Page last updated: 2024-08-16

spiperone and yohimbine

spiperone has been researched along with yohimbine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199019 (52.78)18.7374
1990's13 (36.11)18.2507
2000's2 (5.56)29.6817
2010's2 (5.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Amlaiky, N; Boschert, U; Hen, R; Maroteaux, L; Plassat, JL; Saudou, F1
Branchek, TA; Hartig, PR; Macchi, MJ; Weinshank, RL; Zgombick, JM1
Hamblin, MW; Metcalf, MA1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Bondinell, WE; Hieble, JP; Ruffolo, RR1
Baez, M; Kursar, JD; Nelson, DL; Wainscott, DB1
Billings, J; Chumpradit, S; Kung, HF; Kung, MP; Mach, R1
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Newman, ME1
Harris, LT; King, KA; McCall, RB1
Iuvone, PM; Zawilska, J1
Fujiwara, M; Nishikawa, H; Taniguchi, T; Yokotani, K1
Convents, A; De Backer, JP; De Keyser, J; Ebinger, G; Vanderheyden, P; Vauquelin, G1
Alexander, BS; Broadhurst, AM; Wood, MD1
Greiner, HE; Haase, A; Klockow, M; Schmitges, CJ; Seyfried, C1
Boyajian, CL; Leslie, FM1
Goldstein, M1
de Boer, TH; de Vos, CJ; Maura, G; Pinder, RM; Raiteri, M; Wieringa, J1
Broadhurst, AM; Wyllie, MG1
Nelson, A; Richelson, E1
Costall, B; Lim, SK; Naylor, RJ1
Bischoff, S; Ortmann, R; Waldmeier, PC1
Barbaz, B; Bernard, P; Braunwalder, A; Kim, HS; Liebman, JM; Lovell, RA; Robson, RD; Stone, G; Wasley, JW; Welch, J1
Bradbury, AJ; Costall, B; Naylor, RJ; Neumeyer, JL1
Charlton, KG; Clarke, DE; Hamed, AT; Johnson, TD1
Baldwin, JJ; Martin, GE; McClure, DE; Watling, KJ; Williams, M1
Gudelsky, GA; Meltzer, HY; Simonovic, M1
Docherty, JR; Kearns, S; O'Rourke, M1
Li, L; Schafer, JA1
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K1
Lai, WS; Liao, RM; Lin, JY1

Reviews

1 review(s) available for spiperone and yohimbine

ArticleYear
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1995

Other Studies

35 other study(ies) available for spiperone and yohimbine

ArticleYear
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Apr-01, Volume: 89, Issue:7

    Topics: 3T3 Cells; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cerebellum; Corpus Striatum; Gene Expression; Genes; GTP-Binding Proteins; Mice; Molecular Sequence Data; Nucleic Acid Hybridization; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Purkinje Cells; Receptors, Serotonin; RNA, Messenger; Serotonin

1992
Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Apr-15, Volume: 89, Issue:8

    Topics: Amino Acid Sequence; Animals; Brain; Cattle; Cell Membrane; Cloning, Molecular; DNA Probes; Female; Gene Library; Humans; Kinetics; Molecular Sequence Data; Multigene Family; Placenta; Pregnancy; Receptors, Serotonin; Recombinant Proteins; Sequence Homology, Nucleic Acid

1992
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.
    Molecular pharmacology, 1991, Volume: 40, Issue:2

    Topics: Amino Acid Sequence; Base Sequence; Cloning, Molecular; Cyclic AMP; GTP-Binding Proteins; Humans; Molecular Sequence Data; Pertussis Toxin; Receptors, Serotonin; Virulence Factors, Bordetella

1991
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Molecular cloning, functional expression, and mRNA tissue distribution of the human 5-hydroxytryptamine2B receptor.
    Molecular pharmacology, 1994, Volume: 46, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; DNA, Complementary; Humans; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution

1994
Fluorinated and iodinated dopamine agents: D2 imaging agents for PET and SPECT.
    Journal of medicinal chemistry, 1993, Jan-22, Volume: 36, Issue:2

