spiperone has been researched along with ergoline in 104 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 54 (51.92) | 18.7374 |
1990's | 49 (47.12) | 18.2507 |
2000's | 1 (0.96) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Battista, AF; Fuxe, K; Goldstein, M; Lew, JY; Lieberman, A; Nakamura, S | 1 |
Cote, T; Kebabian, J; Munemura, M | 1 |
Battista, AF; Goldstein, M; Lew, JY; Nakamura, S | 1 |
Fuller, RW; Snoddy, HD | 3 |
Fujita, N; Saito, K; Yonehara, N; Yoshida, H | 1 |
Jenner, P; Marsden, CD; Rose, S; Thomas, KL | 1 |
Esterle, TM; Sanders-Bush, E | 1 |
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD | 1 |
Lucki, I; McGonigle, P; Subramaniam, S | 1 |
DeSouza, EB; Grigoriadis, DE; Levant, B | 2 |
LaHoste, GJ; Marshall, JF | 1 |
Kozlowski, MR; Neve, KA; Rosser, MP | 1 |
Pawlikowski, M; Pisarek, H; Stepien, H | 1 |
Aulakh, CS; Hill, JL; Murphy, DL | 1 |
Choudhary, MS; Craigo, S; Roth, BL | 1 |
Todd, RD | 1 |
Boroni, F; Castelletti, L; Memo, M; Missale, C; Spano, P | 1 |
Gong, L; Kostrzewa, RM | 1 |
Michel, AD; Nunes, JL; Sharif, NA; Whiting, RL | 1 |
Schaus, JM; Seeman, P | 1 |
Brus, R; Kalbfleisch, J; Kostrzewa, RM | 1 |
Bourque, CW; Renaud, LP; Yang, CR | 1 |
Aghajanian, GK; Sheldon, PW | 1 |
Courtney, ND; Howlett, AC; Westfall, TC | 1 |
Bancroft, C; Dong, KW; McChesney, R; Roberts, JL; Sealfon, SC; Tsutsumi, M | 1 |
Hashimoto, T; Katsura, M; Kuriyama, K | 1 |
Linseman, MA | 1 |
Nowak, JZ; Schorderet, M | 1 |
Axel, R; Huang, KN; Jessell, TM; Julius, D; Livelli, TJ | 1 |
Gessa, GL; Olianas, MC; Onali, P | 1 |
Iuvone, PM | 1 |
Beaulieu, M; Felder, R; Kebabian, JW | 1 |
Cohen, ML; Kurz, KD; Schenck, KW | 1 |
Brazell, C; Dourish, CT; King, BH; Middlemiss, DN | 1 |
Doty, RL; Risser, JM | 1 |
Segawa, T; Zhang, X | 1 |
Allin, R; Reyneke, L; Russell, VA; Taljaard, JJ | 1 |
Klimek, V; Maj, J | 1 |
Dlabac, A; Dobrovský, K; Krejcí, I; Valchár, M | 1 |
Chojnacka-Wójcik, E; Jaros, T; Kłodzińska, A; Maj, J | 1 |
Fuller, RW; Hemrick-Luecke, SK; Perry, KW; Toomey, RE | 1 |
Arnt, J; Hyttel, J | 1 |
Crocker, AD; Faunt, JE | 2 |
Battaglia, G; Creese, I; Hess, EJ; Norman, AB | 1 |
Kidric, M; Petrović, J; Soskić, V; Trajković, D | 1 |
Beart, PM; Bridge, S; Christie, MJ | 1 |
Amedro, J; Brown, L; Smith, D; Williams, G | 1 |
Ares, J; Chang, YA; Farooqui, T; Miller, D; Uretsky, N; Wallace, L; Wallace, RA | 1 |
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW | 1 |
Arnt, J; Hyttel, J; Nowak, G | 1 |
Burchill, SA; Thody, AJ | 1 |
Bondy, SC; Breese, GR; Duncan, GE; Iorio, LC; Mueller, RA; Napier, TC | 1 |
Nakagawa, K; Sekihara, S; Somei, M; Watanabe, H; Yamada, F | 1 |
