sr 95531 has been researched along with 5-(4-piperidyl)isoxazol-3-ol in 3 studies
Studies (sr 95531) | Trials (sr 95531) | Recent Studies (post-2010) (sr 95531) | Studies (5-(4-piperidyl)isoxazol-3-ol) | Trials (5-(4-piperidyl)isoxazol-3-ol) | Recent Studies (post-2010) (5-(4-piperidyl)isoxazol-3-ol) |
---|---|---|---|---|---|
610 | 0 | 209 | 21 | 0 | 4 |
Protein | Taxonomy | sr 95531 (IC50) | 5-(4-piperidyl)isoxazol-3-ol (IC50) |
---|---|---|---|
Plasminogen | Homo sapiens (human) | 2.8 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Engblom, C; Frølund, B; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Tagmose, L | 1 |
Maksay, G; McKernan, R | 1 |
Ebert, B; Fjalland, B; Hansen, SL; Kristiansen, U | 1 |
3 other study(ies) available for sr 95531 and 5-(4-piperidyl)isoxazol-3-ol
Article | Year |
---|---|
A novel class of potent 3-isoxazolol GABA(A) antagonists: design, synthesis, and pharmacology.
Topics: Animals; Brain; Cells, Cultured; GABA Antagonists; Isoxazoles; Models, Molecular; Muscimol; Neurons; Patch-Clamp Techniques; Piperidines; Radioligand Assay; Rats; Receptors, GABA-A; Structure-Activity Relationship; Synaptic Membranes | 2000 |
Entropy as the predominant driving force of binding to human recombinant alpha(x)beta(3)gamma(2) GABA(A) receptors.
Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Entropy; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; L Cells; Membranes; Mice; Muscimol; Piperidines; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Temperature; Tritium | 2001 |
Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Cerebral Cortex; Electrophysiology; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Receptors, GABA-A; Xenopus laevis | 2001 |