Page last updated: 2024-09-03

sr 46349b and mdl 100907

sr 46349b has been researched along with mdl 100907 in 14 studies

Compound Research Comparison

Studies
(sr 46349b)
Trials
(sr 46349b)
Recent Studies (post-2010)
(sr 46349b)
Studies
(mdl 100907)
Trials
(mdl 100907)
Recent Studies (post-2010) (mdl 100907)
51171,24165539

Protein Interaction Comparison

ProteinTaxonomysr 46349b (IC50)mdl 100907 (IC50)
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0048

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.14)18.2507
2000's7 (50.00)29.6817
2010's6 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Marcoli, M; Maura, G; Raiteri, M; Tortarolo, M1
Alboszta, AR; Bonaccorso, S; Dai, J; Ichikawa, J; Li, Z; Meltzer, HY1
Gray, JA; Joseph, MH; McDonald, LM; Moran, PM; Stephenson, JD; Vythelingum, GN1
Auclair, A; Blanc, G; Glowinski, J; Tassin, JP1
Bourin, M; Dailly, E; Hascoët, M; Masse, F1
Miyamoto, M; Terao, A1
Blessing, WW; Nalivaiko, E; Ootsuka, Y1
Baumert, M; Beig, MI; Day, TA; Nalivaiko, E; Walker, FR1
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA1
Lanfumey, L; Maldonado, R; Orejarena, MJ; Robledo, P1
Arnt, J; Ebdrup, BH; Glenthøj, B; Rasmussen, H1
Alonso, R; Avenet, P; Beeské, S; Decobert, M; Françon, D; Griebel, G; Jacquet, A; Laufrais, C1
Dougherty, JP; Oristaglio, J1
Ootsuka, Y; Sinh, V1

Reviews

2 review(s) available for sr 46349b and mdl 100907

ArticleYear
[Recent and potential drugs for treatment of insomnia].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2007, Volume: 129, Issue:1

    Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Diphenhydramine; Drug Design; Fluorobenzenes; GABA-A Receptor Agonists; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Indenes; Orexin Receptors; Phenols; Piperazines; Pyridines; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Serotonin 5-HT2 Receptor Antagonists; Sleep Initiation and Maintenance Disorders; Thiophenes; Zolpidem

2007
Serotonin 2A receptor antagonists for treatment of schizophrenia.
    Expert opinion on investigational drugs, 2011, Volume: 20, Issue:9

    Topics: Antipsychotic Agents; Brain; Fluorobenzenes; Humans; Phenols; Piperidines; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin 5-HT2 Receptor Antagonists; Urea

2011

Other Studies

12 other study(ies) available for sr 46349b and mdl 100907

ArticleYear
Serotonin inhibition of the NMDA receptor/nitric oxide/cyclic GMP pathway in rat cerebellum: involvement of 5-hydroxytryptamine2C receptors.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebellum; Cyclic GMP; Excitatory Amino Acid Agonists; Fluorobenzenes; Indoles; Male; N-Methylaspartate; Nitric Oxide; Organ Culture Techniques; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Urea; Yohimbine

1997
SR46349-B, a 5-HT(2A/2C) receptor antagonist, potentiates haloperidol-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 27, Issue:3

    Topics: Analysis of Variance; Animals; Dopamine; Dopamine Antagonists; Drug Synergism; Fluorobenzenes; Haloperidol; Male; Nucleus Accumbens; Phenols; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Telencephalon

2002
Enhancement of latent inhibition by two 5-HT2A receptor antagonists only when given at both pre-exposure and conditioning.
    Psychopharmacology, 2003, Volume: 169, Issue:3-4

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Amphetamine; Analysis of Variance; Animals; Association Learning; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Classical; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; Inhibition, Psychological; Male; Phencyclidine; Phenols; Quinolines; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Stereotyped Behavior

2003
Role of serotonin 2A receptors in the D-amphetamine-induced release of dopamine: comparison with previous data on alpha1b-adrenergic receptors.
    Journal of neurochemistry, 2004, Volume: 91, Issue:2

    Topics: Animals; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Antagonism; Extracellular Fluid; Fluorobenzenes; Male; Microdialysis; Motor Activity; Neurons; Nucleus Accumbens; Phenols; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Ventral Tegmental Area

2004
Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzylamines; Brain; Cyclopropanes; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Flumazenil; Fluorobenzenes; Idazoxan; Indoles; Ketanserin; Male; Mice; Milnacipran; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenols; Prazosin; Punishment; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Selective blockade of 5-HT2A receptors attenuates the increased temperature response in brown adipose tissue to restraint stress in rats.
    Stress (Amsterdam, Netherlands), 2008, Volume: 11, Issue:2

    Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Fluorobenzenes; Male; Phenols; Rats; Rats, Wistar; Restraint, Physical; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological; Tachycardia; Tail; Vasoconstriction

2008
Blockade of 5-HT2A receptors suppresses hyperthermic but not cardiovascular responses to psychosocial stress in rats.
    Neuroscience, 2009, Mar-31, Volume: 159, Issue:3

    Topics: Analysis of Variance; Animals; Blood Pressure; Body Temperature; Cardiovascular System; Electrocardiography; Fever; Fluorobenzenes; Heart Rate; Male; Phenols; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Social Dominance; Stress, Psychological; Tachycardia

2009
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
    Chemical biology & drug design, 2010, Volume: 76, Issue:4

    Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists

2010
Involvement of 5-HT2A receptors in MDMA reinforcement and cue-induced reinstatement of MDMA-seeking behaviour.
    The international journal of neuropsychopharmacology, 2011, Volume: 14, Issue:7

    Topics: Animals; Behavior, Addictive; Cues; Dopamine; Dose-Response Relationship, Drug; Extinction, Psychological; Female; Fluorobenzenes; Locomotion; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Norepinephrine; Nucleus Accumbens; Phenols; Prefrontal Cortex; Receptor, Serotonin, 5-HT2A; Reinforcement, Psychology; Self Administration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2011
Further evidence for the sleep-promoting effects of 5-HT₂A receptor antagonists and demonstration of synergistic effects with the hypnotic, zolpidem in rats.
    Neuropharmacology, 2013, Volume: 70

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hypnotics and Sedatives; Male; Phenols; Piperidines; Pyridines; Rats; Serotonin Antagonists; Sleep Stages; Wakefulness; Zolpidem

2013
Chronic treatment with the serotonin 2A/2C receptor antagonist SR 46349B enhances the retention and efficiency of rule-guided behavior in mice.
    Neurobiology of learning and memory, 2013, Volume: 103

    Topics: Animals; Behavior, Animal; Fluorobenzenes; Male; Maze Learning; Memory; Mice; Phenols; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Reversal Learning; Serotonin 5-HT2 Receptor Antagonists

2013
Blockade of 5-HT2A receptors inhibits emotional hyperthermia in mice.
    The journal of physiological sciences : JPS, 2019, Volume: 69, Issue:6

    Topics: Animals; Fever; Fluorobenzenes; Heart Rate; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phenols; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological

2019