Fuller, RW; Hemrick-Luecke, SK | 1 |
Dlabac, A; Krejcí, I; Valchár, M; Vrsecká, M | 1 |
Anderson, D; Gordon, J; Herbster, G; Koller, W; Wack, R | 1 |
Brunello, N; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC | 1 |
Bymaster, FP; Kornfeld, EC; Nichols, CL; Reid, LR; Wong, DT | 1 |
Arnt, J | 1 |
Liskowsky, DR; Potter, LT | 1 |
Cohen, ML; Fuller, RW; Garbrecht, WL; Kurz, KD; Marzoni, GP; Mason, NR | 1 |
Dow, RC; Hill, AG; McQueen, JK | 1 |
Hruska, RE; Silbergeld, EK | 1 |
Filburn, CR; Joseph, JA; Roth, GS | 1 |
Fuller, RW; Hemrick-Luecke, SK; Perry, KW | 1 |
Beart, PM; McDonald, D | 1 |
Ferrer, JM; Mora, F; Sanguinetti, AM; Vives, F | 1 |
Creese, I; De Lean, A; Sibley, DR | 1 |
Beart, PM; Gundlach, AL; Krstich, M | 1 |
Koller, WC | 1 |
Hruska, RE; Silbergeld, EK; Weir, RL | 1 |
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K | 1 |
Asano, T; Goldstein, M; Lew, JY; Lieberman, A; Makman, MH; Rosenfeld, MR | 1 |
Reynolds, GP; Riederer, P | 1 |
Battaglia, G; Titeler, M | 1 |
Senogles, SE | 1 |
Bancroft, C; Fischberg, DJ | 1 |
Barrett, RJ; Caul, WF; Huffman, EM; Jones, JR; Strand, EJ | 1 |
Erol, DD; Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD; Smith, LA | 1 |
Abarca, J; Bustos, G; Gysling, K; Roth, RH | 1 |
Chaouche-Teyara, K; Dabiré, H; Fournier, B; Safar, M | 1 |
Katz, JL; Witkin, JM | 1 |
Contestabile, A; Dall'Olio, R; Facchinetti, F; Gandolfi, O | 1 |
Guo, J; Kostrzewa, FP; Kostrzewa, RM | 1 |
Bernard, A; Cavegn, C; Chabert, C; Mills, A | 1 |
Dall'Olio, R; Gandolfi, O; Rimondini, R | 1 |
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD | 1 |
Bole-Vunduk, B; Budihna, MV; Krisch, I; Lavric, B; Ocvirk, A; Pepelnak, M; Sket, D | 1 |
Nowak, JZ; Zawilska, JB | 1 |
Burnham, P; Louis, JC; Magal, E; Varon, S | 1 |
Dall'Olio, R; Gandolfi, O | 1 |
Aloyo, VJ; Chen, JF; Weiss, B | 1 |
Ball, S; Boyfield, I; Coldwell, MC; Cook, T; Gloger, IS; Herrity, N; McHale, M; Robinson, JH; Winn, FM | 1 |
Craig, DA; Martin, GR | 1 |
Allard, S; Falardeau, P; Lapointe, S | 1 |
Allet, B; Bernard, A; Brandt, E; Cavegn, C; Chabert, C; Chollet, A; Kawashima, E; Mills, A | 1 |
Felder, RA; Jose, PA; Walk, SF; Yamaguchi, I | 1 |
Cheng, CC; Leonard, NL; Levant, B; Moehlenkamp, JD; Morgan, KA | 1 |
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP | 1 |
Clifton, PG; Dourish, CT; Kennett, GA; Lee, MD; Somerville, EM | 1 |
1 review(s) available for spiperone and ergoline
Article | Year |
---|---|
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates | 1990 |
103 other study(ies) available for spiperone and ergoline
Article | Year |
---|---|
Dopaminephilic properties of ergot alkaloids.
