sr 46349b has been researched along with fluorobenzenes in 50 studies
Studies (sr 46349b) | Trials (sr 46349b) | Recent Studies (post-2010) (sr 46349b) | Studies (fluorobenzenes) | Trials (fluorobenzenes) | Recent Studies (post-2010) (fluorobenzenes) |
---|---|---|---|---|---|
51 | 1 | 7 | 3,032 | 581 | 1,214 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 21 (42.00) | 18.2507 |
2000's | 21 (42.00) | 29.6817 |
2010's | 8 (16.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Breliere, JC; Congy, C; Gautret, B; Labeeuw, B; Le Fur, G; Neliat, G; Rinaldi-Carmona, M; Santucci, V; Simiand, J; Soubrie, P | 1 |
Di Pasquale, E; Hilaire, G; Monteau, R | 1 |
Bouaboula, M; Casellas, P; Herbert, JM; Le Fur, G; Poinot-Chazel, C; Prabonnaud, V; Rinaldi-Carmona, M | 1 |
Brelière, JC; Congy, C; Le Fur, G; Pointeau, P; Rinaldi-Carmona, M; Vidal, H | 1 |
Bouaboula, M; Brelière, JC; Casellas, P; Congy, C; Le Fur, G; Oury-Donat, F; Rinaldi-Carmona, M; Shire, D; Simiand, J; Soubrié, P | 1 |
Breliere, JC; Congy, C; Le Fur, G; Oury-Donat, F; Rinaldi-Carmona, M; Simiand, J; Soubrie, P | 1 |
Barthelemy, G; Bernat, A; Dol, F; Herbert, JM; Rinaldi, M | 1 |
Bernat, A; Dol, F; Herbert, JM; Rinaldi, M; Sainte-Marie, M | 1 |
Alexoff, DL; Fowler, JS; Gatley, SJ; King, P; Schlyer, DJ; Shea, C; Wolf, AP | 1 |
Ashworth, S; Hume, SP; Lammertsma, AA; Opacka-Juffry, J; Pike, VW; Shah, F | 1 |
Callas, D; Fareed, J; Herbert, JM; Yang, LH | 1 |
Marcoli, M; Maura, G; Raiteri, M; Tortarolo, M | 1 |
Chaouloff, F; Kulikov, A; Mormède, P | 1 |
Aguerre, S; Chaouloff, F; Gauffre, JC; Mormède, P | 1 |
Berthemy, A; Buhrman, D; Burton, R; Kealy, M; Newton, J; Simpson, H; Wells, D; Wu, D | 1 |
Hjemdahl, P; Ladjevardi, M; Li, N; Wallén, NH | 1 |
Darmani, NA | 1 |
Darmani, NA; Zhao, W | 1 |
Cruz, AP; Morato, S; Motta, VA; Pinheiro, AP; Setem, J | 1 |
De Deurwaerdére, P; Di Giovanni, G; Di Mascio, M; Di Matteo, V; Esposito, E; Spampinato, U | 1 |
Achermann, P; Borbély, AA; Burgess, HJ; Cattelin, F; Finelli, LA; Landolt, HP; Meier, V | 1 |
Caccia, S; De Deurwaerdère, P; Lucas, G | 1 |
Bou-Flores, C; De Maeyer, E; Hilaire, G; Lajard, AM; Lanoir, J; Monteau, R; Seif, I | 1 |
Hashimoto, K; Higuchi, T; Iyo, M; Minabe, Y; Shirayama, Y; Watanabe, K | 1 |
Darmani, NA; Pandya, DK | 1 |
Besson, MJ; Durand, C; Mathieu-Kia, AM; Penit-Soria, J | 1 |
Alboszta, AR; Bonaccorso, S; Dai, J; Ichikawa, J; Li, Z; Meltzer, HY | 1 |
Gray, JA; Joseph, MH; McDonald, LM; Moran, PM; Stephenson, JD; Vythelingum, GN | 2 |
Bubar, MJ; Cunningham, KA; Filip, M | 2 |
Blessing, WW; Nalivaiko, E; Ootsuka, Y | 2 |
Auclair, A; Blanc, G; Glowinski, J; Tassin, JP | 1 |
Blessing, WW; Ootsuka, Y | 1 |
Auclair, A; Cotecchia, S; Drouin, C; Glowinski, J; Tassin, JP | 1 |
Bourin, M; Dailly, E; Hascoët, M; Masse, F | 1 |
Ball, KT; Rebec, GV | 1 |
Miyamoto, M; Terao, A | 1 |
Blanc, G; Gingrich, J; Godeheu, G; Lanteri, C; Salomon, L; Tassin, JP | 1 |
Doucet, EL; Godeheu, G; Hernández Vallejo, SJ; Houades, V; Lanteri, C; Salomon, L; Tassin, JP; Torrens, Y | 1 |
Baumert, M; Beig, MI; Day, TA; Nalivaiko, E; Walker, FR | 1 |
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA | 1 |
