Page last updated: 2024-08-16

spiperone and raclopride

spiperone has been researched along with raclopride in 85 studies

Research

Studies (85)

Timeframe	Studies, this research(%)	All Research%
pre-1990	12 (14.12)	18.7374
1990's	49 (57.65)	18.2507
2000's	18 (21.18)	29.6817
2010's	6 (7.06)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P	1
Billings, J; Kung, HF; Kung, MP; Murphy, RA	1
Guo, YZ; Kasliwal, R; Kung, HF; Kung, MP; Mach, RH; Pan, SG	1
Bervoets, K; Brocco, M; Dacquet, C; Girardon, S; Gobert, A; Millan, MJ; Newman-Tancredi, A; Peglion, JL; Rivet, JM; Vian, J	1
Billings, J; Chumpradit, S; Kung, HF; Kung, MP; Mach, R	1
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L	1
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X	1
Benachour, N; Vanderheyden, PML	1
Civelli, O; Guan, HC; Niznik, HB; Seeman, P; Sunahara, RK; Van Tol, HH	1
Wong, DF	1
Csöregh, I; de Paulis, T; Hall, H; Högberg, T; Lundin, K; Ogren, SO; Stensland, B; Ström, P	1
Inoue, O; Itoh, T; Kobayashi, K; Langstrom, B; Tsukada, H	1
Bengtsson, S; Hall, H; Halldin, C; Högberg, T; Wedel, I	1
Chen, C; Goldman, S; Matsumura, K; Minkin, E; Scheffel, U; Wagner, HN; Wong, DF; Young, LT	1
Ekman, A; Eriksson, E	1
Braff, DL; Geyer, MA; Keith, VA; Swerdlow, NR	1
Farde, L; Hall, H; Halldin, C; Högberg, T; Ohlberger, A; Solin, O; Ström, P	1
Bengtsson, S; de Paulis, T; Hall, H; Högberg, T; Johansson, L; Ogren, SO; Ström, P	1
Andersen, PH; Jansen, JA	1
Farde, L; Hall, H; Halldin, C; Kopp, J; Wedel, I	1
Långström, B	1
Gallager, DW; Goldman-Rakic, PS; Lidow, MS; Rakic, P	1
Guan, HC; Niznik, HB; Seeman, P	2
Lannoye, GS; Moerlein, SM; Parkinson, D; Welch, MJ	1
Dewar, KM; Grondin, L; Montreuil, B; Reader, TA	1
Hidaka, K; Nakamura, Y; Terai, M	1
Hall, H; Sällemark, M	1
Hall, H; Wedel, I	1
Andersen, PH; Nielsen, EB	1
Karlsson-Boethius, G; Köhler, C	1
Andreasen, NC; Carson, R; Diksic, M; Evans, A; Farde, L; Gjedde, A; Hakim, A; Lal, S; Nair, N; Sedvall, G	1
Arnt, J; Hyttel, J; Nowak, G	1
Axelsson, S; Eckernäs, SA; Ekblom, B; Fasth, KJ; Gullberg, P; Hartvig, P; Långström, B; Lindström, L; Lundqvist, H	1
Angeby-Möller, K; de Paulis, T; Hall, H; Johansson, L; Kumar, Y; Ogren, SO; Rämsby, S; Sällemark, M	1
Durcan, MJ; Morgan, PF; Norman, MH; Rigdon, GC	1
Farde, L; Halldin, C; Karlsson, P; Nordström, AL; Nyberg, S; Sedvall, G	1
Asghari, V; Buchwaldt, S; Jovanovic, V; Paterson, A; Sanyal, S; Van Tol, HH	1
Farde, L; Halldin, C; Nordström, AL	1
Nobrega, JN; Seeman, P	1
Korf, J; Vaalburg, W; van der Worp, H; Visser, GM; Wiegman, T; Zijlstra, S	1
Carlsson, A; Haadsma-Svensson, SR; Smith, MW; Svensson, K; Waters, N	1
Guan, HC; Niznik, HB; Seeman, P; Van Tol, HH	1
Fowler, JS; Hitzemann, RJ; MacGregor, RR; Schlyer, DJ; Shea, CE; Volkow, ND; Wang, GJ; Wolf, AP	1
Högberg, T; Jackson, DM; Malmberg, A; Mohell, N; Rosqvist, S; Sällemark, M	1
Fukuda, T; Futamura, T; Haga, K; Ohashi, Y; Takahashi, Y; Yano, K	1
Fowler, JS; Gatley, SJ; Hitzemann, R; Logan, J; MacGregor, RR; Schlyer, DJ; Volkow, ND; Wang, GJ; Wolf, AP	1
Dannals, RF; Kao, PF; Kim, S; Lever, JR; Ravert, HT; Wagner, HN	1
Inoue, O; Kobayashi, K; Långström, B; Onoe, H; Watanabe, Y	1
Creese, I; Florijn, WJ; Tarazi, FI	1
Cravchik, A; Gejman, PV; Hietala, J; Någren, K; Pohjalainen, T; Rinne, J; Syvälahti, E	1
al-Tikriti, MS; Baldwin, RM; Charney, DS; Kessler, RM; Kung, HF; Laruelle, M; Malison, RT; Sybirska, E; Zea-Ponce, Y; Zoghbi, SS	1
Bjurling, P; Fasth, KJ; Hartvig, P; Långström, B; Tedroff, J; Torstenson, R; Watanabe, Y	1
Lima, L; Obregón, F; Urbina, M	1
Fosbraey, P; Kitchen, I; Ridd, MJ	1
Bobirnac, I; Bruinvels, AT; Danzeisen, M; Gazi, L; Geisse, S; Hoyer, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M	1
Bergström, M; Gefvert, O; Hagberg, G; Långström, B; Lindström, L; Wiesel, FA; Wieselgren, IM	1
Gee, A; Hosoi, R; Inoue, O; Kobayashi, K	1
Chu, A; Schetz, JA; Sibley, DR	1
Gee, A; Inoue, O; Kobayashi, K; Wakahara, S	1
Eriksson, B; Farde, L; Halldin, C; Nyberg, S; Oxenstierna, G	1
Endo, K; Hayakawa, N; Ishiwata, K; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H	1
Kaasinen, V; Lehikoinen, P; Någren, K; Oikonen, V; Rinne, JO; Ruottinen, HM	1
Gee, A; Hosoi, R; Inoue, O; Kobayashi, K; Yamaguchi, M	1
Ferré, S; Finnman, UB; Fuxe, K; Owman, C; Rinken, A; Terasmaa, A	1
Alberts, GL; Im, WB; Pregenzer, JF	1
Armstrong, D; Strange, PG	1
Dewey, SL; Fowler, JS; Gatley, SJ; Logan, J; Volkow, ND	1
Endo, K; Hayakawa, N; Ishiwata, K; Nagaoka, T; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H; Umegaki, H	1
Gee, A; Hosoi, R; Inoue, O; Ishikawa, M; Kobayashi, K; Yamaguchi, M	1
Ginovart, N; Kapur, S; Ko, F; Seeman, P; Sun, W	1
Hosoi, R; Inoue, O; Ishida, J; Kobayashi, K; Yamaguchi, M	1
Ko, F; Seeman, P; Tallerico, T	1
Cumming, P; Gjedde, A; Jensen, SB; Munk, OL; Olsen, AK; Rosa-Neto, P; Watanabe, H	1
Lin, H; Strange, PG; Vivo, M	1
Durand, CJ; Lan, H; Neve, KA; Teeter, MM	1
