Page last updated: 2024-09-03

sr 46349b and fluorobenzenes

sr 46349b has been researched along with fluorobenzenes in 50 studies

Compound Research Comparison

Studies
(sr 46349b)
Trials
(sr 46349b)
Recent Studies (post-2010)
(sr 46349b)
Studies
(fluorobenzenes)
Trials
(fluorobenzenes)
Recent Studies (post-2010) (fluorobenzenes)
51173,0325811,214

Research

Studies (50)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's21 (42.00)18.2507
2000's21 (42.00)29.6817
2010's8 (16.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Breliere, JC; Congy, C; Gautret, B; Labeeuw, B; Le Fur, G; Neliat, G; Rinaldi-Carmona, M; Santucci, V; Simiand, J; Soubrie, P1
Di Pasquale, E; Hilaire, G; Monteau, R1
Bouaboula, M; Casellas, P; Herbert, JM; Le Fur, G; Poinot-Chazel, C; Prabonnaud, V; Rinaldi-Carmona, M1
Brelière, JC; Congy, C; Le Fur, G; Pointeau, P; Rinaldi-Carmona, M; Vidal, H1
Bouaboula, M; Brelière, JC; Casellas, P; Congy, C; Le Fur, G; Oury-Donat, F; Rinaldi-Carmona, M; Shire, D; Simiand, J; Soubrié, P1
Breliere, JC; Congy, C; Le Fur, G; Oury-Donat, F; Rinaldi-Carmona, M; Simiand, J; Soubrie, P1
Barthelemy, G; Bernat, A; Dol, F; Herbert, JM; Rinaldi, M1
Bernat, A; Dol, F; Herbert, JM; Rinaldi, M; Sainte-Marie, M1
Alexoff, DL; Fowler, JS; Gatley, SJ; King, P; Schlyer, DJ; Shea, C; Wolf, AP1
Ashworth, S; Hume, SP; Lammertsma, AA; Opacka-Juffry, J; Pike, VW; Shah, F1
Callas, D; Fareed, J; Herbert, JM; Yang, LH1
Marcoli, M; Maura, G; Raiteri, M; Tortarolo, M1
Chaouloff, F; Kulikov, A; Mormède, P1
Aguerre, S; Chaouloff, F; Gauffre, JC; Mormède, P1
Berthemy, A; Buhrman, D; Burton, R; Kealy, M; Newton, J; Simpson, H; Wells, D; Wu, D1
Hjemdahl, P; Ladjevardi, M; Li, N; Wallén, NH1
Darmani, NA1
Darmani, NA; Zhao, W1
Cruz, AP; Morato, S; Motta, VA; Pinheiro, AP; Setem, J1
De Deurwaerdére, P; Di Giovanni, G; Di Mascio, M; Di Matteo, V; Esposito, E; Spampinato, U1
Achermann, P; Borbély, AA; Burgess, HJ; Cattelin, F; Finelli, LA; Landolt, HP; Meier, V1
Caccia, S; De Deurwaerdère, P; Lucas, G1
Bou-Flores, C; De Maeyer, E; Hilaire, G; Lajard, AM; Lanoir, J; Monteau, R; Seif, I1
Hashimoto, K; Higuchi, T; Iyo, M; Minabe, Y; Shirayama, Y; Watanabe, K1
Darmani, NA; Pandya, DK1
Besson, MJ; Durand, C; Mathieu-Kia, AM; Penit-Soria, J1
Alboszta, AR; Bonaccorso, S; Dai, J; Ichikawa, J; Li, Z; Meltzer, HY1
Gray, JA; Joseph, MH; McDonald, LM; Moran, PM; Stephenson, JD; Vythelingum, GN2
Bubar, MJ; Cunningham, KA; Filip, M2
Blessing, WW; Nalivaiko, E; Ootsuka, Y2
Auclair, A; Blanc, G; Glowinski, J; Tassin, JP1
Blessing, WW; Ootsuka, Y1
Auclair, A; Cotecchia, S; Drouin, C; Glowinski, J; Tassin, JP1
Bourin, M; Dailly, E; Hascoët, M; Masse, F1
Ball, KT; Rebec, GV1
Miyamoto, M; Terao, A1
Blanc, G; Gingrich, J; Godeheu, G; Lanteri, C; Salomon, L; Tassin, JP1
Doucet, EL; Godeheu, G; Hernández Vallejo, SJ; Houades, V; Lanteri, C; Salomon, L; Tassin, JP; Torrens, Y1
Baumert, M; Beig, MI; Day, TA; Nalivaiko, E; Walker, FR1
Herth, MM; Knudsen, GM; Kramer, V; Palner, M; Rösch, F; Santini, MA1
Aloyo, VJ; Harvey, JA; Scarlota, LC1
Lanfumey, L; Maldonado, R; Orejarena, MJ; Robledo, P1
Arnt, J; Ebdrup, BH; Glenthøj, B; Rasmussen, H1
Alonso, R; Avenet, P; Beeské, S; Decobert, M; Françon, D; Griebel, G; Jacquet, A; Laufrais, C1
Dougherty, JP; Oristaglio, J1
Goto, T; Kohari, D; Okayama, T; Otabi, H; Toyoda, A1
Ootsuka, Y; Sinh, V1

