Page last updated: 2024-08-16

spiperone and n-n-propylnorapomorphine

spiperone has been researched along with n-n-propylnorapomorphine in 81 studies

Research

Studies (81)

TimeframeStudies, this research(%)All Research%
pre-199061 (75.31)18.7374
1990's17 (20.99)18.2507
2000's2 (2.47)29.6817
2010's1 (1.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Seeman, P; Titeler, M1
De Boer, T; Florijn, WJ; Tonnaer, JA; Versteeg, DH1
Inoue, O; Itoh, T; Suhara, T; Tsukada, H; Yamasaki, T; Yonezawa, H1
Elazar, Z; Fuchs, S1
De Boer, T; Florijn, WJ; Tonnaer, JA; Van Nispen, JW; Versteeg, DH1
Grol, CJ; Hacksell, U; Johansson, AM; Nordvall, G1
Bouvier, C; Collu, R; Lagacé, G; Potier, M1
Carlsson, A; Fredriksson, K; Grol, CJ; Hacksell, U; Johansson, AM; Sundell, S; Svensson, K1
Heyer, EJ1
Fuchs, S; Kanety, H1
Elazar, Z; Fuchs, S; Siegel, G1
George, SR; Seeman, P; Watanabe, M2
Allikmets, LKh; Maĭmets, MO; Nurk, AM; Vasar, EE1
Hall, H; Jerning, E; Sällemark, M1
Bajwa, SB; Johnson, RL; Mishra, RK; Srivastava, LK1
Allikmets, L; Maimets, M; Nurk, A; Soosaar, A; Vasar, E1
Grol, CJ; Hacksell, U; Johansson, AM; Karlén, A; Kenne, L; Sundell, S1
Andersen, PH; Nielsen, EB1
Battaglia, G; Creese, I; Norman, AB1
Lin, C; McGonigle, P; Molinoff, PB1
Beauregard, G; Bouvier, C; Collu, R; Lafond, J; Lagacé, G; Potier, M1
Karlsson-Boethius, G; Köhler, C1
Martin, JR; Takemori, AE1
Wreggett, KA1
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Schweitzer, JW1
Grigoriadis, D; Seeman, P1
Kohjimoto, Y; Kuwaki, T; Nomura, Y; Ono, T; Satoh, H; Shibayama, F; Shirakawa, K1
Korf, J; Sebens, JB; Van der Werf, JF1
Cullen, M; Kazmi, SM; Mishra, RK; Rajakumar, G; Ramwani, J; Ross, GM; Srivastava, LK1
Brann, MR; Young, WS1
Ozaki, L; Stern, N; Tuck, ML1
Gredal, O; Nielsen, M1
Blengio, M; Bosco, MC; Eva, C; Ferretti, C; Ghi, P; Portaleone, P1
Flentge, F; Korf, J; Sebens, JB; van der Werf, JF1
Fleminger, S; Hall, MD; Jenner, P; Kilpatrick, G; Mann, S; Marsden, CD; Rupniak, NM2
Costall, B; Lim, SK; Naylor, RJ1
Battaglia, G; Titeler, M1
Fleminger, S; Hall, MD; Jenner, P; Kerwin, R; Marsden, CD; Murugaiah, K; Rupniak, NM1
Fuxe, K; Köhler, C; Ogren, SO1
Agnati, LF; Celani, MF; Fuxe, K; Martire, M; Zini, I; Zoli, M1
Chivers, JK; Hall, MD; Jenner, P; Kelly, E; Marsden, CD1
Angeby, K; Florvall, L; Hall, H; Köhler, C; Lindbom, LO; Magnusson, O; Ogren, SO1
Hall, MD; Jenner, P; Marsden, CD2
Kuno, T; Tanaka, C1
MacKenzie, RG; Zigmond, MJ1
Agnati, LF; Celani, MF; Fuxe, K1
Randall, PK; Severson, JA1
Hall, MD; Jenner, P; Kelly, E; Marsden, CD1
Hall, MD; Jenner, P; Kilpatrick, G; Marsden, CD; Rupniak, NM1
Battaini, F; Govoni, S; Rius, RA; Spano, PF; Trabucchi, M1
Caron, MG; Kilpatrick, BF; Sibley, DR1
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M1
Fuller, RW; Hemrick-Luecke, SK; Snoddy, HD1
Riffee, WH; Smith, RV; Vaughn, DM; Wilcox, RE1
Creese, I; Sibley, DR2
Creese, I; Mahan, LC; Sibley, DR1
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K1
Creese, I; Segal, DS; Sibley, DR; Weinberger, S1
Caron, MG; De Lean, A; Kilpatrick, BF3
Mahler, HR; Near, JA1
Adams, L; Creese, I; Hyttel, J; Leff, S1
Senogles, SE1
Bhatia, M; Borrelli, E; Ceraline, J; Guiramand, J; Montmayeur, JP1
Bruhwyler, J; Damas, J; Delarge, J; Geczy, J; Liégeois, JF; Masereel, B; Rogister, F1
Grol, CJ; Hacksell, U; Johansson, AM; Karlén, A1
Di Paolo, T; Lévesque, D1
DeSouza, EB; Grigoriadis, DE; Levant, B1
Allard, S; Falardeau, P; Lapointe, S1
Andersson, K; Bjelke, B; Chen, Y; Gross, J; Herrera-Marschitz, M; Hillefors-Berglund, M; von Euler, G1
Geurts, M; Hermans, E; Maloteaux, JM1
Lin, H; Roberts, DJ; Strange, PG1
Cho, EY; Kim, JH; Kim, KM; Min, C; Park, JH1
Halldin, C; Hong, J; Innis, RB; Liow, JS; Pike, VW; Seneca, N; Sibley, DR; Skinbjerg, M; Weinshenker, D1
Dumbrille-Ross, A; Elmaleh, DR; Guan, JH; Neumeyer, JL; Niznik, HB; Padmanabhan, S; Seeman, P1