Aloyo, VJ; Harvey, JA; Scarlota, LC | 1 |
Lanfumey, L; Maldonado, R; Orejarena, MJ; Robledo, P | 1 |
Arnt, J; Ebdrup, BH; Glenthøj, B; Rasmussen, H | 1 |
Alonso, R; Avenet, P; Beeské, S; Decobert, M; Françon, D; Griebel, G; Jacquet, A; Laufrais, C | 1 |
Dougherty, JP; Oristaglio, J | 1 |
Goto, T; Kohari, D; Okayama, T; Otabi, H; Toyoda, A | 1 |
Ootsuka, Y; Sinh, V | 1 |
2 review(s) available for sr 46349b and fluorobenzenes
Article | Year |
---|---|
[Recent and potential drugs for treatment of insomnia].
Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Diphenhydramine; Drug Design; Fluorobenzenes; GABA-A Receptor Agonists; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Indenes; Orexin Receptors; Phenols; Piperazines; Pyridines; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Serotonin 5-HT2 Receptor Antagonists; Sleep Initiation and Maintenance Disorders; Thiophenes; Zolpidem | 2007 |
Serotonin 2A receptor antagonists for treatment of schizophrenia.
Topics: Antipsychotic Agents; Brain; Fluorobenzenes; Humans; Phenols; Piperidines; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin 5-HT2 Receptor Antagonists; Urea | 2011 |
1 trial(s) available for sr 46349b and fluorobenzenes
Article | Year |
---|---|
Effects of serotonin on platelet activation in whole blood.
Topics: Adenosine Diphosphate; Adult; Analysis of Variance; Female; Flow Cytometry; Fluorobenzenes; Humans; Male; Middle Aged; Phenols; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Reference Values; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Thrombin | 1997 |
47 other study(ies) available for sr 46349b and fluorobenzenes
Article | Year |
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Biochemical and pharmacological properties of SR 46349B, a new potent and selective 5-hydroxytryptamine2 receptor antagonist.
Topics: Animals; Brain; Electroencephalography; Escape Reaction; Female; Fluorobenzenes; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Phenols; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sleep | 1992 |
Further evidence that various 5-HT receptor subtypes modulate central respiratory activity: in vitro studies with SR 46349B.
Topics: Animals; Brain; Fluorobenzenes; Phenols; Rats; Receptors, Serotonin; Respiration; Serotonin Antagonists | 1994 |
Regulation of 5-hydroxytryptamine2 (5-HT2) receptor expression in cultured rat aortic smooth muscle cells by SR 46349B, a selective 5-HT2 receptor antagonist.
Topics: Amphetamines; Animals; Aorta; Base Sequence; Binding Sites; Cells, Cultured; DNA Primers; Fluorobenzenes; Gene Expression Regulation; Ketanserin; Molecular Sequence Data; Muscle, Smooth, Vascular; Phenols; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists | 1994 |
Identification of binding sites for SR 46349B, a 5-hydroxytryptamine2 receptor antagonist, in rodent brain.
Topics: Animals; Binding, Competitive; Brain; Fluorobenzenes; In Vitro Techniques; Ketanserin; Male; Mice; Phenols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1994 |
Up-regulation of 5-HT2 receptors in the rat brain by repeated administration of SR 46349B, a selective 5-HT2 receptor antagonist.
