spiperone has been researched along with n-n-propylnorapomorphine in 81 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 61 (75.31) | 18.7374 |
1990's | 17 (20.99) | 18.2507 |
2000's | 2 (2.47) | 29.6817 |
2010's | 1 (1.23) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH | 1 |
Seeman, P; Titeler, M | 1 |
De Boer, T; Florijn, WJ; Tonnaer, JA; Versteeg, DH | 1 |
Inoue, O; Itoh, T; Suhara, T; Tsukada, H; Yamasaki, T; Yonezawa, H | 1 |
Elazar, Z; Fuchs, S | 1 |
De Boer, T; Florijn, WJ; Tonnaer, JA; Van Nispen, JW; Versteeg, DH | 1 |
Grol, CJ; Hacksell, U; Johansson, AM; Nordvall, G | 1 |
Bouvier, C; Collu, R; Lagacé, G; Potier, M | 1 |
Carlsson, A; Fredriksson, K; Grol, CJ; Hacksell, U; Johansson, AM; Sundell, S; Svensson, K | 1 |
Heyer, EJ | 1 |
Fuchs, S; Kanety, H | 1 |
Elazar, Z; Fuchs, S; Siegel, G | 1 |
George, SR; Seeman, P; Watanabe, M | 2 |
Allikmets, LKh; Maĭmets, MO; Nurk, AM; Vasar, EE | 1 |
Hall, H; Jerning, E; Sällemark, M | 1 |
Bajwa, SB; Johnson, RL; Mishra, RK; Srivastava, LK | 1 |
Allikmets, L; Maimets, M; Nurk, A; Soosaar, A; Vasar, E | 1 |
Grol, CJ; Hacksell, U; Johansson, AM; Karlén, A; Kenne, L; Sundell, S | 1 |
Andersen, PH; Nielsen, EB | 1 |
Battaglia, G; Creese, I; Norman, AB | 1 |
Lin, C; McGonigle, P; Molinoff, PB | 1 |
Beauregard, G; Bouvier, C; Collu, R; Lafond, J; Lagacé, G; Potier, M | 1 |
Karlsson-Boethius, G; Köhler, C | 1 |
Martin, JR; Takemori, AE | 1 |
Wreggett, KA | 1 |
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Schweitzer, JW | 1 |
Grigoriadis, D; Seeman, P | 1 |
Kohjimoto, Y; Kuwaki, T; Nomura, Y; Ono, T; Satoh, H; Shibayama, F; Shirakawa, K | 1 |
Korf, J; Sebens, JB; Van der Werf, JF | 1 |
Cullen, M; Kazmi, SM; Mishra, RK; Rajakumar, G; Ramwani, J; Ross, GM; Srivastava, LK | 1 |
Brann, MR; Young, WS | 1 |
Ozaki, L; Stern, N; Tuck, ML | 1 |
Gredal, O; Nielsen, M | 1 |
Blengio, M; Bosco, MC; Eva, C; Ferretti, C; Ghi, P; Portaleone, P | 1 |
Flentge, F; Korf, J; Sebens, JB; van der Werf, JF | 1 |
Fleminger, S; Hall, MD; Jenner, P; Kilpatrick, G; Mann, S; Marsden, CD; Rupniak, NM | 2 |
Costall, B; Lim, SK; Naylor, RJ | 1 |
Battaglia, G; Titeler, M | 1 |
Fleminger, S; Hall, MD; Jenner, P; Kerwin, R; Marsden, CD; Murugaiah, K; Rupniak, NM | 1 |
Fuxe, K; Köhler, C; Ogren, SO | 1 |
Agnati, LF; Celani, MF; Fuxe, K; Martire, M; Zini, I; Zoli, M | 1 |
Chivers, JK; Hall, MD; Jenner, P; Kelly, E; Marsden, CD | 1 |
Angeby, K; Florvall, L; Hall, H; Köhler, C; Lindbom, LO; Magnusson, O; Ogren, SO | 1 |
Hall, MD; Jenner, P; Marsden, CD | 2 |
Kuno, T; Tanaka, C | 1 |
MacKenzie, RG; Zigmond, MJ | 1 |
Agnati, LF; Celani, MF; Fuxe, K | 1 |
Randall, PK; Severson, JA | 1 |
Hall, MD; Jenner, P; Kelly, E; Marsden, CD | 1 |
Hall, MD; Jenner, P; Kilpatrick, G; Marsden, CD; Rupniak, NM | 1 |
Battaini, F; Govoni, S; Rius, RA; Spano, PF; Trabucchi, M | 1 |
Caron, MG; Kilpatrick, BF; Sibley, DR | 1 |
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M | 1 |
Fuller, RW; Hemrick-Luecke, SK; Snoddy, HD | 1 |
Riffee, WH; Smith, RV; Vaughn, DM; Wilcox, RE | 1 |
Creese, I; Sibley, DR | 2 |
Creese, I; Mahan, LC; Sibley, DR | 1 |
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K | 1 |
Creese, I; Segal, DS; Sibley, DR; Weinberger, S | 1 |