Topics: Acetonitriles; Animals; Bromocriptine; Corpus Striatum; Ergolines; Ergot Alkaloids; Haplorhini; Humans; Levodopa; Parkinson Disease; Receptors, Dopamine; Spiperone; Substantia Nigra; Synaptosomes; Tremor; Tyrosine 3-Monooxygenase | 1978 |
Lisuride hydrogen maleate: an ergoline with beta-adrenergic antagonist activity.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding Sites; Cerebellum; Dihydroalprenolol; Ergolines; Isoproterenol; Lisuride; Rabbits; Spiperone | 1979 |
Dopamine agonist potencies of ergolines.
Topics: Animals; Cattle; Corpus Striatum; Dopamine; Ergolines; Haplorhini; Humans; Neural Pathways; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra; Tegmentum Mesencephali; Tremor | 1979 |
The effects of metergoline and other serotonin receptor antagonists on serum corticosterone in rats.
Topics: Animals; Corticosterone; Cyproheptadine; Ergolines; Male; Metergoline; Methysergide; Rats; Serotonin Antagonists; Spiperone; Structure-Activity Relationship | 1979 |
Lisuride inhibits 3H-spiroperidol binding to membranes isolated from striatum.
Topics: Animals; Butyrophenones; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Ergolines; In Vitro Techniques; Lisuride; Male; Membranes; Rats; Spiperone | 1978 |
Dissociation of the striatal D-2 dopamine receptor from adenylyl cyclase following 6-hydroxydopamine-induced denervation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Denervation; Dopamine; Ergolines; Female; Homovanillic Acid; Oxidopamine; Prosencephalon; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1992 |
Serotonin agonists increase transferrin levels via activation of 5-HT1C receptors in choroid plexus epithelium.
Topics: Amino Acid Isomerases; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Choroid Plexus; Cyclosporins; Epithelium; Ergolines; Fibroblasts; Kinetics; Male; Mianserin; Peptidylprolyl Isomerase; Phosphatidylinositols; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA Probes; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Thymidine; Time Factors; Transferrin | 1992 |
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone | 1992 |
Effects of chronic treatment with selective agonists on the subtypes of dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Body Temperature Regulation; Brain; Caudate Nucleus; Dopamine Agents; Drug Interactions; Ergolines; Kinetics; Male; Nucleus Accumbens; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reference Values; Spiperone; Substantia Nigra | 1992 |
Characterization of [3H]quinpirole binding to D2-like dopamine receptors in rat brain.
Topics: Animals; Binding Sites; Brain; Culture Techniques; Dopamine Agents; Dopamine Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone | 1992 |
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium | 1992 |
Dopamine D2 receptor stimulation of Na+/H+ exchange assessed by quantification of extracellular acidification.
Topics: Amiloride; Animals; Carrier Proteins; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Glioma; Hydrogen-Ion Concentration; Kinetics; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Sodium-Hydrogen Exchangers; Spiperone; Tumor Cells, Cultured | 1992 |
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.
Topics: Animals; Antiparkinson Agents; Bromocriptine; Diethylstilbestrol; Dose-Response Relationship, Drug; Ergolines; Female; Hyperplasia; Hyperprolactinemia; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Time Factors; Tritium | 1992 |
Effects of various serotonin receptor subtype-selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
Topics: Animals; Corticosterone; Ergolines; Male; Metergoline; Mianserin; Neurosecretory Systems; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1992 |
Identification of receptor domains that modify ligand binding to 5-hydroxytryptamine2 and 5-hydroxytryptamine1c serotonin receptors.
Topics: Base Sequence; Binding, Competitive; Ergolines; Haloperidol; In Vitro Techniques; Ketanserin; Molecular Sequence Data; Oligodeoxyribonucleotides; Receptors, Serotonin; Recombinant Fusion Proteins; Spiperone; Structure-Activity Relationship; Transfection | 1992 |
Neural development is regulated by classical neurotransmitters: dopamine D2 receptor stimulation enhances neurite outgrowth.
