Page last updated: 2024-08-16

spiperone and fluphenazine

spiperone has been researched along with fluphenazine in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-199025 (71.43)18.7374
1990's7 (20.00)18.2507
2000's0 (0.00)29.6817
2010's3 (8.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Choudhary, MS; Craigo, SC; Meltzer, HY; Monsma, FJ; Roth, BL; Shen, Y; Sibley, DR; Uluer, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brouillette, WJ; Brown, GB; Zha, C1
Dismukes, K; Mulder, AH1
Hanin, I; Sherman, KA; Zigmond, MJ1
Creese, I; Snyder, SH; Stewart, K1
Klimek, V; Maj, J; Rawlów, A; Sarnek, J1
Baran, L; Sarnek, J1
Greenshaw, AJ; Juorio, AV; Paterson, IA; Zhu, MY1
De Vivo, M; Maayani, S1
Boyson, SJ; McGonigle, P; Molinoff, PB; Reuter, S1
Hietala, J; Röyttä, M; Syvälahti, E1
Aravagiri, M; Ellison, GD; See, RE1
Madras, BK; Seeman, P1
Finch, CE; Morgan, DG1
Agui, T; Amlaiky, N; Caron, MG; Kebabian, JW1
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW1
Wreggett, KA1
Thermos, K; Weiss, B; Winkler, JD1
Fong, JC1
Dakshinamurti, K; Paulose, CS1
Burchinsky, SG1
Bacopoulos, NG2
Benson, DI; Kuhn, CM; Meyerson, LR; Stanley, M; Virgilio, J; Wazer, D1
Cote, TE; Frey, EA; Grewe, CW; Kebabian, JW1
De Vries, J; Dijkstra, D; Horn, AS; Mulder, AH1
Misra, CH; Shelat, H; Smith, RC1
Misra, CH; Smith, RC1
Chuang, YC; Huang, WT; Lin, MT; Liu, HS; Won, SJ1
Ashizawa, T; Saito, T; Takahata, N1
Bradley, RJ; Dwyer, DS; Liu, Y1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1

Reviews

1 review(s) available for spiperone and fluphenazine

ArticleYear
Neurotransmitter receptors in the central nervous system and aging: pharmacological aspect (review).
    Experimental gerontology, 1984, Volume: 19, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Brain; Desipramine; Dopamine; Dopamine Antagonists; Female; Fluphenazine; Haloperidol; Humans; Male; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Cholinergic; Receptors, Dopamine; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Serotonin; Reserpine; Scopolamine; Spiperone; Tetrahydronaphthalenes; Tissue Distribution; Tritium

1984

Other Studies

34 other study(ies) available for spiperone and fluphenazine

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:3

    Topics: Animals; Antipsychotic Agents; Cell Line; Molecular Structure; Rats; Receptors, Serotonin

1994
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
Effects of neuroleptics on release of 3H-dopamine from slices of rat corpus striatum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 297, Issue:1

    Topics: Animals; Antipsychotic Agents; Apomorphine; Chlorpromazine; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; Fluphenazine; Haloperidol; Male; Rats; Spiperone

1977
The effect of neuroleptics on acetylcholine concentration and choline uptake in striatum: Implications for regulation of acetylcholine metabolism.
    The Journal of pharmacology and experimental therapeutics, 1978, Volume: 206, Issue:3

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Brain Chemistry; Cerebral Cortex; Choline; Corpus Striatum; Fluphenazine; Haloperidol; Male; Rats; Spiperone

1978
Species variation in dopamine receptor binding.
    European journal of pharmacology, 1979, Nov-23, Volume: 60, Issue:1

    Topics: Animals; Apomorphine; Binding, Competitive; Brain; Cattle; Caudate Nucleus; Fluphenazine; Haloperidol; Humans; In Vitro Techniques; Male; Rats; Receptors, Dopamine; Species Specificity; Spiperone; Tetrahydronaphthalenes

1979
On the anticataleptic action of cyproheptadine.
    Pharmacology, biochemistry, and behavior, 1976, Volume: 5, Issue:2

