Page last updated: 2024-09-02

sr 95531 and 2-amino-5-phosphonovalerate

sr 95531 has been researched along with 2-amino-5-phosphonovalerate in 52 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(2-amino-5-phosphonovalerate)
Trials
(2-amino-5-phosphonovalerate)
Recent Studies (post-2010) (2-amino-5-phosphonovalerate)
61002094,3931539

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)2-amino-5-phosphonovalerate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.29

Research

Studies (52)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (5.77)18.2507
2000's23 (44.23)29.6817
2010's26 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Mody, I; Soltesz, I1
Ashworth-Preece, M; Jarrott, B; Krstew, E; Lawrence, AJ1
Chéry, N; de Koninck, Y1
Chéry, N; de Koninck, Y; Yu, XH1
Keller, A; Laaris, N1
Auerbach, SB; Tao, R1
Baxi, S; Evans, C; Irnaten, M; Mendelowitz, D; Venkatesan, P; Wang, J; Wang, X1
Christie, JM; Westbrook, GL1
Midtgaard, J; Pinato, G1
Bonhoeffer, T; Finski, A; Lohmann, C1
Holmes, GL; Isaev, D; Isaeva, E; Khazipov, R1
Bevan, MD; Hallworth, NE1
Maher, BJ; Westbrook, GL1
Barski, JJ; Bearzatto, B; Cheron, G; Dan, B; De Saedeleer, C; Dumont, M; Schiffmann, SN; Schwaller, B; Servais, L1
Ghosh, A; Hall, BJ; Hu, SC; Huganir, RL; Ince-Dunn, G; Olson, JM; Ripley, B; Tapscott, SJ1
Pressler, RT; Strowbridge, BW1
Capogna, M; Kerr, AM1
Li, DP; Pan, HL1
Ennis, M; Hayar, A1
Adelman, JP; Lin, MT; Luján, R; Maylie, J; Watanabe, M1
Gutiérrez, R; Heinemann, U; Romo-Parra, H; Treviño, M1
Both, M; Draguhn, A; Lopantsev, V1
Bollmann, JH; Engert, F1
Jean, A; Lebrun, B; Roux, J; Trouslard, J; Wanaverbecq, N1
Blankenship, AG; Copenhagen, DR; Edwards, RH; Feller, MB; Ford, KJ; Johnson, J; Seal, RP1
Kwag, J; Paulsen, O1
Arisi, I; Brandi, R; Capsoni, S; Cattaneo, A; Cherubini, E; D'Onofrio, M; Franzot, J; Lagostena, L; Rosato-Siri, M1
Bayliss, DA; Chen, X; Kapur, J; Schwartz, LC; Shu, S; Sun, C1
Bisogno, T; Brussaard, AB; Burnashev, N; Canto, CB; Di Marzo, V; Heistek, TS; Lodder, JC; Mansvelder, HD; Min, R; Testa-Silva, G1
Dergacheva, O; Jameson, H; Lovett-Barr, MR; Mendelowitz, D; Wang, X1
Gire, DH; Pandipati, S; Schoppa, NE1
Doengi, M; Gaburro, S; Häring, M; Kamprath, K; Lutz, B; Pape, HC; Romo-Parra, H1
Li, WC; Roberts, A; Soffe, SR1
Hall, WC; Isa, T; Lee, PH; Mizuno, F; Phongphanphanee, P; Yanagawa, Y1
Menzler, J; Zeck, G1
Adelman, JP; Maylie, J; Wu, WW1
Charpak, S; De Saint Jan, D; Grandes, P; Najac, M; Reguero, L1
Oswald, MJ; Reynolds, JN; Schulz, JM1
Andresen, MC; Jin, YH1
Kernig, K; Kirschstein, T; Köhling, R; Rohde, M; Würdemann, T1
Bolze, F; Kaifosh, P; Lee, PH; Losonczy, A; Lovett-Barron, M; Nicoud, JF; Sternson, SM; Sun, XH; Turi, GF; Zemelman, BV1
Hou, Q; Jerome, D; Yuan, Q1
Bargas, J; Carrillo-Reid, L; Drucker-Colin, R; Fiordelisio, T; Galarraga, E; López-Huerta, VG; Tapia, D1
Maccaferri, G; Quattrocolo, G1
Becker, D; Deller, T; Diesmann, M; Helias, M; Vlachos, A1
Jackson, MB; Wright, BJ1
Gale, SD; Murphy, GJ1
Anderson, CT; Borges, K; Joshi, A; Middleton, JW; Shepherd, GM; Suter, BA; Tzounopoulos, T1
Cai, R; Caspary, DM1
Crunelli, V; David, F; Lambert, RC; Leresche, N1
Bandara, SB; Llano, DA; Sadowski, RN; Schantz, SL; Slater, BJ; Stebbings, KA1
Johnson, JW; Povysheva, NV1

