Page last updated: 2024-09-02

sr 95531 and bis(7)-tacrine

sr 95531 has been researched along with bis(7)-tacrine in 1 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(bis(7)-tacrine)
Trials
(bis(7)-tacrine)
Recent Studies (post-2010) (bis(7)-tacrine)
610020937020

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)bis(7)-tacrine (IC50)
Gamma-aminobutyric acid receptor subunit piHomo sapiens (human)6
Gamma-aminobutyric acid receptor subunit deltaHomo sapiens (human)6
AcetylcholinesteraseElectrophorus electricus (electric eel)0.0007
Amyloid-beta precursor proteinHomo sapiens (human)8.4
CholinesteraseHomo sapiens (human)0.0142
Cytochrome P450 3A4Homo sapiens (human)0.0053
AromataseHomo sapiens (human)2.9
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit beta-1Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)6
AcetylcholinesteraseMus musculus (house mouse)0.0019
AcetylcholinesteraseHomo sapiens (human)0.0011
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiens (human)6
Cytochrome P450 2C19Homo sapiens (human)0.0053
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiens (human)6
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0158
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit alpha-4Homo sapiens (human)6
Beta-secretase 1Homo sapiens (human)7.5
Gamma-aminobutyric acid receptor subunit epsilonHomo sapiens (human)6
CholinesteraseEquus caballus (horse)0.0051
CholinesteraseMus musculus (house mouse)0.0091
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiens (human)6
Nitric oxide synthase, endothelial Rattus norvegicus (Norway rat)2.9
Gamma-aminobutyric acid receptor subunit gamma-1Homo sapiens (human)6
Gamma-aminobutyric acid receptor subunit gamma-3Homo sapiens (human)6
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.1675
Carboxylic ester hydrolase Equus caballus (horse)0.01
Gamma-aminobutyric acid receptor subunit thetaHomo sapiens (human)6

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chebib, M; Johnston, GA1

Reviews

1 review(s) available for sr 95531 and bis(7)-tacrine

ArticleYear
GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology.
    Journal of medicinal chemistry, 2000, Apr-20, Volume: 43, Issue:8

    Topics: Animals; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Ion Channels; Ligands; Receptors, GABA; Receptors, GABA-A; Structure-Activity Relationship

2000