nervous System; Vigabatrin

2008
Potentiating effect of eszopiclone on GABA(A) receptor-mediated responses in pedunculopontine neurons.
    Sleep, 2009, Volume: 32, Issue:7

    Topics: Anesthetics, Local; Animals; Animals, Newborn; Azabicyclo Compounds; Drug Synergism; Electric Stimulation; Eszopiclone; GABA Agonists; GABA Antagonists; Hypnotics and Sedatives; Isonicotinic Acids; Neurons; Patch-Clamp Techniques; Pedunculopontine Tegmental Nucleus; Piperazines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tetrodotoxin; Time Factors

2009
In the adult hippocampus, chronic nerve growth factor deprivation shifts GABAergic signaling from the hyperpolarizing to the depolarizing direction.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antibodies, Neutralizing; Biophysics; Bumetanide; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Hippocampus; In Vitro Techniques; Ion Channel Gating; Isonicotinic Acids; K Cl- Cotransporters; Mice; Mice, Transgenic; Nerve Growth Factor; Neurons; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Receptors, Nicotinic; RNA, Messenger; Sodium Potassium Chloride Symporter Inhibitors; Symporters

2010
Regulation of spike timing-dependent plasticity of olfactory inputs in mitral cells in the rat olfactory bulb.
    PloS one, 2012, Volume: 7, Issue:4

    Topics: Action Potentials; Animals; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABAergic Neurons; In Vitro Techniques; Isonicotinic Acids; Neural Inhibition; Neuronal Plasticity; Neurons; Olfactory Bulb; Olfactory Nerve; Pyridazines; Rats; Rats, Sprague-Dawley

2012
GABA in Paraventricular Nucleus Regulates Adipose Afferent Reflex in Rats.
    PloS one, 2015, Volume: 10, Issue:8

    Topics: Adipose Tissue, White; Afferent Pathways; Animals; Baclofen; gamma-Aminobutyric Acid; Isonicotinic Acids; Kidney; Male; Organophosphorus Compounds; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Vigabatrin

2015