Other Studies

52 other study(ies) available for sr 95531 and 2-amino-5-phosphonovalerate

ArticleYear
Patch-clamp recordings reveal powerful GABAergic inhibition in dentate hilar neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Chlorides; Electrophysiology; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Neurons; Picrotoxin; Pyridazines; Quinoxalines; Rats; Rats, Wistar; Receptors, GABA-A; Tetrodotoxin; Time Factors

1994
Functional GABAA receptors on rat vagal afferent neurones.
    British journal of pharmacology, 1997, Volume: 120, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Autoradiography; Bicuculline; Brain Stem; Denervation; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Image Processing, Computer-Assisted; In Vitro Techniques; Isonicotinic Acids; Male; Neurons, Afferent; Nodose Ganglion; Presynaptic Terminals; Pyridazines; Rats; Rats, Inbred WKY; Receptors, GABA-A; Vagus Nerve

1997
Junctional versus extrajunctional glycine and GABA(A) receptor-mediated IPSCs in identified lamina I neurons of the adult rat spinal cord.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Sep-01, Volume: 19, Issue:17

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Evoked Potentials; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Strychnine; Sucrose; Tetrodotoxin

1999
Visualization of lamina I of the dorsal horn in live adult rat spinal cord slices.
    Journal of neuroscience methods, 2000, Mar-15, Volume: 96, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Evoked Potentials; Image Processing, Computer-Assisted; Immunohistochemistry; In Vitro Techniques; Male; Microscopy, Video; Patch-Clamp Techniques; Posterior Horn Cells; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Strychnine; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin

2000
Functional independence of layer IV barrels.
    Journal of neurophysiology, 2002, Volume: 87, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Anesthetics, Local; Animals; Electric Stimulation; Excitatory Amino Acid Antagonists; Fluorescent Dyes; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Neurons; Pyridazines; Pyridinium Compounds; Receptors, N-Methyl-D-Aspartate; Somatosensory Cortex; Tetrodotoxin; Vibrissae

2002
Influence of inhibitory and excitatory inputs on serotonin efflux differs in the dorsal and median raphe nuclei.
    Brain research, 2003, Jan-24, Volume: 961, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Animals; Bicuculline; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Motor Activity; Neural Inhibition; Pyridazines; Quinoxalines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Serotonin

2003
Endogenous acetylcholine and nicotine activation enhances GABAergic and glycinergic inputs to cardiac vagal neurons.
    Journal of neurophysiology, 2003, Volume: 89, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Cholinesterase Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Heart; Neostigmine; Neurons; Nicotine; Nicotinic Agonists; Parasympathetic Nervous System; Picrotoxin; Pyridazines; Rats; Strychnine; Synaptic Transmission; Vagus Nerve

2003
Regulation of backpropagating action potentials in mitral cell lateral dendrites by A-type potassium currents.
    Journal of neurophysiology, 2003, Volume: 89, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 4-Aminopyridine; Action Potentials; Animals; Axons; Calcium Signaling; Dendrites; Excitatory Amino Acid Antagonists; In Vitro Techniques; Membrane Potentials; Olfactory Bulb; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Pyridazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetrodotoxin

2003
Dendritic sodium spikelets and low-threshold calcium spikes in turtle olfactory bulb granule cells.
    Journal of neurophysiology, 2005, Volume: 93, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Calcium Channel Blockers; Dendrites; Diagnostic Imaging; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Membrane Potentials; Mibefradil; Models, Neurological; Neurons; Nickel; Olfactory Bulb; Patch-Clamp Techniques; Pyridazines; Sodium; Synaptic Transmission; Tetrodotoxin; Time Factors; Turtles; Valine