Iwata, Y; Minabe, Y; Mori, N; Nakamura, K; Okada, H; Ouchi, Y; Sekine, Y; Sugihara, G; Suzuki, K; Takei, N; Tsuchiya, KJ; Yoshikawa, E	1
Michaelides, M; Piyis, YK; Thanos, PK; Volkow, ND; Wang, GJ	1
Seeman, P	1
De Backer, JP; Packeu, A; Van Liefde, I; Vanderheyden, PM; Vauquelin, G	1
Alstrup, AK; Cumming, P; Doudet, D; Gramsbergen, JB; Jensen, SB; Minuzzi, L; Ostergaard, SD; Pedersen, K	1
De Backer, JP; Packeu, A; Vauquelin, G	1
Ishibashi, K; Ishii, K; Ishiwata, K; Mizusawa, H; Oda, K	1
Nutt, DJ; Parker, CA; Quelch, DR; Tyacke, RJ; Withey, SL	1
Cho, J; Delis, F; Kim, R; Rocco, MJ; Thanos, PK; Volkow, ND	1

Reviews

3 review(s) available for spiperone and raclopride

Article	Year
Influence of the cellular environment on ligand binding kinetics at membrane-bound targets. Bioorganic & medicinal chemistry letters, 2017, 08-15, Volume: 27, Issue:16 Topics: Angiotensin II Type 1 Receptor Blockers; Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Humans; Kinetics; Ligands; Protein Binding; Receptor, Angiotensin, Type 1; Receptors, Cell Surface; Signal Transduction	2017
Design of molecules labeled with beta+ emitters for use in multitracer investigations using positron emission tomography. Acta radiologica. Supplementum, 1990, Volume: 374 Topics: Beta Particles; Humans; Isotope Labeling; Levodopa; Methionine; Neurotransmitter Agents; Nomifensine; Raclopride; Salicylamides; Spiperone; Tomography, Emission-Computed	1990
Workshop on schizophrenia, PET, and dopamine D2 receptors in the human neostriatum. Schizophrenia bulletin, 1988, Volume: 14, Issue:3 Topics: Adult; Corpus Striatum; Haloperidol; Humans; National Institute of Mental Health (U.S.); Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Schizophrenia; Schizophrenic Psychology; Spiperone; Tomography, Emission-Computed; United States	1988

Trials

4 trial(s) available for spiperone and raclopride

Article	Year
High 5-HT2 receptor occupancy in clozapine treated patients demonstrated by PET. Psychopharmacology, 1993, Volume: 110, Issue:3 Topics: Adult; Antipsychotic Agents; Clozapine; Dopamine Agonists; Female; Humans; Male; Middle Aged; Prefrontal Cortex; Psychotic Disorders; Raclopride; Receptors, Serotonin; Salicylamides; Schizophrenia; Spiperone; Tomography, Emission-Computed	1993
N-[11C]methylspiperone PET, in contrast to [11C]raclopride, fails to detect D2 receptor occupancy by an atypical neuroleptic. Psychiatry research, 1998, Jun-30, Volume: 82, Issue:3 Topics: Adult; Antipsychotic Agents; Caudate Nucleus; Cerebellum; Dibenzothiazepines; Dopamine; Dose-Response Relationship, Drug; Humans; Male; Putamen; Quetiapine Fumarate; Raclopride; Receptors, Dopamine D2; Salicylamides; Schizophrenia; Spiperone; Tomography, Emission-Computed	1998
Suggested minimal effective dose of risperidone based on PET-measured D2 and 5-HT2A receptor occupancy in schizophrenic patients. The American journal of psychiatry, 1999, Volume: 156, Issue:6 Topics: Adult; Antipsychotic Agents; Basal Ganglia Diseases; Brain; Carbon Radioisotopes; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Psychiatric Status Rating Scales; Raclopride; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Schizophrenia; Schizophrenic Psychology; Spiperone; Tomography, Emission-Computed; Treatment Outcome	1999
Perospirone is a new generation antipsychotic: evidence from a positron emission tomography study of serotonin 2 and D2 receptor occupancy in the living human brain. Journal of clinical psychopharmacology, 2006, Volume: 26, Issue:5 Topics: Adult; Antipsychotic Agents; Binding, Competitive; Brain; Humans; Indoles; Isoindoles; Male; Positron-Emission Tomography; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Reference Values; Spiperone; Thiazoles	2006

Other Studies

78 other study(ies) available for spiperone and raclopride

Article	Year
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics. Nature, 1990, Sep-13, Volume: 347, Issue:6289 Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution	1990
Synthesis and characterization of iodobenzamide analogues: potential D-2 dopamine receptor imaging agents. Journal of medicinal chemistry, 1990, Volume: 33, Issue:1 Topics: Animals; Benzofurans; Binding, Competitive; Chemical Phenomena; Chemistry; Corpus Striatum; Iodine Radioisotopes; Isotope Labeling; Male; Molecular Structure; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Tissue Distribution	1990
Dopamine D-2 receptor imaging radiopharmaceuticals: synthesis, radiolabeling, and in vitro binding of (R)-(+)- and (S)-(-)-3-iodo-2-hydroxy-6-methoxy-N- [(1-ethyl-2-pyrrolidinyl)methyl]benzamide. Journal of medicinal chemistry, 1988, Volume: 31, Issue:5 Topics: Animals; Benzamides; Chemical Phenomena; Chemistry; Corpus Striatum; In Vitro Techniques; Iodine Radioisotopes; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship	1988
