Page last updated: 2024-08-16

spiperone and mianserin

spiperone has been researched along with mianserin in 59 studies

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-199029 (49.15)18.7374
1990's21 (35.59)18.2507
2000's8 (13.56)29.6817
2010's1 (1.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Amlaiky, N; Boschert, U; Hen, R; Maroteaux, L; Plassat, JL; Saudou, F1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Glennon, RA2
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Andrews, PR; Craik, DJ; Martin, JL1
Amlaiky, N; Hen, R; Plassat, JL1
Arrang, JM; Diaz, J; Leurs, R; Ruat, M; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Dokhan, R; el Ahmad, Y; Laurent, E; Maillet, P; Ollivier, R; Talab, A; Teste, JF; Tran, G1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB1
Egan, CT; Herrick-Davis, K; Teitler, M1
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD1
Benhamú, B; Lavandera, JL; López-Rodríguez, ML; Morcillo, MJ; Porras, E; Ramos, JA1
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R1
Benhamú, B; Campillo, M; Lavandera, JL; López-Rodríguez, ML; Morcillo, MJ; Olivella, M; Pardo, L; Porras, E; Ramos, JA; Soto, LJ1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Esterle, TM; Sanders-Bush, E1
Aulakh, CS; Hill, JL; Murphy, DL1
Barker, EL; Burris, KD; Sanders-Bush, E1
Albrecht, S; Walter, RD1
Gallager, DW; Goldman-Rakic, PS; Lidow, MS; Rakic, P1
De Vivo, M; Maayani, S1
Laing, JC; Young, RJ1
Fermanian, J; Frances, H; Lienard, C1
Jenner, P; Marsden, CD; Stewart, BR1
Convents, A; De Keyser, J; Ebinger, G; Vauquelin, G; Walraevens, H1
Klimek, V; Maj, J1
Chojnacka-Wójcik, E; Jaros, T; Kłodzińska, A; Maj, J1
Conn, PJ; Hartig, PR; Hoffman, BJ; Sanders-Bush, E1
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN1
de Boer, TH; de Vos, CJ; Maura, G; Pinder, RM; Raiteri, M; Wieringa, J1
Penney, JB; Richfield, EK; Young, AB1
Blurton, PA; Wood, MD1
Chester, NA; Menking, D; Shih, TM; Valdes, JJ; Whalley, C1
Peroutka, SJ; Snyder, SH2
Fuller, RW; Snoddy, HD1
Barbaz, B; Bernard, P; Braunwalder, A; Kim, HS; Liebman, JM; Lovell, RA; Robson, RD; Stone, G; Wasley, JW; Welch, J1
Helmeste, DM; Tang, SW1
Mayer, RJ; Strange, PG; Withy, RM2
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS1
Goodwin, GM; Green, AR; Johnson, P1
Coscina, DV; Dumbrille-Ross, A; Tang, SW1
Hall, H; Ross, SB; Sällemark, M1
Köhler, C1
Kendall, DA; Nahorski, SR1
Boehme, RE; Ciaranello, RD1
Chan, B; Madras, BK1
Hartig, PR; Hoffman, BJ; Kaufman, MJ1
Ageel, AM; Alhaider, AA; Ginawi, OT1
Currie, PJ; Saxena, N; Tu, AY1
Huang, XF; Zavitsanou, K1
Clifton, PG; Dourish, CT; Kennett, GA; Lee, MD; Somerville, EM1

Reviews

2 review(s) available for spiperone and mianserin

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

57 other study(ies) available for spiperone and mianserin

ArticleYear
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Apr-01, Volume: 89, Issue:7

    Topics: 3T3 Cells; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cerebellum; Corpus Striatum; Gene Expression; Genes; GTP-Binding Proteins; Mice; Molecular Sequence Data; Nucleic Acid Hybridization; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Purkinje Cells; Receptors, Serotonin; RNA, Messenger; Serotonin

1992
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Sep-15, Volume: 90, Issue:18

    Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Northern; Brain; CHO Cells; Cricetinae; Cyclic AMP; DNA; Genomic Library; Kinetics; Lysergic Acid Diethylamide; Mianserin; Molecular Sequence Data; Multigene Family; Oligodeoxyribonucleotides; Organ Specificity; Rats; Receptors, Serotonin; Restriction Mapping; Serotonin; Serotonin Receptor Agonists; Transfection

1993
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
New benzocycloalkylpiperazines, potent and selective 5-HT1A receptor ligands.
    Journal of medicinal chemistry, 1997, Mar-14, Volume: 40, Issue:6

    Topics: Adenylyl Cyclases; Animals; Behavior, Animal; Binding, Competitive; Colforsin; Cyclic AMP; Electrophysiology; Enzyme Activation; Kinetics; Magnetic Resonance Spectroscopy; Molecular Conformation; Molecular Structure; Piperazines; Protein Binding; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship

1997
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine

1998
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Animals; Antipsychotic Agents; COS Cells; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship

1998
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
    Journal of medicinal chemistry, 1999, Aug-12, Volume: 42, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes

1999
First pharmacophoric hypothesis for 5-HT7 antagonism.
    Bioorganic & medicinal chemistry letters, 2000, May-15, Volume: 10, Issue:10

    Topics: Animals; Cell Membrane; Drug Design; Drug Evaluation, Preclinical; Hypothalamus; Models, Molecular; Rats; Receptors, Serotonin; Reproducibility of Results; Serotonin Antagonists; Structure-Activity Relationship

2000
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:2

    Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

2001
Optimization of the pharmacophore model for 5-HT7R antagonism. Design and synthesis of new naphtholactam and naphthosultam derivatives.
    Journal of medicinal chemistry, 2003, Dec-18, Volume: 46, Issue:26

    Topics: Animals; Binding, Competitive; Computer Simulation; Drug Design; Hypothalamus; In Vitro Techniques; Lactams; Ligands; Male; Models, Molecular; Molecular Conformation; Naphthalenes; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides; Thiazoles

2003
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Serotonin agonists increase transferrin levels via activation of 5-HT1C receptors in choroid plexus epithelium.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: Amino Acid Isomerases; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Choroid Plexus; Cyclosporins; Epithelium; Ergolines; Fibroblasts; Kinetics; Male; Mianserin; Peptidylprolyl Isomerase; Phosphatidylinositols; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA Probes; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Thymidine; Time Factors; Transferrin

1992
Effects of various serotonin receptor subtype-selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Corticosterone; Ergolines; Male; Metergoline; Mianserin; Neurosecretory Systems; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1992
Phosphoinositide hydrolysis linked 5-HT2 receptors in fibroblasts from choroid plexus.
    Brain research, 1991, Jun-28, Volume: 552, Issue:2

    Topics: Animals; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fibroblasts; Haloperidol; Hydrolysis; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Serotonin; Serotonin; Spiperone

1991
Hallucinogenic and neuroleptic drug interactions with potential neurotransmitter receptors in parasitic nematodes.
    Molecular and biochemical parasitology, 1991, Volume: 45, Issue:2

    Topics: Animals; Antipsychotic Agents; Ascaris; Binding, Competitive; Diethylamines; Haloperidol; Lysergic Acid Diethylamide; Mianserin; Onchocerca; Receptors, Neurotransmitter; Spiperone

1991
Distribution of dopaminergic receptors in the primate cerebral cortex: quantitative autoradiographic analysis using [3H]raclopride, [3H]spiperone and [3H]SCH23390.
    Neuroscience, 1991, Volume: 40, Issue:3

    Topics: Animals; Benzazepines; Brain Mapping; Cerebral Cortex; Ketanserin; Macaca mulatta; Mianserin; Raclopride; Receptors, Dopamine; Salicylamides; Species Specificity; Spiperone

1991
Stimulation and inhibition of adenylyl cyclase by distinct 5-hydroxytryptamine receptors.
    Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Membrane; Cerebral Cortex; Colforsin; Drug Interactions; Enzyme Activation; Fluphenazine; Guinea Pigs; Hippocampus; Mathematics; Mianserin; Pindolol; Piperazines; Rats; Receptors, Serotonin; Spiperone

1990
Biogenic amine binding sites in rabbit spermatozoa.
    Biochemistry international, 1990, Volume: 21, Issue:4

    Topics: Animals; Binding Sites; Biogenic Amines; Epinephrine; Haloperidol; In Vitro Techniques; Male; Mianserin; Rabbits; Sperm Head; Sperm Tail; Spermatozoa; Spiperone

1990
Improvement of the isolation-induced social behavioural deficit involves activation of the 5-HT1B receptors.
    Progress in neuro-psychopharmacology & biological psychiatry, 1990, Volume: 14, Issue:1

    Topics: Animals; Cyproheptadine; Escape Reaction; Indoles; Male; Mianserin; Mice; Mice, Inbred Strains; Penbutolol; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Social Behavior; Social Isolation; Spiperone; Tropisetron

1990
Induction of purposeless chewing behaviour in rats by 5-HT agonist drugs.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Male; Methiothepin; Methoxydimethyltryptamines; Mianserin; Parasympatholytics; Piperazines; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1989
[3H]SCH 23390 labels a novel 5-hydroxytryptamine binding site in human blood platelet membranes.
    European journal of pharmacology, 1989, Mar-29, Volume: 162, Issue:3

    Topics: Antipsychotic Agents; Benzazepines; Binding, Competitive; Blood Platelets; Cell Membrane; Cerebral Cortex; Humans; In Vitro Techniques; Mianserin; Radioligand Assay; Receptors, Serotonin; Spiperone

