Page last updated: 2024-08-16

spiperone and quinpirole

spiperone has been researched along with quinpirole in 90 studies

Research

Studies (90)

TimeframeStudies, this research(%)All Research%
pre-199022 (24.44)18.7374
1990's49 (54.44)18.2507
2000's18 (20.00)29.6817
2010's1 (1.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bunzow, JR; Civelli, O; Guan, HC; Niznik, HB; Seeman, P; Sunahara, RK; Van Tol, HH1
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P1
Bervoets, K; Brocco, M; Dacquet, C; Girardon, S; Gobert, A; Millan, MJ; Newman-Tancredi, A; Peglion, JL; Rivet, JM; Vian, J1
Billings, J; Chumpradit, S; Kung, HF; Kung, MP; Mach, R1
Doll, MK; Kilts, JD; Lawler, CP; Lewis, MM; Mailman, RB; Nichols, DE; Prioleau, C1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Jenner, P; Marsden, CD; Rose, S; Thomas, KL1
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD1
Lucki, I; McGonigle, P; Subramaniam, S1
DeSouza, EB; Grigoriadis, DE; Levant, B2
LaHoste, GJ; Marshall, JF1
Kozlowski, MR; Neve, KA; Rosser, MP1
Todd, RD1
Boroni, F; Castelletti, L; Memo, M; Missale, C; Spano, P1
Gong, L; Kostrzewa, RM1
Michel, AD; Nunes, JL; Sharif, NA; Whiting, RL1
Schaus, JM; Seeman, P1
Brus, R; Kalbfleisch, J; Kostrzewa, RM1
Bourque, CW; Renaud, LP; Yang, CR1
Courtney, ND; Howlett, AC; Westfall, TC1
Linseman, MA1
Nowak, JZ; Schorderet, M1
Gessa, GL; Olianas, MC; Onali, P1
Iuvone, PM1
Beaulieu, M; Felder, R; Kebabian, JW1
Doty, RL; Risser, JM1
Segawa, T; Zhang, X1
Allin, R; Reyneke, L; Russell, VA; Taljaard, JJ1
Klimek, V; Maj, J1
Arnt, J; Hyttel, J1
Crocker, AD; Faunt, JE2
Battaglia, G; Creese, I; Hess, EJ; Norman, AB1
Beart, PM; Bridge, S; Christie, MJ1
Ares, J; Chang, YA; Farooqui, T; Miller, D; Uretsky, N; Wallace, L; Wallace, RA1
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW1
Arnt, J; Hyttel, J; Nowak, G1
Burchill, SA; Thody, AJ1
Bondy, SC; Breese, GR; Duncan, GE; Iorio, LC; Mueller, RA; Napier, TC1
Fuller, RW; Hemrick-Luecke, SK1
Anderson, D; Gordon, J; Herbster, G; Koller, W; Wack, R1
Brunello, N; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC1
Liskowsky, DR; Potter, LT1
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K1
Senogles, SE1
Bancroft, C; Fischberg, DJ1
Barrett, RJ; Caul, WF; Huffman, EM; Jones, JR; Strand, EJ1
Erol, DD; Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD; Smith, LA1
Abarca, J; Bustos, G; Gysling, K; Roth, RH1
Katz, JL; Witkin, JM1
Contestabile, A; Dall'Olio, R; Facchinetti, F; Gandolfi, O1
Guo, J; Kostrzewa, FP; Kostrzewa, RM1
Bernard, A; Cavegn, C; Chabert, C; Mills, A1
Dall'Olio, R; Gandolfi, O; Rimondini, R2
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD1
Nowak, JZ; Zawilska, JB1
Burnham, P; Louis, JC; Magal, E; Varon, S1
Dall'Olio, R; Gandolfi, O1
Aloyo, VJ; Chen, JF; Weiss, B1
Ball, S; Boyfield, I; Coldwell, MC; Cook, T; Gloger, IS; Herrity, N; McHale, M; Robinson, JH; Winn, FM1
Allard, S; Falardeau, P; Lapointe, S1
Allet, B; Bernard, A; Brandt, E; Cavegn, C; Chabert, C; Chollet, A; Kawashima, E; Mills, A1
Felder, RA; Jose, PA; Walk, SF; Yamaguchi, I1
Cheng, CC; Leonard, NL; Levant, B; Moehlenkamp, JD; Morgan, KA1
Domae, M; Furukawa, T; Inoue, T; Kurashima, M; Nagashima, M; Shirakawa, K; Yamada, K1
Bancroft, GN; Levant, B1
Kuzhikandathil, EV; Oxford, GS; Yu, W1
Cook, CD; Picker, MJ; Rodefer, JS1
Hu, JY; Jin, GZ2
Jaliffa, CO; Lacoste, FF; Llomovatte, DW; Rosenstein, RE; Sarmiento, MI1
Cypess, AM; Graber, SG; Kazmi, MA; Sakmar, TP; Snyder, LA1
Kumar, U; Lange, DC; Patel, RC; Patel, SC; Patel, YC; Rocheville, M1
Alper, RH; Gilliland, SL; Levant, B1
Armogida, M; Chiacchio, S; Colzi, A; Corsini, GU; DeMontis, MG; Maggio, R; Scarselli, M1
Baik, JH; Borrelli, E; Dierich, A; LeMeur, M; Piazza, PV; Picetti, R; Rougé-Pont, F; Usiello, A1
Bridges, SR; Thompson, TL; Weirs, WJ1
Einsiedel, J; Gmeiner, P; Hübner, H1
Ahlgren-Beckendorf, JA; Chen, K; Grandy, DK; Levant, B; Morgan, KA; Seif, I; Shih, JC1
Chesneau, D; de la Riva, C; Fabre-Nys, C; Hinton, MR; Kendrick, KM; Locatelli, A; Ohkura, S1
Jaliffa, CO; Keller Sarmiento, MI; Minces, L; Rosenstein, RE; Sacca, GB; Sáenz, DA1
Lau, YS; Meredith, GE; Petroske, E; Wang, JQ1
Ebadi, M; Govitrapong, P; Santanavanich, C1
Buck, DC; Macey, TA; Neve, KA; Wang, C; Yang, R1
Cleland, TA; Linster, C; Wei, CJ1
Cho, EY; Kim, JH; Kim, KM; Min, C; Park, JH1
Culver, KE; Levant, B; Szechtman, H1
Antipov, A; Blessing, WW; Brizuela, M; Ootsuka, Y1