Reviews

2 review(s) available for sr 46349b and fluorobenzenes

ArticleYear
[Recent and potential drugs for treatment of insomnia].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2007, Volume: 129, Issue:1

    Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Diphenhydramine; Drug Design; Fluorobenzenes; GABA-A Receptor Agonists; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Indenes; Orexin Receptors; Phenols; Piperazines; Pyridines; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Serotonin 5-HT2 Receptor Antagonists; Sleep Initiation and Maintenance Disorders; Thiophenes; Zolpidem

2007
Serotonin 2A receptor antagonists for treatment of schizophrenia.
    Expert opinion on investigational drugs, 2011, Volume: 20, Issue:9

    Topics: Antipsychotic Agents; Brain; Fluorobenzenes; Humans; Phenols; Piperidines; Positron-Emission Tomography; Receptor, Serotonin, 5-HT2A; Schizophrenia; Serotonin 5-HT2 Receptor Antagonists; Urea

2011

Trials

1 trial(s) available for sr 46349b and fluorobenzenes

ArticleYear
Effects of serotonin on platelet activation in whole blood.
    Blood coagulation & fibrinolysis : an international journal in haemostasis and thrombosis, 1997, Volume: 8, Issue:8

    Topics: Adenosine Diphosphate; Adult; Analysis of Variance; Female; Flow Cytometry; Fluorobenzenes; Humans; Male; Middle Aged; Phenols; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Reference Values; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Thrombin

1997

Other Studies

47 other study(ies) available for sr 46349b and fluorobenzenes

ArticleYear
Biochemical and pharmacological properties of SR 46349B, a new potent and selective 5-hydroxytryptamine2 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Animals; Brain; Electroencephalography; Escape Reaction; Female; Fluorobenzenes; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Phenols; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sleep

1992
Further evidence that various 5-HT receptor subtypes modulate central respiratory activity: in vitro studies with SR 46349B.
    European journal of pharmacology, 1994, Jun-23, Volume: 259, Issue:1

    Topics: Animals; Brain; Fluorobenzenes; Phenols; Rats; Receptors, Serotonin; Respiration; Serotonin Antagonists

1994
Regulation of 5-hydroxytryptamine2 (5-HT2) receptor expression in cultured rat aortic smooth muscle cells by SR 46349B, a selective 5-HT2 receptor antagonist.
    The Journal of biological chemistry, 1994, Jan-07, Volume: 269, Issue:1

    Topics: Amphetamines; Animals; Aorta; Base Sequence; Binding Sites; Cells, Cultured; DNA Primers; Fluorobenzenes; Gene Expression Regulation; Ketanserin; Molecular Sequence Data; Muscle, Smooth, Vascular; Phenols; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists

1994
Identification of binding sites for SR 46349B, a 5-hydroxytryptamine2 receptor antagonist, in rodent brain.
    Life sciences, 1994, Volume: 54, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Fluorobenzenes; In Vitro Techniques; Ketanserin; Male; Mice; Phenols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1994
Up-regulation of 5-HT2 receptors in the rat brain by repeated administration of SR 46349B, a selective 5-HT2 receptor antagonist.
    European journal of pharmacology, 1993, Jun-15, Volume: 246, Issue:1

    Topics: Amphetamines; Animals; Base Sequence; Blotting, Southern; Brain Chemistry; Cerebral Cortex; Fluorobenzenes; In Vitro Techniques; Inosine Monophosphate; Ketanserin; Male; Molecular Sequence Data; Phenols; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; RNA, Messenger; Second Messenger Systems; Serotonin Antagonists; Serotonin Receptor Agonists; Up-Regulation

1993
Repeated administration of SR 46349B, a selective 5-hydroxytryptamine2 antagonist, up-regulates 5-hydroxytryptamine2 receptors in mouse brain.
    Molecular pharmacology, 1993, Volume: 43, Issue:1

    Topics: 5-Hydroxytryptophan; Amphetamines; Animals; Brain Chemistry; Fluorobenzenes; In Vitro Techniques; Inositol Phosphates; Ketanserin; Male; Mice; Phenols; Receptors, Serotonin; Serotonin Antagonists; Up-Regulation

1993
Antithrombotic activity of SR 46349, a novel, potent and selective 5-HT2 receptor antagonist.
    Thrombosis and haemostasis, 1993, Mar-01, Volume: 69, Issue:3

    Topics: Animals; Bleeding Time; Coronary Circulation; Depression, Chemical; Disease Models, Animal; Dogs; Fibrinolytic Agents; Fluorobenzenes; Humans; Ketanserin; Phenols; Platelet Aggregation; Platelet Aggregation Inhibitors; Rabbits; Serotonin Antagonists; Species Specificity; Thrombosis; Vasoconstriction

1993
Potentiating effect of clopidogrel and SR 46349, a novel 5-HT2 antagonist, on streptokinase-induced thrombolysis in the rabbit.
    Thrombosis and haemostasis, 1993, Mar-01, Volume: 69, Issue:3

    Topics: Animals; Bleeding Time; Clopidogrel; Drug Synergism; Fibrinolytic Agents; Fluorobenzenes; Jugular Veins; Male; Phenols; Platelet Aggregation Inhibitors; Rabbits; Serotonin Antagonists; Streptokinase; Thrombolytic Therapy; Thrombosis; Ticlopidine

1993
Plasma input function determination for PET using a commercial laboratory robot.
    Nuclear medicine and biology, 1995, Volume: 22, Issue:7

    Topics: Animals; Benztropine; Blood Chemical Analysis; Carbon Radioisotopes; Cocaine; Fluorobenzenes; Humans; Methylphenidate; Papio; Phenols; Radioisotopes; Reproducibility of Results; Robotics; Selegiline; Tomography, Emission-Computed

1995
Development of central 5-HT2A receptor radioligands for PET: comparison of [3H]RP 62203 and [3H]SR 46349B kinetics in rat brain.
    Nuclear medicine and biology, 1996, Volume: 23, Issue:3

    Topics: Animals; Brain; Cyclic S-Oxides; Fluorobenzenes; Kinetics; Male; Models, Theoretical; Naphthalenes; Phenols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Substrate Specificity; Tissue Distribution; Tomography, Emission-Computed; Tritium

1996
Modulation of platelet function and vascular smooth muscle contractile actions by a novel, selective, highly potent 5-HT2 antagonist (SR46349).
    Thrombosis research, 1996, Mar-01, Volume: 81, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Fluorobenzenes; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phenols; Platelet Aggregation; Rabbits; Rats; Rats, Sprague-Dawley; Serotonin Antagonists

