Page last updated: 2024-08-16

spiperone and nomifensine

spiperone has been researched along with nomifensine in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19907 (58.33)18.7374
1990's3 (25.00)18.2507
2000's1 (8.33)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Långström, B1
Allin, R; Reyneke, L; Russell, VA; Taljaard, JJ1
Leenders, KL1
Kilbourn, MR1
O'Boyle, KM; Waddington, JL1
Brenner, M; Dandridge, PA; Davis, LD; Foley, JJ; Gaitanopoulos, D; Kaiser, C; Sarau, HM; Webb, RL1
Lee, T; Tang, SW1
Cantuti-Castelvetri, I; Joseph, JA1
Bridges, S; Miller, C; Thompson, TL1

Reviews

2 review(s) available for spiperone and nomifensine

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993
Design of molecules labeled with beta+ emitters for use in multitracer investigations using positron emission tomography.
    Acta radiologica. Supplementum, 1990, Volume: 374

    Topics: Beta Particles; Humans; Isotope Labeling; Levodopa; Methionine; Neurotransmitter Agents; Nomifensine; Raclopride; Salicylamides; Spiperone; Tomography, Emission-Computed

1990

Other Studies

10 other study(ies) available for spiperone and nomifensine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Lack of effect of chronic desipramine treatment on dopaminergic activity in the nucleus accumbens of the rat.
    Neurochemical research, 1989, Volume: 14, Issue:7

    Topics: Acetylcholine; Animals; Benzazepines; Desipramine; Dopamine; Dopamine Agents; Dopamine Antagonists; Electric Stimulation; Ergolines; Male; Nomifensine; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Septal Nuclei; Spiperone

1989
Parkinson's disease and PET tracer studies.
    Journal of neural transmission. Supplementum, 1988, Volume: 27

    Topics: Animals; Carbon Radioisotopes; Cerebrovascular Circulation; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Energy Metabolism; Fluorine Radioisotopes; Humans; Ligands; Nomifensine; Parkinson Disease; Receptors, Dopamine; Selegiline; Spiperone; Tomography, Emission-Computed

1988
In vivo binding of [18F]GBR 13119 to the brain dopamine uptake system.
    Life sciences, 1988, Volume: 42, Issue:14

    Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Dopamine; Flupenthixol; Kinetics; Mazindol; Nomifensine; Piperazines; Rats; Rats, Inbred Strains; Spiperone

1988
New substituted 1-phenyl-3-benzazepine analogues of SK&F 38393 and N-methyl-thienopyridine analogues of dihydroxynomifensine with selective affinity for the D-1 dopamine receptor in human post-mortem brain.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Binding, Competitive; Brain Chemistry; Humans; In Vitro Techniques; Kinetics; Ligands; Nomifensine; Putamen; Pyridines; Receptors, Dopamine; Spiperone; Thiophenes

1987
Synthesis, resolution, absolute stereochemistry, and enantioselectivity of 3',4'-dihydroxynomifensine.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:1

    Topics: Adenylyl Cyclases; Animals; Biological Assay; Caudate Nucleus; Cerebral Cortex; Circular Dichroism; Clonidine; Imidazoline Receptors; Indicators and Reagents; Isoquinolines; Kinetics; Models, Molecular; Molecular Conformation; Nomifensine; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-2; Receptors, Dopamine; Spiperone; Stereoisomerism; Structure-Activity Relationship

1984
Reduced presynaptic dopamine receptor density after chronic antidepressant treatment in rats.
    Psychiatry research, 1982, Volume: 7, Issue:1

    Topics: Animals; Corpus Striatum; Desipramine; Dopamine; Isoquinolines; Male; Nomifensine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Synapses

1982
Differential effect of dopamine catabolism and uptake inhibition on dopamine-induced calcium dysregulation and viability loss.
    Free radical biology & medicine, 1999, Volume: 27, Issue:11-12

    Topics: Animals; Calcium; Caspase 3; Caspases; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Fluorescent Dyes; Free Radicals; Homeostasis; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nomifensine; Pargyline; PC12 Cells; Rats; Reactive Oxygen Species; Receptors, Dopamine D2; Spiperone

1999
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.
    Neuroscience letters, 2001, Oct-26, Volume: 312, Issue:3

    Topics: Animals; Antipsychotic Agents; Carbazoles; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Ligands; Neurons; Nomifensine; Nucleus Accumbens; Phenazocine; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, sigma; Spiperone; Sulpiride; Synaptosomes; Tritium

2001