    Topics: Animals; Benzamides; Dopamine Agents; Dopamine D2 Receptor Antagonists; Fluorine Radioisotopes; Iodine Radioisotopes; Macaca fascicularis; Male; Pyrrolidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon

1993
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
    The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31

    Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction

1993
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine

1998
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Serotonin inhibits adenylate cyclase in human platelet membranes.
    European journal of pharmacology, 1992, Aug-03, Volume: 226, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Binding Sites; Blood Platelets; Colforsin; Dose-Response Relationship, Drug; Humans; Methysergide; Quinoxalines; Receptors, Serotonin; Serotonin; Spiperone; Yohimbine

1992
Sympatholytic action of yohimbine mediated by 5-HT1A receptors.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Heart Rate; Injections, Intravenous; Receptors, Serotonin; Spiperone; Sympathetic Nervous System; Tetrahydronaphthalenes; Yohimbine

1991
Catecholamine receptors regulating serotonin N-acetyltransferase activity and melatonin content of chicken retina and pineal gland: D2-dopamine receptors in retina and alpha-2 adrenergic receptors in pineal gland.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: Acetyltransferases; Adrenergic beta-Antagonists; Animals; Apomorphine; Arylamine N-Acetyltransferase; Chickens; Clonidine; Darkness; Dopamine Antagonists; Light; Male; Melatonin; Pineal Gland; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Reference Values; Retina; Spiperone; Yohimbine

1989
The bindings of 3H-prazosin and 3H-yohimbine to alpha adrenoceptors in the guinea-pig stomach.
    Life sciences, 1988, Volume: 42, Issue:23

    Topics: Animals; Apomorphine; Binding, Competitive; Cell Membrane; Domperidone; Dopamine; Gastric Mucosa; Guinea Pigs; Male; Prazosin; Receptors, Adrenergic, alpha; Spiperone; Sympatholytics; Sympathomimetics; Tritium; Yohimbine

1988
Subtypes of adrenergic and dopaminergic receptors in bovine cerebral blood vessels.
    Neuroscience letters, 1988, Feb-29, Volume: 85, Issue:2

    Topics: Animals; Benzazepines; Cattle; Cerebral Arteries; Dihydroalprenolol; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine; Spiperone; Yohimbine

1988
Heterogeneous 3H-rauwolscine binding sites in rat cortex: two alpha 2-adrenoceptor subtypes or an additional non-adrenergic interaction?
    Life sciences, 1988, Volume: 43, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Creatinine; Dioxanes; Drug Combinations; Hippocampus; Ketanserin; Male; Methysergide; Phentolamine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spiperone; Spiro Compounds; Yohimbine

1988
Studies on the receptor profile of bisoprolol.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bisoprolol; Cattle; Dihydroalprenolol; Domperidone; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Prazosin; Propanolamines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Histamine; Receptors, Muscarinic; Spiperone; Tetrahydronaphthalenes; Yohimbine

1986
Pharmacological evidence for alpha-2 adrenoceptor heterogeneity: differential binding properties of [3H]rauwolscine and [3H]idazoxan in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Dioxanes; Dioxins; Dopamine; Epinephrine; Idazoxan; Kinetics; Lung; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spiperone; Tissue Distribution; Yohimbine

1987
Ergot alkaloids and central monoaminergic receptors.
    Journal de pharmacologie, 1985, Volume: 16 Suppl 3

    Topics: Animals; Antiparkinson Agents; Biogenic Amines; Central Nervous System; Dioxanes; Dopamine; Drug Interactions; Ergot Alkaloids; Guanosine Triphosphate; Humans; Receptors, Adrenergic, alpha; Receptors, Drug; Spiperone; Yohimbine

1985
Neurochemical and autonomic pharmacological profiles of the 6-aza-analogue of mianserin, Org 3770 and its enantiomers.
    Neuropharmacology, 1988, Volume: 27, Issue:4

    Topics: Animals; Antidepressive Agents, Tricyclic; Autonomic Nervous System; Binding, Competitive; Cerebral Cortex; Corpus Striatum; In Vitro Techniques; Male; Mianserin; Mirtazapine; Norepinephrine; Prazosin; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Stereoisomerism; Synaptosomes; Yohimbine