Caron, MG; De Lean, A; Kilpatrick, BF | 3 |
Mahler, HR; Near, JA | 1 |
Adams, L; Creese, I; Hyttel, J; Leff, S | 1 |
Senogles, SE | 1 |
Bhatia, M; Borrelli, E; Ceraline, J; Guiramand, J; Montmayeur, JP | 1 |
Bruhwyler, J; Damas, J; Delarge, J; Geczy, J; Liégeois, JF; Masereel, B; Rogister, F | 1 |
Grol, CJ; Hacksell, U; Johansson, AM; Karlén, A | 1 |
Di Paolo, T; Lévesque, D | 1 |
DeSouza, EB; Grigoriadis, DE; Levant, B | 1 |
Allard, S; Falardeau, P; Lapointe, S | 1 |
Andersson, K; Bjelke, B; Chen, Y; Gross, J; Herrera-Marschitz, M; Hillefors-Berglund, M; von Euler, G | 1 |
Geurts, M; Hermans, E; Maloteaux, JM | 1 |
Lin, H; Roberts, DJ; Strange, PG | 1 |
Cho, EY; Kim, JH; Kim, KM; Min, C; Park, JH | 1 |
Halldin, C; Hong, J; Innis, RB; Liow, JS; Pike, VW; Seneca, N; Sibley, DR; Skinbjerg, M; Weinshenker, D | 1 |
Dumbrille-Ross, A; Elmaleh, DR; Guan, JH; Neumeyer, JL; Niznik, HB; Padmanabhan, S; Seeman, P | 1 |
81 other study(ies) available for spiperone and n-n-propylnorapomorphine
Article | Year |
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Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection | 1991 |
Antiparkinsonian drug doses and neuroleptic receptors.
Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Cattle; Caudate Nucleus; Haloperidol; In Vitro Techniques; Receptors, Dopamine; Spiperone; Tritium | 1978 |
Characterization of the inhibitory effect of adrenocorticotropin/melanocyte-stimulating hormone-like peptides on the binding of dopamine receptor ligands to the dopamine D2 receptor in vitro.
Topics: Adrenocorticotropic Hormone; Age Factors; Animals; Apomorphine; Binding, Competitive; Dopamine D2 Receptor Antagonists; Guanylyl Imidodiphosphate; Ligands; Male; Melanocyte-Stimulating Hormones; Peptides; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Temperature; Time Factors | 1992 |
Effect of lithium and anesthetics on in vivo binding of dopamine receptors.
Topics: Animals; Apomorphine; Benzazepines; Ketamine; Lithium; Male; Mice; Mice, Inbred C3H; Pentobarbital; Rats; Receptors, Dopamine; Spiperone | 1991 |
Vanadate inhibits agonist binding to D2 dopamine receptor.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Corpus Striatum; Dopamine Agents; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Vanadates | 1991 |
ACTH/MSH-like peptides inhibit the binding of dopaminergic ligands to the dopamine D2 receptor in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Amino Acid Sequence; Animals; Apomorphine; Cosyntropin; Dopamine Agents; In Vitro Techniques; Kinetics; Ligands; Male; Melanocyte-Stimulating Hormones; Molecular Sequence Data; Peptide Fragments; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes | 1991 |
5-Oxygenated N-alkyl- and N,N-Dialkyl-2-amino-1-methyltetralins. Effects of structure and stereochemistry on dopamine-D2-receptor affinity.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Computer Simulation; Corpus Striatum; Culture Techniques; Dopamine Agents; Oxygen; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium | 1991 |
Structural differences between dopamine D2 receptors present in a rat pituitary adenoma and in transplantable rat pituitary tumors 7315a and MtTW15.
