spiperone has been researched along with thiophenes in 12 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (66.67) | 18.7374 |
1990's | 1 (8.33) | 18.2507 |
2000's | 2 (16.67) | 29.6817 |
2010's | 1 (8.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cass, WA; Zahniser, NR | 1 |
Farooqui, T; Harrold, MW; Miller, DD; Uretsky, N; Wallace, LJ; Wallace, RA | 1 |
Butler, R; Christopher, WL; Cipollina, JA; New, JS; Schlemmer, RF; VanderMaelen, CP; Yevich, JP | 1 |
Grigoriadis, D; Horn, AS; Seeman, P; Tepper, P; Van der Weide, J; Watanabe, M | 1 |
Katzenellenbogen, BS; Toney, TW | 1 |
Beart, PM; Cincotta, M; Cook, CJ; de Vries, DJ; Dijkstra, D; Horn, AS; Tepper, P | 1 |
O'Boyle, KM; Waddington, JL | 1 |
De Vries, JB; Horn, AS; Tepper, PG; Van der Weide, J | 1 |
Dell, HD; Schöllnhammer, G; Seidel, PR | 1 |
Akunne, HC; Cooke, LW; Davis, MD; Georgic, LM; Heffner, TG; MacKenzie, RG; Meltzer, LT; Pugsley, TA; Shih, YH; Whetzel, SZ; Wise, LD; Wustrow, DJ; Zoski, KT | 1 |
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L | 1 |
Feng, Z; Hou, T; Li, Y | 1 |
12 other study(ies) available for spiperone and thiophenes
Article | Year |
---|---|
Inhibition of striatal dopamine release by the selective D-2 dopamine receptor agonist N-0437 is blocked by quinine.
Topics: Animals; Binding, Competitive; Corpus Striatum; Dopamine; In Vitro Techniques; Male; Naphthalenes; Quinine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tetrahydronaphthalenes; Thiophenes | 1990 |
Synthesis and D2 dopaminergic activity of pyrrolidinium, tetrahydrothiophenium, and tetrahydrothiophene analogues of sulpiride.
Topics: Acetylcholine; Animals; Apomorphine; Cell Membrane; Chemical Phenomena; Chemistry; Corpus Striatum; Dopamine Antagonists; Potassium; Pyrrolidines; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes | 1989 |
The thieno[3,2-c]pyridine and furo[3,2-c]pyridine rings: new pharmacophores with potential antipsychotic activity.
Topics: Amphetamines; Animals; Avoidance Learning; Binding, Competitive; Catalepsy; Chemical Phenomena; Chemistry; Dioxanes; Female; Furans; Macaca; Male; Mice; Molecular Structure; Motor Activity; Piperazines; Psychoses, Substance-Induced; Psychotic Disorders; Pyridines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Stereotyped Behavior; Structure-Activity Relationship; Thiophenes | 1989 |
Synthesis and radioreceptor binding activity of N-0437, a new, extremely potent and selective D2 dopamine receptor agonist.
Topics: Animals; Binding, Competitive; In Vitro Techniques; Naphthalenes; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Swine; Tetrahydronaphthalenes; Thiophenes; Tritium | 1985 |
An evaluation of the interactions of antiestrogens with pituitary and striatal dopamine receptors.
Topics: Animals; Binding, Competitive; Cell Membrane; Corpus Striatum; Diethylamines; Estrogen Antagonists; Female; Nitromifene; Pituitary Gland, Anterior; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tamoxifen; Thiophenes | 1987 |
Radioreceptor binding reveals the potencies of N,N-disubstituted 2-aminotetralins as D2 dopamine agonists.
Topics: Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Corpus Striatum; Guanosine Triphosphate; Male; Naphthalenes; Phenethylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tetrahydronaphthalenes; Thiophenes | 1987 |
New substituted 1-phenyl-3-benzazepine analogues of SK&F 38393 and N-methyl-thienopyridine analogues of dihydroxynomifensine with selective affinity for the D-1 dopamine receptor in human post-mortem brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Binding, Competitive; Brain Chemistry; Humans; In Vitro Techniques; Kinetics; Ligands; Nomifensine; Putamen; Pyridines; Receptors, Dopamine; Spiperone; Thiophenes | 1987 |
In vitro binding of the very potent and selective D-2 dopamine agonist, [3H]N-0437 to calf caudate membranes.
Topics: Animals; Cattle; Caudate Nucleus; Corpus Striatum; In Vitro Techniques; Kinetics; Membranes; Naphthalenes; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Thiophenes | 1987 |
[Biochemical studies on tienocarbine and related compounds].
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Binding, Competitive; Brain Chemistry; Catecholamines; Caudate Nucleus; Dopamine; Homovanillic Acid; Hydroxyindoleacetic Acid; Indoles; Male; Norepinephrine; Putamen; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Structure-Activity Relationship; Thiophenes | 1984 |
PD 158771, a potential antipsychotic agent with D(2)/D(3) partial agonist and 5-HT(1A) agonist actions. I. Neurochemical effects.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Benzazepines; Biogenic Amines; Brain Chemistry; Cells, Cultured; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Humans; Male; Membranes; Neostriatum; Piperazines; Pyrimidines; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Spiperone; Tetrahydronaphthalenes; Thiophenes | 2000 |
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction | 2004 |
Structure-based drug design for dopamine D3 receptor.
Topics: Animals; Combinatorial Chemistry Techniques; Drug Design; Haloperidol; Humans; Indoles; Mice; Models, Molecular; Molecular Structure; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptors, Dopamine D3; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes | 2012 |