2005
Local calcium transients regulate the spontaneous motility of dendritic filopodia.
    Nature neuroscience, 2005, Volume: 8, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Boron Compounds; Calcium; Calcium Signaling; Cell Movement; Cells, Cultured; Dendrites; Diagnostic Imaging; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; Glycine; Hippocampus; Immunohistochemistry; In Vitro Techniques; Indoles; Pseudopodia; Pyramidal Cells; Pyridazines; Quinoxalines; Rats; Synapses; Time Factors

2005
Anticonvulsant action of GABA in the high potassium-low magnesium model of ictogenesis in the neonatal rat hippocampus in vivo and in vitro.
    Journal of neurophysiology, 2005, Volume: 94, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Bicuculline; Disease Models, Animal; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isonicotinic Acids; Lipoproteins; Magnesium; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Pyridazines; Rats; Seizures

2005
Globus pallidus neurons dynamically regulate the activity pattern of subthalamic nucleus neurons through the frequency-dependent activation of postsynaptic GABAA and GABAB receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Lysine; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Neurons; Parkinson Disease; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Quinoxalines; Receptors, GABA-A; Receptors, GABA-B; Subthalamic Nucleus; Synapses; Tetrodotoxin

2005
SK channel regulation of dendritic excitability and dendrodendritic inhibition in the olfactory bulb.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Animals, Newborn; Apamin; Cadmium; Calcium; Dendrites; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Magnesium; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Olfactory Bulb; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Pyridazines; Quinoxalines; Synaptic Transmission; Tetraethylammonium; Tetrodotoxin; Time Factors

2005
Mono- and dual-frequency fast cerebellar oscillation in mice lacking parvalbumin and/or calbindin D-28k.
    The European journal of neuroscience, 2005, Volume: 22, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Analysis of Variance; Animals; Calbindin 2; Calbindins; Carbenoxolone; Cerebellum; Evoked Potentials; Excitatory Amino Acid Antagonists; Fourier Analysis; GABA Antagonists; Immunohistochemistry; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Parvalbumins; Periodicity; Purkinje Cells; Pyridazines; S100 Calcium Binding Protein G; Time Factors

2005
Regulation of thalamocortical patterning and synaptic maturation by NeuroD2.
    Neuron, 2006, Mar-02, Volume: 49, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Amino Acid Sequence; Amino Acids; Animals; Animals, Newborn; Basic Helix-Loop-Helix Transcription Factors; Blotting, Western; Calcium Channel Blockers; Cells, Cultured; Chelating Agents; Chloramphenicol O-Acetyltransferase; CREB-Binding Protein; Drug Interactions; Egtazic Acid; Electric Stimulation; Embryo, Mammalian; Excitatory Amino Acid Antagonists; GABA Antagonists; Gene Expression; Immunohistochemistry; In Vitro Techniques; Membrane Potentials; Mice; Mice, Knockout; Models, Biological; Nerve Growth Factors; Neural Pathways; Neurons; Neuropeptides; Nimodipine; Patch-Clamp Techniques; Phosphopyruvate Hydratase; Potassium Chloride; Pyridazines; Pyridinium Compounds; Quinoxalines; Receptors, AMPA; S100 Calcium Binding Protein beta Subunit; S100 Proteins; Somatosensory Cortex; Synapses; Thalamus; Transcriptional Activation; Transfection; Vibrissae

2006
Blanes cells mediate persistent feedforward inhibition onto granule cells in the olfactory bulb.
    Neuron, 2006, Mar-16, Volume: 49, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Cadmium; Chelating Agents; Diagnostic Imaging; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Lighting; Membrane Potentials; Models, Neurological; Nerve Net; Neural Inhibition; Olfactory Bulb; Organic Chemicals; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time

2006
Unitary IPSPs enhance hilar mossy cell gain in the rat hippocampus.
    The Journal of physiology, 2007, Jan-15, Volume: 578, Issue:Pt 2

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Bridged Bicyclo Compounds; Cell Membrane; Electric Capacitance; Electric Impedance; Excitatory Postsynaptic Potentials; Hippocampus; Inhibitory Postsynaptic Potentials; Interneurons; Male; Mossy Fibers, Hippocampal; Neurons; Patch-Clamp Techniques; Pilocarpine; Pyridazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium Channels; Synaptic Transmission; Tetrodotoxin