Reviews

1 review(s) available for spiperone and quinpirole

ArticleYear
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates

1990

Other Studies

89 other study(ies) available for spiperone and quinpirole

ArticleYear
Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cloning, Molecular; Clozapine; Gene Library; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Neuroblastoma; Organ Specificity; Protein Conformation; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
    Nature, 1990, Sep-13, Volume: 347, Issue:6289

    Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution

1990
Functional correlates of dopamine D3 receptor activation in the rat in vivo and their modulation by the selective antagonist, (+)-S 14297: 1. Activation of postsynaptic D3 receptors mediates hypothermia, whereas blockade of D2 receptors elicits prolactin
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: 2-Naphthylamine; Animals; Body Temperature Regulation; Catalepsy; CHO Cells; Cricetinae; Dopamine Antagonists; Furans; Humans; Male; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins; Stereoisomerism

1995
Fluorinated and iodinated dopamine agents: D2 imaging agents for PET and SPECT.
    Journal of medicinal chemistry, 1993, Jan-22, Volume: 36, Issue:2

    Topics: Animals; Benzamides; Dopamine Agents; Dopamine D2 Receptor Antagonists; Fluorine Radioisotopes; Iodine Radioisotopes; Macaca fascicularis; Male; Pyrrolidines; Radionuclide Imaging; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon

1993
Synthesis and dopaminergic properties of benzo-fused analogues of quinpirole and quinelorane.
    Journal of medicinal chemistry, 1999, Mar-11, Volume: 42, Issue:5

