spiperone has been researched along with guanylyl imidodiphosphate in 44 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 32 (72.73) | 18.7374 |
1990's | 10 (22.73) | 18.2507 |
2000's | 2 (4.55) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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De Boer, T; Florijn, WJ; Tonnaer, JA; Versteeg, DH | 1 |
O'Boyle, KM; Waddington, JL | 1 |
Barton, AC; Monsma, FJ; Sibley, DR | 1 |
Johnson, RL; Mishra, RK; Srivastava, LK | 1 |
Badia, A; Casas, M; Ferré, S; Guix, T; Herrera-Marschitz, M; Jané, F; Parra, P; Sallés, J; Ungerstedt, U | 1 |
Agui, T; Munemura, M; Sibley, DR | 1 |
De Backer, JP; De Keyser, J; Ebinger, G; Vauquelin, G; Walraevens, H | 1 |
George, SR; Seeman, P; Watanabe, M | 2 |
Crooke, ST; Flaim, KE; Gessner, GW; Sarau, HM; Weinstock, J | 1 |
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P | 1 |
Hall, H; Sällemark, M | 1 |
Bajwa, SB; Johnson, RL; Mishra, RK; Srivastava, LK | 1 |
Battaglia, G; Creese, I; Norman, AB | 1 |
Dumbrille-Ross, A; Seeman, P | 1 |
Besselievre, R; Cossery, JM; el Mestikawy, S; Emerit, MB; Gozlan, H; Hamon, M; Marquet, A | 1 |
Beauregard, G; Bouvier, C; Collu, R; Lafond, J; Lagacé, G; Potier, M | 1 |
Agui, T; Amlaiky, N; Caron, MG; Kebabian, JW | 1 |
Bhatnagar, RK; Chatterjee, TK; Scott, CE; Vazquez, DM | 1 |
Bernier, MA; Di Paolo, T | 1 |
Cullen, M; Kazmi, SM; Mishra, RK; Rajakumar, G; Ramwani, J; Ross, GM; Srivastava, LK | 1 |
Penney, JB; Richfield, EK; Young, AB | 1 |
Blurton, PA; Wood, MD | 1 |
Cote, TE; Frey, EA; Sekura, RD | 1 |
Fujita, M; Nishio, H; Nomura, Y; Segawa, T; Taguchi, J | 1 |
Creese, I; De Lean, A; Sibley, DR | 1 |
MacKenzie, RG; Zigmond, MJ | 1 |
Seeman, P; Wreggett, KA | 1 |
Hancock, AA; Marsh, CL | 1 |
Cote, TE; Frey, EA; Grewe, CW; Kebabian, JW | 2 |
Andorn, AC; Kohagen, KR | 1 |
Battaglia, G; Shannon, M; Titeler, M | 1 |
Amlaiky, N; Caron, MG; Kilpatrick, BF | 1 |
Caron, MG; Kilpatrick, BF | 1 |
Marshall, AM; Mishra, RK; Ramwani, J | 1 |
Caron, MG; De Lean, A; Kilpatrick, BF | 1 |
Hatta, S; Hatta, Y; Saito, T | 1 |
Nobrega, JN; Seeman, P | 1 |
Grünewald, S; Michel, H; Reiländer, H | 1 |
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL | 1 |
Braun, K; Poeggel, G; Reiser, M; Schnabel, R; Schröder, H | 1 |
George, SR; Liu, IS; Seeman, P | 1 |
Ginovart, N; Kapur, S; Ko, F; Seeman, P; Sun, W | 1 |
44 other study(ies) available for spiperone and guanylyl imidodiphosphate
Article | Year |
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Characterization of the inhibitory effect of adrenocorticotropin/melanocyte-stimulating hormone-like peptides on the binding of dopamine receptor ligands to the dopamine D2 receptor in vitro.