Functional correlates of dopamine D3 receptor activation in the rat in vivo and their modulation by the selective antagonist, (+)-S 14297: 1. Activation of postsynaptic D3 receptors mediates hypothermia, whereas blockade of D2 receptors elicits prolactin The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2 Topics: 2-Naphthylamine; Animals; Body Temperature Regulation; Catalepsy; CHO Cells; Cricetinae; Dopamine Antagonists; Furans; Humans; Male; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins; Stereoisomerism	1995
Fluorinated and iodinated dopamine agents: D2 imaging agents for PET and SPECT. Journal of medicinal chemistry, 1993, Jan-22, Volume: 36, Issue:2 Topics: Animals; Benzamides; Dopamine Agents; Dopamine D2 Receptor Antagonists; Fluorine Radioisotopes; Iodine Radioisotopes; Macaca fascicularis; Male; Pyrrolidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon	1993
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study. European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3 Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes	1998
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach. Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21 Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water	2003
The cloned dopamine D2 receptor reveals different densities for dopamine receptor antagonist ligands. Implications for human brain positron emission tomography. European journal of pharmacology, 1992, Oct-01, Volume: 227, Issue:2 Topics: Antipsychotic Agents; Benzamides; Brain Chemistry; Cloning, Molecular; Dopamine D2 Receptor Antagonists; Humans; Pituitary Gland, Anterior; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1992
PET studies of neuroreceptors in schizophrenia. Commentary on "The current status of PET scanning with respect to schizophrenia". Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1992, Volume: 7, Issue:1 Topics: Brain; Carbon Radioisotopes; Dopamine Antagonists; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Schizophrenia; Spiperone; Tomography, Emission-Computed; Tritium	1992
Potential antipsychotic agents. 9. Synthesis and stereoselective dopamine D-2 receptor blockade of a potent class of substituted (R)-N-[(1-benzyl-2-pyrrolidinyl)methyl]benzamides. Relations to other side chain congeners. Journal of medicinal chemistry, 1991, Volume: 34, Issue:3 Topics: Animals; Antipsychotic Agents; Benzamides; Benzyl Compounds; Chemical Phenomena; Chemistry; Corpus Striatum; Dopamine Antagonists; Male; Molecular Conformation; Molecular Structure; Pyrrolidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction	1991
Difference in in vivo receptor binding between [3H]N-methylspiperone and [3H]raclopride in reserpine-treated mouse brain. Journal of neural transmission. General section, 1991, Volume: 85, Issue:1 Topics: Animals; Cerebellum; Corpus Striatum; Dopamine Agents; Male; Mice; Raclopride; Receptors, Dopamine; Reserpine; Salicylamides; Spiperone	1991
Synthesis and binding properties of the fluorinated substituted benzamide [3H]NCQ 115, a new selective dopamine D2 receptor ligand. European journal of pharmacology, 1991, Aug-16, Volume: 201, Issue:1 Topics: Animals; Benzamides; Binding, Competitive; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine Agents; Dopamine Antagonists; In Vitro Techniques; Kinetics; Magnetic Resonance Spectroscopy; Pyrrolidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Sodium; Spiperone; Stereoisomerism	1991
Effects of endogenous dopamine on kinetics of [3H]N-methylspiperone and [3H]raclopride binding in the rat brain. Synapse (New York, N.Y.), 1991, Volume: 9, Issue:3 Topics: Amphetamine; Animals; Brain; Dopamine; Dopamine Antagonists; Kinetics; Male; Raclopride; Rats; Reserpine; Salicylamides; Spiperone; Tomography, Emission-Computed; Tritium	1991
Pituitary and brain D2 receptor density measured in vitro and in vivo in EEDQ treated male rats. Life sciences, 1991, Volume: 48, Issue:4 Topics: 4-Butyrolactone; Animals; Brain; Cell Membrane; Corpus Striatum; Kinetics; Limbic System; Male; Pituitary Gland; Quinolines; Raclopride; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Tritium	1991
Effects of spiperone, raclopride, SCH 23390 and clozapine on apomorphine inhibition of sensorimotor gating of the startle response in the rat. The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2 Topics: Analysis of Variance; Animals; Apomorphine; Benzazepines; Clozapine; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reflex, Startle; Salicylamides; Schizophrenia; Spiperone	1991
A comparative PET-study of five carbon-11 or fluorine-18 labelled salicylamides. Preparation and in vitro dopamine D-2 receptor binding. International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology, 1991, Volume: 18, Issue:8 Topics: Animals; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine Antagonists; Fluorine Radioisotopes; In Vitro Techniques; Isotope Labeling; Macaca fascicularis; Male; Potentiometry; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1991
