Page last updated: 2024-09-02

sr 140333 and cp 99994

sr 140333 has been researched along with cp 99994 in 3 studies

Compound Research Comparison

Studies
(sr 140333)
Trials
(sr 140333)
Recent Studies (post-2010)
(sr 140333)
Studies
(cp 99994)
Trials
(cp 99994)
Recent Studies (post-2010) (cp 99994)
236012231219

Protein Interaction Comparison

ProteinTaxonomysr 140333 (IC50)cp 99994 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 2Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 3Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 4Rattus norvegicus (Norway rat)0.0006
Substance-P receptorHomo sapiens (human)0.0004

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowery, NG; Malcangio, M1
Belmonte, KE; Costello, RW; Fryer, AD; Jacoby, DB1
Bornstein, JC; Burcher, E; Johnson, PJ1

Other Studies

3 other study(ies) available for sr 140333 and cp 99994

ArticleYear
Effect of the tachykinin NK1 receptor antagonists, RP 67580 and SR 140333, on electrically-evoked substance P release from rat spinal cord.
    British journal of pharmacology, 1994, Volume: 113, Issue:2

    Topics: Amino Acid Sequence; Analgesics; Animals; Biphenyl Compounds; Calcitonin Gene-Related Peptide; Electric Stimulation; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Isoindoles; Male; Molecular Sequence Data; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Spinal Cord; Substance P

1994
Effects of tachykinin NK1 receptor antagonists on vagal hyperreactivity and neuronal M2 muscarinic receptor function in antigen challenged guinea-pigs.
    British journal of pharmacology, 1998, Volume: 124, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biphenyl Compounds; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Electric Stimulation; Eosinophilia; Guinea Pigs; Lung; Neurokinin A; Neurokinin-1 Receptor Antagonists; Ovalbumin; Peptide Fragments; Pilocarpine; Piperidines; Quinuclidines; Receptor, Muscarinic M2; Receptors, Muscarinic; Receptors, Tachykinin; Specific Pathogen-Free Organisms; Substance P; Trachea; Vagus Nerve

1998
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998