Topics: Adrenocorticotropic Hormone; Age Factors; Animals; Apomorphine; Binding, Competitive; Dopamine D2 Receptor Antagonists; Guanylyl Imidodiphosphate; Ligands; Male; Melanocyte-Stimulating Hormones; Peptides; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Temperature; Time Factors | 1992 |
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1992 |
Expression of functional D2 dopamine receptors following differentiation of Y-79 human retinoblastoma cells.
Topics: Adenylyl Cyclase Inhibitors; Binding, Competitive; Cell Membrane; Colforsin; Dopamine; Dopamine Agents; Dopamine Antagonists; Eye Neoplasms; Guanylyl Imidodiphosphate; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Retinoblastoma; Spiperone; Tumor Cells, Cultured | 1990 |
Modulation of high-affinity CNS dopamine D2 receptor by L-pro-L-leu-glycinamide (PLG) analogue 3(R)-(N-L-prolylamino)-2-oxo-1-pyrrolidineacetamide.
Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Kinetics; MSH Release-Inhibiting Hormone; Pyrrolidinones; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1990 |
Paraxanthine displaces the binding of [3H]SCH 23390 from rat striatal membranes.
Topics: Animals; Benzazepines; Binding, Competitive; Brain; Caffeine; Corpus Striatum; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Membranes; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Theophylline | 1990 |
Chronic estrogen treatment promotes a functional uncoupling of the D2 dopamine receptor in rat anterior pituitary gland.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Binding, Competitive; Cell Membrane; Diethylstilbestrol; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Male; Organ Size; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Vasoactive Intestinal Peptide | 1989 |
D2 dopamine receptors in the human brain: heterogeneity based on differences in guanine nucleotide effect on agonist binding, and their presence on corticostriatal nerve terminals.
Topics: Adult; Aged; Aged, 80 and over; Benzazepines; Brain; Cerebral Cortex; Corpus Striatum; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Male; Middle Aged; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1989 |
Dopamine D2 receptors in the anterior pituitary: a single population without reciprocal antagonist/agonist states.
Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; Butyrophenones; Dopamine; Dopamine Antagonists; Guanylyl Imidodiphosphate; Norepinephrine; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Serotonin; Sodium Chloride; Spiperone; Swine; Tetrahydronaphthalenes | 1985 |
Binding of a novel dopaminergic agonist radioligand [3H]-fenoldopam (SKF 82526) to D-1 receptors in rat striatum.
Topics: Adenylyl Cyclase Inhibitors; Animals; Benzazepines; Binding, Competitive; Caudate Nucleus; Fenoldopam; Flupenthixol; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Putamen; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Sodium; Spiperone | 1985 |
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes | 1985 |
Effects of chronic neuroleptic treatment on agonist affinity states of the dopamine-D2 receptor in the rat brain.
Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Brain Chemistry; Guanylyl Imidodiphosphate; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Salicylamides; Spiperone | 1987 |
Interaction of L-prolyl-L-leucyl glycinamide with dopamine D2 receptor: evidence for modulation of agonist affinity states in bovine striatal membranes.
Topics: Animals; Apomorphine; Cattle; Corpus Striatum; Guanylyl Imidodiphosphate; MSH Release-Inhibiting Hormone; Osmolar Concentration; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1988 |
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone | 1987 |
Dopamine agonist high-affinity state in solubilized D2 receptors in striatum, but not in anterior pituitary.
Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Chromatography, High Pressure Liquid; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone | 1987 |
Photoaffinity labelling and solubilization on the central 5-HT1A receptor binding site.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Affinity Labels; Animals; Azides; Binding Sites; Cations; Detergents; Guanylyl Imidodiphosphate; Hippocampus; Male; Photolysis; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Solubility; Spiperone; Tetrahydronaphthalenes | 1987 |
Characterization of D2 dopamine receptors in dopamine-resistant prolactin-secreting rat pituitary tumors 7315a and MtTW15.