Potential antipsychotic agents 5. Synthesis and antidopaminergic properties of substituted 5,6-dimethoxysalicylamides and related compounds. Journal of medicinal chemistry, 1990, Volume: 33, Issue:4 Topics: Animals; Antipsychotic Agents; Apomorphine; Binding Sites; Chemical Phenomena; Chemistry; Dopamine Antagonists; Male; Raclopride; Rats; Rats, Inbred Strains; Salicylamides; Spiperone; Structure-Activity Relationship	1990
Dopamine receptor agonists: selectivity and dopamine D1 receptor efficacy. European journal of pharmacology, 1990, Jun-12, Volume: 188, Issue:6 Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Benzazepines; Blood-Brain Barrier; Corpus Striatum; Dopamine Agents; Guanosine Triphosphate; In Vitro Techniques; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone; Stimulation, Chemical; Structure-Activity Relationship	1990
Comparison of the in vitro receptor binding properties of N-[3H]methylspiperone and [3H]raclopride to rat and human brain membranes. Journal of neurochemistry, 1990, Volume: 55, Issue:6 Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Humans; Male; Membranes; Putamen; Raclopride; Rats; Salicylamides; Spiperone; Tritium	1990
Distribution of dopaminergic receptors in the primate cerebral cortex: quantitative autoradiographic analysis using [3H]raclopride, [3H]spiperone and [3H]SCH23390. Neuroscience, 1991, Volume: 40, Issue:3 Topics: Animals; Benzazepines; Brain Mapping; Cerebral Cortex; Ketanserin; Macaca mulatta; Mianserin; Raclopride; Receptors, Dopamine; Salicylamides; Species Specificity; Spiperone	1991
Elevation of dopamine D2 receptors in schizophrenia is underestimated by radioactive raclopride. Archives of general psychiatry, 1990, Volume: 47, Issue:12 Topics: Animals; Brain; Carbon Radioisotopes; Caudate Nucleus; Cerebellum; Corpus Striatum; Dopamine; Dopamine Antagonists; Humans; Putamen; Raclopride; Receptors, Dopamine; Salicylamides; Schizophrenia; Spiperone; Tomography, Emission-Computed; Tritium	1990
N-fluoroalkylated and N-alkylated analogues of the dopaminergic D-2 receptor antagonist raclopride. Journal of medicinal chemistry, 1990, Volume: 33, Issue:9 Topics: Animals; Brain; Dopamine Antagonists; Female; Ligands; Macaca nemestrina; Male; Raclopride; Radiochemistry; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone	1990
Endogenous dopamine lowers the dopamine D2 receptor density as measured by [3H]raclopride: implications for positron emission tomography of the human brain. Synapse (New York, N.Y.), 1989, Volume: 3, Issue:1 Topics: Animals; Corpus Striatum; Dopamine; Humans; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1989
Dopamine D2 receptors labeled with [3H]raclopride in rat and rabbit brains. Equilibrium binding, kinetics, distribution and selectivity. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:2 Topics: Animals; Binding, Competitive; Corpus Striatum; Kinetics; Male; Rabbits; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Sodium; Species Specificity; Spiperone; Tritium	1989
Comparison of [3H]YM-09151-2 with [3H]spiperone and [3H]raclopride for dopamine d-2 receptor binding to rat striatum. European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3 Topics: Animals; Antipsychotic Agents; Benzamides; Corpus Striatum; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone	1989
Effects of chronic neuroleptic treatment on agonist affinity states of the dopamine-D2 receptor in the rat brain. Pharmacology & toxicology, 1987, Volume: 60, Issue:5 Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Brain Chemistry; Guanylyl Imidodiphosphate; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Salicylamides; Spiperone	1987
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum. Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:5 Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride	1986
The benzazepine, SCH 23390, inhibits 3H-NPA binding in mouse brain in vivo. Acta pharmacologica et toxicologica, 1986, Volume: 59, Issue:4 Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Male; Mice; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Spiperone	1986
In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain. Journal of neural transmission, 1988, Volume: 73, Issue:2 Topics: Animals; Apomorphine; Binding, Competitive; Brain; Kinetics; Male; Organ Specificity; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Stereoisomerism	1988
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors. European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3 Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone	1988