Other Studies

81 other study(ies) available for spiperone and n-n-propylnorapomorphine

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Antiparkinsonian drug doses and neuroleptic receptors.
    Experientia, 1978, Nov-15, Volume: 34, Issue:11

    Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Cattle; Caudate Nucleus; Haloperidol; In Vitro Techniques; Receptors, Dopamine; Spiperone; Tritium

1978
Characterization of the inhibitory effect of adrenocorticotropin/melanocyte-stimulating hormone-like peptides on the binding of dopamine receptor ligands to the dopamine D2 receptor in vitro.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Adrenocorticotropic Hormone; Age Factors; Animals; Apomorphine; Binding, Competitive; Dopamine D2 Receptor Antagonists; Guanylyl Imidodiphosphate; Ligands; Male; Melanocyte-Stimulating Hormones; Peptides; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Temperature; Time Factors

1992
Effect of lithium and anesthetics on in vivo binding of dopamine receptors.
    Acta radiologica. Supplementum, 1991, Volume: 376

    Topics: Animals; Apomorphine; Benzazepines; Ketamine; Lithium; Male; Mice; Mice, Inbred C3H; Pentobarbital; Rats; Receptors, Dopamine; Spiperone

1991
Vanadate inhibits agonist binding to D2 dopamine receptor.
    Journal of molecular neuroscience : MN, 1991, Volume: 3, Issue:1

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Corpus Striatum; Dopamine Agents; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Vanadates

1991
ACTH/MSH-like peptides inhibit the binding of dopaminergic ligands to the dopamine D2 receptor in vitro.
    European journal of pharmacology, 1991, May-25, Volume: 207, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Amino Acid Sequence; Animals; Apomorphine; Cosyntropin; Dopamine Agents; In Vitro Techniques; Kinetics; Ligands; Male; Melanocyte-Stimulating Hormones; Molecular Sequence Data; Peptide Fragments; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes

1991
5-Oxygenated N-alkyl- and N,N-Dialkyl-2-amino-1-methyltetralins. Effects of structure and stereochemistry on dopamine-D2-receptor affinity.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:7

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Computer Simulation; Corpus Striatum; Culture Techniques; Dopamine Agents; Oxygen; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium

1991
Structural differences between dopamine D2 receptors present in a rat pituitary adenoma and in transplantable rat pituitary tumors 7315a and MtTW15.
    Journal of neurochemistry, 1990, Volume: 54, Issue:3

    Topics: Adenoma; Animals; Apomorphine; Binding, Competitive; Carrier Proteins; Chemical Phenomena; Chemistry; Dopamine Agents; Ethylmaleimide; Neoplasm Transplantation; Pituitary Neoplasms; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone

1990
Synthesis and pharmacology of the enantiomers of cis-7-hydroxy-3-methyl-2-(dipropylamino)tetralin.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:10

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Binding, Competitive; Cattle; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Crystallography; Dihydroxyphenylalanine; Dopamine Antagonists; In Vitro Techniques; Isomerism; Male; Molecular Conformation; Molecular Structure; Motor Activity; Rats; Reserpine; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; X-Ray Diffraction

1990
Dopamine antagonists reduce spontaneous electrical activity in cultured mammalian neurons from ventral mesencephalon.
    Brain research, 1986, Sep-24, Volume: 382, Issue:2

    Topics: Action Potentials; Animals; Apomorphine; Butaclamol; Cells, Cultured; Dibenzocycloheptenes; Dopamine Antagonists; Fetus; Haloperidol; Membrane Potentials; Mesencephalon; Mice; Mice, Inbred ICR; Neurons; Receptors, Dopamine; Spinal Cord; Spiperone

1986
Immuno-photoaffinity labeling of the D2-dopamine receptor.
    Biochemical and biophysical research communications, 1988, Sep-15, Volume: 155, Issue:2

    Topics: Affinity Labels; Animals; Apomorphine; Azides; Butaclamol; Cattle; Corpus Striatum; Haloperidol; Immunologic Techniques; Kinetics; Molecular Weight; Photochemistry; Receptors, Dopamine; Spiperone

1988
Association of two pertussis toxin-sensitive G-proteins with the D2-dopamine receptor from bovine striatum.
    The EMBO journal, 1989, Volume: 8, Issue:8

    Topics: Adenosine Diphosphate; Animals; Apomorphine; Blotting, Western; Cattle; Chromatography, Affinity; Corpus Striatum; Dopamine Agents; GTP Phosphohydrolases; GTP-Binding Proteins; Guanine Nucleotides; Kinetics; Membranes; Pertussis Toxin; Receptors, Dopamine; Solubility; Spiperone; Virulence Factors, Bordetella

1989
Dopamine D2 receptors in the anterior pituitary: a single population without reciprocal antagonist/agonist states.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; Butyrophenones; Dopamine; Dopamine Antagonists; Guanylyl Imidodiphosphate; Norepinephrine; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Serotonin; Sodium Chloride; Spiperone; Swine; Tetrahydronaphthalenes

1985
[Stimulation by cerulein--an analog of the octapeptide cholecystokinin--of 3H-spiroperidol binding after the long-term administration of neuroleptics].
    Biulleten' eksperimental'noi biologii i meditsiny, 1985, Volume: 99, Issue:1

    Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Butyrophenones; Ceruletide; Drug Interactions; Male; Mice; Spiperone; Stimulation, Chemical; Time Factors; Tritium

1985
Effects of remoxipride and some related new substituted salicylamides on rat brain receptors.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:1

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Benzamides; Brain; Domperidone; Dopamine; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Remoxipride; Salicylamides; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium

1986
Interaction of L-prolyl-L-leucyl glycinamide with dopamine D2 receptor: evidence for modulation of agonist affinity states in bovine striatal membranes.
    Journal of neurochemistry, 1988, Volume: 50, Issue:3

