Page last updated: 2024-09-02

sr 140333 and sr 142801

sr 140333 has been researched along with sr 142801 in 27 studies

Compound Research Comparison

Studies
(sr 140333)
Trials
(sr 140333)
Recent Studies (post-2010)
(sr 140333)
Studies
(sr 142801)
Trials
(sr 142801)
Recent Studies (post-2010) (sr 142801)
236012127211

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (25.93)18.2507
2000's20 (74.07)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Inoue, H; Koshihara, Y; Nagata, N1
Barthó, L; Heinemann, A; Holzer, P; Lippe, IT1
Bueno, L; Emonds-Alt, X; Fioramonti, J; Mazelin, L; More, J; Theodorou, V1
Bornstein, JC; Burcher, E; Johnson, PJ1
Bueno, L; Emonds-Alt, X; Fioramonti, J; Garcia-Villar, R; Gay, J1
Fisher, L; Lau, WA; Moodley, N; Pennefather, JN; Story, ME1
Bredenbröker, D; Fehmann, H; Klüber, D; Lange, A; Wagner, U; Wichert, P1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L1
Coupar, IM; Kerr, KP; Mitchelson, F1
Kajekar, R; Myers, AC1
Advenier, C; Beerens, D; Gustin, P; Halloy, D; Moreaux, B; Nemmar, A; Vincke, G1
Corinaldesi, R; Crema, F; D'Agostino, G; De Giorgio, R; De Ponti, F; Spelta, V; Stanghellini, V; Sternini, C; Tonini, M1
Gibbins, IL; Jobling, P; Messenger, JP1
Beck, DR; Gebhart, GF; Kamp, EH1
Glowinski, J; Godeheu, G; Kemel, ML; Pérez, S; Soubrié, P1
Crema, A; Crema, F; de Ponti, F; Frigo, G; Moro, E; Nardelli, G1
Furness, JB; Kumano, K; Kunze, WA; Larsson, H; Murr, E; Vogalis, F1
Advenier, C; Alt, XE; D'Agostino, B; Daoui, S; Gallelli, L; Rossi, F1
Hirano, K; Kanaide, H; Naito, S; Nishimura, J; Takahashi, R1
Amadesi, S; Bardella, E; Bunnett, NW; De Giorgio, R; Figueroa, CD; Geppetti, P; Harrison, S; Maggiore, B; Navarra, G; Poblete, MT; Schmidlin, F; Tognetto, M; Trevisani, M; Turini, A1
de Francischi, JN; Lisboa, MC; Santos, JM; Tatsuo, MA; Turchetti-Maia, RM1
Bornstein, JC; Johnson, PJ1
Advenier, C; Boichot, E; Emonds-Alt, X; Guenon, I; Lagente, V; Nenan, S; Veron, M1
Bitel, M; Chodorowski, Z; Ciechanownicz, R; Korolkiewicz, RP; Petrusewicz, J; Sein-Anand, J1
Candenas, ML; Fernández-Sánchez, M; Orea, A; Pintado, CO; Pinto, FM; Ravina, CG; Seda, M1
Appleyard, CB; Morales, M; Santiago, C1
Bornstein, JC; Gwynne, RM1

Other Studies

27 other study(ies) available for sr 140333 and sr 142801

ArticleYear
Effect of the tachykinin receptor antagonists, SR 140333, FK 888, and SR 142801, on capsaicin-induced mouse ear oedema.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:6

    Topics: Animals; Binding Sites; Capsaicin; Dipeptides; Disease Models, Animal; Ear Diseases; Edema; Indoles; Injections, Intravenous; Lethal Dose 50; Male; Mice; Piperidines; Quinuclidines; Receptors, Tachykinin; Skin; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Tachykinin NK1 and NK2 receptor-mediated control of peristaltic propulsion in the guinea-pig small intestine in vitro.
    Neuropharmacology, 1998, Volume: 37, Issue:1

    Topics: Animals; Atropine; Benzamides; Female; Guinea Pigs; Hexamethonium; In Vitro Techniques; Intestine, Small; Male; Neurokinin-1 Receptor Antagonists; Peristalsis; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2

1998
Comparative effects of nonpeptide tachykinin receptor antagonists on experimental gut inflammation in rats and guinea-pigs.
    Life sciences, 1998, Volume: 63, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Body Weight; Colitis; Guinea Pigs; Ileitis; Male; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Tachykinin

1998
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998
Involvement of tachykinin receptors in sensitisation to cow's milk proteins in guinea pigs.
    Gut, 1999, Volume: 44, Issue:4