1996
Serotonin inhibition of the NMDA receptor/nitric oxide/cyclic GMP pathway in rat cerebellum: involvement of 5-hydroxytryptamine2C receptors.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebellum; Cyclic GMP; Excitatory Amino Acid Agonists; Fluorobenzenes; Indoles; Male; N-Methylaspartate; Nitric Oxide; Organ Culture Techniques; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Urea; Yohimbine

1997
Repeated DOI and SR 46349B treatments do not affect elevated plus-maze anxiety despite opposite effects on cortical 5-HT2A receptors.
    European journal of pharmacology, 1997, Sep-03, Volume: 334, Issue:1

    Topics: Amphetamines; Animals; Anxiety; Behavior, Animal; Body Weight; Cerebral Cortex; Female; Fluorobenzenes; Ketanserin; Male; Maze Learning; Phenols; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Cortical [3H]ketanserin binding and 5-HT2A receptor-mediated inositol phosphate production in the spontaneously hypertensive rat and Lewis rat strains.
    Neuroscience letters, 1997, Oct-31, Volume: 236, Issue:2

    Topics: Amphetamines; Animals; Antihypertensive Agents; Cerebral Cortex; Dose-Response Relationship, Drug; Fluorobenzenes; Frontal Lobe; Inositol Phosphates; Ketanserin; Male; Phenols; Rats; Rats, Inbred Lew; Rats, Inbred SHR; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Species Specificity

1997
High throughput liquid chromatography/mass spectrometry bioanalysis using 96-well disk solid phase extraction plate for the sample preparation.
    Rapid communications in mass spectrometry : RCM, 1998, Volume: 12, Issue:2

    Topics: Anti-Asthmatic Agents; Benzamides; Cholinergic Agents; Chromatography, Liquid; Fluorobenzenes; Humans; Indicator Dilution Techniques; Mass Spectrometry; Pharmaceutical Preparations; Phenols; Piperidines; Propylamines; Pyridazines; Receptors, Neurokinin-2; Robotics; Serotonin Antagonists

1998
The silent and selective 5-HT1A antagonist, WAY 100635, produces via an indirect mechanism, a 5-HT2A receptor-mediated behaviour in mice during the day but not at night. Short communication.
    Journal of neural transmission (Vienna, Austria : 1996), 1998, Volume: 105, Issue:6-7

    Topics: Animals; Behavior, Animal; Circadian Rhythm; Dose-Response Relationship, Drug; Fluorobenzenes; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR; Phenols; Piperazines; Pyridines; Receptors, Serotonin; Serotonin Antagonists

1998
Production of serotonin syndrome by 8-OH DPAT in Cryptotis parva.
    Physiology & behavior, 1998, Nov-15, Volume: 65, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Fluorobenzenes; Injections, Intraperitoneal; Male; Phenols; Piperazines; Propranolol; Serotonin Antagonists; Serotonin Receptor Agonists; Serotonin Syndrome; Shrews

1998
Ethopharmacological analysis of 5-HT ligands on the rat elevated plus-maze.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 62, Issue:3

    Topics: Animals; Anxiety; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Cyclic S-Oxides; Exploratory Behavior; Fluorobenzenes; Indoles; Male; Naphthalenes; Phenols; Piperazines; Pyrimidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Risk Assessment; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Selective blockade of serotonin-2C/2B receptors enhances mesolimbic and mesostriatal dopaminergic function: a combined in vivo electrophysiological and microdialysis study.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Electrophysiology; Evoked Potentials; Fluorobenzenes; Indoles; Limbic System; Male; Microdialysis; Neurons; Nucleus Accumbens; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tegmentum Mesencephali

1999
Serotonin-2 receptors and human sleep: effect of a selective antagonist on EEG power spectra.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1999, Volume: 21, Issue:3

    Topics: Adult; Body Temperature; Electroencephalography; Fluorobenzenes; Heart Rate; Humans; Male; Phenols; Receptors, Serotonin; Serotonin Antagonists; Sleep; Sleep Stages