Receptor binding and selectivity of three 11C-labelled dopamine receptor antagonists in the brain of rhesus monkeys studied with positron emission tomography. Acta neurologica Scandinavica, 1988, Volume: 77, Issue:4 Topics: Animals; Brain; Clozapine; Female; Macaca mulatta; Raclopride; Receptors, Dopamine; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed	1988
Potential neuroleptic agents. 4. Chemistry, behavioral pharmacology, and inhibition of [3H]spiperone binding of 3,5-disubstituted N-[(1-ethyl-2-pyrrolidinyl)methyl]-6-methoxysalicylamides. Journal of medicinal chemistry, 1986, Volume: 29, Issue:1 Topics: Animals; Apomorphine; Chemical Phenomena; Chemistry; Corpus Striatum; Haloperidol; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone; Stereotyped Behavior; Structure-Activity Relationship	1986
Is clozapine selective for the dopamine D4 receptor? Life sciences, 1995, Volume: 57, Issue:18 Topics: Binding Sites; Cell Membrane; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone	1995
D1, D2, and 5-HT2 receptor occupancy in relation to clozapine serum concentration: a PET study of schizophrenic patients. The American journal of psychiatry, 1995, Volume: 152, Issue:10 Topics: Adult; Benzazepines; Brain; Clozapine; Female; Humans; Male; Middle Aged; Raclopride; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Schizophrenia; Spiperone; Tomography, Emission-Computed; Treatment Outcome	1995
Modulation of intracellular cyclic AMP levels by different human dopamine D4 receptor variants. Journal of neurochemistry, 1995, Volume: 65, Issue:3 Topics: Animals; Benzamides; Cell Line; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; Dinoprostone; Dopamine; Haloperidol; HeLa Cells; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Transfection	1995
Dopamine D2 receptors mapped in rat brain with [3H](+)PHNO. Synapse (New York, N.Y.), 1994, Volume: 17, Issue:3 Topics: Animals; Autoradiography; Brain; Brain Chemistry; Brain Mapping; Densitometry; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Ligands; Male; Oxazines; Raclopride; Rats; Rats, Wistar; Salicylamides; Spiperone	1994
Synthesis and in vivo distribution in the rat of a dopamine agonist: N-([11C]methyl)norapomorphine. Nuclear medicine and biology, 1993, Volume: 20, Issue:1 Topics: Animals; Apomorphine; Brain; Carbon Radioisotopes; Dopamine Agents; Kidney; Liver; Lung; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone	1993
The dopamine D3-receptor: a postsynaptic receptor inhibitory on rat locomotor activity. Journal of neural transmission. General section, 1993, Volume: 94, Issue:1 Topics: Aminoquinolines; Animals; Apomorphine; CHO Cells; Corpus Striatum; Cricetinae; Dextroamphetamine; Dopamine; Dopamine Antagonists; Drug Interactions; Indans; Male; Methyltyrosines; Models, Biological; Motor Activity; Nucleus Accumbens; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Fusion Proteins; Reserpine; Salicylamides; Spiperone; Stimulation, Chemical	1993
Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata. Synapse (New York, N.Y.), 1993, Volume: 14, Issue:4 Topics: Animals; Benzamides; Corpus Striatum; Dopamine D2 Receptor Antagonists; Humans; In Vitro Techniques; Kinetics; Parkinson Disease; Pituitary Gland, Anterior; Pyrrolidines; Raclopride; Rats; Receptors, Dopamine; Receptors, Dopamine D4; Salicylamides; Schizophrenia; Spiperone; Swine; Tomography, Emission-Computed	1993
Comparison of two PET radioligands for imaging extrastriatal dopamine receptors in the human brain. Synapse (New York, N.Y.), 1993, Volume: 15, Issue:3 Topics: Adult; Brain; Carbon Radioisotopes; Fluorine Radioisotopes; Humans; Kinetics; Male; Middle Aged; Organ Specificity; Pituitary Gland; Raclopride; Radioligand Assay; Receptors, Dopamine; Reference Values; Salicylamides; Spiperone; Tomography, Emission-Computed	1993
Binding characteristics of remoxipride and its metabolites to dopamine D2 and D3 receptors. European journal of pharmacology, 1993, Jul-06, Volume: 238, Issue:1 Topics: Animals; Cell Line; Cloning, Molecular; Corpus Striatum; Fibroblasts; Humans; Mice; Raclopride; Radioligand Assay; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Salicylamides; Spiperone	1993
[The affinities of mosapramine for the dopamine receptor subtypes in human cell lines expressing D2, D3 and D4 receptors]. Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1996, Volume: 107, Issue:5 Topics: Antipsychotic Agents; Benzazepines; Cell Line; Clozapine; Haloperidol; Humans; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Dopamine D5; Risperidone; Salicylamides; Spiperone	1996
Measuring age-related changes in dopamine D2 receptors with 11C-raclopride and 18F-N-methylspiroperidol. Psychiatry research, 1996, May-31, Volume: 67, Issue:1 Topics: Adult; Age Factors; Aged; Aging; Cerebellum; Corpus Striatum; Dopamine Agonists; Female; Humans; Ligands; Male; Middle Aged; Nerve Degeneration; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1996