    Topics: Animals; Apomorphine; Cattle; Corpus Striatum; Guanylyl Imidodiphosphate; MSH Release-Inhibiting Hormone; Osmolar Concentration; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1988
Regulation of anterior pituitary D2 dopamine receptors by magnesium and sodium ions.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Apomorphine; Dopamine; Guanine Nucleotides; Magnesium; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Sodium; Spiperone; Swine

1985
Comparison of motor depressant effects of caerulein and N-propylnorapomorphine in mice.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Animals; Apomorphine; Ceruletide; Depression, Chemical; Exploratory Behavior; Fenclonine; Haloperidol; Hydroxydopamines; Male; Mice; Motor Activity; Nerve Endings; Oxidopamine; Receptors, Dopamine; Receptors, Serotonin; Sincalide; Spiperone

1986
Dopaminergic 2-aminotetralins: affinities for dopamine D2-receptors, molecular structures, and conformational preferences.
    Molecular pharmacology, 1986, Volume: 30, Issue:3

    Topics: Apomorphine; Magnetic Resonance Spectroscopy; Molecular Conformation; Naphthalenes; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium; X-Ray Diffraction

1986
The benzazepine, SCH 23390, inhibits 3H-NPA binding in mouse brain in vivo.
    Acta pharmacologica et toxicologica, 1986, Volume: 59, Issue:4

    Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Male; Mice; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Spiperone

1986
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:5

    Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone

1987
Characterization of D-2 dopamine receptors in a tumor of the rat anterior pituitary gland.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Apomorphine; Colforsin; Dopamine; Female; Guanosine Triphosphate; Pituitary Gland, Anterior; Pituitary Neoplasms; Rats; Rats, Inbred BUF; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1987
Characterization of D2 dopamine receptors in dopamine-resistant prolactin-secreting rat pituitary tumors 7315a and MtTW15.
    Journal of neurochemistry, 1987, Volume: 49, Issue:5

    Topics: Affinity Labels; Animals; Apomorphine; Cell Membrane; Dopamine; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Female; Guanylyl Imidodiphosphate; Molecular Weight; Neoplasm Transplantation; Photochemistry; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred BUF; Rats, Inbred WF; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone

1987
In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain.
    Journal of neural transmission, 1988, Volume: 73, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Brain; Kinetics; Male; Organ Specificity; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Stereoisomerism

1988
Increased sensitivity to dopamine agonists following a single dose of morphine or levorphanol in mice.
    European journal of pharmacology, 1985, Dec-10, Volume: 119, Issue:1-2

    Topics: Animals; Apomorphine; Brain; Brain Stem; Cerebral Cortex; Chlorides; Corpus Striatum; Dextrorphan; Drug Synergism; Hippocampus; Levorphanol; Lithium; Lithium Chloride; Male; Mice; Morphine; Motor Activity; Naloxone; Narcotics; Receptors, Dopamine; Spiperone

1985
Alkylation of the bovine anterior pituitary D2-dopamine receptor: inconsistency with predictions of the ternary complex model.
    Biochemical and biophysical research communications, 1987, Sep-30, Volume: 147, Issue:3

    Topics: Alkylation; Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Computer Simulation; Dopamine Antagonists; Fluphenazine; GTP-Binding Proteins; In Vitro Techniques; Ligands; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Structure-Activity Relationship

1987
Chronic haloperidol does not alter agonist affinity for dopamine receptors in vitro.
    European journal of pharmacology, 1985, Mar-12, Volume: 109, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Haloperidol; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide.
    Journal of neurochemistry, 1985, Volume: 44, Issue:6

    Topics: Animals; Apomorphine; Brain; Guanine Nucleotides; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Tetrahydronaphthalenes; Tritium