Topics: Affinity Labels; Animals; Apomorphine; Cell Membrane; Dopamine; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Female; Guanylyl Imidodiphosphate; Molecular Weight; Neoplasm Transplantation; Photochemistry; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred BUF; Rats, Inbred WF; Receptors, Dopamine; Receptors, Dopamine D2; Solubility; Spiperone | 1987 |
Binding of [125I]-N-(p-aminophenethyl)spiroperidol to the D-2 dopamine receptor in the neurointermediate lobe of the rat pituitary gland: a thermodynamic study.
Topics: Animals; Apomorphine; Female; Fluphenazine; Guanylyl Imidodiphosphate; In Vitro Techniques; Iodine Radioisotopes; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Thermodynamics | 1988 |
Interaction of [3H]spiperone with rat striatal dopamine D-2 receptors: kinetic evidence for antagonist-induced formation of ternary complex.
Topics: Algorithms; Animals; Bromocriptine; Corpus Striatum; Guanylyl Imidodiphosphate; Kinetics; Male; Pertussis Toxin; Polymers; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Virulence Factors, Bordetella | 1988 |
Estradiol and guanine nucleotide modulation of dopamine receptor agonist and antagonist binding sites in 7315a pituitary tumors.
Topics: Animals; Binding Sites; Estradiol; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred BUF; Receptors, Dopamine; Sodium Chloride; Spiperone | 1988 |
Characterization of high-affinity dopamine D2 receptors and modulation of affinity states by guanine nucleotides in cholate-solubilized bovine striatal preparations.
Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cholic Acid; Cholic Acids; Computers; Corpus Striatum; Domperidone; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Receptors, Dopamine; Solubility; Spiperone | 1986 |
Properties of D2 dopamine receptor autoradiography: high percentage of high-affinity agonist sites and increased nucleotide sensitivity in tissue sections.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1986 |
Identification of multiple binding sites for [3H]5-hydroxytryptamine in the rat CNS.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Calcium; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Hippocampus; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Tissue Distribution | 1986 |
Dependence of dopamine receptor conversion from agonist high- to low-affinity state on temperature and sodium ions.
Topics: Animals; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Receptors, Dopamine; Sodium; Spiperone; Swine; Temperature; Tritium | 1985 |
Altered activity of the inhibitory guanyl nucleotide-binding component (Ni) induced by pertussis toxin. Uncoupling of Ni from receptor with continued coupling of Ni to the catalytic unit.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bacterial Toxins; Cell Membrane; Cholera Toxin; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Pertussis Toxin; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Virulence Factors, Bordetella | 1984 |
Factors regulating ligand binding to 5-hydroxytryptamine receptors in rat brain.
Topics: Animals; Ascorbic Acid; Bicarbonates; Female; Frontal Lobe; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Lipid Peroxides; Male; Manganese; Oxidation-Reduction; Rats; Receptors, Serotonin; Sodium Bicarbonate; Spiperone | 1984 |
Anterior pituitary dopamine receptors. Demonstration of interconvertible high and low affinity states of the D-2 dopamine receptor.
Topics: Animals; Binding, Competitive; Butaclamol; Cattle; Cell Membrane; Computers; Ergolines; Guanylyl Imidodiphosphate; Kinetics; Pergolide; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1982 |
High- and low-affinity states of striatal D2 receptors are not affected by 6-hydroxydopamine or chronic haloperidol treatment.
Topics: Animals; Apomorphine; Butaclamol; Cinanserin; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1984 |
Agonist high- and low-affinity states of the D2-dopamine receptor in calf brain. Partial conversion by guanine nucleotide.
Topics: Animals; Binding, Competitive; Cattle; Caudate Nucleus; Cell Membrane; Guanylyl Imidodiphosphate; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tetrahydronaphthalenes | 1984 |
Distinctions between ligand-binding sites for [3H]dopamine and D2 dopaminergic receptors characterized with [3H]spiroperidol.
Topics: Animals; Binding Sites; Binding, Competitive; Butyrophenones; Cell Membrane; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Kinetics; Male; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1984 |
Evidence that the D-2 dopamine receptor in the intermediate lobe of the rat pituitary gland is associated with an inhibitory guanyl nucleotide component.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Cholera Toxin; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Pituitary Gland; Rats; Receptors, Adrenergic, beta; Receptors, Dopamine; Spiperone | 1983 |
Guanyl nucleotides decrease antagonist binding at high affinity dopamine receptors.
