sr 140333 has been researched along with thiorphan in 3 studies
Studies (sr 140333) | Trials (sr 140333) | Recent Studies (post-2010) (sr 140333) | Studies (thiorphan) | Trials (thiorphan) | Recent Studies (post-2010) (thiorphan) |
---|---|---|---|---|---|
236 | 0 | 12 | 665 | 50 | 82 |
Protein | Taxonomy | sr 140333 (IC50) | thiorphan (IC50) |
---|---|---|---|
Thermolysin | Bacillus thermoproteolyticus | 9.5 | |
Neprilysin | Rattus norvegicus (Norway rat) | 0.0058 | |
Neprilysin | Oryctolagus cuniculus (rabbit) | 0.0085 | |
Neprilysin | Homo sapiens (human) | 0.0024 | |
Angiotensin-converting enzyme | Homo sapiens (human) | 0.2281 | |
Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | 0.42 | |
Neprilysin | Sus scrofa (pig) | 0.0062 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (66.67) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Advenier, C; Emonds-Alt, X; Girard, V; Yavo, JC | 1 |
Giuliani, S; Maggi, CA | 1 |
Coupar, IM; Kerr, KP; Thai, B | 1 |
3 other study(ies) available for sr 140333 and thiorphan
Article | Year |
---|---|
The tachykinin NK2 receptor antagonist SR 48968 inhibits citric acid-induced airway hyperresponsiveness in guinea pigs.
Topics: Acetylcholine; Aerosols; Animals; Benzamides; Bronchial Hyperreactivity; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Codeine; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Guinea Pigs; Injections, Intraperitoneal; Injections, Intravenous; Male; Narcotics; Piperidines; Protease Inhibitors; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Stereoisomerism; Tachykinins; Thiorphan | 1996 |
Characterization of the apamin- and L-nitroarginine-resistant NANC inhibitory transmission to the circular muscle of guinea-pig colon.
Topics: Adrenergic Agents; Animals; Apamin; Atropine; Autonomic Nervous System; Colon; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Guanethidine; Guinea Pigs; Humans; Indoles; Male; Muscarinic Antagonists; Muscle Relaxation; Muscle, Smooth; Nitroarginine; Piperidines; Protease Inhibitors; Quinuclidines; Thiorphan; Vasoactive Intestinal Peptide | 1996 |
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan | 2000 |