1985
Effect of long-term dosing with tiapride on brain dopamine receptors and metabolism in rats. Comparative study with sulpiride and haloperidol.
    Japanese journal of pharmacology, 1987, Volume: 44, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Apomorphine; Benzamides; Brain Chemistry; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride; Tiapamil Hydrochloride

1987
Tracer and maximal specific binding of tritiated spiperone or N-n-propylnorapomorphine to quantify dopamine receptors in rat brain regions in vivo.
    Life sciences, 1986, Jul-14, Volume: 39, Issue:2

    Topics: Animals; Apomorphine; Brain; Brain Mapping; Butyrophenones; Rats; Receptors, Dopamine; Spiperone

1986
Characterization of high-affinity dopamine D2 receptors and modulation of affinity states by guanine nucleotides in cholate-solubilized bovine striatal preparations.
    Journal of neurochemistry, 1986, Volume: 47, Issue:5

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cholic Acid; Cholic Acids; Computers; Corpus Striatum; Domperidone; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Receptors, Dopamine; Solubility; Spiperone

1986
Dopamine receptors are located on rods in bovine retina.
    Neuroscience letters, 1986, Sep-12, Volume: 69, Issue:3

    Topics: Animals; Apomorphine; Autoradiography; Cattle; Photoreceptor Cells; Receptors, Dopamine; Retina; Spiperone

1986
Evidence for dopaminergic binding sites in the human adrenal cortex.
    Metabolism: clinical and experimental, 1986, Volume: 35, Issue:12

    Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors

1986
In situ molecular size of agonist dopamine D-2 binding sites in rat striatum.
    Journal of neurochemistry, 1987, Volume: 48, Issue:2

    Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Guanosine Triphosphate; Kinetics; Male; Molecular Weight; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium Chloride; Spiperone

1987
The effects of a long term dihydroergotoxine treatment on agonist and antagonist striatal dopamine binding sites are dose and age related.
    Pharmacological research communications, 1986, Volume: 18, Issue:10

    Topics: Aging; Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dihydroergotoxine; Dose-Response Relationship, Drug; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1986
Occupation of dopamine receptors by N-n-propylnorapomorphine or spiperone and acetylcholine levels in the rat striatum.
    Journal of neurochemistry, 1985, Volume: 44, Issue:1

    Topics: Acetylcholine; Animals; Apomorphine; Binding Sites; Butyrophenones; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Time Factors

1985
Chronic treatment with clozapine, unlike haloperidol, does not induce changes in striatal D-2 receptor function in the rat.
    Biochemical pharmacology, 1985, Aug-01, Volume: 34, Issue:15

    Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Male; Mastication; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes; Tritium

1985
Characterisation of the mechanisms by which purported dopamine agonists reduce spontaneous locomotor activity of mice.
    European journal of pharmacology, 1981, Jul-17, Volume: 73, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Bromocriptine; Catecholamines; Dopamine; Dose-Response Relationship, Drug; Imidazolines; Male; Mice; Motor Activity; Prazosin; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine

1981
[3H]N-propylapomorphine and [3H]spiperone binding in brain indicate two states of the D2-dopamine receptor.
    European journal of pharmacology, 1982, Jul-16, Volume: 81, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Butyrophenones; Catecholamines; Cattle; Caudate Nucleus; Cyclic AMP; Ergot Alkaloids; Guanosine Triphosphate; In Vitro Techniques; Kinetics; Receptors, Dopamine; Spiperone

1982
Long-term adaptive changes in striatal dopamine function in response to chronic neuroleptic intake in rats.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Glutamates; Glutamic Acid; Haloperidol; Rats; Receptors, Dopamine; Spiperone; Sulpiride

1983
Studies on the mechanism of action of substituted benzamide drugs.
    Acta psychiatrica Scandinavica. Supplementum, 1984, Volume: 311

    Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Brain; Catalepsy; Corpus Striatum; Humans; Hyperkinesis; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra; Sulpiride; Tritium

1984
l-Glutamate reduces the affinity of [3H]N-propylnorapomorphine binding sites in striatal membranes.
    European journal of pharmacology, 1984, Apr-13, Volume: 100, Issue:1