Topics: Adenoma; Animals; Apomorphine; Binding, Competitive; Carrier Proteins; Chemical Phenomena; Chemistry; Dopamine Agents; Ethylmaleimide; Neoplasm Transplantation; Pituitary Neoplasms; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone | 1990 |
Synthesis and pharmacology of the enantiomers of cis-7-hydroxy-3-methyl-2-(dipropylamino)tetralin.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Binding, Competitive; Cattle; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Crystallography; Dihydroxyphenylalanine; Dopamine Antagonists; In Vitro Techniques; Isomerism; Male; Molecular Conformation; Molecular Structure; Motor Activity; Rats; Reserpine; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; X-Ray Diffraction | 1990 |
Dopamine antagonists reduce spontaneous electrical activity in cultured mammalian neurons from ventral mesencephalon.
Topics: Action Potentials; Animals; Apomorphine; Butaclamol; Cells, Cultured; Dibenzocycloheptenes; Dopamine Antagonists; Fetus; Haloperidol; Membrane Potentials; Mesencephalon; Mice; Mice, Inbred ICR; Neurons; Receptors, Dopamine; Spinal Cord; Spiperone | 1986 |
Immuno-photoaffinity labeling of the D2-dopamine receptor.
Topics: Affinity Labels; Animals; Apomorphine; Azides; Butaclamol; Cattle; Corpus Striatum; Haloperidol; Immunologic Techniques; Kinetics; Molecular Weight; Photochemistry; Receptors, Dopamine; Spiperone | 1988 |
Association of two pertussis toxin-sensitive G-proteins with the D2-dopamine receptor from bovine striatum.
Topics: Adenosine Diphosphate; Animals; Apomorphine; Blotting, Western; Cattle; Chromatography, Affinity; Corpus Striatum; Dopamine Agents; GTP Phosphohydrolases; GTP-Binding Proteins; Guanine Nucleotides; Kinetics; Membranes; Pertussis Toxin; Receptors, Dopamine; Solubility; Spiperone; Virulence Factors, Bordetella | 1989 |
Dopamine D2 receptors in the anterior pituitary: a single population without reciprocal antagonist/agonist states.
Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; Butyrophenones; Dopamine; Dopamine Antagonists; Guanylyl Imidodiphosphate; Norepinephrine; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Serotonin; Sodium Chloride; Spiperone; Swine; Tetrahydronaphthalenes | 1985 |
[Stimulation by cerulein--an analog of the octapeptide cholecystokinin--of 3H-spiroperidol binding after the long-term administration of neuroleptics].
Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Butyrophenones; Ceruletide; Drug Interactions; Male; Mice; Spiperone; Stimulation, Chemical; Time Factors; Tritium | 1985 |
Effects of remoxipride and some related new substituted salicylamides on rat brain receptors.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Benzamides; Brain; Domperidone; Dopamine; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Remoxipride; Salicylamides; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium | 1986 |
Interaction of L-prolyl-L-leucyl glycinamide with dopamine D2 receptor: evidence for modulation of agonist affinity states in bovine striatal membranes.
Topics: Animals; Apomorphine; Cattle; Corpus Striatum; Guanylyl Imidodiphosphate; MSH Release-Inhibiting Hormone; Osmolar Concentration; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1988 |
Regulation of anterior pituitary D2 dopamine receptors by magnesium and sodium ions.
Topics: Animals; Apomorphine; Dopamine; Guanine Nucleotides; Magnesium; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Sodium; Spiperone; Swine | 1985 |
Comparison of motor depressant effects of caerulein and N-propylnorapomorphine in mice.