    Topics: Animals; Binding, Competitive; Dopamine Agonists; In Vitro Techniques; Isoquinolines; Male; Naphthols; Neostriatum; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Structure-Activity Relationship

1999
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Dissociation of the striatal D-2 dopamine receptor from adenylyl cyclase following 6-hydroxydopamine-induced denervation.
    Biochemical pharmacology, 1992, Jul-07, Volume: 44, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Denervation; Dopamine; Ergolines; Female; Homovanillic Acid; Oxidopamine; Prosencephalon; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1992
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Dec-15, Volume: 89, Issue:24

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone

1992
Effects of chronic treatment with selective agonists on the subtypes of dopamine receptors.
    Brain research, 1992, Feb-07, Volume: 571, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Body Temperature Regulation; Brain; Caudate Nucleus; Dopamine Agents; Drug Interactions; Ergolines; Kinetics; Male; Nucleus Accumbens; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reference Values; Spiperone; Substantia Nigra

1992
Characterization of [3H]quinpirole binding to D2-like dopamine receptors in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Binding Sites; Brain; Culture Techniques; Dopamine Agents; Dopamine Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone

1992
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
    Synapse (New York, N.Y.), 1992, Volume: 12, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium

1992
Dopamine D2 receptor stimulation of Na+/H+ exchange assessed by quantification of extracellular acidification.
    The Journal of biological chemistry, 1992, Dec-25, Volume: 267, Issue:36

    Topics: Amiloride; Animals; Carrier Proteins; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Glioma; Hydrogen-Ion Concentration; Kinetics; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Sodium-Hydrogen Exchangers; Spiperone; Tumor Cells, Cultured

1992
Neural development is regulated by classical neurotransmitters: dopamine D2 receptor stimulation enhances neurite outgrowth.
    Biological psychiatry, 1992, Apr-15, Volume: 31, Issue:8

    Topics: Animals; Base Sequence; Brain; Cells, Cultured; Cerebral Cortex; Ergolines; Female; Male; Mental Disorders; Models, Biological; Molecular Sequence Data; Nerve Growth Factors; Neurites; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; RNA, Messenger; Salicylamides; Spiperone

1992
Epidermal growth factor induces the functional expression of dopamine receptors in the GH3 cell line.
    Endocrinology, 1991, Volume: 128, Issue:1

    Topics: Animals; Binding, Competitive; Cell Line; Cells, Cultured; Dopamine Agents; Epidermal Growth Factor; Ergolines; Kinetics; Pituitary Gland, Anterior; Pituitary Neoplasms; Potassium; Prolactin; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1991
Supersensitized D1 receptors mediate enhanced oral activity after neonatal 6-OHDA.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Mouth; Movement; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1991
Dopamine D2-receptors mediate hypothermia in mice: ICV and IP effects of agonists and antagonists.
    Neurochemical research, 1991, Volume: 16, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Body Temperature Regulation; Cerebral Ventricles; Domperidone; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1991
Dopamine receptors labelled by [3H]quinpirole.
    European journal of pharmacology, 1991, Oct-02, Volume: 203, Issue:1

    Topics: Animals; Corpus Striatum; Dogs; Dopamine Agents; Dopamine Antagonists; Ergolines; Guanine Nucleotides; Haloperidol; In Vitro Techniques; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1991
Ontogenetic homologous sensitization to the antinociceptive action of quinpirole in rats.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Aging; Analgesics; Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Female; Pain Measurement; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1991
Dopamine D2 receptor activation depolarizes rat supraoptic neurones in hypothalamic explants.
    The Journal of physiology, 1991, Volume: 443

    Topics: Animals; Calcium; Dopamine; Dopamine Agents; Ergolines; Membrane Potentials; Neurons; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Sulpiride; Supraoptic Nucleus

1991
Dopaminergic regulation of dopamine release from PC12 cells via a pertussis toxin-sensitive G protein.
    Neuroscience letters, 1991, Jan-28, Volume: 122, Issue:2