Topics: Animals; Base Sequence; Brain; Cells, Cultured; Cerebral Cortex; Ergolines; Female; Male; Mental Disorders; Models, Biological; Molecular Sequence Data; Nerve Growth Factors; Neurites; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; RNA, Messenger; Salicylamides; Spiperone | 1992 |
Epidermal growth factor induces the functional expression of dopamine receptors in the GH3 cell line.
Topics: Animals; Binding, Competitive; Cell Line; Cells, Cultured; Dopamine Agents; Epidermal Growth Factor; Ergolines; Kinetics; Pituitary Gland, Anterior; Pituitary Neoplasms; Potassium; Prolactin; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1991 |
Supersensitized D1 receptors mediate enhanced oral activity after neonatal 6-OHDA.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Mouth; Movement; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1991 |
Dopamine D2-receptors mediate hypothermia in mice: ICV and IP effects of agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Body Temperature Regulation; Cerebral Ventricles; Domperidone; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1991 |
Dopamine receptors labelled by [3H]quinpirole.
Topics: Animals; Corpus Striatum; Dogs; Dopamine Agents; Dopamine Antagonists; Ergolines; Guanine Nucleotides; Haloperidol; In Vitro Techniques; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1991 |
Ontogenetic homologous sensitization to the antinociceptive action of quinpirole in rats.
Topics: Aging; Analgesics; Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Female; Pain Measurement; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1991 |
Dopamine D2 receptor activation depolarizes rat supraoptic neurones in hypothalamic explants.
Topics: Animals; Calcium; Dopamine; Dopamine Agents; Ergolines; Membrane Potentials; Neurons; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Sulpiride; Supraoptic Nucleus | 1991 |
Excitatory responses to serotonin (5-HT) in neurons of the rat piriform cortex: evidence for mediation by 5-HT1C receptors in pyramidal cells and 5-HT2 receptors in interneurons.
Topics: Animals; Electrophysiology; Ergolines; Interneurons; Limbic System; Male; Neurons; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone | 1991 |
Dopaminergic regulation of dopamine release from PC12 cells via a pertussis toxin-sensitive G protein.
Topics: Adrenal Gland Neoplasms; Animals; Apomorphine; Cell Line; Dopamine; Dopamine Antagonists; Ergolines; GTP-Binding Proteins; Haloperidol; Nicotine; Pertussis Toxin; Pheochromocytoma; Potassium; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Virulence Factors, Bordetella | 1991 |
Either isoform of the dopamine D2 receptor can mediate dopaminergic repression of the rat prolactin promoter.
Topics: Animals; Cell Line; Ergolines; Female; Hysterectomy; Ovariectomy; Pituitary Neoplasms; Plasmids; Prolactin; Prolactinoma; Promoter Regions, Genetic; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D1; RNA, Messenger; Signal Transduction; Spiperone; Transcription, Genetic | 1991 |
On the mechanism of mergocryptine-induced suppression of dopamine turnover in the rat striatum.
Topics: Animals; Apomorphine; Benzazepines; Corpus Striatum; Dopamine; Ergolines; Half-Life; Male; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1991 |
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1990 |
The 5HT2 receptor defines a family of structurally distinct but functionally conserved serotonin receptors.
Topics: Amino Acid Sequence; Animals; Antiparkinson Agents; Brain; DNA; Ergolines; Fibroblasts; Gene Library; Genes; Mice; Molecular Sequence Data; Organ Specificity; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Nucleic Acid; Spiperone; Transfection; Type C Phospholipases | 1990 |
Characterization of dopamine receptors mediating inhibition of adenylate cyclase activity in rat striatum.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butaclamol; Corpus Striatum; Dopamine; Enzyme Activation; Ergolines; Guanine Nucleotides; Norepinephrine; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Sulpiride | 1985 |
Evidence for a D2 dopamine receptor in frog retina that decreases cyclic AMP accumulation and serotonin N-acetyltransferase activity.