    Topics: Animals; Benzamides; Female; Food Hypersensitivity; Guinea Pigs; Immunoglobulin E; Immunoglobulin G; Jejunum; Lactoglobulins; Mast Cells; Passive Cutaneous Anaphylaxis; Piperidines; Quinuclidines; Receptors, Tachykinin

1999
NK2 receptors mediate tachykinin-induced contractions of rat uterus during the oestrous cycle.
    European journal of pharmacology, 1999, Jul-02, Volume: 376, Issue:1-2

    Topics: Animals; Anti-Bacterial Agents; Benzamides; Diestrus; Estrus; Female; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptides; Piperidines; Proestrus; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Tachykinins; Uterine Contraction

1999
Effects of selective tachykinin-receptor antagonists on tachykinin-induced airway mucus secretion in the rat.
    Neuropeptides, 1999, Volume: 33, Issue:1

    Topics: Animals; Benzamides; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mucosa; Substance P; Tachykinins; Trachea

1999
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium

2000
Tachykinins play a minor role in mediating the third phase of the contractile response to vagal nerve stimulation of the guinea-pig oesophagus.
    Neuropeptides, 2000, Volume: 34, Issue:1

    Topics: Animals; Benzamides; Electric Stimulation; Esophagus; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Vagus Nerve

2000
Effect of bradykinin on membrane properties of guinea pig bronchial parasympathetic ganglion neurons.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 278, Issue:3

    Topics: Animals; Bradykinin; Bronchi; Cyclooxygenase Inhibitors; Electrophysiology; Ganglia, Parasympathetic; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Membrane Potentials; Membranes; Neurokinin-1 Receptor Antagonists; Neurons; Piperidines; Quinuclidines; Reaction Time; Receptors, Neurokinin-3

2000
Role of substance P and tachykinin receptor antagonists in citric acid-induced cough in pigs.
    European journal of pharmacology, 2000, Nov-24, Volume: 408, Issue:3

    Topics: Animals; Benzamides; Citric Acid; Cough; Female; Lung; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Reflex; Substance P; Swine, Miniature

2000
Tachykinin-dependent and -independent components of peristalsis in the guinea pig isolated distal colon.
    Gastroenterology, 2001, Volume: 120, Issue:4

    Topics: Animals; Colon; Drug Combinations; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Nicotinic Antagonists; Peptides, Cyclic; Peristalsis; Piperidines; Quinuclidines; Scopolamine; Tachykinins

2001
Differential expression of functionally identified and immunohistochemically identified NK(1) receptors on sympathetic neurons.
    Journal of neurophysiology, 2001, Volume: 85, Issue:5

    Topics: Action Potentials; Animals; Biotin; Coloring Agents; Enzyme Inhibitors; Female; Ganglia, Sympathetic; Guinea Pigs; Image Processing, Computer-Assisted; Immune Sera; Male; Microelectrodes; Nerve Tissue Proteins; Neurons; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Protein Kinase C; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Sympathetic Fibers, Postganglionic; Tachykinins

2001
Combinations of neurokinin receptor antagonists reduce visceral hyperalgesia.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:1

    Topics: Animals; Benzamides; Biomarkers; Colitis; Drug Interactions; Hyperalgesia; Injections, Spinal; Male; Motor Activity; Neurokinin-1 Receptor Antagonists; Pain Measurement; Peroxidase; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Zymosan

2001
Facilitation by endogenous tachykinins of the NMDA-evoked release of acetylcholine after acute and chronic suppression of dopaminergic transmission in the matrix of the rat striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Mar-01, Volume: 22, Issue:5

    Topics: Acetylcholine; Animals; Benzamides; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Inhibitors; In Vitro Techniques; Male; N-Methylaspartate; Neural Inhibition; Neurons; Oxidopamine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Synaptic Transmission; Tachykinins; Time Factors

2002
Role of tachykininergic and cholinergic pathways in modulating canine gastric tone and compliance in vivo.
    Pharmacological research, 2002, Volume: 45, Issue:4

    Topics: Animals; Atropine; Autonomic Pathways; Benzamides; Compliance; Dogs; Female; Muscarinic Antagonists; Muscle Tonus; Muscle, Smooth; Parasympathetic Nervous System; Piperidines; Pressure; Quinuclidines; Receptors, Tachykinin; Stomach; Tachykinins

2002
Sensitization of enteric reflexes in the rat colon in vitro.
    Autonomic neuroscience : basic & clinical, 2002, Apr-18, Volume: 97, Issue:1

    Topics: Animals; Area Under Curve; Carbachol; Cholinergic Agonists; Colon; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Hexamethonium; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Neurons, Afferent; Nicotinic Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Tachykinin; Serotonin Antagonists; Time Factors

