Page last updated: 2024-08-23

sq-11725 and albuterol

sq-11725 has been researched along with albuterol in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.56)18.7374
1990's5 (27.78)18.2507
2000's8 (44.44)29.6817
2010's4 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; el Tayar, N; Testa, B; Van de Waterbeemd, H1
Topliss, JG; Yoshida, F1
Baker, JG1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Lipworth, BJ; McDevitt, DG; McFarlane, LC; Wheeldon, NM1
Lipworth, BJ; McDevitt, DG; Wheeldon, NM2
Kalish, R; Kydonieus, A; Wille, JJ; Wood, JA1
Azevedo, ER; Newton, GE; Parker, JD1
Horinouchi, T; Koike, K1
Montpetit, CJ; Perry, SF1
Bond, RA; Dickey, BF; Franklin, AE; Garner, WJ; Hanania, NA; Lipworth, BJ; Mannava, B; Williamson, PA1

Reviews

1 review(s) available for sq-11725 and albuterol

ArticleYear
Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:11

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Models, Molecular; Receptors, Adrenergic, beta; Structure-Activity Relationship

1988

Trials

3 trial(s) available for sq-11725 and albuterol

ArticleYear
Beta-adrenoceptor subtypes mediating the metabolic effects of BRL 35135 in man.
    Clinical science (London, England : 1979), 1994, Volume: 86, Issue:3

    Topics: Adrenergic beta-Agonists; Adult; Albuterol; Basal Metabolism; Bisoprolol; Blood Glucose; Fatty Acids, Nonesterified; Glycerol; Humans; Insulin; Lactates; Lactic Acid; Male; Nadolol; Phenethylamines; Potassium; Single-Blind Method

1994
Cardiac effects of the beta 3-adrenoceptor agonist BRL35135 in man.
    British journal of clinical pharmacology, 1994, Volume: 37, Issue:4

    Topics: Administration, Oral; Adrenergic beta-Agonists; Adult; Albuterol; Bisoprolol; Drug Interactions; Hemodynamics; Humans; Male; Myocardial Contraction; Nadolol; Phenethylamines; Tremor

1994
The effects of lower than conventional doses of oral nadolol on relative beta 1/beta 2-adrenoceptor blockade.
    British journal of clinical pharmacology, 1994, Volume: 38, Issue:2

    Topics: Administration, Oral; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Adult; Albuterol; Cross-Over Studies; Dose-Response Relationship, Drug; Exercise; Female; Humans; Hyperkalemia; Male; Nadolol; Single-Blind Method; Tachycardia; Tremor

1994

Other Studies

14 other study(ies) available for sq-11725 and albuterol

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Sensitization of mice to topically applied drugs: albuterol, chlorpheniramine, clonidine and nadolol.
    Contact dermatitis, 1996, Volume: 35, Issue:2

    Topics: Administration, Cutaneous; Albuterol; Animals; Anti-Asthmatic Agents; Antihypertensive Agents; Biological Availability; Chlorpheniramine; Clonidine; Dermatitis, Allergic Contact; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Delivery Systems; Drug Eruptions; Female; Histamine Agonists; Linear Models; Mice; Mice, Inbred CBA; Nadolol; Skin Absorption; Vitamin A

1996
Inotropic and sympathetic responses to the intracoronary infusion of a beta2-receptor agonist: a human in vivo study.
    Circulation, 1999, May-11, Volume: 99, Issue:18

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Albuterol; Atenolol; Cardiac Catheterization; Chest Pain; Coronary Disease; Coronary Vessels; Female; Heart; Heart Ventricles; Hemodynamics; Humans; Infusions, Intra-Arterial; Male; Middle Aged; Myocardial Contraction; Nadolol; Norepinephrine; Sympathetic Nervous System; Sympathomimetics

1999
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism

2001
Adrenergic regulation of catecholamine secretion from trout (Oncorhynchus mykiss) chromaffin cells.
    The Journal of endocrinology, 2002, Volume: 173, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Albuterol; Analysis of Variance; Angiotensin II; Animals; Carbachol; Catecholamines; Chromaffin Cells; Clonidine; Dobutamine; Electric Stimulation; Epinephrine; Female; Male; Nadolol; Norepinephrine; Oncorhynchus mykiss; Perfusion; Phentolamine; Phenylephrine; Receptors, Cholinergic; Vasoactive Intestinal Peptide

2002
Response to salbutamol in patients with mild asthma treated with nadolol.
    The European respiratory journal, 2010, Volume: 36, Issue:4

    Topics: Adolescent; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Adult; Albuterol; Asthma; Female; Humans; Male; Middle Aged; Nadolol; Propranolol; Respiratory Function Tests; Treatment Outcome

2010