spiperone has been researched along with ym 09151-2 in 32 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (25.00) | 18.7374 |
1990's | 21 (65.63) | 18.2507 |
2000's | 3 (9.38) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD | 1 |
Civelli, O; Guan, HC; Niznik, HB; Seeman, P; Sunahara, RK; Van Tol, HH | 1 |
Kobayashi, T; Shimizu, H; Toru, M | 1 |
Iida, H; Kanno, I; Kondoh, Y; Miura, S; Mizusawa, S; Murakami, M; Nakamichi, H; Sasaki, H; Takahashi, K; Uemura, K | 1 |
Beaulieu, M; Felder, R; Kebabian, JW | 1 |
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K | 1 |
Hidaka, K; Nakamura, Y; Terai, M | 1 |
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P | 1 |
Grigoriadis, D; Seeman, P | 1 |
Jarvie, KR; Niznik, HB; Seeman, P | 1 |
Kuroiwa, I; Maeno, H; Noshiro, O; Terai, M; Usuda, S | 1 |
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M | 1 |
Strange, PG; Vile, JM | 1 |
D'Souza, UM; Strange, PG | 1 |
Asghari, V; Buchwaldt, S; Jovanovic, V; Paterson, A; Sanyal, S; Van Tol, HH | 1 |
AssiƩ, MB; Koek, W; Sleight, AJ | 1 |
Hidaka, K; Matsumoto, M; Tada, S; Tasaki, Y; Yamaguchi, T | 1 |
D'Souza, UM; Strange, PG; Vile, JM | 1 |
Nowak, JZ; Zawilska, JB | 1 |
Javitch, JA; Kaback, J; Karlin, A; Li, X | 1 |
Guan, HC; Niznik, HB; Seeman, P; Van Tol, HH | 1 |
Chen, J; Fu, D; Javitch, JA | 1 |
Deveney, AM; Waddington, JL | 1 |
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Kogure, K; Shuto, K | 1 |
Iida, Y; Kinoshita, T; Magata, Y; Saji, H; Tanahashi, K; Yokoyama, A | 1 |
Creese, I; Florijn, WJ; Tarazi, FI | 1 |
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Shuto, K | 1 |
Endo, K; Hayakawa, N; Ishiwata, K; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H | 1 |
Amenta, F; Bronzetti, E; Felici, L; Ricci, A; Tayebati, SK | 1 |
Castelli, MP; Gessa, GL; Mocci, I; Pani, L; Sanna, AM | 1 |
Endo, K; Hayakawa, N; Ishiwata, K; Nagaoka, T; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H; Umegaki, H | 1 |
Lin, H; Strange, PG; Vivo, M | 1 |
32 other study(ies) available for spiperone and ym 09151-2
Article | Year |
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Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone | 1992 |
The cloned dopamine D2 receptor reveals different densities for dopamine receptor antagonist ligands. Implications for human brain positron emission tomography.
Topics: Antipsychotic Agents; Benzamides; Brain Chemistry; Cloning, Molecular; Dopamine D2 Receptor Antagonists; Humans; Pituitary Gland, Anterior; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed | 1992 |
[The inhibition of dopamine D1 and D2 receptors in human putamen by antipsychotic drugs].
Topics: Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Benzazepines; Chlorpromazine; Depression, Chemical; Female; Haloperidol; Humans; In Vitro Techniques; Putamen; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1990 |
[Systematization of methylation procedure and application to 11C-labeled compounds].
Topics: Benzamides; Carbon Radioisotopes; Clorgyline; Flumazenil; Isotope Labeling; Methionine; Methylation; Nuclear Medicine; Spiperone | 1991 |
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone | 1986 |
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride | 1989 |
Comparison of [3H]YM-09151-2 with [3H]spiperone and [3H]raclopride for dopamine d-2 receptor binding to rat striatum.
Topics: Animals; Antipsychotic Agents; Benzamides; Corpus Striatum; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone | 1989 |
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes | 1985 |
[3H]-domperidone labels only a single population of receptors which convert from high to low affinity for dopamine in rat brain.
Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Brain; Corpus Striatum; Domperidone; Dopamine; In Vitro Techniques; Kinetics; Male; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1986 |
Dopamine D-2 receptors in canine brain: ionic effects on [3H]neuroleptic binding.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Antipsychotic Agents; Benzamides; Dogs; Drug Interactions; Ethylmaleimide; In Vitro Techniques; Osmolar Concentration; Receptors, Dopamine; Spiperone; Visual Cortex | 1987 |
Selective binding of YM-09151-2, a new potent neuroleptic, to D2-dopaminergic receptors.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Benzamides; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Proteins; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1983 |
Effect of a novel benzamide, YM-09151-2, on rat serum prolactin levels.
Topics: Animals; Benzamides; Dose-Response Relationship, Drug; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Time Factors | 1983 |
Comparison of [3H]nemonapride and [3H]spiperone binding to D2(long) dopamine receptors.
Topics: Animals; Benzamides; Binding, Competitive; Butaclamol; CHO Cells; Cricetinae; Dopamine Antagonists; Kinetics; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection; Tritium | 1995 |
pH dependence of ligand binding to D2 dopamine receptors.
Topics: Animals; Benzamides; Binding Sites; Cattle; Caudate Nucleus; CHO Cells; Cricetinae; Dicyclohexylcarbodiimide; Dopamine Antagonists; Hydrogen-Ion Concentration; Kinetics; Ligands; Mathematics; Models, Theoretical; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection | 1995 |
Modulation of intracellular cyclic AMP levels by different human dopamine D4 receptor variants.
