Page last updated: 2024-08-16

spiperone and trifluoperazine

spiperone has been researched along with trifluoperazine in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-199012 (80.00)18.7374
1990's2 (13.33)18.2507
2000's0 (0.00)29.6817
2010's1 (6.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Clow, A; Jenner, P; Marsden, CD; Theodorou, A5
Lee, T; Schmidt, MH1
McMillen, BA1
Ansell, J; Norman, JA; Stone, GA; Wasley, JW; Wennogle, LP1
Dawbarn, D; Pycock, C1
Clow, A; Jenner, P; Mann, S; Marsden, CD; Murugaiah, K; Theodorou, A1
Allikmets, LKh; AvrutskiÄ­, GIa; Beliakov, AV; Neduva, AA; ZharkovskiÄ­, AM1
Clow, A; Gommeren, W; Jenner, P; Leysen, J; Marsden, CD; Theodorou, A1
Chuang, YC; Huang, WT; Lin, MT; Liu, HS; Won, SJ1

Other Studies

15 other study(ies) available for spiperone and trifluoperazine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Striatal dopamine receptors become supersensitive while rats are geven trifluoperazine for six months.
    Nature, 1979, Mar-01, Volume: 278, Issue:5699

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Apomorphine; Corpus Striatum; Dopamine; Homovanillic Acid; Humans; Male; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors; Trifluoperazine

1979
Investigation of striatal dopamine D2 receptor acquisition following prenatal neuroleptic exposure.
    Psychiatry research, 1991, Volume: 36, Issue:3

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Corpus Striatum; Dose-Response Relationship, Drug; Female; Haloperidol; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Thiothixene; Trifluoperazine

1991
Comparative chronic effects of buspirone or neuroleptics on rat brain dopaminergic neurotransmission.
    Journal of neural transmission, 1985, Volume: 64, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Body Weight; Buspirone; Dopamine; Female; Haloperidol; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Synaptic Transmission; Time Factors; Trifluoperazine; Tyrosine 3-Monooxygenase

1985
CGS 9343B, a novel, potent, and selective inhibitor of calmodulin activity.
    Molecular pharmacology, 1987, Volume: 31, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Benzimidazoles; Calmodulin; Cattle; Enzyme Activation; Mice; Protein Kinase C; Receptors, Dopamine; Spiperone; Trifluoperazine

1987
Changes in rat striatal dopamine turnover and receptor activity during one years neuroleptic administration.
    European journal of pharmacology, 1980, May-02, Volume: 63, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Binding Sites; Corpus Striatum; Cyclic AMP; Dopamine; Homovanillic Acid; Male; Rats; Receptors, Dopamine; Spiperone; Thioridazine; Time Factors; Trifluoperazine

1980
Cerebral dopamine function in rats following withdrawal from one year of continuous neuroleptic administration.
    European journal of pharmacology, 1980, May-02, Volume: 63, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Binding Sites; Body Weight; Brain; Corpus Striatum; Dopamine; Homovanillic Acid; Humans; Male; Motor Activity; Mouth; Movement; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substance Withdrawal Syndrome; Thioridazine; Time Factors; Trifluoperazine

1980
Differential sensitivity to neuroleptic drugs of cerebral dopamine receptors following chronic treatment of rats with trifluoperazine.
    European journal of pharmacology, 1981, May-08, Volume: 71, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Brain; Catalepsy; Female; Haloperidol; Humans; Radioligand Assay; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes; Trifluoperazine

1981
Chronic continuous administration of neuroleptic drugs alters cerebral dopamine receptors and increases spontaneous dopaminergic action in the striatum.
    Nature, 1982, Apr-08, Volume: 296, Issue:5857

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Rats; Receptors, Dopamine; Spiperone; Trifluoperazine

1982
[Various methods of overcoming secondary resistance to treatment developing in relation to adaptation to psychotropic drugs during long-term treatment (clinico-experimental study)].
    Zhurnal nevropatologii i psikhiatrii imeni S.S. Korsakova (Moscow, Russia : 1952), 1984, Volume: 84, Issue:8

    Topics: Adult; Animals; Catalepsy; Corpus Striatum; Disease Models, Animal; Drug Therapy, Combination; Drug Tolerance; Haloperidol; Humans; Male; Mice; Receptors, Dopamine; Schizophrenia, Paranoid; Spiperone; Trifluoperazine

1984
A comparison of striatal and mesolimbic dopamine function in the rat during 6-month trifluoperazine administration.
    Psychopharmacology, 1980, Volume: 69, Issue:3

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Binding Sites; Corpus Striatum; Dopamine; Humans; Limbic System; Male; Rats; Spiperone; Stereotyped Behavior; Time Factors; Trifluoperazine

1980
Changes in cerebral dopamine function induced by a year's administration of trifluoperazine or thioridazine and their subsequent withdrawal.
    Advances in biochemical psychopharmacology, 1980, Volume: 24

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Brain; Corpus Striatum; Dopamine; Dyskinesia, Drug-Induced; Humans; Male; Rats; Spiperone; Stereotyped Behavior; Substance Withdrawal Syndrome; Thioridazine; Time Factors; Trifluoperazine

1980
Chronic neuroleptic treatment specifically alters the number of dopamine receptors in rat brain.
    Life sciences, 1981, Apr-06, Volume: 28, Issue:14

    Topics: Animals; Brain; Kinetics; Male; Rats; Receptors, Dopamine; Spiperone; Tissue Distribution; Trifluoperazine

1981
Suppression of natural killer cell activity in mouse spleen lymphocytes by several dopamine receptor antagonists.
    Experientia, 1995, Apr-15, Volume: 51, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cytotoxicity, Immunologic; Dopamine Antagonists; Flupenthixol; Fluphenazine; Killer Cells, Natural; Mice; Mice, Inbred C3H; Pimozide; Spiperone; Spleen; Thiothixene; Trifluoperazine

1995