Page last updated: 2024-08-16

spiperone and phenoxybenzamine

spiperone has been researched along with phenoxybenzamine in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199014 (82.35)18.7374
1990's2 (11.76)18.2507
2000's0 (0.00)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Brouillette, WJ; Brown, GB; Zha, C1
Clark, D; Willner, P1
Giachetti, A; Hefco, E; Jameson, HE; Krulich, L; Marchlewska-Koj, A1
Kordecka, A; Maj, J; Mogilnicka, E1
Barrett, VJ; Leff, P; Martin, GR; Richardson, PJ1
Creese, I; Hamblin, MW1
Crews, FT; Scott, JA; Shorstein, NH1
Hancock, AA; Marsh, CL1
Hall, MD; Jenner, P; Marsden, CD1
Bockaert, J; Marchais, D1
Allen, LE; Ashworth, EM; Becker, JA; Hyslop, DK; Riblet, LA; Taylor, DP1
Clincke, G; Fransen, J; Wauquier, A1
Titeler, M1
Creese, I; Hamblin, M1
Docherty, JR; Kearns, S; O'Rourke, M1
Amobi, N; Coker, C; Guillebaud, J; Mulvin, D; Smith, IC1

Other Studies

17 other study(ies) available for spiperone and phenoxybenzamine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
A reappraisal of the interaction between tricyclic antidepressants and reserpine-like drugs.
    Psychopharmacology, 1978, Jun-15, Volume: 58, Issue:1

    Topics: Animals; Antidepressive Agents, Tricyclic; Conditioning, Operant; Desipramine; Drug Interactions; Male; Motor Activity; Phenoxybenzamine; Phentolamine; Pimozide; Rats; Reserpine; Spiperone; Tetrabenazine; Time Factors

1978
On the role of the central noradrenergic and dopaminergic systems in the regulation of TSH secretion in the rat.
    Endocrinology, 1977, Volume: 100, Issue:2

    Topics: Animals; Apomorphine; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Clonidine; Ditiocarb; Dopamine; Kinetics; Male; Methyltyrosines; Norepinephrine; Phenoxybenzamine; Phentolamine; Pituitary Gland; Propranolol; Rats; Spiperone; Stress, Physiological; Thyrotropin; Thyrotropin-Releasing Hormone

1977
Chronic treatment with antidepressant drugs: potentiation of apomorphine-induced aggressive behaviour in rats.
    Neuroscience letters, 1979, Volume: 13, Issue:3

    Topics: Aggression; Animals; Antidepressive Agents; Apomorphine; Behavior; Drug Interactions; Humans; Male; Metergoline; Phenoxybenzamine; Phentolamine; Rats; Spiperone; Stereotyped Behavior; Time Factors

1979
Pharmacological analysis of the interaction between Bay K 8644 and 5-HT in rabbit aorta.
    British journal of pharmacology, 1986, Volume: 87, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Drug Synergism; In Vitro Techniques; Muscle, Smooth, Vascular; Phenoxybenzamine; Rabbits; Serotonin; Serotonin Antagonists; Spiperone

1986
Phenoxybenzamine treatment differentiates dopaminergic 3H-ligand binding sites in bovine caudate membranes.
    Molecular pharmacology, 1982, Volume: 21, Issue:1

    Topics: Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Cattle; Caudate Nucleus; In Vitro Techniques; Kinetics; Membranes; Phenoxybenzamine; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone

1982
Rapid down-regulation of serotonin2 receptor binding during combined administration of tricyclic antidepressant drugs and alpha 2 antagonists.
    Neuropharmacology, 1983, Volume: 22, Issue:10

    Topics: Adrenergic alpha-Antagonists; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cerebral Cortex; Desipramine; Kinetics; Male; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1983
Distinctions between ligand-binding sites for [3H]dopamine and D2 dopaminergic receptors characterized with [3H]spiroperidol.
    Molecular pharmacology, 1984, Volume: 26, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Butyrophenones; Cell Membrane; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Kinetics; Male; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1984
Turnover of specific [3H]spiperone and [3H]N,n-propylnorapomorphine binding sites in rat striatum following phenoxybenzamine administration.
    Biochemical pharmacology, 1983, Oct-01, Volume: 32, Issue:19

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Butyrophenones; Corpus Striatum; Female; Kinetics; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Is there a connection between high affinity 3H-spiperone binding sites and DA-sensitive adenylate cyclase in corpus striatum?
    Biochemical pharmacology, 1980, May-15, Volume: 29, Issue:10

    Topics: Adenylyl Cyclases; Animals; Binding Sites; Butyrophenones; Corpus Striatum; Dopamine; Guanosine Triphosphate; Haloperidol; In Vitro Techniques; Male; Phenethylamines; Phenoxybenzamine; Rats; Spiperone

1980
Treatment with trazodone plus phenoxybenzamine accelerates development of decreased type 2 serotonin binding in rat cortex.
    Neuropharmacology, 1981, Volume: 20, Issue:5

    Topics: Animals; Cerebral Cortex; Kinetics; Male; Phenoxybenzamine; Piperazines; Rats; Receptors, Serotonin; Spiperone; Trazodone

1981
Brain reinforcement mechanisms: alpha-adrenergic and dopaminergic agonists and antagonists.
    Progress in clinical and biological research, 1981, Volume: 71

    Topics: Animals; Apomorphine; Brain; Clonidine; Electric Stimulation; Hypothalamus; Locus Coeruleus; Neurons; Phenoxybenzamine; Rats; Receptors, Adrenergic; Receptors, Dopamine; Reinforcement, Psychology; Saimiri; Self Stimulation; Spiperone; Substantia Nigra

1981
Irreversible blockade of [3H]spiperone- but not [3H]dopamine-labeled dopamine receptors with phenoxybenzamine.
    Biochemical pharmacology, 1981, Nov-15, Volume: 30, Issue:22

    Topics: Animals; Binding Sites; Binding, Competitive; Butyrophenones; Cattle; Caudate Nucleus; Dopamine; Phenoxybenzamine; Receptors, Dopamine; Spiperone; Tritium

1981
Phenoxybenzamine discriminates multiple dopamine receptors.
    European journal of pharmacology, 1980, Jul-11, Volume: 65, Issue:1

    Topics: Animals; Apomorphine; Binding Sites; Cattle; Dopamine; In Vitro Techniques; Ligands; Phenoxybenzamine; Receptors, Dopamine; Spiperone; Tritium

1980
Investigation of the actions of chloroethylclonidine in rat aorta.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine

1995
Functional characterization of alpha1-adrenoceptor subtypes in longitudinal and circular muscle of human vas deferens.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Alkylating Agents; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Piperazines; Prazosin; Receptors, Adrenergic; Spiperone; Vas Deferens

1999