1988
A reassessment of the binding of [3H]rauwolscine to membranes from the rat cortex.
    Neuropharmacology, 1986, Volume: 25, Issue:3

    Topics: Animals; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Kinetics; Male; Membranes; Prazosin; Rats; Rats, Inbred Strains; Spiperone; Yohimbine

1986
Antagonism by antidepressants of neurotransmitter receptors of normal human brain in vitro.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Antidepressive Agents; Binding, Competitive; Brain; Doxepin; Humans; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Neurotransmitter; Spiperone; Yohimbine

1984
Characterisation of the mechanisms by which purported dopamine agonists reduce spontaneous locomotor activity of mice.
    European journal of pharmacology, 1981, Jul-17, Volume: 73, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Bromocriptine; Catecholamines; Dopamine; Dose-Response Relationship, Drug; Imidazolines; Male; Mice; Motor Activity; Prazosin; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine

1981
Modulation of dopaminergic transmission by alpha-noradrenergic agonists and antagonists: evidence for antidopaminergic properties of some alpha antagonists.
    Experientia, 1982, Oct-15, Volume: 38, Issue:10

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Clonidine; Dopamine; Female; Haloperidol; Homovanillic Acid; Male; Prazosin; Rats; Spiperone; Synaptic Transmission; Yohimbine

1982
CGS 7525A, a new, centrally active alpha 2 adrenoceptor antagonist.
    Life sciences, 1983, Jan-24, Volume: 32, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Benzodiazepines; Chemical Phenomena; Chemistry; Clonidine; Male; Mesencephalon; Mianserin; Norepinephrine; Prazosin; Quinones; Rats; Rats, Inbred Strains; Spiperone; Yohimbine

1983
Motor inhibition induced by aporphine derivatives in the mouse.
    The Journal of pharmacy and pharmacology, 1983, Volume: 35, Issue:8

    Topics: Animals; Aporphines; Corpus Striatum; Drug Interactions; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred Strains; Motor Activity; Prazosin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine

1983
Cardiovascular actions of kynuramine and 5-hydroxykynuramine in pithed rats.
    Journal of neural transmission, 1983, Volume: 57, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Brain; Cerebral Cortex; Decerebrate State; Heart Rate; Kynuramine; Male; Phentolamine; Phenylephrine; Propiophenones; Propranolol; Rats; Receptors, Adrenergic, alpha; Spiperone; Yohimbine

1983
Interaction of the component enantiomers of the putative dopamine autoreceptor agonist, TL-99 (6,7-dihydroxy-2-dimethylamino tetralin) with dopaminergic systems in mammalian brain and teleost retina.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Brain; Female; Fishes; Male; Mice; Motor Activity; Naphthalenes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Retina; Spiperone; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes; Yohimbine

1983
Effect of yohimbine on rat prolactin secretion.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Animals; Dopamine; Female; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Histamine; Reserpine; Spiperone; Yohimbine

1983
Investigation of the actions of chloroethylclonidine in rat aorta.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine

1995
Dopamine inhibits vasopressin-dependent cAMP production in the rat cortical collecting duct.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: Alkaloids; Animals; Arginine Vasopressin; Benzophenanthridines; Clozapine; Cyclic AMP; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Inhibitors; Epinephrine; Fenoldopam; GTP-Binding Proteins; In Vitro Techniques; Kidney Cortex; Kidney Tubules, Collecting; Kinetics; Male; Naphthalenes; Phenanthridines; Pimozide; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D3; Receptors, Dopamine D4; Spiperone; Time Factors; Yohimbine

1998
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
    European journal of pharmacology, 2000, Jan-03, Volume: 387, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine

2000
The role of catecholamines in retention performance of a partially baited radial eight-arm maze for rats.
    The Chinese journal of physiology, 2002, Dec-31, Volume: 45, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Benzazepines; Dopamine; Dopamine Antagonists; Haloperidol; Male; Maze Learning; Memory; Norepinephrine; Prazosin; Propranolol; Rats; Rats, Wistar; Space Perception; Spiperone; Yohimbine

2002