Page last updated: 2024-09-03

sr 2640 and l 663536

sr 2640 has been researched along with l 663536 in 3 studies

Compound Research Comparison

Studies
(sr 2640)
Trials
(sr 2640)
Recent Studies (post-2010)
(sr 2640)
Studies
(l 663536)
Trials
(l 663536)
Recent Studies (post-2010) (l 663536)
31184854138

Protein Interaction Comparison

ProteinTaxonomysr 2640 (IC50)l 663536 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.023
Prostaglandin E synthaseHomo sapiens (human)2.2274
Prostaglandin G/H synthase 1Ovis aries (sheep)8
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiens (human)0.57
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.023
Arachidonate 5-lipoxygenase-activating proteinHomo sapiens (human)0.025
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.023
Prostaglandin G/H synthase 2Homo sapiens (human)2.4
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.023
Leukotriene C4 synthaseHomo sapiens (human)3
Macrophage-expressed gene 1 proteinHomo sapiens (human)2.2
GABA theta subunitRattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.023
Prostaglandin E synthase 2Homo sapiens (human)1.6

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kreft, AF; Musser, JH1
Brooks, CD; Summers, JB1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Reviews

2 review(s) available for sr 2640 and l 663536

ArticleYear
5-lipoxygenase: properties, pharmacology, and the quinolinyl(bridged)aryl class of inhibitors.
    Journal of medicinal chemistry, 1992, Jul-10, Volume: 35, Issue:14

    Topics: Animals; Arachidonate 5-Lipoxygenase; Asthma; Eosinophils; Humans; Inflammation; Leukotriene Antagonists; Lipoxygenase Inhibitors; Lung Diseases; Neutrophils; Quinolines

1992
Modulators of leukotriene biosynthesis and receptor activation.
    Journal of medicinal chemistry, 1996, Jul-05, Volume: 39, Issue:14

    Topics: 5-Lipoxygenase-Activating Proteins; Animals; Carrier Proteins; Forecasting; Humans; Leukotriene B4; Leukotrienes; Lipoxygenase Inhibitors; Membrane Proteins; Molecular Structure; Receptors, Leukotriene

1996

Other Studies

1 other study(ies) available for sr 2640 and l 663536

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009