Page last updated: 2024-09-02

sr 95531 and desoxycorticosterone

sr 95531 has been researched along with desoxycorticosterone in 5 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(desoxycorticosterone)
Trials
(desoxycorticosterone)
Recent Studies (post-2010) (desoxycorticosterone)
61002097,58852284

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)desoxycorticosterone (IC50)
Solute carrier family 22 member 3Rattus norvegicus (Norway rat)8.4
Solute carrier family 22 member 2Rattus norvegicus (Norway rat)1.9

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's2 (40.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Acosta-Burruel, M; Goodnough, DB; Hawkinson, JE; Kimbrough, CL; Wood, PL1
Biggio, G; Concas, A; Marino, G; Minei, R; Mostallino, MC; Pierobon, P; Porcu, P1
Andersson, A; Asztely, F; Heeroma, JH; McEvoy, AW; Rydenhag, B; Scimemi, A; Strandberg, J; Thom, M; Walker, MC1
Amin, J; Hadley, SH1
Bayliss, DA; Chen, X; Kapur, J; Schwartz, LC; Shu, S; Sun, C1

Other Studies

5 other study(ies) available for sr 95531 and desoxycorticosterone

ArticleYear
Steroid inhibition of [3H]SR 95531 binding to the GABAA recognition site.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Cell Membrane; Cerebral Cortex; Desoxycorticosterone; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pregnanolone; Pregnenolone; Protein Binding; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Steroids

1996
Modulation of gamma-aminobutyric acid (GABA) receptors and the feeding response by neurosteroids in Hydra vulgaris.
    Neuroscience, 1998, Volume: 85, Issue:3

    Topics: Anesthetics; Animals; Anti-Anxiety Agents; Bicuculline; Carbolines; Cerebral Cortex; Chemoreceptor Cells; Clonazepam; Desoxycorticosterone; Diazepam; Feeding Behavior; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Glutathione; Hydra; Neurotransmitter Agents; Pregnanolone; Progesterone; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1998
Tonic GABA(A) receptor-mediated currents in human brain.
    The European journal of neuroscience, 2006, Volume: 24, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Dentate Gyrus; Desoxycorticosterone; Electrophysiology; GABA Antagonists; Humans; Interneurons; Membrane Potentials; Neurons; Picrotoxin; Pyridazines; Receptors, GABA-A

2006
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities.
    The Journal of physiology, 2007, Jun-15, Volume: 581, Issue:Pt 3

    Topics: Action Potentials; Animals; beta-Alanine; Bicuculline; Crotonates; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Furosemide; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Microinjections; Mutation; Neural Inhibition; Neurons; Oocytes; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Sesterterpenes; Taurine; Xenopus laevis; Zinc

2007
Homeostatic regulation of synaptic excitability: tonic GABA(A) receptor currents replace I(h) in cortical pyramidal neurons of HCN1 knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Desoxycorticosterone; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Agents; Homeostasis; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Neurological; Patch-Clamp Techniques; Potassium Channels; Protein Subunits; Pyramidal Cells; Pyridazines; Pyrimidines; Receptors, GABA-A; Sodium Channel Blockers; Synapses; Tetrodotoxin; Up-Regulation; Valine

2010