Page last updated: 2024-09-03

sr 48692 and glutamic acid

sr 48692 has been researched along with glutamic acid in 9 studies

Compound Research Comparison

Studies
(sr 48692)
Trials
(sr 48692)
Recent Studies (post-2010)
(sr 48692)
Studies
(glutamic acid)
Trials
(glutamic acid)
Recent Studies (post-2010) (glutamic acid)
20333641,75745212,876

Protein Interaction Comparison

ProteinTaxonomysr 48692 (IC50)glutamic acid (IC50)
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2Rattus norvegicus (Norway rat)0.821
Chain A, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Chain B, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Metabotropic glutamate receptor 8Homo sapiens (human)0.0057
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.07
Glutamate receptor 1Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 2Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 3Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 4Rattus norvegicus (Norway rat)0.5885
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.38
Glutamate receptor 1Homo sapiens (human)0.613
Glutamate receptor 2Homo sapiens (human)0.613
Glutamate receptor 3Homo sapiens (human)0.613
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.38
Excitatory amino acid transporter 1Homo sapiens (human)207
Glutamate receptor 4Homo sapiens (human)0.613
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.1533

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's6 (66.67)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Antonelli, T; Ferraro, L; Fuxe, K; O'Connor, WT; Soubrié, P; Tanganelli, S1
Antonelli, T; Bebe, BW; Fernandez, M; Ferraro, L; Fuxe, K; Glennon, JC; O'Connor, WT; Tanganelli, S; Tomasini, MC1
Antonelli, T; Calzà, L; Ferraro, L; Finetti, S; Fuxe, K; Giardino, L; Soubriè, P; Tanganelli, S; Tomasini, MC1
Fukui, R; Higashi, H; Matsuyama, S; Nishi, A1
Antonelli, T; De Mattei, M; Ferraro, L; Finetti, S; Fournier, J; Fuxe, K; Tanganelli, S; Tomasini, MC1
Chen, L; Yung, KK; Yung, WH1
Della Corte, L; Mayer, A; Petkova-Kirova, P; Radomirov, R; Rakovska, A; Zaekova, G1
Hugel, S; Kadiri, N; Rodeau, JL; Schlichter, R1
Bonci, A; Cho, SL; de Lecea, L; Deisseroth, K; Kempadoo, KA; Leinninger, GM; Magnani, F; Myers, MG; Stuber, GD; Tourino, C; Zhang, F1

Other Studies

9 other study(ies) available for sr 48692 and glutamic acid

ArticleYear
The striatal neurotensin receptor modulates striatal and pallidal glutamate and GABA release: functional evidence for a pallidal glutamate-GABA interaction via the pallidal-subthalamic nucleus loop.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Sep-01, Volume: 18, Issue:17

    Topics: Animals; Bicuculline; Corpus Striatum; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Glutamic Acid; Injections; Male; Microdialysis; Perfusion; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Synaptic Transmission; Thalamic Nuclei

1998
Nigral neurotensin receptor regulation of nigral glutamate and nigroventral thalamic GABA transmission: a dual-probe microdialysis study in intact conscious rat brain.
    Neuroscience, 2001, Volume: 102, Issue:1

    Topics: Animals; Consciousness; Dopamine Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Neural Pathways; Neurons; Neurotensin; Peptide Fragments; Pyrazoles; Quinolines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Substantia Nigra; Synaptic Transmission; Tetrodotoxin; Ventral Thalamic Nuclei

2001
Neurotensin enhances glutamate excitotoxicity in mesencephalic neurons in primary culture.
    Journal of neuroscience research, 2002, Dec-15, Volume: 70, Issue:6

    Topics: Animals; Cells, Cultured; Dopamine; Embryo, Mammalian; Enzyme Inhibitors; Glutamic Acid; Immunohistochemistry; Mesencephalon; Naphthalenes; Nerve Degeneration; Neurons; Neuroprotective Agents; Neurotensin; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Tyrosine 3-Monooxygenase

2002
Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Anesthetics, Local; Animals; Benzazepines; Dizocilpine Maleate; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Histamine H1 Antagonists; Immunoblotting; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Piperidines; Pyrazoles; Quinolines; Raclopride; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin; Threonine; Time Factors

2003
Neurotensin enhances endogenous extracellular glutamate levels in primary cultures of rat cortical neurons: involvement of neurotensin receptor in NMDA induced excitotoxicity.
    Cerebral cortex (New York, N.Y. : 1991), 2004, Volume: 14, Issue:4

    Topics: Animals; Bisbenzimidazole; Calcium; Cells, Cultured; Cerebral Cortex; Chromatin; Coloring Agents; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Extracellular Space; Glutamic Acid; N-Methylaspartate; Naphthalenes; Neurons; Neurotensin; Neurotoxicity Syndromes; Peptide Fragments; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin

2004
Neurotensin selectively facilitates glutamatergic transmission in globus pallidus.
    Neuroscience, 2006, Sep-15, Volume: 141, Issue:4

    Topics: Anesthetics, Local; Animals; Animals, Newborn; Bicuculline; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Estrenes; Excitatory Postsynaptic Potentials; GABA Antagonists; Globus Pallidus; Glutamic Acid; In Vitro Techniques; Neural Inhibition; Neurons; Neurotensin; Patch-Clamp Techniques; Pyrazoles; Pyrrolidinones; Quinolines; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Tetrodotoxin

2006
Neurotensin modulation of acetylcholine, GABA, and aspartate release from rat prefrontal cortex studied in vivo with microdialysis.
    Brain research bulletin, 2008, Sep-30, Volume: 77, Issue:2-3

    Topics: Acetylcholine; Animals; Aspartic Acid; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Motor Activity; Neurotensin; Prefrontal Cortex; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin; Sodium Channel Blockers; Taurine; Tetrodotoxin

2008
Neurotensin inhibits background K+ channels and facilitates glutamatergic transmission in rat spinal cord dorsal horn.
    The European journal of neuroscience, 2011, Volume: 34, Issue:8

    Topics: Animals; Benzophenanthridines; Excitatory Postsynaptic Potentials; Glutamic Acid; Neurotensin; Oligopeptides; Patch-Clamp Techniques; Pertussis Toxin; Piperidines; Posterior Horn Cells; Potassium Channels; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Signal Transduction; Synapses; Synaptic Transmission

2011
Hypothalamic neurotensin projections promote reward by enhancing glutamate transmission in the VTA.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, May-01, Volume: 33, Issue:18

    Topics: Animals; Bacterial Proteins; Channelrhodopsins; Conditioning, Operant; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Hypothalamus; In Vitro Techniques; Light; Luminescent Proteins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutation; Neural Pathways; Neurotensin; Pyrazoles; Quinolines; Quinoxalines; Receptors, Neurotensin; Reward; Self Stimulation; Signal Transduction; Tyrosine 3-Monooxygenase; Valine; Ventral Tegmental Area

2013