    Topics: Animals; Antiparkinson Agents; Apomorphine; Aspartic Acid; Binding Sites; Cell Membrane; Corpus Striatum; Glutamates; Glutamic Acid; Male; N-Methylaspartate; Neuromuscular Depolarizing Agents; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Spiperone

1984
Dopamine receptor binding sites in the rat superior colliculus.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:7

    Topics: Animals; Apomorphine; In Vitro Techniques; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Superior Colliculi

1984
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Binding, Competitive; Brain Chemistry; Catalepsy; Chlorpromazine; Dogs; Female; Haloperidol; Histocytochemistry; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Spiperone; Sulpiride; Thioridazine; Vomiting

1984
Differential labelling of dopamine receptors in rat brain in vivo: comparison of [3H]piribedil, [3H]S 3608 and [3H]N,n-propylnorapomorphine.
    European journal of pharmacology, 1983, Jan-28, Volume: 87, Issue:1

    Topics: Animals; Apomorphine; Brain; Butaclamol; Corpus Striatum; Female; Nucleus Accumbens; Piperazines; Piribedil; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Correspondency between different affinity states and target size of the bovine striatal D2 dopamine receptor.
    Biochemical and biophysical research communications, 1983, Nov-30, Volume: 117, Issue:1

    Topics: Acetylcholinesterase; Animals; Apomorphine; Butaclamol; Cattle; Cell Membrane; Corpus Striatum; Dopamine; Guanosine Triphosphate; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Sulpiride

1983
High- and low-affinity states of striatal D2 receptors are not affected by 6-hydroxydopamine or chronic haloperidol treatment.
    Journal of neurochemistry, 1984, Volume: 43, Issue:5

    Topics: Animals; Apomorphine; Butaclamol; Cinanserin; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1984
Cholecystokinin peptides in vitro modulate the characteristics of the striatal 3H-N-propylnorapomorphine sites.
    Acta physiologica Scandinavica, 1983, Volume: 118, Issue:1

    Topics: Animals; Apomorphine; Cell Membrane; Corpus Striatum; Gastrins; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide; Spiperone; Tetragastrin

1983
Localization of [3H]N-propylnorapomorphine binding in mouse striatum.
    Brain research, 1983, Nov-21, Volume: 279, Issue:1-2

    Topics: Afferent Pathways; Animals; Apomorphine; Corpus Striatum; Frontal Lobe; Hydroxydopamines; Kainic Acid; Kinetics; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Neurons; Oxidopamine; Receptors, Dopamine; Spiperone

1983
Differential anatomical location of [3H]-N,n-propylnorapomorphine and [3H]-spiperone binding sites in the striatum and substantia nigra of the rat.
    British journal of pharmacology, 1983, Volume: 79, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Female; Hydroxydopamines; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Substantia Nigra; Tritium

1983
Differential effects of continuous administration for 1 year of haloperidol or sulpiride on striatal dopamine function in the rat.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Corpus Striatum; Haloperidol; Humans; Kinetics; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1984
Differential alterations in striatal dopamine receptor sensitivity induced by repeated administration of clinically equivalent doses of haloperidol, sulpiride or clozapine in rats.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1984
Chronic dihydroergotoxine treatment affects the number of dopamine recognition sites in rat striatum.
    Pharmacological research communications, 1984, Volume: 16, Issue:6

    Topics: Animals; Antiparkinson Agents; Apomorphine; Butyrophenones; Corpus Striatum; Dihydroergotoxine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tritium

1984
Turnover of specific [3H]spiperone and [3H]N,n-propylnorapomorphine binding sites in rat striatum following phenoxybenzamine administration.
    Biochemical pharmacology, 1983, Oct-01, Volume: 32, Issue:19

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Butyrophenones; Corpus Striatum; Female; Kinetics; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Direct radioligand measurement of dopamine receptors in the anterior pituitary gland.
    Methods in enzymology, 1983, Volume: 103