Topics: 5,7-Dihydroxytryptamine; Animals; Apomorphine; Ceruletide; Depression, Chemical; Exploratory Behavior; Fenclonine; Haloperidol; Hydroxydopamines; Male; Mice; Motor Activity; Nerve Endings; Oxidopamine; Receptors, Dopamine; Receptors, Serotonin; Sincalide; Spiperone | 1986 |
Dopaminergic 2-aminotetralins: affinities for dopamine D2-receptors, molecular structures, and conformational preferences.
Topics: Apomorphine; Magnetic Resonance Spectroscopy; Molecular Conformation; Naphthalenes; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Tetrahydronaphthalenes; Tritium; X-Ray Diffraction | 1986 |
The benzazepine, SCH 23390, inhibits 3H-NPA binding in mouse brain in vivo.
Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Male; Mice; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Spiperone | 1986 |
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone | 1987 |
Characterization of D-2 dopamine receptors in a tumor of the rat anterior pituitary gland.
Topics: Adenylyl Cyclase Inhibitors; Animals; Apomorphine; Colforsin; Dopamine; Female; Guanosine Triphosphate; Pituitary Gland, Anterior; Pituitary Neoplasms; Rats; Rats, Inbred BUF; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1987 |
Characterization of D2 dopamine receptors in dopamine-resistant prolactin-secreting rat pituitary tumors 7315a and MtTW15.
Topics: Affinity Labels; Animals; Apomorphine; Cell Membrane; Dopamine; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Female; Guanylyl Imidodiphosphate; Molecular Weight; Neoplasm Transplantation; Photochemistry; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred BUF; Rats, Inbred WF; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone | 1987 |
In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain.
Topics: Animals; Apomorphine; Binding, Competitive; Brain; Kinetics; Male; Organ Specificity; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Stereoisomerism | 1988 |
Increased sensitivity to dopamine agonists following a single dose of morphine or levorphanol in mice.
Topics: Animals; Apomorphine; Brain; Brain Stem; Cerebral Cortex; Chlorides; Corpus Striatum; Dextrorphan; Drug Synergism; Hippocampus; Levorphanol; Lithium; Lithium Chloride; Male; Mice; Morphine; Motor Activity; Naloxone; Narcotics; Receptors, Dopamine; Spiperone | 1985 |
Alkylation of the bovine anterior pituitary D2-dopamine receptor: inconsistency with predictions of the ternary complex model.
Topics: Alkylation; Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Computer Simulation; Dopamine Antagonists; Fluphenazine; GTP-Binding Proteins; In Vitro Techniques; Ligands; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Structure-Activity Relationship | 1987 |
Chronic haloperidol does not alter agonist affinity for dopamine receptors in vitro.
Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Haloperidol; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide.
Topics: Animals; Apomorphine; Brain; Guanine Nucleotides; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Tetrahydronaphthalenes; Tritium | 1985 |
Effect of long-term dosing with tiapride on brain dopamine receptors and metabolism in rats. Comparative study with sulpiride and haloperidol.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Apomorphine; Benzamides; Brain Chemistry; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride; Tiapamil Hydrochloride | 1987 |
Tracer and maximal specific binding of tritiated spiperone or N-n-propylnorapomorphine to quantify dopamine receptors in rat brain regions in vivo.
Topics: Animals; Apomorphine; Brain; Brain Mapping; Butyrophenones; Rats; Receptors, Dopamine; Spiperone | 1986 |
Characterization of high-affinity dopamine D2 receptors and modulation of affinity states by guanine nucleotides in cholate-solubilized bovine striatal preparations.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cholic Acid; Cholic Acids; Computers; Corpus Striatum; Domperidone; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Receptors, Dopamine; Solubility; Spiperone | 1986 |
Dopamine receptors are located on rods in bovine retina.
Topics: Animals; Apomorphine; Autoradiography; Cattle; Photoreceptor Cells; Receptors, Dopamine; Retina; Spiperone | 1986 |
Evidence for dopaminergic binding sites in the human adrenal cortex.
Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors | 1986 |
In situ molecular size of agonist dopamine D-2 binding sites in rat striatum.
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Guanosine Triphosphate; Kinetics; Male; Molecular Weight; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium Chloride; Spiperone | 1987 |
The effects of a long term dihydroergotoxine treatment on agonist and antagonist striatal dopamine binding sites are dose and age related.
Topics: Aging; Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dihydroergotoxine; Dose-Response Relationship, Drug; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1986 |
Occupation of dopamine receptors by N-n-propylnorapomorphine or spiperone and acetylcholine levels in the rat striatum.
Topics: Acetylcholine; Animals; Apomorphine; Binding Sites; Butyrophenones; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Time Factors | 1985 |
Chronic treatment with clozapine, unlike haloperidol, does not induce changes in striatal D-2 receptor function in the rat.
Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Male; Mastication; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes; Tritium | 1985 |
Characterisation of the mechanisms by which purported dopamine agonists reduce spontaneous locomotor activity of mice.
Topics: Animals; Antipsychotic Agents; Apomorphine; Bromocriptine; Catecholamines; Dopamine; Dose-Response Relationship, Drug; Imidazolines; Male; Mice; Motor Activity; Prazosin; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine | 1981 |
[3H]N-propylapomorphine and [3H]spiperone binding in brain indicate two states of the D2-dopamine receptor.
Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Butyrophenones; Catecholamines; Cattle; Caudate Nucleus; Cyclic AMP; Ergot Alkaloids; Guanosine Triphosphate; In Vitro Techniques; Kinetics; Receptors, Dopamine; Spiperone | 1982 |
Long-term adaptive changes in striatal dopamine function in response to chronic neuroleptic intake in rats.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Glutamates; Glutamic Acid; Haloperidol; Rats; Receptors, Dopamine; Spiperone; Sulpiride | 1983 |
Studies on the mechanism of action of substituted benzamide drugs.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Brain; Catalepsy; Corpus Striatum; Humans; Hyperkinesis; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra; Sulpiride; Tritium | 1984 |
l-Glutamate reduces the affinity of [3H]N-propylnorapomorphine binding sites in striatal membranes.
Topics: Animals; Antiparkinson Agents; Apomorphine; Aspartic Acid; Binding Sites; Cell Membrane; Corpus Striatum; Glutamates; Glutamic Acid; Male; N-Methylaspartate; Neuromuscular Depolarizing Agents; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Spiperone | 1984 |
Dopamine receptor binding sites in the rat superior colliculus.
Topics: Animals; Apomorphine; In Vitro Techniques; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Superior Colliculi | 1984 |
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Binding, Competitive; Brain Chemistry; Catalepsy; Chlorpromazine; Dogs; Female; Haloperidol; Histocytochemistry; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Spiperone; Sulpiride; Thioridazine; Vomiting | 1984 |
Differential labelling of dopamine receptors in rat brain in vivo: comparison of [3H]piribedil, [3H]S 3608 and [3H]N,n-propylnorapomorphine.
Topics: Animals; Apomorphine; Brain; Butaclamol; Corpus Striatum; Female; Nucleus Accumbens; Piperazines; Piribedil; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1983 |
Correspondency between different affinity states and target size of the bovine striatal D2 dopamine receptor.
Topics: Acetylcholinesterase; Animals; Apomorphine; Butaclamol; Cattle; Cell Membrane; Corpus Striatum; Dopamine; Guanosine Triphosphate; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Sulpiride | 1983 |
High- and low-affinity states of striatal D2 receptors are not affected by 6-hydroxydopamine or chronic haloperidol treatment.
Topics: Animals; Apomorphine; Butaclamol; Cinanserin; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1984 |
Cholecystokinin peptides in vitro modulate the characteristics of the striatal 3H-N-propylnorapomorphine sites.
Topics: Animals; Apomorphine; Cell Membrane; Corpus Striatum; Gastrins; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide; Spiperone; Tetragastrin | 1983 |
Localization of [3H]N-propylnorapomorphine binding in mouse striatum.
