Page last updated: 2024-09-03

sr 48692 and tetrodotoxin

sr 48692 has been researched along with tetrodotoxin in 11 studies

Compound Research Comparison

Studies
(sr 48692)
Trials
(sr 48692)
Recent Studies (post-2010)
(sr 48692)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
20333612,992111,477

Protein Interaction Comparison

ProteinTaxonomysr 48692 (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0186

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (18.18)18.2507
2000's9 (81.82)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kombian, SB; Pittman, QJ; Saleh, TM; Zidichouski, JA1
Héaulme, M; Le Fur, G; Leyris, R; Soubrié, P1
Castagliuolo, I; Matthews, JB; Pothoulakis, C; Riegler, M; Sogukoglu, T; Wang, C; Wenzl, E; Wlk, M1
Antonelli, T; Bebe, BW; Fernandez, M; Ferraro, L; Fuxe, K; Glennon, JC; O'Connor, WT; Tanganelli, S; Tomasini, MC1
Greengard, P; Higashi, H; Maeda, H; Matsuyama, S; Nishi, A1
Fukui, R; Higashi, H; Matsuyama, S; Nishi, A1
Chen, L; Yung, KK; Yung, WH2
Bubser, M; Carraway, RE; Deutch, AY; Fadel, J; Petrie, KA; Schmidt, D1
Della Corte, L; Mayer, A; Petkova-Kirova, P; Radomirov, R; Rakovska, A; Zaekova, G1
Kawahara, H; Mitchell, VA; Vaughan, CW1

Other Studies

11 other study(ies) available for sr 48692 and tetrodotoxin

ArticleYear
Cholecystokinin and neurotensin inversely modulate excitatory synaptic transmission in the parabrachial nucleus in vitro.
    Neuroscience, 1997, Volume: 77, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cholecystokinin; Devazepide; Electric Conductivity; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hormone Antagonists; Interneurons; N-Methylaspartate; Neural Inhibition; Neurons, Afferent; Neurotensin; Patch-Clamp Techniques; Phenylurea Compounds; Pons; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

1997
Stimulation by neurotensin of (3H)5-hydroxytryptamine (5HT) release from rat frontal cortex slices.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Adamantane; Animals; Corpus Striatum; Dizocilpine Maleate; Dopamine Antagonists; Down-Regulation; Frontal Lobe; Hippocampus; Imidazoles; In Vitro Techniques; Inhibitory Concentration 50; Neurotensin; Peptide Fragments; Potassium; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotensin; Serotonin; Tetrodotoxin

1998
Neurotensin stimulates Cl(-) secretion in human colonic mucosa In vitro: role of adenosine.
    Gastroenterology, 2000, Volume: 119, Issue:2

    Topics: Adamantane; Adenosine; Adenosine Deaminase Inhibitors; Affinity Labels; Anti-Inflammatory Agents, Non-Steroidal; Cells, Cultured; Chlorides; Colon; Electrophysiology; Enteric Nervous System; Enzyme Inhibitors; Guanosine; Histamine; Humans; Imidazoles; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Mast Cells; Membrane Potentials; Neurotensin; Pentostatin; Pyrazoles; Quinolines; Receptors, Neurotensin; Tetrodotoxin; Thioinosine; Thionucleosides

2000
Nigral neurotensin receptor regulation of nigral glutamate and nigroventral thalamic GABA transmission: a dual-probe microdialysis study in intact conscious rat brain.
    Neuroscience, 2001, Volume: 102, Issue:1

    Topics: Animals; Consciousness; Dopamine Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Neural Pathways; Neurons; Neurotensin; Peptide Fragments; Pyrazoles; Quinolines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Substantia Nigra; Synaptic Transmission; Tetrodotoxin; Ventral Thalamic Nuclei

2001
Neurotensin regulates DARPP-32 thr34 phosphorylation in neostriatal neurons by activation of dopamine D1-type receptors.
    Journal of neurochemistry, 2002, Volume: 81, Issue:2

    Topics: Animals; Cobalt; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Glutamine; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Phosphorylation; Piperidines; Pyrazoles; Quinolines; Receptors, Dopamine D1; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin

2002
Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Anesthetics, Local; Animals; Benzazepines; Dizocilpine Maleate; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Histamine H1 Antagonists; Immunoblotting; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Piperidines; Pyrazoles; Quinolines; Raclopride; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin; Threonine; Time Factors

2003
Neurotensin depolarizes globus pallidus neurons in rats via neurotensin type-1 receptor.
    Neuroscience, 2004, Volume: 125, Issue:4

    Topics: Action Potentials; Adamantane; Anesthetics, Local; Animals; Electrophysiology; Globus Pallidus; Imidazoles; Neurons; Neurotensin; Organ Culture Techniques; Patch-Clamp Techniques; Peptide Fragments; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

2004
Neurotensin activates GABAergic interneurons in the prefrontal cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Feb-16, Volume: 25, Issue:7

    Topics: Animals; Axons; Dopamine; Dopamine Agonists; gamma-Aminobutyric Acid; Interneurons; Male; Microdialysis; Neurotensin; Parvalbumins; Prefrontal Cortex; Pyrazoles; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Neurotensin; Schizophrenia; Tetrodotoxin

2005
Neurotensin selectively facilitates glutamatergic transmission in globus pallidus.
    Neuroscience, 2006, Sep-15, Volume: 141, Issue:4

    Topics: Anesthetics, Local; Animals; Animals, Newborn; Bicuculline; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Estrenes; Excitatory Postsynaptic Potentials; GABA Antagonists; Globus Pallidus; Glutamic Acid; In Vitro Techniques; Neural Inhibition; Neurons; Neurotensin; Patch-Clamp Techniques; Pyrazoles; Pyrrolidinones; Quinolines; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Tetrodotoxin

2006
Neurotensin modulation of acetylcholine, GABA, and aspartate release from rat prefrontal cortex studied in vivo with microdialysis.
    Brain research bulletin, 2008, Sep-30, Volume: 77, Issue:2-3

    Topics: Acetylcholine; Animals; Aspartic Acid; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Motor Activity; Neurotensin; Prefrontal Cortex; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin; Sodium Channel Blockers; Taurine; Tetrodotoxin

2008
Neurotensin inhibition of GABAergic transmission via mGluR-induced endocannabinoid signalling in rat periaqueductal grey.
    The Journal of physiology, 2009, Jun-01, Volume: 587, Issue:Pt 11

    Topics: Adamantane; Animals; Cannabinoid Receptor Modulators; Endocannabinoids; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Neural Inhibition; Neurons; Neurotensin; Pain; Periaqueductal Gray; Piperidines; Presynaptic Terminals; Pyrazoles; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin; Time Factors

2009