1989
Repeated administration of antidepressants enhances agonist affinity for mesolimbic D2-receptors.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:8

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Binding, Competitive; Ergolines; Imipramine; Limbic System; Male; Mianserin; Motor Activity; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spiperone

1989
Exploratory hypoactivity induced by m-trifluoromethylphenylpiperazine (TFMPP) and m-chlorophenylpiperazine (m-CPP).
    Journal of neural transmission. Parkinson's disease and dementia section, 1989, Volume: 1, Issue:3

    Topics: Animals; Ergolines; Exploratory Behavior; Male; Metergoline; Mianserin; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1989
A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:11

    Topics: Animals; Cerebral Cortex; Choroid Plexus; In Vitro Techniques; Ketanserin; Mianserin; Phosphatidylinositols; Piperidines; Rats; Receptors, Serotonin; Spiperone

1986
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain.
    Life sciences, 1985, Aug-19, Volume: 37, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution

1985
Neurochemical and autonomic pharmacological profiles of the 6-aza-analogue of mianserin, Org 3770 and its enantiomers.
    Neuropharmacology, 1988, Volume: 27, Issue:4

    Topics: Animals; Antidepressive Agents, Tricyclic; Autonomic Nervous System; Binding, Competitive; Cerebral Cortex; Corpus Striatum; In Vitro Techniques; Male; Mianserin; Mirtazapine; Norepinephrine; Prazosin; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Stereoisomerism; Synaptosomes; Yohimbine

1988
Properties of D2 dopamine receptor autoradiography: high percentage of high-affinity agonist sites and increased nucleotide sensitivity in tissue sections.
    Brain research, 1986, Sep-24, Volume: 383, Issue:1-2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1986
Identification of multiple binding sites for [3H]5-hydroxytryptamine in the rat CNS.
    Journal of neurochemistry, 1986, Volume: 46, Issue:5

    Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Calcium; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Hippocampus; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Tissue Distribution

1986
Regional sensitivity of neuroleptic receptors to sub-acute soman intoxication.
    Brain research bulletin, 1985, Volume: 14, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cerebral Cortex; Corpus Striatum; Haloperidol; Hippocampus; Kinetics; Male; Mianserin; Organophosphorus Compounds; Rats; Receptors, Dopamine; Soman; Spiperone

1985
[3H]Mianserin: differential labeling of serotonin and histamine receptors in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 216, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cerebral Cortex; Dibenzazepines; In Vitro Techniques; Kinetics; Male; Mianserin; Neurotransmitter Agents; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Serotonin; Spiperone; Triprolidine

1981
Elevation of serum corticosterone concentrations in rats by pergolide and other dopamine agonists.
    Endocrinology, 1981, Volume: 109, Issue:4

    Topics: Animals; Antiparkinson Agents; Corticosterone; Domperidone; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Metergoline; Mianserin; Pergolide; Rats; Rats, Inbred Strains; Spiperone

1981
CGS 7525A, a new, centrally active alpha 2 adrenoceptor antagonist.
    Life sciences, 1983, Jan-24, Volume: 32, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Benzodiazepines; Chemical Phenomena; Chemistry; Clonidine; Male; Mesencephalon; Mianserin; Norepinephrine; Prazosin; Quinones; Rats; Rats, Inbred Strains; Spiperone; Yohimbine

1983
Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors.
    Life sciences, 1983, Dec-19, Volume: 33, Issue:25

    Topics: Amoxapine; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Fenclonine; Frontal Lobe; Ketanserin; Loxapine; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1983
[3H] spiroperidol binding to brain neurotransmitter receptors.
    FEBS letters, 1980, Apr-07, Volume: 112, Issue:2

    Topics: Animals; Butaclamol; Butyrophenones; Cattle; Caudate Nucleus; Dopamine; Kinetics; Mianserin; Microsomes; Radioligand Assay; Receptors, Dopamine; Receptors, Serotonin; Spiperone

1980
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
    Brain research, 1984, Jun-11, Volume: 303, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone

1984
5-HT2 receptor characteristics in frontal cortex and 5-HT2 receptor-mediated head-twitch behaviour following antidepressant treatment to mice.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents; Behavior, Animal; Brain; Cerebral Cortex; Desipramine; Frontal Lobe; Kinetics; Male; Mianserin; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Radioligand Assay; Receptors, Serotonin; Spiperone; Tranylcypromine; Zimeldine

1984
[3H]Spiroperidol binding in bovine caudate nucleus [proceedings].
    Biochemical Society transactions, 1980, Volume: 8, Issue:2

    Topics: Animals; Binding, Competitive; Butyrophenones; Cattle; Caudate Nucleus; Kinetics; Mianserin; Receptors, Neurotransmitter; Spiperone

