spiperone has been researched along with u-50488 in 4 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Armstrong, RA; Rooney, KF; Sewell, RD | 1 |
Bhargava, HN; Gulati, A; Ramarao, P | 1 |
Brent, PJ; Bunn, SJ | 1 |
Bhargava, HN; Reddy, PL | 1 |
4 other study(ies) available for spiperone and u-50488
Article | Year |
---|---|
Increased dopamine receptor sensitivity in the rat following acute administration of sufentanil, U50,488H and D-Ala2-D-Leu5-enkephalin.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzazepines; Corpus Striatum; Enkephalin, Leucine-2-Alanine; Fentanyl; In Vitro Techniques; Locomotion; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sufentanil; Tritium | 1991 |
Effect of repeated administration of U-50,488H on the binding of 3H-SCH 23390 and 3H-spiperone to rat brain and spinal cord dopamine receptors.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzazepines; Brain; Drug Tolerance; Kinetics; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spinal Cord; Spiperone | 1990 |
In vivo treatment with mu and delta, but not kappa-selective opioid agonists reduces [3H]spiperone binding to the guinea-pig striatum: autoradiographic evidence.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Autoradiography; Brain; Corpus Striatum; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Guinea Pigs; Male; Morphine; Organ Specificity; Pyrrolidines; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spiperone; Tritium | 1994 |
Effect of chronic administration of U-50,488H, a kappa-opioid receptor agonist, on central dopamine D2 receptors of the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Binding Sites; Brain; Bromocriptine; Drug Tolerance; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Opioid, kappa; Spinal Cord; Spiperone; Up-Regulation | 1993 |