Topics: Amphetamines; Animals; Base Sequence; Blotting, Southern; Brain Chemistry; Cerebral Cortex; Fluorobenzenes; In Vitro Techniques; Inosine Monophosphate; Ketanserin; Male; Molecular Sequence Data; Phenols; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; RNA, Messenger; Second Messenger Systems; Serotonin Antagonists; Serotonin Receptor Agonists; Up-Regulation | 1993 |
Repeated administration of SR 46349B, a selective 5-hydroxytryptamine2 antagonist, up-regulates 5-hydroxytryptamine2 receptors in mouse brain.
Topics: 5-Hydroxytryptophan; Amphetamines; Animals; Brain Chemistry; Fluorobenzenes; In Vitro Techniques; Inositol Phosphates; Ketanserin; Male; Mice; Phenols; Receptors, Serotonin; Serotonin Antagonists; Up-Regulation | 1993 |
Antithrombotic activity of SR 46349, a novel, potent and selective 5-HT2 receptor antagonist.
Topics: Animals; Bleeding Time; Coronary Circulation; Depression, Chemical; Disease Models, Animal; Dogs; Fibrinolytic Agents; Fluorobenzenes; Humans; Ketanserin; Phenols; Platelet Aggregation; Platelet Aggregation Inhibitors; Rabbits; Serotonin Antagonists; Species Specificity; Thrombosis; Vasoconstriction | 1993 |
Potentiating effect of clopidogrel and SR 46349, a novel 5-HT2 antagonist, on streptokinase-induced thrombolysis in the rabbit.
Topics: Animals; Bleeding Time; Clopidogrel; Drug Synergism; Fibrinolytic Agents; Fluorobenzenes; Jugular Veins; Male; Phenols; Platelet Aggregation Inhibitors; Rabbits; Serotonin Antagonists; Streptokinase; Thrombolytic Therapy; Thrombosis; Ticlopidine | 1993 |
Plasma input function determination for PET using a commercial laboratory robot.
Topics: Animals; Benztropine; Blood Chemical Analysis; Carbon Radioisotopes; Cocaine; Fluorobenzenes; Humans; Methylphenidate; Papio; Phenols; Radioisotopes; Reproducibility of Results; Robotics; Selegiline; Tomography, Emission-Computed | 1995 |
Development of central 5-HT2A receptor radioligands for PET: comparison of [3H]RP 62203 and [3H]SR 46349B kinetics in rat brain.
Topics: Animals; Brain; Cyclic S-Oxides; Fluorobenzenes; Kinetics; Male; Models, Theoretical; Naphthalenes; Phenols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Substrate Specificity; Tissue Distribution; Tomography, Emission-Computed; Tritium | 1996 |
Modulation of platelet function and vascular smooth muscle contractile actions by a novel, selective, highly potent 5-HT2 antagonist (SR46349).
Topics: Animals; Dose-Response Relationship, Drug; Fluorobenzenes; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phenols; Platelet Aggregation; Rabbits; Rats; Rats, Sprague-Dawley; Serotonin Antagonists | 1996 |
Serotonin inhibition of the NMDA receptor/nitric oxide/cyclic GMP pathway in rat cerebellum: involvement of 5-hydroxytryptamine2C receptors.
Topics: Adrenergic alpha-Antagonists; Animals; Cerebellum; Cyclic GMP; Excitatory Amino Acid Agonists; Fluorobenzenes; Indoles; Male; N-Methylaspartate; Nitric Oxide; Organ Culture Techniques; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Urea; Yohimbine | 1997 |
Repeated DOI and SR 46349B treatments do not affect elevated plus-maze anxiety despite opposite effects on cortical 5-HT2A receptors.
Topics: Amphetamines; Animals; Anxiety; Behavior, Animal; Body Weight; Cerebral Cortex; Female; Fluorobenzenes; Ketanserin; Male; Maze Learning; Phenols; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
Cortical [3H]ketanserin binding and 5-HT2A receptor-mediated inositol phosphate production in the spontaneously hypertensive rat and Lewis rat strains.
Topics: Amphetamines; Animals; Antihypertensive Agents; Cerebral Cortex; Dose-Response Relationship, Drug; Fluorobenzenes; Frontal Lobe; Inositol Phosphates; Ketanserin; Male; Phenols; Rats; Rats, Inbred Lew; Rats, Inbred SHR; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Species Specificity | 1997 |
High throughput liquid chromatography/mass spectrometry bioanalysis using 96-well disk solid phase extraction plate for the sample preparation.
