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spiroxatrine and spiperone

spiroxatrine has been researched along with spiperone in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19905 (35.71)18.7374
1990's6 (42.86)18.2507
2000's2 (14.29)29.6817
2010's1 (7.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buckingham, J; Glen, RC; Hill, AP; Hyde, RM; Martin, GR; Robertson, AD; Salmon, JA; Woollard, PM1
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB1
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Singer, EA; Valenta, B1
Alexander, BS; Broadhurst, AM; Wood, MD1
Martin, AR; Nelson, DL; Nikam, SS1
Lambert, G; Monroe, PJ; Nelson, DL; Yamamura, HI1
Anderson, EG; Marszalec, W; Scroggs, RS1
Nelson, DL; Taylor, EW1
Wallis, DI; Wang, XC; Wu, J1
Chu, TC; Ogidigben, MJ; Potter, DE1
Johnson, MS; Laurila, JM; Ruuskanen, JO; Scheinin, M; Wissel, G; Xhaard, H1

Other Studies

14 other study(ies) available for spiroxatrine and spiperone

ArticleYear
Computer-aided design and synthesis of 5-substituted tryptamines and their pharmacology at the 5-HT1D receptor: discovery of compounds with potential anti-migraine properties.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Aorta; Computer-Aided Design; Drug Design; Haplorhini; In Vitro Techniques; Migraine Disorders; Models, Chemical; Rabbits; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Saphenous Vein; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines

1995
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine

1998
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
    European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3

    Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes

1998
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:2

    Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

2001
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Hypotensive effects of 8-hydroxy-2-(di-n-propylamino)tetralin and 5-methylurapidil following stereotaxic microinjection into the ventral medulla of the rat.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Blood Pressure; Dioxanes; Dopamine Antagonists; Heart Rate; Male; Medulla Oblongata; Microinjections; Naphthalenes; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Spiperone; Spiro Compounds; Stereotaxic Techniques; Tetrahydronaphthalenes

1990
Heterogeneous 3H-rauwolscine binding sites in rat cortex: two alpha 2-adrenoceptor subtypes or an additional non-adrenergic interaction?
    Life sciences, 1988, Volume: 43, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Creatinine; Dioxanes; Drug Combinations; Hippocampus; Ketanserin; Male; Methysergide; Phentolamine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spiperone; Spiro Compounds; Yohimbine

1988
Serotonergic properties of spiroxatrine enantiomers.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:10

    Topics: Animals; Antipsychotic Agents; Binding Sites; Dioxanes; Dioxins; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Spiro Compounds; Stereoisomerism

1988
[3H]spiroxatrine labels a serotonin1A-like site in the rat hippocampus.
    Life sciences, 1987, Sep-28, Volume: 41, Issue:13

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Cell Membrane; Dioxanes; Dioxins; Dopamine; Guanosine Triphosphate; Haloperidol; Hippocampus; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Spiro Compounds; Tetrahydronaphthalenes; Tritium

1987
Serotonin-induced reduction of the calcium-dependent plateau in frog dorsal root ganglion cells is blocked by serotonergic agents acting at 5-hydroxytryptamine1A sites.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Calcium; Dioxanes; Ganglia, Spinal; Methiothepin; Rana catesbeiana; Receptors, Serotonin; Serotonin; Spiperone; Spiro Compounds; Tetrahydronaphthalenes

1988
Spiroxatrine: a selective serotonin1A receptor antagonist.
    European journal of pharmacology, 1986, May-13, Volume: 124, Issue:1-2

    Topics: Animals; Dioxanes; Dioxins; In Vitro Techniques; Muscle, Smooth, Vascular; Rats; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Spiro Compounds

1986
Is 5-hydroxytryptamine mediating descending inhibition in the neonatal rat spinal cord through different receptor subtypes?
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Animals, Newborn; Citalopram; Dioxanes; Dopamine Antagonists; Electric Stimulation; Ketanserin; Lumbar Vertebrae; Methiothepin; Methysergide; Rats; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Spinal Cord; Spinal Nerve Roots; Spiperone; Spiro Compounds; Sulpiride; Sumatriptan

1993
8OH-DPAT-Induced ocular hypotension: sites and mechanisms of action.
    Experimental eye research, 1999, Volume: 69, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ciliary Body; Cyclic AMP; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Intraocular Pressure; Iris; Norepinephrine; Ocular Hypertension; Rabbits; Serotonin Receptor Agonists; Spiperone; Spiro Compounds

1999
Involvement of the first transmembrane segment of human α(2) -adrenoceptors in the subtype-selective binding of chlorpromazine, spiperone and spiroxatrine.
    British journal of pharmacology, 2011, Volume: 164, Issue:5

    Topics: Adrenergic alpha-2 Receptor Antagonists; Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Cell Culture Techniques; Chlorpromazine; CHO Cells; Cricetinae; Cricetulus; Dioxanes; Humans; Ligands; Models, Molecular; Molecular Sequence Data; Protein Binding; Protein Structure, Secondary; Receptors, Adrenergic, alpha-2; Sequence Alignment; Spiperone; Spiro Compounds; Transfection

2011