1980
Lack of effect of raphe lesions on serotonin S2 receptor changes induced by amitriptyline and desmethylimipramine.
    Psychiatry research, 1982, Volume: 7, Issue:2

    Topics: Amitriptyline; Animals; Brain Stem; Cerebral Cortex; Corpus Striatum; Desipramine; Dopamine; Hypothalamus; Male; Mesencephalon; Mianserin; Norepinephrine; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Synaptic Transmission

1982
Effect of destruction of central noradrenergic and serotonergic nerve terminals by systemic neurotoxins on the long-term effects of antidepressants on beta-adrenoceptors and 5-HT2 binding sites in the rat cerebral cortex.
    Journal of neural transmission, 1984, Volume: 59, Issue:1

    Topics: Alanine; Amines; Animals; Antidepressive Agents; Benzylamines; Binding Sites; Cerebral Cortex; Clenbuterol; Desipramine; Dihydroalprenolol; Male; Mianserin; p-Chloroamphetamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Spiperone; Zimeldine

1984
Autoradiographic mapping of spirodecanone binding-sites in the hippocampal region of the rat. Evidence for a localization on intrinsic neurons.
    Neuroscience letters, 1984, May-04, Volume: 46, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Mapping; Butyrophenones; Haloperidol; Hippocampus; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Serotonin; Spiperone; Tetrahydronaphthalenes

1984
Temperature-dependent 5-hydroxytryptamine (5-HT)-sensitive [3H]spiperone binding to rat cortical membranes: regulation by guanine nucleotide and antidepressant treatment.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:2

    Topics: Animals; Binding Sites; Butyrophenones; Cerebral Cortex; Dibenzazepines; Guanine Nucleotides; Indoles; Iprindole; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Temperature

1983
Genetic control of dopamine and serotonin receptors in brain regions of inbred mice.
    Brain research, 1983, Apr-25, Volume: 266, Issue:1

    Topics: Animals; Brain; Corpus Striatum; Domperidone; Kinetics; Mianserin; Mice; Mice, Inbred Strains; Pituitary Gland; Receptors, Dopamine; Receptors, Serotonin; Species Specificity; Spiperone

1983
[3H]Mianserin binding to solubilized membranes of frontal cortex.
    European journal of pharmacology, 1982, Sep-10, Volume: 83, Issue:1-2

    Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Dibenzazepines; Dogs; In Vitro Techniques; Kinetics; Membranes; Mianserin; Polyethylene Glycols; Spiperone; Time Factors

1982
Two distinct serotonin receptors: regional variations in receptor binding in mammalian brain.
    Brain research, 1981, Mar-16, Volume: 208, Issue:2

    Topics: Animals; Binding Sites; Brain; Brain Mapping; Cattle; Guinea Pigs; Lysergic Acid Diethylamide; Mianserin; Rats; Receptors, Serotonin; Serotonin; Spiperone

1981
Serotonin 5-HT2C receptor stimulates cyclic GMP formation in choroid plexus.
    Journal of neurochemistry, 1995, Volume: 64, Issue:1

    Topics: Animals; Cattle; Choroid Plexus; Cyclic GMP; Ketanserin; Mianserin; Phosphatidylinositols; Receptors, Serotonin; Spiperone; Swine

1995
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes

1993
5-HT(2A/2C) receptor antagonists in the paraventricular nucleus attenuate the action of DOI on NPY-stimulated eating.
    Neuroreport, 1999, Sep-29, Volume: 10, Issue:14

    Topics: Amphetamines; Animals; Appetite Stimulants; Eating; Male; Mianserin; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Ventromedial Hypothalamic Nucleus

1999
Decreased [(3)H]spiperone binding in the anterior cingulate cortex of schizophrenia patients: an autoradiographic study.
    Neuroscience, 2002, Volume: 109, Issue:4

    Topics: Adult; Aged; Antipsychotic Agents; Binding Sites; Binding, Competitive; Butaclamol; Down-Regulation; Gyrus Cinguli; Haloperidol; Humans; Mianserin; Middle Aged; Neurons; Neurotransmitter Agents; Radioligand Assay; Receptors, Neurotransmitter; Risperidone; Schizophrenia; Spiperone; Tritium

2002
Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice.
    Psychopharmacology, 2004, Volume: 176, Issue:1

    Topics: Animals; Binding Sites; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Evaluation, Preclinical; Eating; Ergolines; Fenfluramine; Genotype; Injections, Intraperitoneal; Injections, Subcutaneous; Isomerism; Mianserin; Mice; Mice, Knockout; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Satiation; Satiety Response; Serotonin 5-HT2 Receptor Agonists; Species Specificity; Spiperone; Spiro Compounds; Time Factors; Tritium; United Kingdom

2004