1999
The effect of serotonergic agents on haloperidol-induced striatal dopamine release in vivo: opposite role of 5-HT(2A) and 5-HT(2C) receptor subtypes and significance of the haloperidol dose used.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Fluorobenzenes; Haloperidol; Indoles; Male; Microdialysis; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Abnormal phrenic motoneuron activity and morphology in neonatal monoamine oxidase A-deficient transgenic mice: possible role of a serotonin excess.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Jun-15, Volume: 20, Issue:12

    Topics: Animals; Animals, Newborn; Brain; Dendrites; Female; Fetus; Fluorobenzenes; Medulla Oblongata; Mice; Mice, Inbred C3H; Mice, Knockout; Mice, Transgenic; Monoamine Oxidase; Motor Neurons; Patch-Clamp Techniques; Phenols; Phrenic Nerve; Pregnancy; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Respiratory Mechanics; Serotonin; Serotonin Antagonists; Spinal Cord

2000
3,4-methylenedioxymethamphetamine (MDMA, ecstasy)-induced egr-1 mRNA in rat brain: pharmacological manipulation.
    European journal of pharmacology, 2000, Aug-25, Volume: 402, Issue:3

    Topics: Animals; Benzazepines; Brain Chemistry; Dizocilpine Maleate; DNA-Binding Proteins; Dopamine Antagonists; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Fluorobenzenes; Hallucinogens; Immediate-Early Proteins; Immunohistochemistry; In Situ Hybridization; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Phenols; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Transcription Factors

2000
Involvement of other neurotransmitters in behaviors induced by the cannabinoid CB1 receptor antagonist SR 141716A in naive mice.
    Journal of neural transmission (Vienna, Austria : 1996), 2000, Volume: 107, Issue:8-9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Dronabinol; Excitatory Amino Acid Antagonists; Fluorobenzenes; Glutamic Acid; Head Movements; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR; Neurotransmitter Agents; Phenols; Piperidines; Psychotropic Drugs; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Serotonin Antagonists; Tachykinins

2000
Regulation of striatal neuropeptide mRNAs: effects of the 5-HT(2) antagonist SR46349B in adult rats with a neonatal 6-hydroxydopamine lesion.
    Journal of neuroscience research, 2002, Jan-01, Volume: 67, Issue:1

    Topics: Animals; Animals, Newborn; Denervation; Dopamine; Down-Regulation; Enkephalins; Fluorobenzenes; Neostriatum; Neurons; Neuropeptides; Oxidopamine; Phenols; Protein Precursors; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Sympatholytics; Tachykinins; Up-Regulation

2002
SR46349-B, a 5-HT(2A/2C) receptor antagonist, potentiates haloperidol-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 27, Issue:3

    Topics: Analysis of Variance; Animals; Dopamine; Dopamine Antagonists; Drug Synergism; Fluorobenzenes; Haloperidol; Male; Nucleus Accumbens; Phenols; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Telencephalon

2002
Latent inhibition is attenuated by noise and partially restored by a 5-HT2A receptor antagonist.
    Behavioural pharmacology, 2002, Volume: 13, Issue:8

    Topics: Animals; Conditioning, Operant; Extinction, Psychological; Fluorobenzenes; Male; Noise; Phenols; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reflex, Startle; Serotonin Antagonists; Stress, Psychological

2002
Enhancement of latent inhibition by two 5-HT2A receptor antagonists only when given at both pre-exposure and conditioning.
    Psychopharmacology, 2003, Volume: 169, Issue:3-4

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Amphetamine; Analysis of Variance; Animals; Association Learning; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Classical; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; Inhibition, Psychological; Male; Phencyclidine; Phenols; Quinolines; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Stereotyped Behavior

2003
Contribution of serotonin (5-hydroxytryptamine; 5-HT) 5-HT2 receptor subtypes to the hyperlocomotor effects of cocaine: acute and chronic pharmacological analyses.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 310, Issue:3

    Topics: Amphetamines; Animals; Cocaine; Drug Interactions; Fluorobenzenes; Hyperkinesis; Indoles; Male; Phenols; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