    Topics: Adrenal Gland Neoplasms; Animals; Apomorphine; Cell Line; Dopamine; Dopamine Antagonists; Ergolines; GTP-Binding Proteins; Haloperidol; Nicotine; Pertussis Toxin; Pheochromocytoma; Potassium; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Virulence Factors, Bordetella

1991
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
    Psychopharmacology, 1990, Volume: 100, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1990
Characterization of dopamine receptors mediating inhibition of adenylate cyclase activity in rat striatum.
    Molecular pharmacology, 1985, Volume: 28, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butaclamol; Corpus Striatum; Dopamine; Enzyme Activation; Ergolines; Guanine Nucleotides; Norepinephrine; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Sulpiride

1985
Evidence for a D2 dopamine receptor in frog retina that decreases cyclic AMP accumulation and serotonin N-acetyltransferase activity.
    Life sciences, 1986, Jan-27, Volume: 38, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Bucladesine; Calcium; Circadian Rhythm; Cyclic AMP; Dopamine; Ergolines; Light; Metoclopramide; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Retina; Spiperone; Xenopus laevis

1986
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
Influence of the D-2 dopamine receptor agonist quinpirole on the odor detection performance of rats before and after spiperone administration.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Acetates; Animals; Behavior, Animal; Conditioning, Operant; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Smell; Spiperone

1989
Selective blockade of dopamine D-1 receptor by SCH 23390 affects dopamine agonist binding to 3H-spiperone labeled D-2 receptors in rat striatum.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Guanosine Triphosphate; In Vitro Techniques; Male; Pertussis Toxin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Virulence Factors, Bordetella

1989
Lack of effect of chronic desipramine treatment on dopaminergic activity in the nucleus accumbens of the rat.
    Neurochemical research, 1989, Volume: 14, Issue:7

    Topics: Acetylcholine; Animals; Benzazepines; Desipramine; Dopamine; Dopamine Agents; Dopamine Antagonists; Electric Stimulation; Ergolines; Male; Nomifensine; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Septal Nuclei; Spiperone

1989
Repeated administration of antidepressants enhances agonist affinity for mesolimbic D2-receptors.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:8

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Binding, Competitive; Ergolines; Imipramine; Limbic System; Male; Mianserin; Motor Activity; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spiperone

1989
Differential involvement of dopamine D-1 and D-2 receptors in the circling behaviour induced by apomorphine, SK & F 38393, pergolide and LY 171555 in 6-hydroxydopamine-lesioned rats.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Appetite Depressants; Benzazepines; Electric Stimulation; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical; Time Factors

1985
Adrenocortical hormone status affects responses to dopamine receptor agonists.
    European journal of pharmacology, 1988, Aug-02, Volume: 152, Issue:3

    Topics: Adrenal Cortex Hormones; Adrenalectomy; Animals; Apomorphine; Behavior, Animal; Benzazepines; Body Temperature; Corticosterone; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1988
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
    Neuroscience letters, 1985, Aug-30, Volume: 59, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
No change in neostriatal D-2 dopamine receptors after NMDA lesions of rat prefrontal cortex.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:6

    Topics: Animals; Aspartic Acid; Corpus Striatum; Ergolines; Female; Frontal Lobe; Male; N-Methylaspartate; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tritium

1986
The effects of selective dopamine receptor agonists and antagonists on body temperature in rats.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Temperature; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1987
Interaction of permanently uncharged dopamine analogs with the D-2 dopaminergic receptor.
    Biochemical pharmacology, 1988, May-15, Volume: 37, Issue:10

    Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Ergolines; In Vitro Techniques; Male; Mice; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sodium Chloride; Spiperone; Sulfides

1988
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
    Advances in experimental medicine and biology, 1988, Volume: 235

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
    European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone

1988
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
    The Journal of endocrinology, 1986, Volume: 111, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride

1986
6-hydroxydopamine treatments enhance behavioral responses to intracerebral microinjection of D1- and D2-dopamine agonists into nucleus accumbens and striatum without changing dopamine antagonist binding.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Ergolines; Female; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Microinjections; Motor Activity; Nucleus Accumbens; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone

1987
Decrease in hypothalamic epinephrine concentration and other neurochemical changes produced by quinpirole, a dopamine agonist, in rats.
    Journal of neural transmission, 1985, Volume: 61, Issue:3-4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Epinephrine; Ergolines; Homovanillic Acid; Hypothalamus; Male; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Quinpirole hydrochloride, a potential anti-parkinsonism drug.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: Animals; Benzazepines; Corpus Striatum; Dogs; Dose-Response Relationship, Drug; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride

1987
Absence of [3H]SCH 23390 specific binding sites in anterior pituitary: dissociation from effects on prolactin secretion.
    European journal of pharmacology, 1987, Mar-17, Volume: 135, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Corpus Striatum; Cyproheptadine; Ergolines; Kinetics; Male; Metergoline; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1987
D-2 dopamine receptors in the frontal cortex of rat and human.
    Life sciences, 1985, Apr-22, Volume: 36, Issue:16

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Cinanserin; Dopamine; Ergolines; Humans; Kinetics; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
    Acta physiologica Scandinavica, 1983, Volume: 117, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
    Endocrinology, 1994, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1994
The D2 receptor: blocked transcription in GH3 cells and cellular pathways employed by D2A to regulate prolactin promoter activity.
    Molecular and cellular endocrinology, 1995, Volume: 111, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Cell Line; Chloramphenicol O-Acetyltransferase; DNA-Binding Proteins; Ergolines; Gene Expression Regulation; Pertussis Toxin; Pituitary Gland; Prolactin; Promoter Regions, Genetic; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Thyrotropin-Releasing Hormone; Transcription Factor Pit-1; Transcription Factors; Transcription, Genetic; Transfection; Virulence Factors, Bordetella

1995
D2-specific discriminative stimuli: parameters, blocking, and rebound.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 51, Issue:1

    Topics: Animals; Cues; Discrimination, Psychological; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Food Deprivation; Haloperidol; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Spiperone

1995
Differential anti-parkinsonian effects of benzazepine D1 dopamine agonists with varying efficacies in the MPTP-treated common marmoset.
    Psychopharmacology, 1995, Volume: 117, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antiparkinson Agents; Behavior, Animal; Benzazepines; Binding, Competitive; Callithrix; Dopamine Agonists; Ergolines; In Vitro Techniques; Male; Parkinson Disease, Secondary; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1995
Changes in extracellular levels of glutamate and aspartate in rat substantia nigra induced by dopamine receptor ligands: in vivo microdialysis studies.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aspartic Acid; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Extracellular Space; Glutamic Acid; Kinetics; Ligands; Male; Microdialysis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Substantia Nigra; Tetrodotoxin; Time Factors

1995
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
    Psychopharmacology, 1993, Volume: 113, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone

1993
Chronic neonatal blockade of N-methyl-D-aspartate receptor by CGP 39551 increases dopaminergic function in adult rat.
    Neuroscience, 1994, Volume: 63, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Apomorphine; Behavior, Animal; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Motor Activity; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; Spiperone; Stereotyped Behavior; Time Factors

1994
Ontogenetic quinpirole treatment induces vertical jumping activity in rats.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Injections, Intraperitoneal; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1993
Characterization of the functional activity of dopamine ligands at human recombinant dopamine D4 receptors.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: Animals; Cell Line; Clozapine; DNA; Dopamine; Dopamine Agents; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Ligands; Moths; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Sulfur Radioisotopes; Tritium

1994
D-cycloserine decreases both D1 and D2 dopamine receptors number and their function in rat brain.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Cell Membrane; Cycloserine; Dizocilpine Maleate; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; In Vitro Techniques; Kinetics; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1994
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
    Neuropharmacology, 1994, Volume: 33, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
    Neuroscience, 1993, Volume: 52, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase

1993
Chronic treatment with MK-801 decreases D2 dopamine receptor function in rat striatum.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Grooming; In Vitro Techniques; Kinetics; Ligands; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone

