Page last updated: 2024-08-16

spiperone and ym 09151-2

spiperone has been researched along with ym 09151-2 in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19908 (25.00)18.7374
1990's21 (65.63)18.2507
2000's3 (9.38)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD1
Civelli, O; Guan, HC; Niznik, HB; Seeman, P; Sunahara, RK; Van Tol, HH1
Kobayashi, T; Shimizu, H; Toru, M1
Iida, H; Kanno, I; Kondoh, Y; Miura, S; Mizusawa, S; Murakami, M; Nakamichi, H; Sasaki, H; Takahashi, K; Uemura, K1
Beaulieu, M; Felder, R; Kebabian, JW1
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K1
Hidaka, K; Nakamura, Y; Terai, M1
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P1
Grigoriadis, D; Seeman, P1
Jarvie, KR; Niznik, HB; Seeman, P1
Kuroiwa, I; Maeno, H; Noshiro, O; Terai, M; Usuda, S1
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M1
Strange, PG; Vile, JM1
D'Souza, UM; Strange, PG1
Asghari, V; Buchwaldt, S; Jovanovic, V; Paterson, A; Sanyal, S; Van Tol, HH1
AssiƩ, MB; Koek, W; Sleight, AJ1
Hidaka, K; Matsumoto, M; Tada, S; Tasaki, Y; Yamaguchi, T1
D'Souza, UM; Strange, PG; Vile, JM1
Nowak, JZ; Zawilska, JB1
Javitch, JA; Kaback, J; Karlin, A; Li, X1
Guan, HC; Niznik, HB; Seeman, P; Van Tol, HH1
Chen, J; Fu, D; Javitch, JA1
Deveney, AM; Waddington, JL1
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Kogure, K; Shuto, K1
Iida, Y; Kinoshita, T; Magata, Y; Saji, H; Tanahashi, K; Yokoyama, A1
Creese, I; Florijn, WJ; Tarazi, FI1
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Shuto, K1
Endo, K; Hayakawa, N; Ishiwata, K; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H1
Amenta, F; Bronzetti, E; Felici, L; Ricci, A; Tayebati, SK1
Castelli, MP; Gessa, GL; Mocci, I; Pani, L; Sanna, AM1
Endo, K; Hayakawa, N; Ishiwata, K; Nagaoka, T; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H; Umegaki, H1
Lin, H; Strange, PG; Vivo, M1

Other Studies

32 other study(ies) available for spiperone and ym 09151-2

ArticleYear
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Dec-15, Volume: 89, Issue:24

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone

1992
The cloned dopamine D2 receptor reveals different densities for dopamine receptor antagonist ligands. Implications for human brain positron emission tomography.
    European journal of pharmacology, 1992, Oct-01, Volume: 227, Issue:2

    Topics: Antipsychotic Agents; Benzamides; Brain Chemistry; Cloning, Molecular; Dopamine D2 Receptor Antagonists; Humans; Pituitary Gland, Anterior; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed

1992
[The inhibition of dopamine D1 and D2 receptors in human putamen by antipsychotic drugs].
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1990, Volume: 10, Issue:2

    Topics: Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Benzazepines; Chlorpromazine; Depression, Chemical; Female; Haloperidol; Humans; In Vitro Techniques; Putamen; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1990
[Systematization of methylation procedure and application to 11C-labeled compounds].
    Kaku igaku. The Japanese journal of nuclear medicine, 1991, Volume: 28, Issue:1

    Topics: Benzamides; Carbon Radioisotopes; Clorgyline; Flumazenil; Isotope Labeling; Methionine; Methylation; Nuclear Medicine; Spiperone

1991
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1989, Volume: 30, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride

1989
Comparison of [3H]YM-09151-2 with [3H]spiperone and [3H]raclopride for dopamine d-2 receptor binding to rat striatum.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Benzamides; Corpus Striatum; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone

1989
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes

1985
[3H]-domperidone labels only a single population of receptors which convert from high to low affinity for dopamine in rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Brain; Corpus Striatum; Domperidone; Dopamine; In Vitro Techniques; Kinetics; Male; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1986
Dopamine D-2 receptors in canine brain: ionic effects on [3H]neuroleptic binding.
    European journal of pharmacology, 1987, Dec-01, Volume: 144, Issue:2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Antipsychotic Agents; Benzamides; Dogs; Drug Interactions; Ethylmaleimide; In Vitro Techniques; Osmolar Concentration; Receptors, Dopamine; Spiperone; Visual Cortex

1987
Selective binding of YM-09151-2, a new potent neuroleptic, to D2-dopaminergic receptors.
    Japanese journal of pharmacology, 1983, Volume: 33, Issue:4

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Benzamides; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Proteins; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Effect of a novel benzamide, YM-09151-2, on rat serum prolactin levels.
    Life sciences, 1983, Feb-28, Volume: 32, Issue:9

    Topics: Animals; Benzamides; Dose-Response Relationship, Drug; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Time Factors

1983
Comparison of [3H]nemonapride and [3H]spiperone binding to D2(long) dopamine receptors.
    Biochemical Society transactions, 1995, Volume: 23, Issue:1

    Topics: Animals; Benzamides; Binding, Competitive; Butaclamol; CHO Cells; Cricetinae; Dopamine Antagonists; Kinetics; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection; Tritium

1995
pH dependence of ligand binding to D2 dopamine receptors.
    Biochemistry, 1995, Oct-17, Volume: 34, Issue:41

    Topics: Animals; Benzamides; Binding Sites; Cattle; Caudate Nucleus; CHO Cells; Cricetinae; Dicyclohexylcarbodiimide; Dopamine Antagonists; Hydrogen-Ion Concentration; Kinetics; Ligands; Mathematics; Models, Theoretical; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection

1995
Modulation of intracellular cyclic AMP levels by different human dopamine D4 receptor variants.
    Journal of neurochemistry, 1995, Volume: 65, Issue:3

    Topics: Animals; Benzamides; Cell Line; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; Dinoprostone; Dopamine; Haloperidol; HeLa Cells; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Transfection

1995
Biphasic displacement of [3H]YM-09151-2 binding in the rat brain by thioridazine, risperidone and clozapine, but not by other antipsychotics.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Clozapine; Corpus Striatum; Dopamine D2 Receptor Antagonists; In Vitro Techniques; Isoxazoles; Male; Olfactory Pathways; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Risperidone; Spiperone; Thioridazine

1993
Differential effects of [3H]nemonapride and [3H]spiperone binding on human dopamine D4 receptors.
    Neuroscience letters, 1995, Feb-17, Volume: 186, Issue:2-3

    Topics: Benzamides; Binding Sites; Binding, Competitive; Cells, Cultured; Cloning, Molecular; DNA, Complementary; Dopamine Antagonists; Humans; Polymorphism, Genetic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Repetitive Sequences, Nucleic Acid; Spiperone; Thermodynamics

1995
[3H]nemonapride and [3H]spiperone label equivalent numbers of D2 and D3 dopamine receptors in a range of tissues and under different conditions.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Animals; Benzamides; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Antagonists; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombination, Genetic; Spiperone; Tritium

1995
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Expression and characterization of human dopamine D2 receptor in baculovirus-infected insect cells.
    Journal of receptor research, 1994, Volume: 14, Issue:2

    Topics: Animals; Azides; Baculoviridae; Base Sequence; Benzamides; Cells, Cultured; Humans; Molecular Sequence Data; Moths; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Spiperone

1994
Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:4

    Topics: Animals; Benzamides; Corpus Striatum; Dopamine D2 Receptor Antagonists; Humans; In Vitro Techniques; Kinetics; Parkinson Disease; Pituitary Gland, Anterior; Pyrrolidines; Raclopride; Rats; Receptors, Dopamine; Receptors, Dopamine D4; Salicylamides; Schizophrenia; Spiperone; Swine; Tomography, Emission-Computed

