Page last updated: 2024-09-02

sr 95531 and carbachol

sr 95531 has been researched along with carbachol in 4 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
610020913,91881968

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chuang, DM; Yu, O1
Changeux, JP; Léna, C1
Barbagli, B; Boissard, R; Fort, P; Gervasoni, D; Luppi, PH; Schmidt, MH1
Birabil, CG; Marks, GA; Sachs, OW1

Other Studies

4 other study(ies) available for sr 95531 and carbachol

ArticleYear
Long-term GABA treatment elicits supersensitivity of quisqualate-preferring metabotropic glutamate receptor in cultured rat cerebellar neurons.
    Journal of neurochemistry, 1993, Volume: 61, Issue:2

    Topics: Animals; Baclofen; Carbachol; Cells, Cultured; Cerebellum; Drug Tolerance; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kainic Acid; N-Methylaspartate; Neurons; Potassium Chloride; Pyridazines; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glutamate

1993
Role of Ca2+ ions in nicotinic facilitation of GABA release in mouse thalamus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aconitine; Action Potentials; Alkaloids; Animals; Arousal; Atropine; Azocines; Bacterial Toxins; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Calcium Channel Blockers; Calcium Channels; Carbachol; Cations, Divalent; Cyanobacteria Toxins; Dihydro-beta-Erythroidine; Dimethylphenylpiperazinium Iodide; GABA Antagonists; gamma-Aminobutyric Acid; Ion Transport; Lobeline; Marine Toxins; Mice; Mice, Inbred C57BL; Mice, Knockout; Microcystins; Neurons, Afferent; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium; Pyridazines; Pyridines; Quinolizines; Receptors, GABA-A; Receptors, Nicotinic; Tetrodotoxin; Thalamic Nuclei

1997
The rat ponto-medullary network responsible for paradoxical sleep onset and maintenance: a combined microinjection and functional neuroanatomical study.
    The European journal of neuroscience, 2002, Volume: 16, Issue:10

    Topics: Animals; Bicuculline; Carbachol; Choline O-Acetyltransferase; Cholinergic Agonists; Efferent Pathways; Electroencephalography; Electromyography; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Immunohistochemistry; Kainic Acid; Kynurenic Acid; Male; Medulla Oblongata; Phytohemagglutinins; Pons; Proto-Oncogene Proteins c-fos; Pyridazines; Rats; Rats, Sprague-Dawley; Sleep, REM; Tegmentum Mesencephali; Wakefulness

2002
Blockade of GABA, type A, receptors in the rat pontine reticular formation induces rapid eye movement sleep that is dependent upon the cholinergic system.
    Neuroscience, 2008, Sep-22, Volume: 156, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Bicuculline; Carbachol; Cholinergic Agonists; Cholinergic Fibers; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscarinic Antagonists; Neural Inhibition; Neural Pathways; Pons; Pyridazines; Rats; Rats, Long-Evans; Receptors, GABA-A; Reticular Formation; Sleep, REM; Synaptic Transmission

2008