Page last updated: 2024-09-02

sr 95531 and flunitrazepam

sr 95531 has been researched along with flunitrazepam in 13 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(flunitrazepam)
Trials
(flunitrazepam)
Recent Studies (post-2010) (flunitrazepam)
61002092,697298130

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)flunitrazepam (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0016
GABA theta subunitRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0016

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.69)18.7374
1990's10 (76.92)18.2507
2000's2 (15.38)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Banerjee, PK; Depaulis, A; Hechler, V; Snead, OC; Vergnes, M1
Harris, RA; Leidenheimer, NJ1
Scarth, BA; Shaw, C1
Farb, DH; Farrant, M; Roca, DJ; Rozenberg, I1
Buck, KJ; Harris, RA1
Ikeda, M; Knapp, RJ; Malatynska, E; Yamamura, HI1
Bormann, J; Feigenspan, A1
Alicke, B; Schwartz-Bloom, RD1
Brett, RR; Pratt, JA1
Barnes, EM; Baumgartner, BJ; Tehrani, MH1
Chéry, N; de Koninck, Y1
Bouairi, E; Gorini, C; Kamendi, H; Mendelowitz, D; Wang, X1
Jembrek, MJ; Pericić, D; Strac, DS; Vlainić, J1

Other Studies

13 other study(ies) available for sr 95531 and flunitrazepam

ArticleYear
The GABAA receptor complex in experimental absence seizures in rat: an autoradiographic study.
    Neuroscience letters, 1992, Jun-08, Volume: 140, Issue:1

    Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Epilepsy, Absence; Flunitrazepam; GABA-A Receptor Antagonists; Ion Channels; Ionophores; Male; Membrane Proteins; Muscimol; Organ Specificity; Pyramidal Tracts; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Tritium

1992
A transient osmotic permeabilization method for the introduction of impermeant molecules into functional brain membrane vesicles.
    Journal of neuroscience methods, 1991, Volume: 40, Issue:2-3

    Topics: Alkaline Phosphatase; Animals; Capsules; Carbon Radioisotopes; Cell Membrane; Cell Membrane Permeability; Chloride Channels; Chlorides; Chlorine; Concanavalin A; Flunitrazepam; Hypotonic Solutions; Membrane Proteins; Mice; Mice, Inbred ICR; Muscimol; Pyridazines; Radioisotope Dilution Technique; Radioisotopes; Receptors, Concanavalin A; Receptors, GABA-A; Sucrose; Tritium

1991
Characterization and differential regulation of GABAA and benzodiazepine receptors in rat neocortex.
    Brain research. Molecular brain research, 1991, Volume: 11, Issue:3-4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cerebral Cortex; Clonazepam; Down-Regulation; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Kinetics; Male; Muscimol; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium; Veratridine

1991
Chronic agonist exposure induces down-regulation and allosteric uncoupling of the gamma-aminobutyric acid/benzodiazepine receptor complex.
    Molecular pharmacology, 1990, Volume: 37, Issue:1

    Topics: Allosteric Regulation; Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chick Embryo; Down-Regulation; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A

1990
Benzodiazepine agonist and inverse agonist actions on GABAA receptor-operated chloride channels. II. Chronic effects of ethanol.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Brain; Carbolines; Chloride Channels; Chlorides; Convulsants; Ethanol; Flunitrazepam; GABA Antagonists; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Pyridazines; Receptors, GABA-A; Substance Withdrawal Syndrome; Tritium

1990
Amoxapine inhibition of GABA-stimulated chloride conductance: investigations of potential sites of activity.
    Life sciences, 1989, Volume: 45, Issue:20

    Topics: Amoxapine; Animals; Cerebral Cortex; Chlorides; Dibenzoxazepines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Antagonists; Ligands; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction

1994
Rapid down-regulation of GABAA receptors in the gerbil hippocampus following transient cerebral ischemia.
    Journal of neurochemistry, 1995, Volume: 65, Issue:6

    Topics: Animals; Autoradiography; Down-Regulation; Flunitrazepam; Gerbillinae; Hippocampus; Ischemic Attack, Transient; Male; Pyridazines; Receptors, GABA-A; Tissue Distribution

1995
Changes in benzodiazepine-GABA receptor coupling in an accumbens-habenula circuit after chronic diazepam treatment.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Autoradiography; Binding, Competitive; Diazepam; Drug Implants; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraperitoneal; Male; Maze Learning; Nucleus Accumbens; Pyridazines; Rats; Receptors, GABA-A; Thalamus

1995
Clathrin-coated vesicles from bovine brain contain uncoupled GABAA receptors.
    Brain research, 1997, Nov-21, Volume: 776, Issue:1-2

    Topics: Allosteric Site; Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chloride Channels; Clathrin; Coated Vesicles; Convulsants; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Ligands; Pyridazines; Receptors, GABA-A; Sulfur Radioisotopes; Synaptic Membranes; Tritium

1997
Junctional versus extrajunctional glycine and GABA(A) receptor-mediated IPSCs in identified lamina I neurons of the adult rat spinal cord.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Sep-01, Volume: 19, Issue:17

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Evoked Potentials; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Strychnine; Sucrose; Tetrodotoxin

1999
Multiple types of GABAA receptors mediate inhibition in brain stem parasympathetic cardiac neurons in the nucleus ambiguus.
    Journal of neurophysiology, 2006, Volume: 96, Issue:6

    Topics: Animals; Brain Stem; Choline O-Acetyltransferase; Efferent Pathways; Electrophysiology; Excitatory Postsynaptic Potentials; Flunitrazepam; GABA Antagonists; GABA Modulators; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heart; Immunohistochemistry; In Vitro Techniques; Medulla Oblongata; Neurons; Parasympathetic Nervous System; Patch-Clamp Techniques; Pharyngeal Muscles; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptic Transmission; Vagus Nerve

2006
Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Diazepam; Flumazenil; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Protein Subunits; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Transfection; Up-Regulation

2007