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Cells, Cultured; Ligands; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Spiperone; Swine; Tritium

1983
Interaction of (+)- and (-)-3-PPP with the dopamine receptor in the anterior pituitary gland.
    Life sciences, 1984, Jan-16, Volume: 34, Issue:3

    Topics: Animals; Apomorphine; Binding Sites; Cell Membrane; Depression, Chemical; In Vitro Techniques; Male; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism

1984
Increase in serum corticosterone concentration and decrease in hypothalamic epinephrine concentration by N-propylnorapomorphine in rats.
    Biochemical pharmacology, 1984, Apr-15, Volume: 33, Issue:8

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corticosterone; Epinephrine; Homovanillic Acid; Hypothalamus; Male; Rats; Rats, Inbred Strains; Spiperone

1984
Dopamine receptor sensitivity after chronic dopamine agonists. Striatal 3H-spiroperidol binding in mice after chronic administration of high doses of apomorphine, N-n-propylnorapomorphine and dextroamphetamine.
    Psychopharmacology, 1982, Volume: 77, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Dextroamphetamine; Humans; Male; Mice; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1982
Regulation of ligand binding to pituitary D-2 dopaminergic receptors. Effects of divalent cations and functional group modification.
    The Journal of biological chemistry, 1983, Apr-25, Volume: 258, Issue:8

    Topics: Animals; Apomorphine; Cations, Divalent; Cattle; Dose-Response Relationship, Drug; Ethylmaleimide; Hydroxymercuribenzoates; Kinetics; Male; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone

1983
Dopamine receptor binding on intact cells. Absence of a high-affinity agonist-receptor binding state.
    Molecular pharmacology, 1983, Volume: 23, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Kinetics; Male; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone

1983
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
    Acta physiologica Scandinavica, 1983, Volume: 117, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Multiple daily amphetamine administration decreases both [3H]agonist and [3H]antagonist dopamine receptor binding.
    Experientia, 1982, Oct-15, Volume: 38, Issue:10

    Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Dextroamphetamine; Dopamine; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1982
Guanine nucleotides regulate both dopaminergic agonist and antagonist binding in porcine anterior pituitary.
    Endocrinology, 1982, Volume: 110, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine

1982
Dopamine receptor of the porcine anterior pituitary gland. Evidence for two affinity states discriminated by both agonists and antagonists.
    Molecular pharmacology, 1982, Volume: 22, Issue:2

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Dopamine; Dopamine Antagonists; Female; Guanine Nucleotides; In Vitro Techniques; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine

1982
Dopamine receptor of the porcine anterior pituitary gland. Effects of N-ethylmaleimide and heat on ligand binding mimic the effects of guanine nucleotides.
    Molecular pharmacology, 1982, Volume: 22, Issue:2

    Topics: Animals; Apomorphine; Ethylmaleimide; Female; Guanine Nucleotides; Hot Temperature; In Vitro Techniques; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Spiperone; Swine

1982
Dopamine receptors in subcellular fractions from bovine caudate: enrichment of [3H]spiperone binding in a postsynaptic membrane fraction.
    Journal of neurochemistry, 1981, Volume: 36, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Butyrophenones; Cattle; Caudate Nucleus; Dopamine; In Vitro Techniques; Kinetics; Receptors, Dopamine; Spiperone; Subcellular Fractions; Synaptic Membranes

1981
Kainate lesion dissociates striatal dopamine receptor radioligand binding sites.
    European journal of pharmacology, 1981, Mar-05, Volume: 70, Issue:1

    Topics: Animals; Apomorphine; Benzimidazoles; Corpus Striatum; Domperidone; Flupenthixol; In Vitro Techniques; Kainic Acid; Male; Piperidines; Pyrrolidines; Radioligand Assay; Rats; Receptors, Dopamine; Spiperone