2007
Glutamatergic inputs in the hypothalamic paraventricular nucleus maintain sympathetic vasomotor tone in hypertension.
    Hypertension (Dallas, Tex. : 1979), 2007, Volume: 49, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Blood Pressure; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Heart Rate; Hypertension; Kynurenic Acid; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Pyridazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Sympathetic Nervous System; Vasomotor System

2007
Endogenous GABA and glutamate finely tune the bursting of olfactory bulb external tufted cells.
    Journal of neurophysiology, 2007, Volume: 98, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Neurons; Olfactory Bulb; Pyridazines; Rats; Rats, Sprague-Dawley; Valine

2007
SK2 channel plasticity contributes to LTP at Schaffer collateral-CA1 synapses.
    Nature neuroscience, 2008, Volume: 11, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Disks Large Homolog 4 Protein; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Guanylate Kinases; Hippocampus; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Long-Term Potentiation; Membrane Proteins; Mice; Mice, Inbred C57BL; Microscopy, Immunoelectron; Nerve Fibers; Neuronal Plasticity; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Small-Conductance Calcium-Activated Potassium Channels; Synapses; Synaptic Transmission

2008
GABA actions in hippocampal area CA3 during postnatal development: differential shift from depolarizing to hyperpolarizing in somatic and dendritic compartments.
    Journal of neurophysiology, 2008, Volume: 99, Issue:3

    Topics: Age Factors; Animals; Animals, Newborn; Dendrites; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Rats; Rats, Wistar; Valine

2008
Rapid plasticity at inhibitory and excitatory synapses in the hippocampus induced by ictal epileptiform discharges.
    The European journal of neuroscience, 2009, Volume: 29, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Biophysics; Calcium; Electric Stimulation; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Long-Term Potentiation; Magnesium; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Neuronal Plasticity; Potassium; Pyridazines; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Sodium Channel Blockers; Synapses; Tetrodotoxin; Valine

2009
Subcellular topography of visually driven dendritic activity in the vertebrate visual system.
    Neuron, 2009, Mar-26, Volume: 61, Issue:6

    Topics: Action Potentials; Animals; Brain Mapping; Calcium; Calcium Signaling; Dendrites; Excitatory Amino Acid Antagonists; GABA Antagonists; Imaging, Three-Dimensional; Larva; Light; Microscopy, Confocal; Neurons; Photic Stimulation; Presynaptic Terminals; Pyridazines; Receptors, N-Methyl-D-Aspartate; Subcellular Fractions; Valine; Visual Pathways; Xenopus

2009
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Capsaicin; Efferent Pathways; Endocannabinoids; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Pyridazines; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Tetrodotoxin; Vagus Nerve

2009
Synaptic and extrasynaptic factors governing glutamatergic retinal waves.
    Neuron, 2009, Apr-30, Volume: 62, Issue:2

    Topics: Amino Acid Transport Systems, Acidic; Animals; Animals, Newborn; Aspartic Acid; Calcium; Dihydro-beta-Erythroidine; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; In Vitro Techniques; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Biological; N-Methylaspartate; Neural Inhibition; Nicotinic Antagonists; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Retinal Ganglion Cells; Synapses; Synaptic Transmission; Time Factors; Valine; Vesicular Glutamate Transport Protein 1

2009
The timing of external input controls the sign of plasticity at local synapses.
    Nature neuroscience, 2009, Volume: 12, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Animals, Newborn; Biophysics; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Models, Neurological; Neural Pathways; Neuronal Plasticity; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Rats; Rats, Wistar; Synapses; Time Factors

2009
In the adult hippocampus, chronic nerve growth factor deprivation shifts GABAergic signaling from the hyperpolarizing to the depolarizing direction.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antibodies, Neutralizing; Biophysics; Bumetanide; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Hippocampus; In Vitro Techniques; Ion Channel Gating; Isonicotinic Acids; K Cl- Cotransporters; Mice; Mice, Transgenic; Nerve Growth Factor; Neurons; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Receptors, Nicotinic; RNA, Messenger; Sodium Potassium Chloride Symporter Inhibitors; Symporters