Topics: 1-Methyl-3-isobutylxanthine; Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Bucladesine; Calcium; Circadian Rhythm; Cyclic AMP; Dopamine; Ergolines; Light; Metoclopramide; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Retina; Spiperone; Xenopus laevis | 1986 |
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone | 1986 |
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1988 |
MK-212 increases rat plasma ACTH concentration by activation of the 5-HT1C receptor subtype.
Topics: Adrenocorticotropic Hormone; Animals; Antiparkinson Agents; Ergolines; Ketanserin; Male; Metergoline; Pindolol; Piperazines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone | 1989 |
Influence of the D-2 dopamine receptor agonist quinpirole on the odor detection performance of rats before and after spiperone administration.
Topics: Acetates; Animals; Behavior, Animal; Conditioning, Operant; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Smell; Spiperone | 1989 |
Selective blockade of dopamine D-1 receptor by SCH 23390 affects dopamine agonist binding to 3H-spiperone labeled D-2 receptors in rat striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Guanosine Triphosphate; In Vitro Techniques; Male; Pertussis Toxin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Virulence Factors, Bordetella | 1989 |
Lack of effect of chronic desipramine treatment on dopaminergic activity in the nucleus accumbens of the rat.
Topics: Acetylcholine; Animals; Benzazepines; Desipramine; Dopamine; Dopamine Agents; Dopamine Antagonists; Electric Stimulation; Ergolines; Male; Nomifensine; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Septal Nuclei; Spiperone | 1989 |
Repeated administration of antidepressants enhances agonist affinity for mesolimbic D2-receptors.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Binding, Competitive; Ergolines; Imipramine; Limbic System; Male; Mianserin; Motor Activity; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spiperone | 1989 |
Comparison of (3H)-terguride and (3H)-spiperone binding to dopamine receptors in the rat striatum.
Topics: Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Ergolines; Ergotamines; Lisuride; Male; Rats; Receptors, Dopamine; Spiperone | 1989 |
Exploratory hypoactivity induced by m-trifluoromethylphenylpiperazine (TFMPP) and m-chlorophenylpiperazine (m-CPP).
Topics: Animals; Ergolines; Exploratory Behavior; Male; Metergoline; Mianserin; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone | 1989 |
Pergolide elevation of MHPG sulphate concentration in rat hypothalamus blocked by spiperone and mimicked by other dopamine agonists.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Butyrophenones; Dopamine; Ergolines; Glycols; Homovanillic Acid; Hypothalamus; Male; Methoxyhydroxyphenylglycol; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1985 |
Differential involvement of dopamine D-1 and D-2 receptors in the circling behaviour induced by apomorphine, SK & F 38393, pergolide and LY 171555 in 6-hydroxydopamine-lesioned rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Appetite Depressants; Benzazepines; Electric Stimulation; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical; Time Factors | 1985 |
Adrenocortical hormone status affects responses to dopamine receptor agonists.
Topics: Adrenal Cortex Hormones; Adrenalectomy; Animals; Apomorphine; Behavior, Animal; Benzazepines; Body Temperature; Corticosterone; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1988 |
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Dopaminergic activity of some ergot alkaloid derivatives: relationship to their chemical structure.
Topics: Animals; Cattle; Caudate Nucleus; Dopamine; Ergolines; Ergot Alkaloids; Guanosine Triphosphate; In Vitro Techniques; Molecular Conformation; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Tritium | 1986 |
No change in neostriatal D-2 dopamine receptors after NMDA lesions of rat prefrontal cortex.
Topics: Animals; Aspartic Acid; Corpus Striatum; Ergolines; Female; Frontal Lobe; Male; N-Methylaspartate; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tritium | 1986 |
The effects of selective dopamine receptor agonists and antagonists on body temperature in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Temperature; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1987 |
A pharmacological analysis of the rat spinal cord serotonin (5-HT) autoreceptor.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Male; Piperazines; Potassium; Quipazine; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Spiperone; Tetrahydronaphthalenes; Tritium | 1988 |
Interaction of permanently uncharged dopamine analogs with the D-2 dopaminergic receptor.
Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Ergolines; In Vitro Techniques; Male; Mice; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sodium Chloride; Spiperone; Sulfides | 1988 |
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior | 1988 |
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone | 1988 |
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride | 1986 |
6-hydroxydopamine treatments enhance behavioral responses to intracerebral microinjection of D1- and D2-dopamine agonists into nucleus accumbens and striatum without changing dopamine antagonist binding.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Ergolines; Female; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Microinjections; Motor Activity; Nucleus Accumbens; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone | 1987 |
Dopamine receptor stimulating effects of chanoclavine analogues, tricyclic ergot alkaloids, in the brain.
Topics: 4-Butyrolactone; Animals; Binding, Competitive; Brain; Catechols; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Ergot Alkaloids; In Vitro Techniques; Male; Mice; Rats; Rats, Inbred Strains; Receptors, Dopamine; Rotation; Spiperone; Stereotyped Behavior; Time Factors | 1987 |
Decrease in hypothalamic epinephrine concentration and other neurochemical changes produced by quinpirole, a dopamine agonist, in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Epinephrine; Ergolines; Homovanillic Acid; Hypothalamus; Male; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Binding characteristics of the dopamine agonist/antagonist [3H]terguride (transdihydrolisuride) in the rat striatum.
Topics: Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Kinetics; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1987 |
Quinpirole hydrochloride, a potential anti-parkinsonism drug.
Topics: Animals; Benzazepines; Corpus Striatum; Dogs; Dose-Response Relationship, Drug; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride | 1987 |
Absence of [3H]SCH 23390 specific binding sites in anterior pituitary: dissociation from effects on prolactin secretion.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Corpus Striatum; Cyproheptadine; Ergolines; Kinetics; Male; Metergoline; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1987 |
Elevation of acetylcholine levels in striatum of rat brain by LY163502, trans-(-)-5,5a,6,7,8,9a,10-octahydro-6-propylpyrimido less than 4,5-g greater than quinolin-2-amine dihydrochloride, a potent and stereospecific dopamine (D2) agonist.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Apomorphine; Clonidine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Ergolines; Pergolide; Quinolines; Rats; Receptors, Dopamine; Spiperone | 1986 |
Hyperactivity induced by stimulation of separate dopamine D-1 and D-2 receptors in rats with bilateral 6-OHDA lesions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Benzazepines; Clopenthixol; Dopamine; Dose-Response Relationship, Drug; Ergolines; Flupenthixol; Hydroxydopamines; Hypothalamus; Male; Motor Activity; Oxidopamine; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1985 |
D-2 dopamine receptors in the frontal cortex of rat and human.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Cinanserin; Dopamine; Ergolines; Humans; Kinetics; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1985 |
Pharmacological activity of the isomers of LY53857, potent and selective 5-HT2 receptor antagonists.
Topics: Animals; Blood Pressure; Cerebral Cortex; Corticosterone; Decerebrate State; Ergolines; Isomerism; Male; Mathematics; Quipazine; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Time Factors | 1985 |
Proceedings: Effects of some dopamine receptor stimulants on cobalt-induced epilepsy in the rat.
Topics: Amphetamine; Animals; Apomorphine; Cobalt; Dopamine; Electroencephalography; Epilepsy; Ergolines; Male; Rats; Receptors, Adrenergic; Spiperone; Stimulation, Chemical | 1974 |
Inhibition of neurotransmitter receptor binding by ergot derivatives.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Bromocriptine; Dioxanes; Ergolines; Ergot Alkaloids; gamma-Aminobutyric Acid; Lysergic Acid Diethylamide; Male; Metergoline; Organ Specificity; Quinuclidinyl Benzilate; Rats; Receptors, Neurotransmitter; Serotonin; Spiperone; Structure-Activity Relationship; Synapses | 1981 |
Development of dopamine receptor denervation supersensitivity in the neostriatum of the senescent rat.