Topics: Animals; Benzamides; Cell Line; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; Dinoprostone; Dopamine; Haloperidol; HeLa Cells; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Transfection | 1995 |
Biphasic displacement of [3H]YM-09151-2 binding in the rat brain by thioridazine, risperidone and clozapine, but not by other antipsychotics.
Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Clozapine; Corpus Striatum; Dopamine D2 Receptor Antagonists; In Vitro Techniques; Isoxazoles; Male; Olfactory Pathways; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Risperidone; Spiperone; Thioridazine | 1993 |
Differential effects of [3H]nemonapride and [3H]spiperone binding on human dopamine D4 receptors.
Topics: Benzamides; Binding Sites; Binding, Competitive; Cells, Cultured; Cloning, Molecular; DNA, Complementary; Dopamine Antagonists; Humans; Polymorphism, Genetic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Repetitive Sequences, Nucleic Acid; Spiperone; Thermodynamics | 1995 |
[3H]nemonapride and [3H]spiperone label equivalent numbers of D2 and D3 dopamine receptors in a range of tissues and under different conditions.
Topics: Animals; Benzamides; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Antagonists; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombination, Genetic; Spiperone; Tritium | 1995 |
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride | 1994 |
Expression and characterization of human dopamine D2 receptor in baculovirus-infected insect cells.
Topics: Animals; Azides; Baculoviridae; Base Sequence; Benzamides; Cells, Cultured; Humans; Molecular Sequence Data; Moths; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Spiperone | 1994 |
Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata.
Topics: Animals; Benzamides; Corpus Striatum; Dopamine D2 Receptor Antagonists; Humans; In Vitro Techniques; Kinetics; Parkinson Disease; Pituitary Gland, Anterior; Pyrrolidines; Raclopride; Rats; Receptors, Dopamine; Receptors, Dopamine D4; Salicylamides; Schizophrenia; Spiperone; Swine; Tomography, Emission-Computed | 1993 |
Differentiating dopamine D2 ligands by their sensitivities to modification of the cysteine exposed in the binding-site crevice.
Topics: Benzamides; Binding Sites; Cell Line; Cysteine; Humans; Mutagenesis, Site-Directed; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship | 1996 |
Pharmacological characterization of behavioural responses to SK&F 83959 in relation to 'D1-like' dopamine receptors not linked to adenylyl cyclase.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Behavior, Animal; Benzamides; Benzazepines; Binding, Competitive; Chromans; Dopamine Agonists; Dopamine Antagonists; Enzyme Induction; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tetrahydroisoquinolines | 1995 |
Effects of cerebral ischemia on dopamine receptors in the gerbil striatum.
Topics: Animals; Benzamides; Benzazepines; Brain Ischemia; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dopamine Uptake Inhibitors; Gerbillinae; Male; Mazindol; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1996 |
Synthesis, in vitro binding profile and biodistribution of a 125I-labeled N-benzyl pyrrolidinyl benzamide derivative: a potential radioligand for mapping dopamine D2 receptors.
Topics: Animals; Autoradiography; Benzamides; Chemical Phenomena; Chemistry, Physical; Dopamine Agents; Dopamine Antagonists; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Male; Membranes; Mice; Mice, Inbred Strains; Neostriatum; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Synaptosomes; Tissue Distribution; Tomography, Emission-Computed, Single-Photon | 1996 |
Dopamine receptor subtypes: differential regulation after 8 months treatment with antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Clozapine; Corpus Striatum; Haloperidol; Iodine Radioisotopes; Male; Organ Specificity; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Spiperone; Tetrahydronaphthalenes; Time Factors; Tritium; Up-Regulation | 1997 |
Effect of aging on dopaminergic receptors and uptake sites in the rat brain studied by receptor autoradiography.
Topics: Aging; Animals; Autoradiography; Benzamides; Benzazepines; Brain Chemistry; Dopamine Antagonists; Dopamine Uptake Inhibitors; Male; Mazindol; Rats; Rats, Inbred F344; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tritium | 1997 |
Comparison of three PET dopamine D2-like receptor ligands, [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone, in rats.
Topics: Animals; Benzamides; Brain; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Ligands; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed; Visual Cortex | 1999 |
Dopamine D2-like receptors on human peripheral blood lymphocytes: a radioligand binding assay and immunocytochemical study.
Topics: Benzamides; Binding, Competitive; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Immune Sera; Immunohistochemistry; In Vitro Techniques; Lymphocytes; Protein Binding; Radioligand Assay; Receptors, Dopamine D2; Solubility; Spiperone; Tetrahydronaphthalenes | 1999 |
(-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors.
Topics: Amisulpride; Animals; Benzamides; Binding, Competitive; Cell Line; DNA, Recombinant; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereoisomerism; Sulpiride; Tritium | 2001 |
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone.
Topics: Animals; Autoradiography; Benzamides; Dopamine Antagonists; Glucose; Magnetic Resonance Imaging; Male; Neostriatum; Neurotoxins; Quinolinic Acid; Raclopride; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Tomography, Emission-Computed | 2002 |
Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor.
Topics: Animals; Benzamides; Cell Line; Dopamine Antagonists; Ligands; Protein Binding; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone | 2006 |