2010
Homeostatic regulation of synaptic excitability: tonic GABA(A) receptor currents replace I(h) in cortical pyramidal neurons of HCN1 knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Desoxycorticosterone; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Agents; Homeostasis; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Neurological; Patch-Clamp Techniques; Potassium Channels; Protein Subunits; Pyramidal Cells; Pyridazines; Pyrimidines; Receptors, GABA-A; Sodium Channel Blockers; Synapses; Tetrodotoxin; Up-Regulation; Valine

2010
Diacylglycerol lipase is not involved in depolarization-induced suppression of inhibition at unitary inhibitory connections in mouse hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: Animals; Animals, Newborn; Benzoxazines; Cyclohexanones; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; Green Fluorescent Proteins; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lipoprotein Lipase; Lysine; Mice; Mice, Inbred C57BL; Mice, Knockout; Morpholines; Naphthalenes; Neocortex; Neural Inhibition; Neurons; Pyridazines; Quinoxalines; Receptor, Cannabinoid, CB1; Valine

2010
The lateral paragigantocellular nucleus modulates parasympathetic cardiac neurons: a mechanism for rapid eye movement sleep-dependent changes in heart rate.
    Journal of neurophysiology, 2010, Volume: 104, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Biophysics; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Heart; Heart Rate; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Medulla Oblongata; N-Methylaspartate; Neurons; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Sleep, REM; Time Factors; Vagus Nerve; Valine

2010
Adrenergic receptor-mediated disinhibition of mitral cells triggers long-term enhancement of synchronized oscillations in the olfactory bulb.
    Journal of neurophysiology, 2010, Volume: 104, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Agonists; Animals; Animals, Newborn; Bicuculline; Biological Clocks; Biophysical Phenomena; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; N-Methylaspartate; Neurons; Norepinephrine; Olfactory Bulb; Pyridazines; Quinoxalines; Rats; Receptors, Adrenergic; Valine

2010
Short-term adaptation of conditioned fear responses through endocannabinoid signaling in the central amygdala.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:3

    Topics: Action Potentials; Adaptation, Psychological; Amygdala; Animals; Behavior, Animal; Cannabinoid Receptor Modulators; Conditioning, Psychological; Electric Stimulation; Endocannabinoids; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; GABA Antagonists; Gene Expression Regulation; In Vitro Techniques; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphinic Acids; Piperidines; Propanolamines; Pyrazoles; Pyridazines; Quinoxalines; Receptor, Cannabinoid, CB1; Sensory Receptor Cells; Signal Transduction; Time Factors; Valine

2011
Specific brainstem neurons switch each other into pacemaker mode to drive movement by activating NMDA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Dec-08, Volume: 30, Issue:49

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Biological Clocks; Brain Stem; Cadmium Chloride; Dihydro-beta-Erythroidine; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Glycyrrhetinic Acid; Humans; In Vitro Techniques; Larva; Models, Biological; Movement; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Periodicity; Pyridazines; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Swimming; Xenopus

2010
A circuit model for saccadic suppression in the superior colliculus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Feb-09, Volume: 31, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Genetically Modified; Animals, Newborn; Biophysics; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Membrane Potentials; Mice; Mice, Inbred C57BL; Models, Neurological; Nerve Net; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Reaction Time; Saccades; Sodium Channel Blockers; Superior Colliculi; Tetrodotoxin; Valine; Wheat Germ Agglutinin-Horseradish Peroxidase Conjugate

2011
Network oscillations in rod-degenerated mouse retinas.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Feb-09, Volume: 31, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Age Factors; Animals; Carbenoxolone; Cyclooxygenase Inhibitors; Disease Models, Animal; Evoked Potentials, Visual; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Gap Junctions; Glutamic Acid; Glycine; In Vitro Techniques; Light; Male; Meclofenamic Acid; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Neurologic Mutants; Nerve Net; Neural Inhibition; Periodicity; Pyridazines; Quinoxalines; Retinal Degeneration; Retinal Rod Photoreceptor Cells; Sodium Channel Blockers; Statistics as Topic; Tetrodotoxin

2011
Ovarian hormone deficiency reduces intrinsic excitability and abolishes acute estrogen sensitivity in hippocampal CA1 pyramidal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Feb-16, Volume: 31, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Analysis of Variance; Animals; Biophysics; Electric Stimulation; Estrogens; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Ovariectomy; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Rats; Time Factors; Valine

