Page last updated: 2024-08-16

spiperone and quipazine

spiperone has been researched along with quipazine in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-199011 (45.83)18.7374
1990's9 (37.50)18.2507
2000's4 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA2
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Boggan, WO; Buckholtz, NS; Meyer, JS1
Byrd, LD; Howell, LL1
Jeffrey, JJ; Rydelek-Fitzgerald, L; Wilcox, BD1
Done, CJ; Sharp, T1
Fukuda, T; Inaba, K; Kawakita, T; Kuroita, T; Sano, M; Tahara, T; Yasumoto, M1
Jenner, P; Marsden, CD; Stewart, BR1
Eison, AS; Yocca, FD1
Amedro, J; Brown, L; Smith, D; Williams, G1
Gorzalka, BB; Mendelson, SD1
Cohen, ML; Fuller, RW; Garbrecht, WL; Kurz, KD; Marzoni, GP; Mason, NR1
Bartness, T; Carlton, J; Rowland, N; Smith, G1
Barrett, RJ; Friedman, RL; Sanders-Bush, E1
Martin, LL; Sanders-Bush, E1
Cohen, ML; Fuller, RW; Wiley, KS1
Ageel, AM; Alhaider, AA; Ginawi, OT1
Jeffrey, JJ; Rydelek-Fitzgerald, L; Teitler, M; Wilcox, BD1
Knowles, ID; Ramage, AG1
Hernandez, E; Hernandez, J; Manjarrez, G; Robles, A1

Reviews

2 review(s) available for spiperone and quipazine

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

22 other study(ies) available for spiperone and quipazine

ArticleYear
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Serotonergic stimulation of pituitary-adrenal activity in the mouse.
    Neuroendocrinology, 1978, Volume: 26, Issue:5

    Topics: 5-Hydroxytryptophan; Animals; Atropine; Benserazide; Carbidopa; Carbolines; Corticosterone; Cyproheptadine; Female; Fenclonine; Indoles; Metergoline; Mice; Pargyline; Phenyl Ethers; Pituitary-Adrenal System; Propylamines; Quinolines; Quipazine; Spiperone; Tryptophan

1978
Enhanced sensitivity to the behavioral effects of cocaine after chronic administration of D2-selective dopamine antagonists in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Fluoxetine; Infusion Pumps; Male; Quipazine; Receptors, Dopamine; Receptors, Dopamine D2; Saimiri; Spiperone

1992
Regulation of collagenase gene expression by serotonin and progesterone in rat uterine smooth muscle cells.
    The Journal of biological chemistry, 1992, Oct-15, Volume: 267, Issue:29

    Topics: Amphetamines; Animals; Cell Nucleus; Cells, Cultured; Collagenases; DNA Probes; Female; Gene Expression Regulation, Enzymologic; Ketanserin; Kinetics; Muscle, Smooth; Myometrium; Progesterone; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Spiperone; Tetradecanoylphorbol Acetate; Transcription, Genetic; Uterus

1992
Evidence that 5-HT2 receptor activation decreases noradrenaline release in rat hippocampus in vivo.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electrophysiology; Hippocampus; Male; Neurons; Norepinephrine; p-Chloroamphetamine; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Receptor Agonists; Spiperone; Sulpiride

1992
Synthesis and pharmacology of 3,4-dihydro-3-oxo-1,4-benzoxazine-8-carboxamide derivatives, a new class of potent serotonin-3 (5-HT3) receptor antagonists.
    Chemical & pharmaceutical bulletin, 1992, Volume: 40, Issue:3

    Topics: Animals; Antiemetics; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Cyclophosphamide; Doxorubicin; Magnetic Resonance Spectroscopy; Male; Oxazines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Spiperone; Structure-Activity Relationship

1992
Induction of purposeless chewing behaviour in rats by 5-HT agonist drugs.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Male; Methiothepin; Methoxydimethyltryptamines; Mianserin; Parasympatholytics; Piperazines; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1989
Reduction in cortical 5HT2 receptor sensitivity after continuous gepirone treatment.
    European journal of pharmacology, 1985, May-20, Volume: 111, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Dose-Response Relationship, Drug; Female; Humans; Male; Pyrimidines; Quipazine; Rats; Receptors, Serotonin; Spiperone; Stereotyped Behavior

1985
A pharmacological analysis of the rat spinal cord serotonin (5-HT) autoreceptor.
    European journal of pharmacology, 1988, Jan-12, Volume: 145, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Male; Piperazines; Potassium; Quipazine; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Spiperone; Tetrahydronaphthalenes; Tritium

1988
A facilitatory role for serotonin in the sexual behavior of the female rat.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone

1985
Pharmacological activity of the isomers of LY53857, potent and selective 5-HT2 receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Blood Pressure; Cerebral Cortex; Corticosterone; Decerebrate State; Ergolines; Isomerism; Male; Mathematics; Quipazine; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Time Factors

1985
Effect of chronic administration of fenfluramine and quipazine on body weight gain after ovariectomy and on brain serotonin receptor binding.
    Behavioral neuroscience, 1983, Volume: 97, Issue:3

    Topics: Animals; Appetite; Body Weight; Brain; Castration; Female; Fenfluramine; Muridae; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone

1983
Discriminative stimulus properties of quipazine: mediation by serotonin2 binding sites.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:3

    Topics: Animals; Cues; Discrimination Learning; Dose-Response Relationship, Drug; Lysergic Acid Diethylamide; Male; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1984
The serotonin autoreceptor: antagonism by quipazine.
    Neuropharmacology, 1982, Volume: 21, Issue:5

    Topics: Animals; Calcium; Fluoxetine; Hypothalamus; In Vitro Techniques; Male; Methiothepin; Phentolamine; Potassium; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1982
Evidence for 5-HT2 receptors mediating contraction in vascular smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 218, Issue:2

    Topics: Animals; Aorta; In Vitro Techniques; Jugular Veins; Male; Muscle Contraction; Muscle, Smooth, Vascular; Quipazine; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1981
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes

1993
Serotonin-mediated 5-HT2 receptor gene regulation in rat myometrial smooth muscle cells.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Biguanides; Cells, Cultured; Cycloheximide; Female; Gene Expression Regulation; Ketanserin; Medroxyprogesterone Acetate; Myometrium; Piperazines; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sulpiride; Transcription, Genetic; Up-Regulation

1993
Evidence for a role for central 5-HT2B as well as 5-HT2A receptors in cardiovascular regulation in anaesthetized rats.
    British journal of pharmacology, 1999, Volume: 128, Issue:3

    Topics: Amidines; Amphetamines; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine Derivatives; Blood Pressure; Cardiovascular Physiological Phenomena; Cinanserin; Injections, Intraventricular; Male; Polyethylene Glycols; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Spiperone

1999
N1/P2 component of auditory evoked potential reflect changes of the brain serotonin biosynthesis in rats.
    Nutritional neuroscience, 2005, Volume: 8, Issue:4

    Topics: Animals; Auditory Cortex; Brain; Electrophysiology; Evoked Potentials, Auditory; Male; Quipazine; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tryptophan

2005