2004
Spinal 5-HT2A receptors regulate cutaneous sympathetic vasomotor outflow in rabbits and rats; relevance for cutaneous vasoconstriction elicited by MDMA (3,4-methylenedioxymethamphetamine, "Ecstasy") and its reversal by clozapine.
    Brain research, 2004, Jul-16, Volume: 1014, Issue:1-2

    Topics: Animals; Clozapine; Ear, External; Fluorobenzenes; Injections, Intravenous; N-Methyl-3,4-methylenedioxyamphetamine; Phenols; Rabbits; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Skin; Spine; Tail; Ultrasonography, Doppler, Pulsed; Vasoconstriction; Vasomotor System

2004
Role of serotonin 2A receptors in the D-amphetamine-induced release of dopamine: comparison with previous data on alpha1b-adrenergic receptors.
    Journal of neurochemistry, 2004, Volume: 91, Issue:2

    Topics: Animals; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Antagonism; Extracellular Fluid; Fluorobenzenes; Male; Microdialysis; Motor Activity; Neurons; Nucleus Accumbens; Phenols; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Ventral Tegmental Area

2004
Activation of slowly conducting medullary raphe-spinal neurons, including serotonergic neurons, increases cutaneous sympathetic vasomotor discharge in rabbit.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2005, Volume: 288, Issue:4

    Topics: Anesthesia; Animals; Axons; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Fluorobenzenes; Injections, Spinal; Kynurenic Acid; Male; Medulla Oblongata; Neural Conduction; Neural Pathways; Neurons; Phenols; Rabbits; Raphe Nuclei; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Skin; Spinal Cord; Sympathetic Nervous System; Trigeminal Nerve

2005
5-HT2A and alpha1b-adrenergic receptors entirely mediate dopamine release, locomotor response and behavioural sensitization to opiates and psychostimulants.
    The European journal of neuroscience, 2004, Volume: 20, Issue:11

    Topics: Adrenergic alpha-Antagonists; Anesthetics, Local; Animals; Behavior, Animal; Brain Chemistry; Central Nervous System Stimulants; Cocaine; Corpus Striatum; Dextroamphetamine; Dopamine; Drug Administration Schedule; Drug Interactions; Fluorobenzenes; Male; Mice; Mice, Knockout; Microdialysis; Motor Activity; Narcotics; Phenols; Prazosin; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Time Factors

2004
Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzylamines; Brain; Cyclopropanes; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Flumazenil; Fluorobenzenes; Idazoxan; Indoles; Ketanserin; Male; Mice; Milnacipran; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenols; Prazosin; Punishment; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Role of 5-HT2A and 5-HT2C/B receptors in the acute effects of 3,4-methylenedioxymethamphetamine (MDMA) on striatal single-unit activity and locomotion in freely moving rats.
    Psychopharmacology, 2005, Volume: 181, Issue:4

    Topics: Amphetamine-Related Disorders; Animals; Corpus Striatum; Dopamine; Electroencephalography; Fluorobenzenes; Indoles; Male; N-Methyl-3,4-methylenedioxyamphetamine; Neurons; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists

2005
Contribution of serotonin (5-HT) 5-HT2 receptor subtypes to the discriminative stimulus effects of cocaine in rats.
    Psychopharmacology, 2006, Volume: 183, Issue:4

    Topics: Animals; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Fluorobenzenes; Indoles; Male; Naphthyridines; Phenols; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Reinforcement Schedule; Serotonin Antagonists; Serotonin Receptor Agonists; Stimulation, Chemical; Urea

2006
Paradoxical constitutive behavioral sensitization to amphetamine in mice lacking 5-HT2A receptors.
    Psychopharmacology, 2007, Volume: 194, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Behavior, Animal; Central Nervous System Stimulants; Dextroamphetamine; Dose-Response Relationship, Drug; Fluorobenzenes; Histamine H2 Antagonists; Mice; Mice, Knockout; Motor Activity; Phenols; Prazosin; Receptor, Serotonin, 5-HT2A