2011
Monosynaptic and polysynaptic feed-forward inputs to mitral cells from olfactory sensory neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jun-15, Volume: 31, Issue:24

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Animals, Newborn; Biophysics; Chromones; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; In Vitro Techniques; Luminescent Proteins; Male; Mice; Mice, Transgenic; Nerve Net; Neurons; Olfactory Bulb; Patch-Clamp Techniques; Pyridazines; Synapses

2011
Visual-induced excitation leads to firing pauses in striatal cholinergic interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Aug-03, Volume: 31, Issue:31

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Bicuculline; Cholinergic Agents; Corpus Striatum; Dose-Response Relationship, Drug; Electric Stimulation; Electroencephalography; Evoked Potentials, Visual; Excitatory Amino Acid Antagonists; Functional Laterality; GABA-A Receptor Antagonists; In Vitro Techniques; Interneurons; Light; Male; Models, Biological; Phosphinic Acids; Photic Stimulation; Propanolamines; Pyridazines; Rats; Rats, Long-Evans; Regression Analysis; Statistics, Nonparametric; Thalamus; Valine; Visual Pathways

2011
GABA(B) restrains release from singly-evoked GABA terminals.
    Neuroscience, 2011, Oct-13, Volume: 193

    Topics: Analysis of Variance; Animals; Benzylamines; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neurons; Phosphinic Acids; Pyridazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Sodium Channel Blockers; Solitary Nucleus; Synapses; Tetrodotoxin; Valine

2011
The afterhyperpolarizing potential following a train of action potentials is suppressed in an acute epilepsy model in the rat Cornu Ammonis 1 area.
    Neuroscience, 2012, Jan-10, Volume: 201

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; CA1 Region, Hippocampal; Disease Models, Animal; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Epilepsy; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Isoquinolines; Male; Neural Inhibition; Neurons; Pyridazines; Rats; Rats, Wistar; Statistics, Nonparametric; Sulfonamides; Time Factors

2012
Regulation of neuronal input transformations by tunable dendritic inhibition.
    Nature neuroscience, 2012, Jan-15, Volume: 15, Issue:3

    Topics: Animals; Biophysics; Cerebral Cortex; Channelrhodopsins; Dependovirus; DNA-Binding Proteins; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; In Vitro Techniques; Interneurons; Ligand-Gated Ion Channels; Luminescent Proteins; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Models, Neurological; Mutation; Neural Inhibition; Parvalbumins; Patch-Clamp Techniques; Photic Stimulation; Pyramidal Cells; Pyridazines; Receptors, Glycine; RNA, Small Interfering; Synapses; Synaptic Transmission; Transcription Factors; Transduction, Genetic; Valine

2012
Interaction of NMDA receptors and L-type calcium channels during early odor preference learning in rats.
    The European journal of neuroscience, 2012, Volume: 36, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Dendrites; Gene Expression; Isoproterenol; Learning; Neuronal Plasticity; Nimodipine; Odorants; Olfactory Bulb; Olfactory Perception; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapsins; Transcription, Genetic

2012
The balance of striatal feedback transmission is disrupted in a model of parkinsonism.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-13, Volume: 33, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adrenergic Agents; Anesthetics, Local; Animals; Animals, Newborn; Bicuculline; Biophysics; Calcium; Disease Models, Animal; Electric Stimulation; Excitatory Amino Acid Antagonists; Feedback, Physiological; GABA Antagonists; gamma-Aminobutyric Acid; Green Fluorescent Proteins; In Vitro Techniques; Lidocaine; Lysine; Male; Mice; Mice, Transgenic; Monte Carlo Method; Neostriatum; Neural Inhibition; Neural Pathways; Neurons; Oxidopamine; Parkinsonian Disorders; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Receptors, Dopamine D2; Synaptic Transmission; Time Factors; Valine

2013
Novel GABAergic circuits mediating excitation/inhibition of Cajal-Retzius cells in the developing hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-27, Volume: 33, Issue:13

    Topics: Age Factors; Animals; Animals, Newborn; Biophysics; Channelrhodopsins; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Hippocampus; In Vitro Techniques; Interneurons; Light; Male; Membrane Potentials; Methoxyhydroxyphenylglycol; Mice; Mice, Transgenic; Mutation; Nerve Net; Neural Inhibition; Optogenetics; Patch-Clamp Techniques; Proteins; Pyridazines; Quinoxalines; Receptors, CXCR4; RNA, Untranslated; Sodium Channel Blockers; Somatostatin; Synaptic Potentials; Tetrodotoxin; Valine