2002
Tachykinins and airway microvascular leakage induced by HCl intra-oesophageal instillation.
    The European respiratory journal, 2002, Volume: 20, Issue:2

    Topics: Animals; Asthma; Capillary Permeability; Disease Models, Animal; Esophagus; Female; Gastroesophageal Reflux; Guinea Pigs; Hydrochloric Acid; Instillation, Drug; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-3

2002
The mechanisms for tachykinin-induced contractions of the rabbit corpus cavernosum.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Animals; Benzamides; Calcium; Dose-Response Relationship, Drug; Glycopeptides; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Penis; Permeability; Piperidines; Quinuclidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Type C Phospholipases

2002
Bradykinin B2 receptors mediate contraction in the normal and inflamed human gallbladder in vitro.
    Gastroenterology, 2003, Volume: 125, Issue:1

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Antipsychotic Agents; Atropine; Benzamides; Bradykinin; Bradykinin Receptor Antagonists; Cyclooxygenase Inhibitors; Female; Gallbladder; Gallbladder Emptying; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Indomethacin; Male; Middle Aged; Muscarinic Antagonists; Piperidines; Quinuclidines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Reverse Transcriptase Polymerase Chain Reaction; Tritium

2003
Leukocyte recruitment to peritoneal cavity of rats following formalin injection: role of tachykinin receptors.
    Journal of pharmacological sciences, 2004, Volume: 94, Issue:4

    Topics: Animals; Benzamides; Cell Movement; Dose-Response Relationship, Drug; Female; Formaldehyde; Injections, Intraperitoneal; Leukocytes; Models, Biological; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peritoneal Cavity; Peritoneal Lavage; Piperidines; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Time Factors

2004
Neurokinin-1 and -3 receptor blockade inhibits slow excitatory synaptic transmission in myenteric neurons and reveals slow inhibitory input.
    Neuroscience, 2004, Volume: 126, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Excitatory Postsynaptic Potentials; Female; Guinea Pigs; Male; Myenteric Plexus; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Phentolamine; Piperazines; Piperidines; Quinuclidines; Reaction Time; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Substance P; Synaptic Transmission

2004
Interactions of tachykinin receptor antagonists with lipopolysaccharide-induced airway inflammation in mice.
    Clinical and experimental pharmacology & physiology, 2004, Volume: 31, Issue:9

    Topics: Aerosols; Animals; Benzamides; Bronchitis; Bronchoalveolar Lavage Fluid; Interleukin-6; Lipopolysaccharides; Male; Matrix Metalloproteinase 9; Mice; Mice, Inbred BALB C; Neurokinin-1 Receptor Antagonists; Piperidines; Pulmonary Alveoli; Quinuclidines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Time Factors; Tumor Necrosis Factor-alpha

2004
Salutary effects of tachykinin receptor antagonists in a rat model of postoperative ileus.
    The Journal of surgical research, 2006, Jun-15, Volume: 133, Issue:2

    Topics: Anesthetics, Inhalation; Animals; Antipsychotic Agents; Benzamides; Disease Models, Animal; Ether; Gastrointestinal Motility; Ileus; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Postoperative Complications; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin

2006
A role for tachykinins in the regulation of human sperm motility.
    Human reproduction (Oxford, England), 2007, Volume: 22, Issue:6

    Topics: Benzamides; Humans; Immunohistochemistry; Male; Neurokinin A; Neurokinin B; Piperidines; Quinuclidines; Receptors, Tachykinin; Sperm Motility; Spermatozoa; Substance P; Tachykinins

2007
Chronic inflammation alters the contribution of neurokinin receptor subtypes to epithelial function in rat colon.
    Digestive diseases and sciences, 2008, Volume: 53, Issue:1

    Topics: Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antipsychotic Agents; Benzamides; Colitis; Disease Models, Animal; Indomethacin; Intestinal Mucosa; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Stereoisomerism; Substance P; Tetrodotoxin; Trinitrobenzenesulfonic Acid

2008
Electrical stimulation of the mucosa evokes slow EPSPs mediated by NK1 tachykinin receptors and by P2Y1 purinoceptors in different myenteric neurons.
    American journal of physiology. Gastrointestinal and liver physiology, 2009, Volume: 297, Issue:1

    Topics: Adenosine Diphosphate; Animals; Electric Stimulation; Evoked Potentials; Excitatory Postsynaptic Potentials; Female; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Intestinal Mucosa; Jejunum; Kinetics; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Nitrergic Neurons; Nitric Oxide Synthase Type I; Piperidines; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Quinuclidines; Receptors, Neurokinin-1; Receptors, Purinergic P2; Receptors, Purinergic P2Y1

2009