Topics: Anti-Asthmatic Agents; Benzamides; Cholinergic Agents; Chromatography, Liquid; Fluorobenzenes; Humans; Indicator Dilution Techniques; Mass Spectrometry; Pharmaceutical Preparations; Phenols; Piperidines; Propylamines; Pyridazines; Receptors, Neurokinin-2; Robotics; Serotonin Antagonists | 1998 |
The silent and selective 5-HT1A antagonist, WAY 100635, produces via an indirect mechanism, a 5-HT2A receptor-mediated behaviour in mice during the day but not at night. Short communication.
Topics: Animals; Behavior, Animal; Circadian Rhythm; Dose-Response Relationship, Drug; Fluorobenzenes; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR; Phenols; Piperazines; Pyridines; Receptors, Serotonin; Serotonin Antagonists | 1998 |
Production of serotonin syndrome by 8-OH DPAT in Cryptotis parva.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Fluorobenzenes; Injections, Intraperitoneal; Male; Phenols; Piperazines; Propranolol; Serotonin Antagonists; Serotonin Receptor Agonists; Serotonin Syndrome; Shrews | 1998 |
Ethopharmacological analysis of 5-HT ligands on the rat elevated plus-maze.
Topics: Animals; Anxiety; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Cyclic S-Oxides; Exploratory Behavior; Fluorobenzenes; Indoles; Male; Naphthalenes; Phenols; Piperazines; Pyrimidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Risk Assessment; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Selective blockade of serotonin-2C/2B receptors enhances mesolimbic and mesostriatal dopaminergic function: a combined in vivo electrophysiological and microdialysis study.
Topics: Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Electrophysiology; Evoked Potentials; Fluorobenzenes; Indoles; Limbic System; Male; Microdialysis; Neurons; Nucleus Accumbens; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tegmentum Mesencephali | 1999 |
Serotonin-2 receptors and human sleep: effect of a selective antagonist on EEG power spectra.
Topics: Adult; Body Temperature; Electroencephalography; Fluorobenzenes; Heart Rate; Humans; Male; Phenols; Receptors, Serotonin; Serotonin Antagonists; Sleep; Sleep Stages | 1999 |
The effect of serotonergic agents on haloperidol-induced striatal dopamine release in vivo: opposite role of 5-HT(2A) and 5-HT(2C) receptor subtypes and significance of the haloperidol dose used.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Fluorobenzenes; Haloperidol; Indoles; Male; Microdialysis; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Abnormal phrenic motoneuron activity and morphology in neonatal monoamine oxidase A-deficient transgenic mice: possible role of a serotonin excess.
Topics: Animals; Animals, Newborn; Brain; Dendrites; Female; Fetus; Fluorobenzenes; Medulla Oblongata; Mice; Mice, Inbred C3H; Mice, Knockout; Mice, Transgenic; Monoamine Oxidase; Motor Neurons; Patch-Clamp Techniques; Phenols; Phrenic Nerve; Pregnancy; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Respiratory Mechanics; Serotonin; Serotonin Antagonists; Spinal Cord | 2000 |
3,4-methylenedioxymethamphetamine (MDMA, ecstasy)-induced egr-1 mRNA in rat brain: pharmacological manipulation.
Topics: Animals; Benzazepines; Brain Chemistry; Dizocilpine Maleate; DNA-Binding Proteins; Dopamine Antagonists; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Fluorobenzenes; Hallucinogens; Immediate-Early Proteins; Immunohistochemistry; In Situ Hybridization; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Phenols; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Transcription Factors | 2000 |
Involvement of other neurotransmitters in behaviors induced by the cannabinoid CB1 receptor antagonist SR 141716A in naive mice.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Dronabinol; Excitatory Amino Acid Antagonists; Fluorobenzenes; Glutamic Acid; Head Movements; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR; Neurotransmitter Agents; Phenols; Piperidines; Psychotropic Drugs; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Serotonin Antagonists; Tachykinins | 2000 |
Regulation of striatal neuropeptide mRNAs: effects of the 5-HT(2) antagonist SR46349B in adult rats with a neonatal 6-hydroxydopamine lesion.