2013
NMDA-receptor inhibition increases spine stability of denervated mouse dentate granule cells and accelerates spine density recovery following entorhinal denervation in vitro.
    Neurobiology of disease, 2013, Volume: 59

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Computer Simulation; Dendritic Spines; Denervation; Dentate Gyrus; Entorhinal Cortex; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; Green Fluorescent Proteins; Male; Mice; Mice, Transgenic; Models, Biological; Neurons; Organ Culture Techniques; Pyridazines; Receptors, N-Methyl-D-Aspartate; Sodium Channel Blockers; Tetrodotoxin

2013
Long-term potentiation in hilar circuitry modulates gating by the dentate gyrus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Jul-16, Volume: 34, Issue:29

    Topics: Analysis of Variance; Animals; Biophysics; Dentate Gyrus; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Long-Term Potentiation; Male; Nerve Net; Neurons; Pyridazines; Rats; Rats, Sprague-Dawley; Valine; Voltage-Sensitive Dye Imaging

2014
Distinct representation and distribution of visual information by specific cell types in mouse superficial superior colliculus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Oct-01, Volume: 34, Issue:40

    Topics: Action Potentials; Animals; Channelrhodopsins; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; Glutamate Decarboxylase; Green Fluorescent Proteins; Luminescent Proteins; Male; Mice; Mice, Transgenic; Neurons; Pyridazines; Quinoxalines; Receptors, Neurotensin; Superior Colliculi; Valine; Vesicular Inhibitory Amino Acid Transport Proteins; Visual Fields; Visual Pathways

2014
Cell-specific activity-dependent fractionation of layer 2/3→5B excitatory signaling in mouse auditory cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, Feb-18, Volume: 35, Issue:7

    Topics: Animals; Animals, Newborn; Auditory Cortex; Auditory Pathways; Excitatory Amino Acid Antagonists; Female; Flavoproteins; GABA Antagonists; In Vitro Techniques; Inferior Colliculi; Male; Mice; Mice, Inbred ICR; Models, Neurological; Nerve Net; Neurons; Patch-Clamp Techniques; Pyridazines; Quinoxalines; Synaptic Potentials; Valine

2015
GABAergic inhibition shapes SAM responses in rat auditory thalamus.
    Neuroscience, 2015, Jul-23, Volume: 299

    Topics: Acoustic Stimulation; Animals; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Geniculate Bodies; Male; Neural Inhibition; Neurons; Pyridazines; Rats; Receptors, N-Methyl-D-Aspartate; Sound; Synaptic Transmission; Valine

2015
Dynamic Analysis of the Conditional Oscillator Underlying Slow Waves in Thalamocortical Neurons.
    Frontiers in neural circuits, 2016, Volume: 10

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzamides; Calcium; Calcium Channel Blockers; Cats; Cerebral Cortex; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Geniculate Bodies; In Vitro Techniques; Membrane Potentials; Models, Neurological; Neurons; Nonlinear Dynamics; Organophosphorus Compounds; Patch-Clamp Techniques; Piperidines; Pyridazines

2016
Developmental exposure to PCBs alters the activation of the auditory cortex in response to GABA
    Neurotoxicology, 2016, Volume: 56

    Topics: Afferent Pathways; Animals; Animals, Newborn; Auditory Cortex; Electric Stimulation; Environmental Pollutants; Excitatory Amino Acid Antagonists; Female; GABA-A Receptor Antagonists; Male; Polychlorinated Biphenyls; Pregnancy; Prenatal Exposure Delayed Effects; Pyridazines; Rats; Rats, Long-Evans; Valine

2016
Effects of memantine on the excitation-inhibition balance in prefrontal cortex.
    Neurobiology of disease, 2016, Volume: 96

    Topics: Animals; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Glutamate Decarboxylase; Green Fluorescent Proteins; Inhibitory Postsynaptic Potentials; Male; Memantine; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neurons; Parvalbumins; Patch-Clamp Techniques; Prefrontal Cortex; Pyridazines; Valine

2016