Assessing neuroreceptor occupancy by continuous infusion of carbon-11 labeled radioligands. European journal of nuclear medicine, 1996, Volume: 23, Issue:2 Topics: Adult; Brain; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Fentanyl; Humans; Infusion Pumps; Male; Raclopride; Radioligand Assay; Radionuclide Imaging; Receptors, Opioid; Salicylamides; Spiperone	1996
Difference in response of D2 receptor binding between 11C-N-methylspiperone and 11C-raclopride against anesthetics in rhesus monkey brain. Journal of neural transmission. General section, 1995, Volume: 100, Issue:2 Topics: Anesthetics; Animals; Brain; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Female; Isoflurane; Ketamine; Macaca mulatta; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1995
Dopamine receptor subtypes: differential regulation after 8 months treatment with antipsychotic drugs. The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2 Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Clozapine; Corpus Striatum; Haloperidol; Iodine Radioisotopes; Male; Organ Specificity; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Spiperone; Tetrahydronaphthalenes; Time Factors; Tritium; Up-Regulation	1997
Antagonist binding characteristics of the Ser311-->Cys variant of human dopamine D2 receptor in vivo and in vitro. Biochemical and biophysical research communications, 1997, Mar-06, Volume: 232, Issue:1 Topics: Adult; Aged; Aged, 80 and over; Animals; CHO Cells; Cricetinae; Cysteine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Heterozygote; Humans; Male; Middle Aged; Protein Binding; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Salicylamides; Serine; Spiperone	1997
Comparison of three high affinity SPECT radiotracers for the dopamine D2 receptor. Nuclear medicine and biology, 1994, Volume: 21, Issue:2 Topics: Animals; Benzamides; Benzofurans; Brain; Contrast Media; Dextroamphetamine; Dopamine Agents; Female; Iodine Radioisotopes; Papio; Pyrrolidines; Raclopride; Receptors, Dopamine D2; Ritanserin; Salicylamides; Serotonin Antagonists; Spiperone; Tissue Distribution; Tomography, Emission-Computed, Single-Photon	1994
Amphetamine effects on dopamine release and synthesis rate studied in the Rhesus monkey brain by positron emission tomography. Journal of neural transmission (Vienna, Austria : 1996), 1997, Volume: 104, Issue:4-5 Topics: Amphetamine; Animals; Brain; Cerebrovascular Circulation; Decarboxylation; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Female; Levodopa; Macaca mulatta; Raclopride; Salicylamides; Spiperone; Tomography, Emission-Computed	1997
[3H]raclopride and [3H]spiroperidol binding to retinal membranes of the teleost Eugerres plumieri: effect of light and dark adaptation. Neurochemistry international, 1997, Volume: 31, Issue:4 Topics: Adaptation, Ocular; Animals; Binding Sites; Dark Adaptation; Dopamine; Dopamine Antagonists; Fishes; Membranes; Raclopride; Retina; Salicylamides; Spiperone; Tritium	1997
The effect of acute kainic acid treatment on dopamine D2 receptors in rat brain. Neuroscience research, 1998, Volume: 30, Issue:3 Topics: Animals; Brain; Iodine Radioisotopes; Isotope Labeling; Kainic Acid; Male; Neurons; Protein Binding; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride; Tritium	1998
The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4 receptor. British journal of pharmacology, 1998, Volume: 124, Issue:5 Topics: Aminopyridines; Antipsychotic Agents; Cell Line; Clozapine; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Humans; Kidney; Piperidines; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone	1998
Changes in apparent in vivo binding of [3H]raclopride and [3H]N-methylspiperone induced by oxotremorine. Journal of neural transmission (Vienna, Austria : 1996), 1998, Volume: 105, Issue:10-12 Topics: Animals; Brain; Male; Mice; Mice, Inbred Strains; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Salicylamides; Scopolamine; Spiperone; Tritium	1998
Zinc modulates antagonist interactions with D2-like dopamine receptors through distinct molecular mechanisms. The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2 Topics: Algorithms; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Kinetics; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Salicylamides; Sodium; Spiperone; Thermodynamics; Zinc	1999
Enhancement of 3H-N-methylspiperone binding but not 3H-raclopride binding in mouse striatum by MK-801: evidence that factors other than competition by endogenous dopamine are responsible for changes in D2 receptor binding in vivo. Short communication. Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:2 Topics: Animals; Binding Sites; Cerebellum; Cerebral Cortex; Dizocilpine Maleate; Dopamine; Dopamine Agonists; Dopamine Antagonists; Kinetics; Mice; Models, Biological; Neostriatum; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone	1999
