Page last updated: 2024-08-26

sr 48968 and sb 223412

sr 48968 has been researched along with sb 223412 in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's5 (71.43)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brawner, ME; Elshourbagy, NA; Foley, JJ; Giardina, GA; Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Potts, W; Sarau, HM; Schmidt, DB; Webb, EF1
Hey, JA; Rizzo, CA1
Oh, EJ; Thompson, LP; Weinreich, D1
Chapple, CR; Chess-Williams, R; Hay, DP; Rosario, DJ; Sellers, DJ; Templeman, L1
Chapple, CR; Chess-Williams, R; Sellers, DJ; W Hay, DP1
Corboz, MR; Fernandez, X; Hey, JA1
Imanishi, A; Kawamoto, M; Mizojiri, G; Nakamura, A; Tanaka, T; Toyoda, M; Tsukimi, Y1

Other Studies

7 other study(ies) available for sr 48968 and sb 223412

ArticleYear
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:3

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Dogs; Humans; Mice; Piperidines; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin

1997
Activity of nonpeptide tachykinin antagonists on neurokinin a induced contractions in dog urinary bladder.
    The Journal of urology, 2000, Volume: 163, Issue:6

    Topics: Animals; Benzamides; Dogs; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Piperidines; Quinolines; Receptors, Neurokinin-2; Stereoisomerism; Urinary Bladder

2000
Sexually dimorphic regulation of NK-1 receptor-mediated electrophysiological responses in vagal primary afferent neurons.
    Journal of neurophysiology, 2000, Volume: 84, Issue:1

    Topics: Animals; Benzamides; Electrophysiology; Estradiol; Female; Gonadal Steroid Hormones; Guinea Pigs; Male; Membrane Potentials; Neurons, Afferent; Nodose Ganglion; Orchiectomy; Ovariectomy; Piperidines; Pregnancy; Quinolines; Receptors, Neurokinin-1; Serotonin; Sex Characteristics; Substance P; Testosterone

2000
Investigation of neurokinin-2 and -3 receptors in the human and pig bladder.
    BJU international, 2003, Volume: 92, Issue:7

    Topics: Animals; Benzamides; Dose-Response Relationship, Drug; Humans; Muscle Contraction; Neurokinin A; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Urinary Bladder

2003
Depressed contractile responses to neurokinin A in idiopathic but not neurogenic overactive human detrusor muscle.
    European urology, 2006, Volume: 49, Issue:3

    Topics: Benzamides; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neurokinin A; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Urinary Bladder

2006
Increased blocking activity of combined tachykinin NK1- and NK2-receptor antagonists on hyperventilation-induced bronchoconstriction in the guinea pig.
    Pulmonary pharmacology & therapeutics, 2008, Volume: 21, Issue:1

    Topics: Administration, Oral; Animals; Benzamides; Bronchoconstriction; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Hyperventilation; Injections, Intravenous; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Respiratory Function Tests

2008
Bidirectional regulation of human colonic smooth muscle contractility by tachykinin NK(2) receptors.
    Journal of pharmacological sciences, 2011, Volume: 117, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Benzamides; Cell Line, Tumor; Colon; Female; Humans; In Vitro Techniques; Isometric Contraction; Male; Middle Aged; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Quinolines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Tachykinins

2011