Topics: Animals; Binding, Competitive; Corpus Striatum; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Magnesium; Rats; Receptors, Dopamine; Spiperone | 1984 |
Guanine nucleotides modulate cortical S2 serotonin receptors.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone | 1984 |
A novel radioiodinated high affinity ligand for the D2-dopamine receptor. Characterization of its binding in bovine anterior pituitary membranes.
Topics: Animals; Binding, Competitive; Butyrophenones; Cattle; Guanylyl Imidodiphosphate; Kinetics; Membranes; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Spiperone | 1984 |
Agonist binding promotes a guanine nucleotide reversible increase in the apparent size of the bovine anterior pituitary dopamine receptors.
Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Chromatography, High Pressure Liquid; Dopamine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Molecular Weight; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone | 1983 |
Factors affecting solubilized dopamine-sensitive adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cattle; Chlorpromazine; Corpus Striatum; Dopamine; Enzyme Activation; Guanylyl Imidodiphosphate; Haloperidol; Lipids; Magnesium; Solubility; Spiperone | 1983 |
Guanine nucleotides regulate both dopaminergic agonist and antagonist binding in porcine anterior pituitary.
Topics: Animals; Apomorphine; Binding, Competitive; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine | 1982 |
[3H]spiroperidol identifies a D-2 dopamine receptor inhibiting adenylate cyclase activity in the intermediate lobe of the rat pituitary gland.
Topics: Adenylyl Cyclase Inhibitors; Animals; Apomorphine; Binding, Competitive; Butyrophenones; Cholera Toxin; Fluphenazine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride | 1982 |
Effects of ceruletide on the dopamine receptor-adenylate cyclase system in striatum and frontal cortex of rats chronically treated with haloperidol.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Ceruletide; Frontal Lobe; Guanylyl Imidodiphosphate; Haloperidol; Male; Neostriatum; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1993 |
Dopamine D2 receptors mapped in rat brain with [3H](+)PHNO.
Topics: Animals; Autoradiography; Brain; Brain Chemistry; Brain Mapping; Densitometry; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Ligands; Male; Oxazines; Raclopride; Rats; Rats, Wistar; Salicylamides; Spiperone | 1994 |
In vivo reconstitution of dopamine D2S receptor-mediated G protein activation in baculovirus-infected insect cells: preferred coupling to Gi1 versus Gi2.
Topics: Adenosine Triphosphate; Animals; Apomorphine; Baculoviridae; Binding, Competitive; Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Receptors, Dopamine D2; Spiperone; Spodoptera | 1996 |
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1998 |
Effect of social experience on dopamine-stimulated adenylyl cyclase activity and G protein composition in chick forebrain.
Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Benzazepines; Chickens; Colforsin; Cyclic AMP; Dopamine; Dopamine Antagonists; Enzyme Activation; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Imprinting, Psychological; In Vitro Techniques; Prosencephalon; Receptors, Dopamine D1; Receptors, Dopamine D2; Social Isolation; Spiperone; Stimulation, Chemical | 1999 |
The human dopamine D2(Longer) receptor has a high-affinity state and inhibits adenylyl cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alternative Splicing; Animals; Binding, Competitive; CHO Cells; Colforsin; Cricetinae; Dopamine; Dopamine Antagonists; Enzyme Activation; Guanylyl Imidodiphosphate; Humans; Receptors, Dopamine D2; Spiperone; Thermodynamics | 2000 |
In vivo evidence for dopamine-mediated internalization of D2-receptors after amphetamine: differential findings with [3H]raclopride versus [3H]spiperone.
Topics: Amphetamine; Animals; Binding Sites; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Endocytosis; Guanylyl Imidodiphosphate; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Time Factors; Tritium | 2003 |