Topics: Animals; Animals, Newborn; Denervation; Dopamine; Down-Regulation; Enkephalins; Fluorobenzenes; Neostriatum; Neurons; Neuropeptides; Oxidopamine; Phenols; Protein Precursors; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Sympatholytics; Tachykinins; Up-Regulation | 2002 |
SR46349-B, a 5-HT(2A/2C) receptor antagonist, potentiates haloperidol-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
Topics: Analysis of Variance; Animals; Dopamine; Dopamine Antagonists; Drug Synergism; Fluorobenzenes; Haloperidol; Male; Nucleus Accumbens; Phenols; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Telencephalon | 2002 |
Latent inhibition is attenuated by noise and partially restored by a 5-HT2A receptor antagonist.
Topics: Animals; Conditioning, Operant; Extinction, Psychological; Fluorobenzenes; Male; Noise; Phenols; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reflex, Startle; Serotonin Antagonists; Stress, Psychological | 2002 |
Enhancement of latent inhibition by two 5-HT2A receptor antagonists only when given at both pre-exposure and conditioning.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Amphetamine; Analysis of Variance; Animals; Association Learning; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Classical; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; Inhibition, Psychological; Male; Phencyclidine; Phenols; Quinolines; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Stereotyped Behavior | 2003 |
Contribution of serotonin (5-hydroxytryptamine; 5-HT) 5-HT2 receptor subtypes to the hyperlocomotor effects of cocaine: acute and chronic pharmacological analyses.
Topics: Amphetamines; Animals; Cocaine; Drug Interactions; Fluorobenzenes; Hyperkinesis; Indoles; Male; Phenols; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes | 2004 |
Spinal 5-HT2A receptors regulate cutaneous sympathetic vasomotor outflow in rabbits and rats; relevance for cutaneous vasoconstriction elicited by MDMA (3,4-methylenedioxymethamphetamine, "Ecstasy") and its reversal by clozapine.
Topics: Animals; Clozapine; Ear, External; Fluorobenzenes; Injections, Intravenous; N-Methyl-3,4-methylenedioxyamphetamine; Phenols; Rabbits; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Skin; Spine; Tail; Ultrasonography, Doppler, Pulsed; Vasoconstriction; Vasomotor System | 2004 |
Role of serotonin 2A receptors in the D-amphetamine-induced release of dopamine: comparison with previous data on alpha1b-adrenergic receptors.
Topics: Animals; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Antagonism; Extracellular Fluid; Fluorobenzenes; Male; Microdialysis; Motor Activity; Neurons; Nucleus Accumbens; Phenols; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Ventral Tegmental Area | 2004 |
Activation of slowly conducting medullary raphe-spinal neurons, including serotonergic neurons, increases cutaneous sympathetic vasomotor discharge in rabbit.
Topics: Anesthesia; Animals; Axons; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Fluorobenzenes; Injections, Spinal; Kynurenic Acid; Male; Medulla Oblongata; Neural Conduction; Neural Pathways; Neurons; Phenols; Rabbits; Raphe Nuclei; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Skin; Spinal Cord; Sympathetic Nervous System; Trigeminal Nerve | 2005 |
5-HT2A and alpha1b-adrenergic receptors entirely mediate dopamine release, locomotor response and behavioural sensitization to opiates and psychostimulants.
Topics: Adrenergic alpha-Antagonists; Anesthetics, Local; Animals; Behavior, Animal; Brain Chemistry; Central Nervous System Stimulants; Cocaine; Corpus Striatum; Dextroamphetamine; Dopamine; Drug Administration Schedule; Drug Interactions; Fluorobenzenes; Male; Mice; Mice, Knockout; Microdialysis; Motor Activity; Narcotics; Phenols; Prazosin; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Time Factors | 2004 |
Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzylamines; Brain; Cyclopropanes; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Flumazenil; Fluorobenzenes; Idazoxan; Indoles; Ketanserin; Male; Mice; Milnacipran; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenols; Prazosin; Punishment; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2005 |
Role of 5-HT2A and 5-HT2C/B receptors in the acute effects of 3,4-methylenedioxymethamphetamine (MDMA) on striatal single-unit activity and locomotion in freely moving rats.
