Page last updated: 2024-09-03

sr 46349b and ritanserin

sr 46349b has been researched along with ritanserin in 3 studies

Compound Research Comparison

Studies
(sr 46349b)
Trials
(sr 46349b)
Recent Studies (post-2010)
(sr 46349b)
Studies
(ritanserin)
Trials
(ritanserin)
Recent Studies (post-2010) (ritanserin)
51177357571

Protein Interaction Comparison

ProteinTaxonomysr 46349b (IC50)ritanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.001
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.047
Diacylglycerol kinase alphaHomo sapiens (human)9
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.047
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.047
D(2) dopamine receptorRattus norvegicus (Norway rat)0.012

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brelière, JC; Congy, C; Le Fur, G; Pointeau, P; Rinaldi-Carmona, M; Vidal, H1
Bouaboula, M; Brelière, JC; Casellas, P; Congy, C; Le Fur, G; Oury-Donat, F; Rinaldi-Carmona, M; Shire, D; Simiand, J; Soubrié, P1
De Deurwaerdére, P; Di Giovanni, G; Di Mascio, M; Di Matteo, V; Esposito, E; Spampinato, U1

Other Studies

3 other study(ies) available for sr 46349b and ritanserin

ArticleYear
Identification of binding sites for SR 46349B, a 5-hydroxytryptamine2 receptor antagonist, in rodent brain.
    Life sciences, 1994, Volume: 54, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Fluorobenzenes; In Vitro Techniques; Ketanserin; Male; Mice; Phenols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1994
Up-regulation of 5-HT2 receptors in the rat brain by repeated administration of SR 46349B, a selective 5-HT2 receptor antagonist.
    European journal of pharmacology, 1993, Jun-15, Volume: 246, Issue:1

    Topics: Amphetamines; Animals; Base Sequence; Blotting, Southern; Brain Chemistry; Cerebral Cortex; Fluorobenzenes; In Vitro Techniques; Inosine Monophosphate; Ketanserin; Male; Molecular Sequence Data; Phenols; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; RNA, Messenger; Second Messenger Systems; Serotonin Antagonists; Serotonin Receptor Agonists; Up-Regulation

1993
Selective blockade of serotonin-2C/2B receptors enhances mesolimbic and mesostriatal dopaminergic function: a combined in vivo electrophysiological and microdialysis study.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Electrophysiology; Evoked Potentials; Fluorobenzenes; Indoles; Limbic System; Male; Microdialysis; Neurons; Nucleus Accumbens; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tegmentum Mesencephali

1999