    Topics: Animals; Atropine; Catalepsy; Clomipramine; Cyproheptadine; Desipramine; Female; Fluphenazine; Humans; Imipramine; Male; Methyltyrosines; Pilocarpine; Pimozide; Promethazine; Rats; Reserpine; Spiperone

1976
The effect of 5-hydroxytrytamine synthesis inhibitors on neuroleptic-induced catalepsy in rats.
    Archivum immunologiae et therapiae experimentalis, 1975, Volume: 23, Issue:4

    Topics: Amphetamines; Catalepsy; Fluphenazine; Humans; p-Chloroamphetamine; Pimozide; Reserpine; Serotonin; Spiperone; Tranquilizing Agents

1975
The effects of some neuroleptics and d-amphetamine on striatal 2-phenylethylamine in the mouse.
    General pharmacology, 1991, Volume: 22, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Chlorpromazine; Corpus Striatum; Dextroamphetamine; Dopamine; Fluphenazine; Homovanillic Acid; In Vitro Techniques; Male; Mice; Monoamine Oxidase Inhibitors; Pargyline; Phenethylamines; Selegiline; Spiperone; Synaptic Transmission

1991
Stimulation and inhibition of adenylyl cyclase by distinct 5-hydroxytryptamine receptors.
    Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Membrane; Cerebral Cortex; Colforsin; Drug Interactions; Enzyme Activation; Fluphenazine; Guinea Pigs; Hippocampus; Mathematics; Mianserin; Pindolol; Piperazines; Rats; Receptors, Serotonin; Spiperone

1990
Effects of chronic treatment with selective and nonselective antagonists on the subtypes of dopamine receptors.
    Synapse (New York, N.Y.), 1989, Volume: 3, Issue:1

    Topics: Animals; Benzazepines; Corpus Striatum; Fluphenazine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1989
Dopamine D2 and muscarinic receptor binding characteristics in rat brain after withdrawal of subchronic fluphenazine and sulpiride treatment.
    Progress in neuro-psychopharmacology & biological psychiatry, 1989, Volume: 13, Issue:1-2

    Topics: Animals; Cerebral Cortex; Corpus Striatum; Fluphenazine; Kinetics; Male; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Muscarinic; Reference Values; Spiperone; Substance Withdrawal Syndrome; Sulpiride

1989
Chronic neuroleptic treatment in rats produces persisting changes in GABAA and dopamine D-2, but not dopamine D-1 receptors.
    Life sciences, 1989, Volume: 44, Issue:3

    Topics: Animals; Autoradiography; Behavior, Animal; Benzazepines; Brain; Disease Models, Animal; Dyskinesia, Drug-Induced; Female; Fluphenazine; Haloperidol; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone

1989
Drug potencies on partially purified brain D2 dopamine receptors.
    Journal of neurochemistry, 1985, Volume: 44, Issue:3

    Topics: Animals; Butaclamol; Chlorpromazine; Corpus Striatum; Dogs; Fluphenazine; Haloperidol; Isoelectric Focusing; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Time Factors

1985
[3H]Fluphenazine binding to brain membranes: simultaneous measurement of D-1 and D-2 receptor sites.
    Journal of neurochemistry, 1986, Volume: 46, Issue:5

    Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Brain; Cell Membrane; Corpus Striatum; Fluphenazine; Kinetics; Male; Mice; Mice, Inbred C57BL; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tissue Distribution

1986
Binding of [125I]-N-(p-aminophenethyl)spiroperidol to the D-2 dopamine receptor in the neurointermediate lobe of the rat pituitary gland: a thermodynamic study.
    Molecular pharmacology, 1988, Volume: 33, Issue:2

    Topics: Animals; Apomorphine; Female; Fluphenazine; Guanylyl Imidodiphosphate; In Vitro Techniques; Iodine Radioisotopes; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Thermodynamics

1988
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
    Advances in experimental medicine and biology, 1988, Volume: 235

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
Alkylation of the bovine anterior pituitary D2-dopamine receptor: inconsistency with predictions of the ternary complex model.
    Biochemical and biophysical research communications, 1987, Sep-30, Volume: 147, Issue:3

    Topics: Alkylation; Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Computer Simulation; Dopamine Antagonists; Fluphenazine; GTP-Binding Proteins; In Vitro Techniques; Ligands; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Structure-Activity Relationship

