Page last updated: 2024-08-16

spiperone and piflutixol

spiperone has been researched along with piflutixol in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199017 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
O'Boyle, KM; Waddington, JL4
Hong, M; Jenner, P; Kilpatrick, GJ; Marsden, CD1
Henry, JM; Joseph, JA; Kochman, K; Roth, GS1
Boyce, S; Davis, A; Fleminger, S; Jenner, P; Kelly, E; Marsden, CD1
Jenner, P; Marsden, CD; Rupniak, NM1
Jenner, P; Kilpatrick, GJ; Marsden, CD1
Fleminger, S; Hall, MD; Jenner, P; Kilpatrick, G; Mann, S; Marsden, CD; Rupniak, NM1
Christensen, AV; Hyttel, J1
Fleminger, S; Hall, MD; Jenner, P; Marsden, CD; Rupniak, NM1
Cross, AJ; Johnson, JA; Mashal, RD; Owen, F1
Cross, A; Rossor, M1
Hyttel, J; Klimek, V; Nielsen, M1
Bohmaker, K; Friedhoff, AJ; Meller, E1
Fleminger, S; Jenner, P; Marsden, CD; Murugaiah, K; Theodorou, A1

Other Studies

17 other study(ies) available for spiperone and piflutixol

ArticleYear
Structural determinants of selective affinity for brain D-1 dopamine receptors within a series of 1-phenyl-1H-3-benzazepine analogues of SK&F 38393 and SCH 23390.
    European journal of pharmacology, 1985, Sep-24, Volume: 115, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Brain; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Thioxanthenes

1985
Effects of continuous administration for 12 months of amine-depleting drugs and chlorpromazine on striatal dopamine function in the rat.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: Animals; Apomorphine; Body Weight; Chlorpromazine; Corpus Striatum; Dopamine; Homovanillic Acid; Indoles; Kinetics; Male; Motor Activity; Piperazines; Rats; Rats, Inbred Strains; Reserpine; Spiperone; Stereotyped Behavior; Thioxanthenes

1987
Effect of aging on striatal dopamine receptor subtype recovery following N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline blockade and relation to motor function in Wistar rats.
    Brain research, 1987, Aug-25, Volume: 418, Issue:2

    Topics: Aging; Animals; Corpus Striatum; Male; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Thioxanthenes

1987
SCH 23390 may alter dopamine-mediated motor behaviour via striatal D-1 receptors.
    Biochemical pharmacology, 1985, May-15, Volume: 34, Issue:10

    Topics: 3,4-Dihydroxyphenylacetic Acid; Acetylcholine; Animals; Apomorphine; Benzazepines; Corpus Striatum; Cyclic AMP; Dopamine; Female; Humans; In Vitro Techniques; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes

1985
Differential alteration of striatal D-1 and D-2 receptors induced by the long-term administration of haloperidol, sulpiride or clozapine to rats.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Dose-Response Relationship, Drug; Haloperidol; Humans; Kinetics; Long-Term Care; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sulpiride; Thioxanthenes

1985
Specific [3H]piflutixol binding to CHAPS-solubilised rat striatal preparations involves dopamine D-2 but not D-1 binding sites.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Cholic Acids; Chromatography, Gel; Corpus Striatum; Flupenthixol; Isomerism; Kinetics; Rats; Receptors, Dopamine; Solubility; Spiperone; Sulpiride; Thioxanthenes

1986
Chronic treatment with clozapine, unlike haloperidol, does not induce changes in striatal D-2 receptor function in the rat.
    Biochemical pharmacology, 1985, Aug-01, Volume: 34, Issue:15

    Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Male; Mastication; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes; Tritium

1985
Biochemical and pharmacological differentiation of neuroleptic effect on dopamine D-1 and D-2 receptors.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Flupenthixol; Haloperidol; Rats; Receptors, Dopamine; Spiperone; Thioxanthenes

1983
Changes in apomorphine-induced stereotypy as a result of subacute neuroleptic treatment correlates with increased D-2 receptors, but not with increases in D-1 receptors.
    Biochemical pharmacology, 1983, Oct-01, Volume: 32, Issue:19

    Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Drug Synergism; Flupenthixol; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sulpiride; Thioxanthenes

1983
Preferential inhibition of ligand binding to calf striatal dopamine D1 receptors by SCH 23390.
    Neuropharmacology, 1983, Volume: 22, Issue:11

    Topics: Animals; Benzazepines; Binding, Competitive; Cattle; Corpus Striatum; In Vitro Techniques; Neurotransmitter Agents; Receptors, Dopamine; Receptors, Dopamine D1; Spiperone; Thioxanthenes

1983
Selective and stereospecific interactions of R-SK & F 38393 with [3H]piflutixol but not [3H]spiperone binding to striatal D1 and D2 dopamine receptors: comparisons with SCH 23390.
    European journal of pharmacology, 1984, Mar-02, Volume: 98, Issue:3-4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Binding, Competitive; Butyrophenones; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism; Thioxanthenes

1984
Loss of rat striatal dopamine receptors with ageing is selective for D-2 but not D-1 sites: association with increased non-specific binding of the D-1 ligand [3H]piflutixol.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: Adenylyl Cyclases; Aging; Animals; Antipsychotic Agents; Corpus Striatum; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Thioxanthenes

1984
Dopamine D-1 and D-2 receptors in Huntington's disease.
    European journal of pharmacology, 1983, Mar-25, Volume: 88, Issue:2-3

    Topics: Aged; Brain; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Kinetics; Male; Middle Aged; Putamen; Receptors, Dopamine; Spiperone; Substantia Nigra; Thioxanthenes

1983
Distinct target size of dopamine D-1 and D-2 receptors in rat striatum.
    Life sciences, 1984, Jul-16, Volume: 35, Issue:3

    Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Electrons; Male; Molecular Weight; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Thioxanthenes

1984
Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Thioxanthenes

1984
Differential effects of chronic clorgyline and amfonelic acid on desensitization of striatal dopamine receptors.
    Life sciences, 1984, Oct-29, Volume: 35, Issue:18

    Topics: Animals; Apomorphine; Behavior, Animal; Cerebral Cortex; Clorgyline; Corpus Striatum; Dihydroalprenolol; Haloperidol; Male; Monoamine Oxidase Inhibitors; Nalidixic Acid; Naphthyridines; Propylamines; Rats; Receptors, Dopamine; Spiperone; Thioxanthenes

1984
Persistent increase in striatal dopamine stimulated adenylate cyclase activity persists for more than 6 months but disappears after 1 year following withdrawal from 18 months cis-flupenthixol intake.
    Biochemical pharmacology, 1983, Sep-01, Volume: 32, Issue:17

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Binding Sites; Corpus Striatum; Dopamine; Flupenthixol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes; Time Factors

1983