1993
Continuous treatment with the D2 dopamine receptor agonist quinpirole decreases D2 dopamine receptors, D2 dopamine receptor messenger RNA and proenkephalin messenger RNA, and increases mu opioid receptors in mouse striatum.
    Neuroscience, 1993, Volume: 54, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Behavior, Animal; Blotting, Northern; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Down-Regulation; Enkephalins; Ergolines; Image Processing, Computer-Assisted; Male; Mice; Nucleic Acid Hybridization; Oligonucleotide Probes; Protein Precursors; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Spiperone; Up-Regulation

1993
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone

1993
Expression and functional characterisation of a synthetic version of the human D4 dopamine receptor in a stable human cell line.
    FEBS letters, 1994, May-30, Volume: 345, Issue:2-3

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Binding, Competitive; Cell Line; Chlorocebus aethiops; Colforsin; DNA; Ergolines; Genes, Synthetic; Humans; Kidney; Kinetics; Molecular Sequence Data; Plasmids; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; Spiperone; Transfection

1994
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
    Biochemical and biophysical research communications, 1993, Jun-15, Volume: 193, Issue:2

    Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1993
Expression and characterization of human D4 dopamine receptors in baculovirus-infected insect cells.
    FEBS letters, 1993, Apr-05, Volume: 320, Issue:2

    Topics: Animals; Baculoviridae; Base Sequence; Cell Line; Ergolines; Genetic Vectors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Introns; Molecular Sequence Data; Moths; Occlusion Body Matrix Proteins; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Fusion Proteins; Spiperone; Viral Proteins; Viral Structural Proteins

1993
Dopamine D2L receptors stimulate Na+/K(+)-ATPase activity in murine LTK- cells.
    Molecular pharmacology, 1996, Volume: 49, Issue:2

    Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dideoxyadenosine; Dopamine Agonists; Ergolines; Kinetics; L Cells; Mice; Ouabain; Pertussis Toxin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Rubidium; Sodium-Potassium-Exchanging ATPase; Spiperone; Transfection; Virulence Factors, Bordetella

1996
Modulation of [3H]quinpirole binding in brain by monoamine oxidase inhibitors: evidence for a potential novel binding site.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone

1996
Inhibitory effects of putative dopamine D3 receptor agonists, 7-OH-DPAT and quinpirole, on prolactin secretion in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: alpha-Methyltyrosine; Animals; Body Temperature; Depression, Chemical; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estradiol; Male; Methyltyrosines; Prolactin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase; Yawning

1996
Effects of competitive and non-competitive NMDA receptor antagonists on behavioral responses induced by 7-OH-DPAT and quinpirole in rats.
    Pharmacological research, 1997, Volume: 36, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Dizocilpine Maleate; Dopamine Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Neostriatum; Nucleus Accumbens; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spiperone; Tetrahydronaphthalenes

1997
Inhibition of [3H]quinpirole binding by a monoamine oxidase inhibitor in subcellular fractions of rat striatum.
    Life sciences, 1998, Volume: 63, Issue:18

    Topics: Animals; Binding, Competitive; Dopamine Agonists; In Vitro Techniques; Male; Monoamine Oxidase Inhibitors; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Ribosomes; Spiperone; Subcellular Fractions; Synaptosomes

1998
Human dopamine D3 and D2L receptors couple to inward rectifier potassium channels in mammalian cell lines.
    Molecular and cellular neurosciences, 1998, Volume: 12, Issue:6

    Topics: Adenosine Triphosphate; Animals; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Gene Expression; Humans; Mammals; Membrane Potentials; Mice; Pertussis Toxin; Pituitary Gland; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Somatostatin; Sodium Chloride; Somatostatin; Spiperone; Transfection; Tritium; Virulence Factors, Bordetella

1998
Selective attenuation of the antinociceptive effects of mu opioids by the putative dopamine D3 agonist 7-OH-DPAT.
    Psychopharmacology, 1999, Volume: 144, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Opioid; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cycloparaffins; Dopamine Agonists; Dopamine Antagonists; Drug Antagonism; Male; Morphine; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Spiperone; Tetrahydronaphthalenes