Comparison of three PET dopamine D2-like receptor ligands, [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone, in rats. Annals of nuclear medicine, 1999, Volume: 13, Issue:3 Topics: Animals; Benzamides; Brain; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Ligands; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed; Visual Cortex	1999
Upregulation of putaminal dopamine D2 receptors in early Parkinson's disease: a comparative PET study with [11C] raclopride and [11C]N-methylspiperone. Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2000, Volume: 41, Issue:1 Topics: Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Female; Humans; Male; Middle Aged; Parkinson Disease; Putamen; Raclopride; Receptors, Dopamine D2; Spiperone; Tomography, Emission-Computed; Up-Regulation	2000
Discrepancies in apparent dopamine D2 receptor occupancy between 3H-raclopride and 3H-N-methylspiperone. Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12 Topics: Animals; Binding Sites; Binding, Competitive; Brain Chemistry; Male; Mice; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone; Tritium	1999
Modulation of [(35)S]GTPgammaS binding to chinese hamster ovary cell membranes by D(2(short)) dopamine receptors. Neuroscience letters, 2000, Feb-18, Volume: 280, Issue:2 Topics: Animals; Binding, Competitive; Butaclamol; CHO Cells; Cricetinae; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Membranes; Raclopride; Radioligand Assay; Rats; Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium	2000
Advantages of heterologous expression of human D2long dopamine receptors in human neuroblastoma SH-SY5Y over human embryonic kidney 293 cells. British journal of pharmacology, 2000, Volume: 131, Issue:3 Topics: Calcium Channels; Cells, Cultured; Cloning, Molecular; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Heterotrimeric GTP-Binding Proteins; Humans; Kidney; Neuroblastoma; Neurons; Raclopride; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Tumor Cells, Cultured	2000
Dopamine D2 receptor dimer formation: evidence from ligand binding. The Journal of biological chemistry, 2001, Jun-22, Volume: 276, Issue:25 Topics: Animals; CHO Cells; Cricetinae; Dimerization; Dopamine Antagonists; Ligands; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone; Tritium	2001
A consideration of the dopamine D2 receptor monomer-dimer equilibrium and the anomalous binding properties of the dopamine D2 receptor ligand, N-methyl spiperone. Journal of neural transmission (Vienna, Austria : 1996), 2001, Volume: 108, Issue:3 Topics: Animals; Binding Sites; Brain; Brain Chemistry; Dimerization; Dopamine Antagonists; Kinetics; Ligands; Models, Biological; Papio; Raclopride; Receptors, Dopamine D2; Spiperone; Tomography, Emission-Computed	2001
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone. Nuclear medicine and biology, 2002, Volume: 29, Issue:3 Topics: Animals; Autoradiography; Benzamides; Dopamine Antagonists; Glucose; Magnetic Resonance Imaging; Male; Neostriatum; Neurotoxins; Quinolinic Acid; Raclopride; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Tomography, Emission-Computed	2002
Effects of rolipram on in vivo dopamine receptor binding. Journal of neural transmission (Vienna, Austria : 1996), 2002, Volume: 109, Issue:9 Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Benzazepines; Binding Sites; Brain; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Mice; Neurons; Phosphodiesterase Inhibitors; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Rolipram; Spiperone	2002
In vivo evidence for dopamine-mediated internalization of D2-receptors after amphetamine: differential findings with [3H]raclopride versus [3H]spiperone. Molecular pharmacology, 2003, Volume: 63, Issue:2 Topics: Amphetamine; Animals; Binding Sites; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Endocytosis; Guanylyl Imidodiphosphate; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Time Factors; Tritium	2003
Effect of sabcomeline on muscarinic and dopamine receptor binding in intact mouse brain. Annals of nuclear medicine, 2003, Volume: 17, Issue:2 Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Diagnostic Techniques, Radioisotope; Dose-Response Relationship, Drug; Imines; Male; Metabolic Clearance Rate; Mice; Mice, Inbred Strains; Organ Specificity; Piperidines; Protein Binding; Quinuclidines; Quinuclidinyl Benzilate; Raclopride; Radionuclide Imaging; Radiopharmaceuticals; Receptors, Dopamine; Spiperone; Tissue Distribution; Tritium	2003
Dopamine displaces [3H]domperidone from high-affinity sites of the dopamine D2 receptor, but not [3H]raclopride or [3H]spiperone in isotonic medium: Implications for human positron emission tomography. Synapse (New York, N.Y.), 2003, Sep-15, Volume: 49, Issue:4 Topics: Animals; Domperidone; Dopamine; Dopamine Antagonists; Isotonic Solutions; Raclopride; Rats; Receptors, Dopamine D2; Sodium; Spiperone; Tomography, Emission-Computed; Tritium	2003