1987
Comparison of the effects of fluphenazine-N-mustard on dopamine binding sites and on behavior induced by apomorphine in supersensitive mice.
    Neuropharmacology, 1987, Volume: 26, Issue:10

    Topics: Animals; Apomorphine; Binding, Competitive; Fluphenazine; Hydroxydopamines; Male; Mice; Oxidopamine; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1987
Preferential adsorption of dopamine antagonist binding sites by fluphenazine-agarose.
    Proceedings of the National Science Council, Republic of China. Part B, Life sciences, 1986, Volume: 10, Issue:2

    Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Chromatography, Affinity; Corpus Striatum; Dopamine; Dopamine Antagonists; Fluphenazine; Kinetics; Receptors, Dopamine; Spiperone

1986
Effect of pyridoxine deficiency in young rats on high-affinity serotonin and dopamine receptors.
    Journal of neuroscience research, 1985, Volume: 14, Issue:2

    Topics: Animals; Body Weight; Brain Chemistry; Cerebral Cortex; Corpus Striatum; Fluphenazine; Organ Size; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Spiperone; Vitamin B 6 Deficiency

1985
Antipsychotic drug effects on dopamine and serotonin receptors: in vitro binding and in vivo turnover studies.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 219, Issue:3

    Topics: Animals; Antipsychotic Agents; Brain; Butaclamol; Catalepsy; Dopamine; Fluphenazine; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Spiperone

1981
Lack of potency of metoclopramide's metabolites in various dopaminergic models.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:2

    Topics: Animals; Apomorphine; Dopamine; Fluphenazine; Haloperidol; Homovanillic Acid; Humans; Male; Metoclopramide; Prolactin; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes

1983
[3H]spiroperidol identifies a D-2 dopamine receptor inhibiting adenylate cyclase activity in the intermediate lobe of the rat pituitary gland.
    Endocrinology, 1982, Volume: 110, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Apomorphine; Binding, Competitive; Butyrophenones; Cholera Toxin; Fluphenazine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride

1982
Is TL-99 a selective presynaptic dopamine receptor agonist?
    European journal of pharmacology, 1982, Sep-10, Volume: 83, Issue:1-2

    Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Female; Fluphenazine; Male; Motor Activity; Naphthalenes; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Time Factors

1982
Age affects dopamine receptor changes during chronic administration of fluphenazine.
    European journal of pharmacology, 1982, Dec-03, Volume: 85, Issue:3-4

    Topics: Age Factors; Animals; Fluphenazine; Rats; Rats, Inbred F344; Receptors, Dopamine; Spiperone

1982
Biochemical mechanism of tolerance to neuroleptic drugs; regional differences in rat brain.
    European journal of pharmacology, 1981, Apr-09, Volume: 70, Issue:4

    Topics: Animals; Butyrophenones; Caudate Nucleus; Cerebral Cortex; Dopamine; Drug Tolerance; Fluphenazine; Haloperidol; Homovanillic Acid; Rats; Spiperone

1981
Effects of age on dopaminergic supersensitivity induced by chronic fluphenazine.
    Communications in psychopharmacology, 1980, Volume: 4, Issue:5

    Topics: Aging; Animals; Corpus Striatum; Dopamine; Fluphenazine; Kinetics; Rats; Rats, Inbred F344; Spiperone

1980
Suppression of natural killer cell activity in mouse spleen lymphocytes by several dopamine receptor antagonists.
    Experientia, 1995, Apr-15, Volume: 51, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cytotoxicity, Immunologic; Dopamine Antagonists; Flupenthixol; Fluphenazine; Killer Cells, Natural; Mice; Mice, Inbred C3H; Pimozide; Spiperone; Spleen; Thiothixene; Trifluoperazine

1995
Effects of ceruletide on perioral movements and the dopamine receptor-adenylate cyclase system in rats chronically treated with fluphenazine.
    Psychopharmacology, 1996, Volume: 125, Issue:3

    Topics: Adenylyl Cyclases; Animals; Behavior, Animal; Benzazepines; Ceruletide; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Electromyography; Fluphenazine; Male; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1996
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
    Neuroscience letters, 1999, Oct-29, Volume: 274, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium

1999
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016