1999
Effect of tetrahydropalmatine analogs on Fos expression induced by formalin-pain.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:3

    Topics: Analgesics, Non-Narcotic; Animals; Berberine; Berberine Alkaloids; Brain; Dopamine Agonists; Dopamine Antagonists; Formaldehyde; Male; Pain; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Sprague-Dawley; Spinal Cord; Spiperone

1999
Supraspinal D2 receptor involved in antinociception induced by l-tetrahydropalmatine.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Non-Narcotic; Animals; Benzazepines; Berberine Alkaloids; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Injections, Spinal; Male; Pain Threshold; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1999
Dopamine decreases melatonin content in golden hamster retina.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Chromatography, High Pressure Liquid; Circadian Rhythm; Clozapine; Cricetinae; Cyclic AMP; Depression, Chemical; Dopamine; Dopamine Agonists; Dopamine Antagonists; Kinetics; Male; Melatonin; Mesocricetus; Quinpirole; Receptors, Dopamine; Retina; Spiperone

2000
Selective reconstitution of human D4 dopamine receptor variants with Gi alpha subtypes.
    Biochemistry, 2000, Apr-04, Volume: 39, Issue:13

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amino Acid Sequence; Animals; Calcium; Cell Line; COS Cells; Cytoplasm; Gene Expression; Genes, Synthetic; Genetic Variation; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Mice; Molecular Sequence Data; Peptide Fragments; Protein Binding; Protein Engineering; Protein Structure, Secondary; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Fusion Proteins; Recombinant Proteins; Spiperone

2000
Receptors for dopamine and somatostatin: formation of hetero-oligomers with enhanced functional activity.
    Science (New York, N.Y.), 2000, Apr-07, Volume: 288, Issue:5463

    Topics: Animals; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Dimerization; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Humans; Ligands; Male; Neurons; Pyramidal Cells; Quinpirole; Rats; Receptor Cross-Talk; Receptors, Dopamine D2; Receptors, Somatostatin; Somatostatin; Spiperone; Sulpiride; Transfection

2000
Pharmacology of quinpirole-stimulated [35S]GTPgammaS binding: discrepancy with receptor binding profile.
    European journal of pharmacology, 2000, Mar-31, Volume: 392, Issue:3

    Topics: Animals; Benzazepines; Binding, Competitive; Clorgyline; Clozapine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Membranes; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Selegiline; Spiperone; Sulfur Radioisotopes; Thiazoles

2000
Reconstitution of functional dopamine D(2s) receptor by co-expression of amino- and carboxyl-terminal receptor fragments.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Animals; Apomorphine; Binding, Competitive; Clozapine; Colforsin; COS Cells; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gene Expression; Haloperidol; Membranes; Peptide Fragments; Pergolide; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Transfection; Tritium

2000
Distinct functions of the two isoforms of dopamine D2 receptors.
    Nature, 2000, Nov-09, Volume: 408, Issue:6809

    Topics: Animals; Apomorphine; Benzazepines; Catalepsy; Chimera; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutagenesis; Protein Isoforms; Quinpirole; Receptors, Dopamine D2; Signal Transduction; Spiperone; Synapses

2000
Alteration of dopamine transport in the striatum and nucleus accumbens of ovariectomized and estrogen-primed rats following N-(p-isothiocyanatophenethyl) spiperone (NIPS) treatment.
    Brain research bulletin, 2001, Volume: 54, Issue:6

    Topics: Animals; Carrier Proteins; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Drug Interactions; Estrogens; Estrus; Female; Guanosine 5'-O-(3-Thiotriphosphate); Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Nucleus Accumbens; Ovariectomy; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Synaptosomes; Tritium

2001
Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179).
    Bioorganic & medicinal chemistry letters, 2001, Sep-17, Volume: 11, Issue:18

    Topics: Animals; Biochemistry; Cattle; CHO Cells; Clozapine; Cricetinae; Cysteine; Dopamine Antagonists; Drug Design; Humans; In Vitro Techniques; Indoles; Magnetic Resonance Spectroscopy; Molecular Structure; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Serine; Spiperone; Stereoisomerism; Structure-Activity Relationship; Threonine