MDMA-evoked changes in [11C]raclopride and [11C]NMSP binding in living pig brain. Synapse (New York, N.Y.), 2004, Sep-15, Volume: 53, Issue:4 Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbon Radioisotopes; Cerebrovascular Circulation; Corpus Striatum; Dopamine; Down-Regulation; Drug Interactions; Female; N-Methyl-3,4-methylenedioxyamphetamine; Presynaptic Terminals; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Serotonin; Spiperone; Sus scrofa; Tomography, Emission-Computed	2004
Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor. Molecular pharmacology, 2006, Volume: 69, Issue:1 Topics: Animals; Benzamides; Cell Line; Dopamine Antagonists; Ligands; Protein Binding; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone	2006
Structural determinants of pharmacological specificity between D(1) and D(2) dopamine receptors. Molecular pharmacology, 2006, Volume: 69, Issue:1 Topics: Alternative Splicing; Animals; Benzazepines; Cell Line; Dopamine Antagonists; Models, Molecular; Mutation; Protein Conformation; Raclopride; Radioligand Assay; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Solvents; Spiperone; Sulpiride	2006
Food restriction markedly increases dopamine D2 receptor (D2R) in a rat model of obesity as assessed with in-vivo muPET imaging ([11C] raclopride) and in-vitro ([3H] spiperone) autoradiography. Synapse (New York, N.Y.), 2008, Volume: 62, Issue:1 Topics: Age Factors; Animals; Apomorphine; Appetite Regulation; Autoradiography; Brain; Disease Models, Animal; Dopamine; Dopamine Agonists; Eating; Food Deprivation; In Vitro Techniques; Male; Motor Activity; Obesity; Positron-Emission Tomography; Raclopride; Rats; Rats, Zucker; Receptors, Dopamine D2; Receptors, Leptin; Spiperone; Tritium	2008
Dopamine D2(High) receptors on intact cells. Synapse (New York, N.Y.), 2008, Volume: 62, Issue:4 Topics: Adenoma; Animals; Binding, Competitive; Corpus Striatum; Domperidone; Dopamine Antagonists; Pituitary Neoplasms; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone	2008
Antagonist-radioligand binding to D2L-receptors in intact cells. Biochemical pharmacology, 2008, Jun-01, Volume: 75, Issue:11 Topics: Animals; CHO Cells; Computer Simulation; Cricetinae; Cricetulus; Deuterium; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Ligands; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone; Time Factors	2008
MDMA-evoked changes in the binding of dopamine D(2) receptor ligands in striatum of rats with unilateral serotonin depletion. Synapse (New York, N.Y.), 2010, Volume: 64, Issue:1 Topics: Animals; Autoradiography; Binding, Competitive; Carbon Radioisotopes; Corpus Striatum; Dopamine Antagonists; Hallucinogens; Image Processing, Computer-Assisted; Ligands; Male; N-Methyl-3,4-methylenedioxyamphetamine; Positron-Emission Tomography; Raclopride; Radioligand Assay; Radiopharmaceuticals; Rats; Rats, Inbred Lew; Receptors, Dopamine D2; Serotonin; Spiperone	2010
Non-competitive interaction between raclopride and spiperone on human D-receptors in intact Chinese hamster ovary cells. Fundamental & clinical pharmacology, 2010, Volume: 24, Issue:3 Topics: Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Humans; Raclopride; Receptors, Dopamine D2; Spiperone	2010
Competition between 11C-raclopride and endogenous dopamine in Parkinson's disease. Nuclear medicine communications, 2010, Volume: 31, Issue:2 Topics: Aged; Binding, Competitive; Carbon Radioisotopes; Case-Control Studies; Dopamine; Female; Humans; Linear Models; Male; Middle Aged; Neostriatum; Nortropanes; Parkinson Disease; Positron-Emission Tomography; Raclopride; Reproducibility of Results; Retrospective Studies; Spiperone; Synapses	2010
The influence of different cellular environments on PET radioligand binding: an application to D2/3-dopamine receptor imaging. Neuropharmacology, 2014, Volume: 85 Topics: Animals; Cell Membrane; Corpus Striatum; Dopamine D2 Receptor Antagonists; Endosomes; Extracellular Space; Kinetics; Male; Positron-Emission Tomography; Raclopride; Radioligand Assay; Radiopharmaceuticals; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Subcellular Fractions; Tritium	2014
Effects of chronic methamphetamine on psychomotor and cognitive functions and dopamine signaling in the brain. Behavioural brain research, 2017, 03-01, Volume: 320 Topics: Animals; Anxiety; Benzazepines; Body Weight; Brain; Carbon Isotopes; Central Nervous System Stimulants; Cognition; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Exploratory Behavior; Male; Methamphetamine; Psychomotor Performance; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recognition, Psychology; Signal Transduction; Spiperone	2017