Page last updated: 2024-08-16

spiperone and pyrilamine

spiperone has been researched along with pyrilamine in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19906 (60.00)18.7374
1990's2 (20.00)18.2507
2000's0 (0.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Andrews, PR; Craik, DJ; Martin, JL1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Feniuk, W; Humphrey, PP; Perren, MJ1
Laduron, PM; Leysen, JE; Van Dun, J; Wouters, W1
Gommeren, W; Janssen, PF; Laduron, PM; Leysen, JE1
Dick, TE; Hughes, MJ; Light, KE1
Berger, D; Burkard, W; Schaffner, W1

Other Studies

10 other study(ies) available for spiperone and pyrilamine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Vascular 5-HT1-like receptors that mediate contraction of the dog isolated saphenous vein and carotid arterial vasoconstriction in anaesthetized dogs are not of the 5-HT1A or 5-HT1D subtype.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Atropine; Carotid Arteries; Dogs; Ganglionic Blockers; In Vitro Techniques; Indoles; Ketanserin; Methiothepin; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Serotonin; Saphenous Vein; Spiperone; Sulfonamides; Sumatriptan; Tetrahydronaphthalenes; Vasoconstriction; Vasoconstrictor Agents

1991
Differential photoaffinity labelling of serotonin-S2 receptors and histamine-H1 receptors using 7-azidoketanserin.
    FEBS letters, 1985, Mar-25, Volume: 182, Issue:2

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Butyrophenones; Cerebellum; Cerebral Cortex; Female; Guinea Pigs; Ketanserin; Photolysis; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Serotonin; Spiperone

1985
In vitro and in vivo binding characteristics of a new long-acting histamine H1 antagonist, astemizole.
    Molecular pharmacology, 1982, Volume: 21, Issue:2

    Topics: Animals; Astemizole; Benzimidazoles; Binding, Competitive; Brain; Guinea Pigs; Histamine Antagonists; Histamine H1 Antagonists; In Vitro Techniques; Lung; Pyrilamine; Rats; Rats, Inbred Strains; Spiperone; Time Factors

1982
Central and peripheral receptors in guinea-pigs exposed to simulated high altitude.
    Neuropharmacology, 1984, Volume: 23, Issue:2A

    Topics: Altitude; Animals; Guinea Pigs; Heart Rate; Kinetics; Male; Myocardium; Norepinephrine; Pyrilamine; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Catecholamine; Receptors, Dopamine; Receptors, Histamine; Receptors, Histamine H1; Spiperone

1984
Influence of Petasites hybridus on dopamine-D2 and histamine-H1 receptors.
    Pharmaceutica acta Helvetiae, 1998, Volume: 72, Issue:6

    Topics: Animals; Asteraceae; Cattle; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Plant Extracts; Plants, Medicinal; Pyrilamine; Radioligand Assay; Receptors, Dopamine D2; Receptors, Histamine H1; Spiperone

1998