1981
Dopamine receptor binding in bovine intermediate lobe pituitary membranes.
    Endocrinology, 1980, Volume: 107, Issue:5

    Topics: Animals; Apomorphine; Butyrophenones; Catecholamines; Cattle; Cell Membrane; Guanosine Triphosphate; Phenothiazines; Pituitary Gland; Receptors, Dopamine; Spiperone

1980
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
    Endocrinology, 1994, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1994
Alternative splicing of the dopamine D2 receptor directs specificity of coupling to G-proteins.
    The Journal of biological chemistry, 1995, Mar-31, Volume: 270, Issue:13

    Topics: Adenylyl Cyclase Inhibitors; Alternative Splicing; Amino Acid Sequence; Animals; Apomorphine; Base Sequence; Cell Line; Cloning, Molecular; Cyclic AMP; Dopamine; Dopamine Agonists; GTP-Binding Proteins; Humans; Isoproterenol; Kinetics; Mice; Molecular Sequence Data; Mutagenesis, Insertional; Receptors, Adrenergic, beta-2; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection

1995
Modulation of the clozapine structure increases its selectivity for the dopamine D4 receptor.
    European journal of pharmacology, 1995, Feb-06, Volume: 273, Issue:3

    Topics: Apomorphine; Binding, Competitive; Cells, Cultured; Clozapine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Spiperone; Structure-Activity Relationship

1995
Dopamine D2 receptor agonists: an analysis of indirect models.
    Drug design and discovery, 1994, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Dopamine Agents; In Vitro Techniques; Models, Chemical; Molecular Conformation; Neostriatum; Receptors, Dopamine D2; Spiperone

1994
Modulation by estradiol and progesterone of the GTP effect on striatal D-2 dopamine receptors.
    Biochemical pharmacology, 1993, Feb-09, Volume: 45, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Estradiol; Female; Guanosine Triphosphate; In Vitro Techniques; Male; Ovariectomy; Progesterone; Rats; Receptors, Dopamine D2; Spiperone

1993
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone

1993
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
    Biochemical and biophysical research communications, 1993, Jun-15, Volume: 193, Issue:2

    Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1993
Perinatal asphyxia induces long-term changes in dopamine D1, D2, and D3 receptor binding in the rat brain.
    Experimental neurology, 1997, Volume: 146, Issue:1

    Topics: Animals; Apomorphine; Asphyxia Neonatorum; Benzazepines; Brain; Cesarean Section; Dopamine Agonists; Female; Humans; Infant, Newborn; Iodine Radioisotopes; Organ Specificity; Pregnancy; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Sulpiride

1997
Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Catalepsy; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium; Up-Regulation

1999
Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptors.
    Biochemical pharmacology, 2004, May-01, Volume: 67, Issue:9

    Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium

2004
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors.
    Archives of pharmacal research, 2008, Volume: 31, Issue:4

    Topics: Amino Acid Motifs; Apomorphine; Arginine; Aspartic Acid; Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Mutation; Protein Conformation; Protein Structure, Tertiary; Protein Transport; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Spiperone; Sulpiride; Transfection

2008
Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:9

    Topics: Animals; Apomorphine; Binding, Competitive; Cerebellum; Dopamine Agonists; Dopamine beta-Hydroxylase; Female; Kinetics; Male; Mice; Mice, Knockout; Neostriatum; Positron-Emission Tomography; Radioligand Assay; Radiopharmaceuticals; Receptors, Dopamine D2; Spiperone

2010
Novel photoaffinity label for the dopamine D2 receptor: synthesis of 4-azido-5-iodo-2-methoxy-N-[1-(phenylmethyl)-4-piperidinyl] benzamide (iodoazidoclebopride, IAC) and the corresponding 125I-labeled analogue (125IAC).
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:4

    Topics: Affinity Labels; Animals; Azides; Benzamides; Iodine Radioisotopes; Photolysis; Rats; Receptors, Dopamine; Receptors, Dopamine D2

1985