2001
Modulation of [3H]quinpirole binding at striatal D2 dopamine receptors by a monoamine oxidaseA-like site: evidence from radioligand binding studies and D2 receptor- and MAO(A)-deficient mice.
    Life sciences, 2001, Nov-30, Volume: 70, Issue:2

    Topics: Animals; Binding Sites; Corpus Striatum; Dopamine Agonists; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Thiazoles; Tritium

2001
Biphasic role of dopamine on female sexual behaviour via D2 receptors in the mediobasal hypothalamus.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Aspartic Acid; Citrulline; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Estradiol; Extracellular Space; Female; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Goats; Hypothalamus, Middle; Luteinizing Hormone; Microdialysis; Norepinephrine; Ovariectomy; Pimozide; Prolactin; Quinpirole; Receptors, Dopamine D2; Serotonin; Sexual Behavior, Animal; Spiperone; Taurine; Time Factors

2003
Photic regulation of heme oxygenase activity in the golden hamster retina: involvement of dopamine.
    Journal of neurochemistry, 2003, Volume: 85, Issue:2

    Topics: Animals; Benzazepines; Bilirubin; Bucladesine; Circadian Rhythm; Clozapine; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Activation; Enzyme Inhibitors; Heme Oxygenase (Decyclizing); In Vitro Techniques; Male; Mesocricetus; Photoperiod; Quinpirole; Retina; Spiperone; Thiobarbituric Acid Reactive Substances

2003
Elevated neuronal nitric oxide synthase expression in chronic haloperidol-treated rats.
    Neuropharmacology, 2003, Volume: 45, Issue:7

    Topics: Animals; Basal Ganglia; Behavior, Animal; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Immunohistochemistry; In Situ Hybridization; Male; Neostriatum; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Spiperone

2003
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
    Journal of pineal research, 2005, Volume: 38, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic

2005
Dopamine D2 receptor stimulation of mitogen-activated protein kinases mediated by cell type-dependent transactivation of receptor tyrosine kinases.
    Journal of neurochemistry, 2005, Volume: 93, Issue:4

    Topics: Animals; Animals, Newborn; Blotting, Western; Cells, Cultured; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Epidermal Growth Factor; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Genetic Vectors; Humans; Indole Alkaloids; Microscopy, Confocal; Neuroblastoma; Piperazines; Platelet-Derived Growth Factor; Quinazolines; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor Protein-Tyrosine Kinases; Receptors, Dopamine D2; Simplexvirus; Spiperone; Transcriptional Activation; Transfection; Tritium; Tyrphostins

2005
Dopamine D(2) receptor activation modulates perceived odor intensity.
    Behavioral neuroscience, 2006, Volume: 120, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Discrimination, Psychological; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Odorants; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Sensory Thresholds; Spiperone

2006
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors.
    Archives of pharmacal research, 2008, Volume: 31, Issue:4

    Topics: Amino Acid Motifs; Apomorphine; Arginine; Aspartic Acid; Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Mutation; Protein Conformation; Protein Structure, Tertiary; Protein Transport; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Spiperone; Sulpiride; Transfection

2008
Altered dopamine D2-like receptor binding in rats with behavioral sensitization to quinpirole: effects of pre-treatment with Ro 41-1049.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: Animals; Behavior, Animal; Dopamine Agonists; Dopamine Antagonists; Kinetics; Male; Monoamine Oxidase Inhibitors; Motor Activity; Neostriatum; Nucleus Accumbens; Quinpirole; Radioligand Assay; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Spiperone; Thiazoles

2008
Activating dopamine D2 receptors reduces brown adipose tissue thermogenesis induced by psychological stress and by activation of the lateral habenula.
    Scientific reports, 2019, 12-20, Volume: 9, Issue:1

    Topics: Adipose Tissue, Brown; Animals; Benzazepines; Dopamine D2 Receptor Antagonists; Habenula; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stress, Psychological; Temperature; Thermogenesis

2019