Page last updated: 2024-08-26

sr 48968 and men 11420

sr 48968 has been researched along with men 11420 in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (36.36)18.2507
2000's6 (54.55)29.6817
2010's1 (9.09)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Giorgio, RD; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Criscuoli, M; Giuliani, S; Lecci, A; Lippi, A; Maggi, CA; Patacchini, R; Santicioli, P; Tramontana, M1
Catalioto, RM; Criscuoli, M; Cucchi, P; Ferrer, C; Giolitti, A; Guelfi, M; Maggi, CA; Renzetti, AR; Rotondaro, L; Warner, FJ1
Cucchi, P; Giolitti, A; Maggi, CA; Renzetti, AR; Rotondaro, L; Zappitelli, S1
Giuliani, S; Maggi, CA; Navarra, G; Patacchini, R; Turini, A1
Buéno, L; Criscuoli, M; Giuliani, S; Guelfi, M; Lecci, A; Maggi, CA; Toulouse, M; Tramontana, M1
Altamura, M; Bellucci, F; Catalani, C; Cucchi, P; Giolitti, A; Giuliani, S; Maggi, CA; Meini, S; Patacchini, R; Rotondaro, L1
Bellucci, F; Candenas, ML; Catalani, C; Catalioto, RM; Faiella, A; Giolitti, A; Giuliani, S; Maggi, CA; Meini, S; Pinto, FM; Quartara, L; Rotondaro, L1
Bellucci, F; Catalani, C; Cucchi, P; Giolitti, A; Giuliani, S; Meini, S; Santicioli, P1
Bechi, P; Catalani, C; Giuliani, S; Maggi, CA; Meini, S; Riccadonna, S; Ringressi, MN; Santicioli, P1

Other Studies

11 other study(ies) available for sr 48968 and men 11420

ArticleYear
Role of tachykinin NK1 and NK2 receptors on colonic motility in anesthetized rats: effect of agonists.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Anesthesia; Animals; Benzamides; Colon; Gastrointestinal Motility; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1997
The role of tachykinin NK1 and NK2 receptors in atropine-resistant colonic propulsion in anaesthetized guinea-pigs.
    British journal of pharmacology, 1998, Volume: 124, Issue:1

    Topics: Anesthesia; Animals; Apamin; Atropine; Benzamides; Colon; Guinea Pigs; Hexamethonium; Male; Models, Biological; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Peristalsis; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2

1998
Characterization of the antibronchoconstrictor activity of MEN 11420, a tachykinin NK2 receptor antagonist, in guinea-pigs.
    European journal of pharmacology, 1998, Jul-10, Volume: 352, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Atropine; Benzamides; Bronchi; Bronchoconstriction; Bronchodilator Agents; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1998
Relevance of aromatic residues in transmembrane segments V to VII for binding of peptide and nonpeptide antagonists to the human tachykinin NK(2) receptor.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:2

    Topics: Animals; Benzamides; Binding, Competitive; CHO Cells; Cricetinae; DNA, Complementary; Humans; Indoles; Mutagenesis, Site-Directed; Mutation; Neurokinin A; Peptides; Peptides, Cyclic; Piperidines; Protein Conformation; Receptors, Neurokinin-2

1999
Molecular determinants of peptide and nonpeptide NK-2 receptor antagonists binding sites of the human tachykinin NK-2 receptor by site-directed mutagenesis.
    Neuropharmacology, 2000, Jun-08, Volume: 39, Issue:8

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Benzamides; Binding Sites; CHO Cells; Cricetinae; Humans; Molecular Sequence Data; Mutagenesis, Site-Directed; Neurokinin A; Peptides, Cyclic; Piperidines; Point Mutation; Protein Binding; Radioligand Assay; Receptors, Neurokinin-2

2000
Effect of nepadutant at tachykinin NK(2) receptors in human intestine and urinary bladder.
    European journal of pharmacology, 2000, Jun-23, Volume: 398, Issue:3

    Topics: Aged; Aged, 80 and over; Benzamides; Colon; Female; Humans; Ileum; Male; Middle Aged; Neurokinin A; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2; Urinary Bladder

2000
Effect of a tachykinin NK(2) receptor antagonist, nepadutant, on cardiovascular and gastrointestinal function in rats and dogs.
    European journal of pharmacology, 2001, Mar-09, Volume: 415, Issue:1

    Topics: Animals; Benzamides; Binding, Competitive; Blood Pressure; Cardiovascular System; Digestive System; Digestive System Physiological Phenomena; Dogs; Dose-Response Relationship, Drug; Fasting; Female; Gastrointestinal Motility; Heart Rate; Injections, Intravenous; Male; Peptides, Cyclic; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Tidal Volume

2001
Mutagenesis at the human tachykinin NK(2) receptor to define the binding site of a novel class of antagonists.
    European journal of pharmacology, 2004, Mar-19, Volume: 488, Issue:1-3

    Topics: Animals; Benzamides; Binding Sites; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; DNA, Complementary; Guinea Pigs; In Vitro Techniques; Ligands; Male; Models, Molecular; Muscle Contraction; Muscle, Smooth; Mutagenesis, Site-Directed; Peptides, Cyclic; Piperidines; Radioligand Assay; Rats; Receptors, Neurokinin-2

2004
Pharmacological evaluation of alpha and beta human tachykinin NK(2) receptor splice variants expressed in CHO cells.
    European journal of pharmacology, 2004, Sep-24, Volume: 499, Issue:3

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Benzamides; Binding, Competitive; Calcium; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Humans; Inositol Phosphates; Intracellular Space; Iodine Radioisotopes; Molecular Sequence Data; Neurokinin A; Peptides, Cyclic; Piperidines; Protein Isoforms; Radioligand Assay; Receptors, Neurokinin-2; Sequence Homology, Amino Acid; Substance P; Transfection; Tritium

2004
Multifaceted approach to determine the antagonist molecular mechanism and interaction of ibodutant ([1-(2-phenyl-1R-[[1-(tetrahydropyran-4-ylmethyl)-piperidin-4-ylmethyl]-carbamoyl]-ethylcarbamoyl)-cyclopentyl]-amide) at the human tachykinin NK2 receptor.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 329, Issue:2

    Topics: Animals; Benzamides; Binding, Competitive; Cell Line; Cloning, Molecular; Cricetinae; Cricetulus; Dipeptides; Dose-Response Relationship, Drug; Humans; Kinetics; Models, Molecular; Peptides, Cyclic; Phosphatidylinositols; Piperidines; Protein Binding; Radioligand Assay; Receptors, Neurokinin-2; Thiophenes; Type C Phospholipases

2009
Characterization of ibodutant at NK(2) receptor in human colon.
    European journal of pharmacology, 2013, Feb-28, Volume: 702, Issue:1-3

    Topics: Aged; Aged, 80 and over; Benzamides; Binding, Competitive; Colon; Dipeptides; Female; Humans; In Vitro Techniques; Male; Middle Aged; Peptides, Cyclic; Piperidines; Radioligand Assay; Receptors, Neurokinin-2; Thiophenes

2013