Topics: Afferent Pathways; Animals; Apomorphine; Corpus Striatum; Frontal Lobe; Hydroxydopamines; Kainic Acid; Kinetics; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Neurons; Oxidopamine; Receptors, Dopamine; Spiperone | 1983 |
Differential anatomical location of [3H]-N,n-propylnorapomorphine and [3H]-spiperone binding sites in the striatum and substantia nigra of the rat.
Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Female; Hydroxydopamines; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Substantia Nigra; Tritium | 1983 |
Differential effects of continuous administration for 1 year of haloperidol or sulpiride on striatal dopamine function in the rat.
Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Corpus Striatum; Haloperidol; Humans; Kinetics; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1984 |
Differential alterations in striatal dopamine receptor sensitivity induced by repeated administration of clinically equivalent doses of haloperidol, sulpiride or clozapine in rats.
Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1984 |
Chronic dihydroergotoxine treatment affects the number of dopamine recognition sites in rat striatum.
Topics: Animals; Antiparkinson Agents; Apomorphine; Butyrophenones; Corpus Striatum; Dihydroergotoxine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tritium | 1984 |
Turnover of specific [3H]spiperone and [3H]N,n-propylnorapomorphine binding sites in rat striatum following phenoxybenzamine administration.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Butyrophenones; Corpus Striatum; Female; Kinetics; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1983 |
Direct radioligand measurement of dopamine receptors in the anterior pituitary gland.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Cells, Cultured; Ligands; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Spiperone; Swine; Tritium | 1983 |
Interaction of (+)- and (-)-3-PPP with the dopamine receptor in the anterior pituitary gland.
Topics: Animals; Apomorphine; Binding Sites; Cell Membrane; Depression, Chemical; In Vitro Techniques; Male; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism | 1984 |
Increase in serum corticosterone concentration and decrease in hypothalamic epinephrine concentration by N-propylnorapomorphine in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corticosterone; Epinephrine; Homovanillic Acid; Hypothalamus; Male; Rats; Rats, Inbred Strains; Spiperone | 1984 |
Dopamine receptor sensitivity after chronic dopamine agonists. Striatal 3H-spiroperidol binding in mice after chronic administration of high doses of apomorphine, N-n-propylnorapomorphine and dextroamphetamine.
Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Dextroamphetamine; Humans; Male; Mice; Receptors, Dopamine; Spiperone; Stereotyped Behavior | 1982 |
Regulation of ligand binding to pituitary D-2 dopaminergic receptors. Effects of divalent cations and functional group modification.
Topics: Animals; Apomorphine; Cations, Divalent; Cattle; Dose-Response Relationship, Drug; Ethylmaleimide; Hydroxymercuribenzoates; Kinetics; Male; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone | 1983 |
Dopamine receptor binding on intact cells. Absence of a high-affinity agonist-receptor binding state.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Kinetics; Male; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone | 1983 |
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1983 |
Multiple daily amphetamine administration decreases both [3H]agonist and [3H]antagonist dopamine receptor binding.
Topics: Animals; Apomorphine; Butyrophenones; Corpus Striatum; Dextroamphetamine; Dopamine; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior | 1982 |
Guanine nucleotides regulate both dopaminergic agonist and antagonist binding in porcine anterior pituitary.
Topics: Animals; Apomorphine; Binding, Competitive; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine | 1982 |
Dopamine receptor of the porcine anterior pituitary gland. Evidence for two affinity states discriminated by both agonists and antagonists.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Dopamine; Dopamine Antagonists; Female; Guanine Nucleotides; In Vitro Techniques; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine | 1982 |
Dopamine receptor of the porcine anterior pituitary gland. Effects of N-ethylmaleimide and heat on ligand binding mimic the effects of guanine nucleotides.
Topics: Animals; Apomorphine; Ethylmaleimide; Female; Guanine Nucleotides; Hot Temperature; In Vitro Techniques; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Spiperone; Swine | 1982 |
Dopamine receptors in subcellular fractions from bovine caudate: enrichment of [3H]spiperone binding in a postsynaptic membrane fraction.