Topics: Amphetamine-Related Disorders; Animals; Corpus Striatum; Dopamine; Electroencephalography; Fluorobenzenes; Indoles; Male; N-Methyl-3,4-methylenedioxyamphetamine; Neurons; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists | 2005 |
Contribution of serotonin (5-HT) 5-HT2 receptor subtypes to the discriminative stimulus effects of cocaine in rats.
Topics: Animals; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Fluorobenzenes; Indoles; Male; Naphthyridines; Phenols; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Reinforcement Schedule; Serotonin Antagonists; Serotonin Receptor Agonists; Stimulation, Chemical; Urea | 2006 |
Paradoxical constitutive behavioral sensitization to amphetamine in mice lacking 5-HT2A receptors.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Behavior, Animal; Central Nervous System Stimulants; Dextroamphetamine; Dose-Response Relationship, Drug; Fluorobenzenes; Histamine H2 Antagonists; Mice; Mice, Knockout; Motor Activity; Phenols; Prazosin; Receptor, Serotonin, 5-HT2A | 2007 |
Selective blockade of 5-HT2A receptors attenuates the increased temperature response in brown adipose tissue to restraint stress in rats.
Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Fluorobenzenes; Male; Phenols; Rats; Rats, Wistar; Restraint, Physical; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological; Tachycardia; Tail; Vasoconstriction | 2008 |
Inhibition of monoamine oxidases desensitizes 5-HT1A autoreceptors and allows nicotine to induce a neurochemical and behavioral sensitization.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Behavior, Animal; Brain Chemistry; Drug Combinations; Fluorobenzenes; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nicotine; Nicotinic Agonists; Phenols; Piperazines; Prazosin; Pyridines; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists; Tranylcypromine | 2009 |
Blockade of 5-HT2A receptors suppresses hyperthermic but not cardiovascular responses to psychosocial stress in rats.
Topics: Analysis of Variance; Animals; Blood Pressure; Body Temperature; Cardiovascular System; Electrocardiography; Fever; Fluorobenzenes; Heart Rate; Male; Phenols; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Social Dominance; Stress, Psychological; Tachycardia | 2009 |
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists | 2010 |
The role of serotonin-2 (5-HT2) and dopamine receptors in the behavioral actions of the 5-HT2A/2C agonist, DOI, and putative 5-HT2C inverse agonist, SR46349B.
Topics: Amphetamines; Animals; Antipsychotic Agents; Fluorobenzenes; Head Movements; Male; Phenols; Rabbits; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists | 2011 |
Involvement of 5-HT2A receptors in MDMA reinforcement and cue-induced reinstatement of MDMA-seeking behaviour.
Topics: Animals; Behavior, Addictive; Cues; Dopamine; Dose-Response Relationship, Drug; Extinction, Psychological; Female; Fluorobenzenes; Locomotion; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Norepinephrine; Nucleus Accumbens; Phenols; Prefrontal Cortex; Receptor, Serotonin, 5-HT2A; Reinforcement, Psychology; Self Administration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2011 |
Further evidence for the sleep-promoting effects of 5-HT₂A receptor antagonists and demonstration of synergistic effects with the hypnotic, zolpidem in rats.
Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hypnotics and Sedatives; Male; Phenols; Piperidines; Pyridines; Rats; Serotonin Antagonists; Sleep Stages; Wakefulness; Zolpidem | 2013 |
Chronic treatment with the serotonin 2A/2C receptor antagonist SR 46349B enhances the retention and efficiency of rule-guided behavior in mice.
Topics: Animals; Behavior, Animal; Fluorobenzenes; Male; Maze Learning; Memory; Mice; Phenols; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Reversal Learning; Serotonin 5-HT2 Receptor Antagonists | 2013 |
The acute social defeat stress and nest-building test paradigm: A potential new method to screen drugs for depressive-like symptoms.
Topics: Animals; Depression; Disease Models, Animal; Dominance-Subordination; Fluorobenzenes; Fluoxetine; Male; Mice; Mice, Inbred C57BL; Nesting Behavior; Phenols; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stress, Psychological | 2017 |
Blockade of 5-HT2A receptors inhibits emotional hyperthermia in mice.
Topics: Animals; Fever; Fluorobenzenes; Heart Rate; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phenols; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological | 2019 |