2007
Selective blockade of 5-HT2A receptors attenuates the increased temperature response in brown adipose tissue to restraint stress in rats.
    Stress (Amsterdam, Netherlands), 2008, Volume: 11, Issue:2

    Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Fluorobenzenes; Male; Phenols; Rats; Rats, Wistar; Restraint, Physical; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological; Tachycardia; Tail; Vasoconstriction

2008
Inhibition of monoamine oxidases desensitizes 5-HT1A autoreceptors and allows nicotine to induce a neurochemical and behavioral sensitization.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Jan-28, Volume: 29, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Behavior, Animal; Brain Chemistry; Drug Combinations; Fluorobenzenes; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nicotine; Nicotinic Agonists; Phenols; Piperazines; Prazosin; Pyridines; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists; Tranylcypromine

2009
Blockade of 5-HT2A receptors suppresses hyperthermic but not cardiovascular responses to psychosocial stress in rats.
    Neuroscience, 2009, Mar-31, Volume: 159, Issue:3

    Topics: Analysis of Variance; Animals; Blood Pressure; Body Temperature; Cardiovascular System; Electrocardiography; Fever; Fluorobenzenes; Heart Rate; Male; Phenols; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Social Dominance; Stress, Psychological; Tachycardia

2009
Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
    Chemical biology & drug design, 2010, Volume: 76, Issue:4

    Topics: Binding, Competitive; Combinatorial Chemistry Techniques; Fluorobenzenes; Hydrophobic and Hydrophilic Interactions; Ketanserin; Ligands; Phenols; Piperidines; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists

2010
The role of serotonin-2 (5-HT2) and dopamine receptors in the behavioral actions of the 5-HT2A/2C agonist, DOI, and putative 5-HT2C inverse agonist, SR46349B.
    Psychopharmacology, 2011, Volume: 213, Issue:2-3

    Topics: Amphetamines; Animals; Antipsychotic Agents; Fluorobenzenes; Head Movements; Male; Phenols; Rabbits; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists

2011
Involvement of 5-HT2A receptors in MDMA reinforcement and cue-induced reinstatement of MDMA-seeking behaviour.
    The international journal of neuropsychopharmacology, 2011, Volume: 14, Issue:7

    Topics: Animals; Behavior, Addictive; Cues; Dopamine; Dose-Response Relationship, Drug; Extinction, Psychological; Female; Fluorobenzenes; Locomotion; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Norepinephrine; Nucleus Accumbens; Phenols; Prefrontal Cortex; Receptor, Serotonin, 5-HT2A; Reinforcement, Psychology; Self Administration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2011
Further evidence for the sleep-promoting effects of 5-HT₂A receptor antagonists and demonstration of synergistic effects with the hypnotic, zolpidem in rats.
    Neuropharmacology, 2013, Volume: 70

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hypnotics and Sedatives; Male; Phenols; Piperidines; Pyridines; Rats; Serotonin Antagonists; Sleep Stages; Wakefulness; Zolpidem

2013
Chronic treatment with the serotonin 2A/2C receptor antagonist SR 46349B enhances the retention and efficiency of rule-guided behavior in mice.
    Neurobiology of learning and memory, 2013, Volume: 103

    Topics: Animals; Behavior, Animal; Fluorobenzenes; Male; Maze Learning; Memory; Mice; Phenols; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Reversal Learning; Serotonin 5-HT2 Receptor Antagonists

2013
The acute social defeat stress and nest-building test paradigm: A potential new method to screen drugs for depressive-like symptoms.
    Behavioural processes, 2017, Volume: 135

    Topics: Animals; Depression; Disease Models, Animal; Dominance-Subordination; Fluorobenzenes; Fluoxetine; Male; Mice; Mice, Inbred C57BL; Nesting Behavior; Phenols; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stress, Psychological

2017
Blockade of 5-HT2A receptors inhibits emotional hyperthermia in mice.
    The journal of physiological sciences : JPS, 2019, Volume: 69, Issue:6

    Topics: Animals; Fever; Fluorobenzenes; Heart Rate; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phenols; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Stress, Psychological

2019