Topics: Animals; Apomorphine; Binding, Competitive; Butyrophenones; Cattle; Caudate Nucleus; Dopamine; In Vitro Techniques; Kinetics; Receptors, Dopamine; Spiperone; Subcellular Fractions; Synaptic Membranes | 1981 |
Kainate lesion dissociates striatal dopamine receptor radioligand binding sites.
Topics: Animals; Apomorphine; Benzimidazoles; Corpus Striatum; Domperidone; Flupenthixol; In Vitro Techniques; Kainic Acid; Male; Piperidines; Pyrrolidines; Radioligand Assay; Rats; Receptors, Dopamine; Spiperone | 1981 |
Dopamine receptor binding in bovine intermediate lobe pituitary membranes.
Topics: Animals; Apomorphine; Butyrophenones; Catecholamines; Cattle; Cell Membrane; Guanosine Triphosphate; Phenothiazines; Pituitary Gland; Receptors, Dopamine; Spiperone | 1980 |
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1994 |
Alternative splicing of the dopamine D2 receptor directs specificity of coupling to G-proteins.
Topics: Adenylyl Cyclase Inhibitors; Alternative Splicing; Amino Acid Sequence; Animals; Apomorphine; Base Sequence; Cell Line; Cloning, Molecular; Cyclic AMP; Dopamine; Dopamine Agonists; GTP-Binding Proteins; Humans; Isoproterenol; Kinetics; Mice; Molecular Sequence Data; Mutagenesis, Insertional; Receptors, Adrenergic, beta-2; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Transfection | 1995 |
Modulation of the clozapine structure increases its selectivity for the dopamine D4 receptor.
Topics: Apomorphine; Binding, Competitive; Cells, Cultured; Clozapine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Spiperone; Structure-Activity Relationship | 1995 |
Dopamine D2 receptor agonists: an analysis of indirect models.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Dopamine Agents; In Vitro Techniques; Models, Chemical; Molecular Conformation; Neostriatum; Receptors, Dopamine D2; Spiperone | 1994 |
Modulation by estradiol and progesterone of the GTP effect on striatal D-2 dopamine receptors.
Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Estradiol; Female; Guanosine Triphosphate; In Vitro Techniques; Male; Ovariectomy; Progesterone; Rats; Receptors, Dopamine D2; Spiperone | 1993 |
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone | 1993 |
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide | 1993 |
Perinatal asphyxia induces long-term changes in dopamine D1, D2, and D3 receptor binding in the rat brain.
Topics: Animals; Apomorphine; Asphyxia Neonatorum; Benzazepines; Brain; Cesarean Section; Dopamine Agonists; Female; Humans; Infant, Newborn; Iodine Radioisotopes; Organ Specificity; Pregnancy; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Sulpiride | 1997 |
Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment.
Topics: Animals; Apomorphine; Binding, Competitive; Catalepsy; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium; Up-Regulation | 1999 |
Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptors.
Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium | 2004 |
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors.
Topics: Amino Acid Motifs; Apomorphine; Arginine; Aspartic Acid; Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Mutation; Protein Conformation; Protein Structure, Tertiary; Protein Transport; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Spiperone; Sulpiride; Transfection | 2008 |
Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding.
Topics: Animals; Apomorphine; Binding, Competitive; Cerebellum; Dopamine Agonists; Dopamine beta-Hydroxylase; Female; Kinetics; Male; Mice; Mice, Knockout; Neostriatum; Positron-Emission Tomography; Radioligand Assay; Radiopharmaceuticals; Receptors, Dopamine D2; Spiperone | 2010 |
Novel photoaffinity label for the dopamine D2 receptor: synthesis of 4-azido-5-iodo-2-methoxy-N-[1-(phenylmethyl)-4-piperidinyl] benzamide (iodoazidoclebopride, IAC) and the corresponding 125I-labeled analogue (125IAC).
Topics: Affinity Labels; Animals; Azides; Benzamides; Iodine Radioisotopes; Photolysis; Rats; Receptors, Dopamine; Receptors, Dopamine D2 | 1985 |