1993
Differentiating dopamine D2 ligands by their sensitivities to modification of the cysteine exposed in the binding-site crevice.
    Molecular pharmacology, 1996, Volume: 49, Issue:4

    Topics: Benzamides; Binding Sites; Cell Line; Cysteine; Humans; Mutagenesis, Site-Directed; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship

1996
Pharmacological characterization of behavioural responses to SK&F 83959 in relation to 'D1-like' dopamine receptors not linked to adenylyl cyclase.
    British journal of pharmacology, 1995, Volume: 116, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Behavior, Animal; Benzamides; Benzazepines; Binding, Competitive; Chromans; Dopamine Agonists; Dopamine Antagonists; Enzyme Induction; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tetrahydroisoquinolines

1995
Effects of cerebral ischemia on dopamine receptors in the gerbil striatum.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Animals; Benzamides; Benzazepines; Brain Ischemia; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dopamine Uptake Inhibitors; Gerbillinae; Male; Mazindol; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1996
Synthesis, in vitro binding profile and biodistribution of a 125I-labeled N-benzyl pyrrolidinyl benzamide derivative: a potential radioligand for mapping dopamine D2 receptors.
    Nuclear medicine and biology, 1996, Volume: 23, Issue:2

    Topics: Animals; Autoradiography; Benzamides; Chemical Phenomena; Chemistry, Physical; Dopamine Agents; Dopamine Antagonists; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Male; Membranes; Mice; Mice, Inbred Strains; Neostriatum; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Synaptosomes; Tissue Distribution; Tomography, Emission-Computed, Single-Photon

1996
Dopamine receptor subtypes: differential regulation after 8 months treatment with antipsychotic drugs.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Clozapine; Corpus Striatum; Haloperidol; Iodine Radioisotopes; Male; Organ Specificity; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Spiperone; Tetrahydronaphthalenes; Time Factors; Tritium; Up-Regulation

1997
Effect of aging on dopaminergic receptors and uptake sites in the rat brain studied by receptor autoradiography.
    Journal of the neurological sciences, 1997, May-29, Volume: 148, Issue:2

    Topics: Aging; Animals; Autoradiography; Benzamides; Benzazepines; Brain Chemistry; Dopamine Antagonists; Dopamine Uptake Inhibitors; Male; Mazindol; Rats; Rats, Inbred F344; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tritium

1997
Comparison of three PET dopamine D2-like receptor ligands, [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone, in rats.
    Annals of nuclear medicine, 1999, Volume: 13, Issue:3

    Topics: Animals; Benzamides; Brain; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Ligands; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed; Visual Cortex

1999
Dopamine D2-like receptors on human peripheral blood lymphocytes: a radioligand binding assay and immunocytochemical study.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:3

    Topics: Benzamides; Binding, Competitive; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Immune Sera; Immunohistochemistry; In Vitro Techniques; Lymphocytes; Protein Binding; Radioligand Assay; Receptors, Dopamine D2; Solubility; Spiperone; Tetrahydronaphthalenes

1999
(-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Amisulpride; Animals; Benzamides; Binding, Competitive; Cell Line; DNA, Recombinant; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereoisomerism; Sulpiride; Tritium

2001
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone.
    Nuclear medicine and biology, 2002, Volume: 29, Issue:3

    Topics: Animals; Autoradiography; Benzamides; Dopamine Antagonists; Glucose; Magnetic Resonance Imaging; Male; Neostriatum; Neurotoxins; Quinolinic Acid; Raclopride; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Tomography, Emission-Computed

2002
Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor.
    Molecular pharmacology, 2006, Volume: 69, Issue:1

    Topics: Animals; Benzamides; Cell Line; Dopamine Antagonists; Ligands; Protein Binding; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone

2006