Topics: Adenylyl Cyclases; Aging; Animals; Corpus Striatum; Dextroamphetamine; Ergolines; Female; Male; Motor Activity; Rats; Receptors, Dopamine; Rotation; Sex Factors; Spiperone | 1981 |
Elevation of serum corticosterone concentrations in rats by pergolide and other dopamine agonists.
Topics: Animals; Antiparkinson Agents; Corticosterone; Domperidone; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Metergoline; Mianserin; Pergolide; Rats; Rats, Inbred Strains; Spiperone | 1981 |
Depletion of epinephrine in rat hypothalamus by a dopamine agonist, pergolide.
Topics: Animals; Antiparkinson Agents; Dopamine Antagonists; Epinephrine; Ergolines; Haloperidol; Hypothalamus; Kinetics; Male; Pergolide; Rats; Rats, Inbred Strains; Spiperone | 1982 |
Neurochemical studies of the mesolimbic dopaminergic pathway: [3H]spiperone labels two bindings sites in homogenates of the nucleus accumbens of rat brain.
Topics: Animals; Antipsychotic Agents; Apomorphine; Butyrophenones; Dopamine; Ergolines; Kinetics; Nucleus Accumbens; Rats; Receptors, Dopamine; Septal Nuclei; Spiperone | 1982 |
Serum corticosterone elevation by pergolide in rats: prevention of tolerance development by spiperone.
Topics: Animals; Butyrophenones; Corticosterone; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Ergolines; Male; Pergolide; Rats; Rats, Inbred Strains; Spiperone | 1982 |
Effects of agonists and antagonists of D1 and D2 dopamine receptors on self-stimulation of the medial prefrontal cortex in the rat.
Topics: Animals; Apomorphine; Bromocriptine; Cerebral Cortex; Dose-Response Relationship, Drug; Ergolines; Functional Laterality; Male; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Self Stimulation; Spiperone; Sulpiride; Synaptic Transmission | 1983 |
Anterior pituitary dopamine receptors. Demonstration of interconvertible high and low affinity states of the D-2 dopamine receptor.
Topics: Animals; Binding, Competitive; Butaclamol; Cattle; Cell Membrane; Computers; Ergolines; Guanylyl Imidodiphosphate; Kinetics; Pergolide; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1982 |
Guanine nucleotides reveal differential actions of ergot derivatives at D-2 receptors labelled by [3H]spiperone in striatal homogenates.
Topics: Animals; Binding, Competitive; Butyrophenones; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Guanine Nucleotides; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tritium | 1983 |
Attenuation by pergolide of haloperidol-induced striatal dopamine receptor density.
Topics: Animals; Corpus Striatum; Ergolines; Guinea Pigs; Haloperidol; Male; Membranes; Pergolide; Receptors, Dopamine; Spiperone | 1984 |
Binding of antiparkinsonian ergot derivatives to the dopamine receptor.
Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Caudate Nucleus; Ergolines; Lisuride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1981 |
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1983 |
Interaction of pergolide with central dopaminergic receptors.
Topics: Adenylyl Cyclases; Animals; Behavior, Animal; Binding, Competitive; Cattle; Cerebral Decortication; Chlorocebus aethiops; Corpus Striatum; Ergolines; Guanosine Triphosphate; Hot Temperature; Male; Pergolide; Rats; Receptors, Dopamine; Spiperone; Tegmentum Mesencephali; Tremor | 1980 |
The effects of lisuride and some other dopaminergic agonists on receptor binding in human brain.
Topics: Brain; Bromocriptine; Ergolines; Humans; Kinetics; Lisuride; Receptors, Dopamine; Spiperone | 1981 |
Direct binding of 3H-lisuride to adrenergic and serotonergic receptors.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Ergolines; Haloperidol; In Vitro Techniques; Kinetics; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Spiperone | 1981 |
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1994 |
The D2 receptor: blocked transcription in GH3 cells and cellular pathways employed by D2A to regulate prolactin promoter activity.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Cell Line; Chloramphenicol O-Acetyltransferase; DNA-Binding Proteins; Ergolines; Gene Expression Regulation; Pertussis Toxin; Pituitary Gland; Prolactin; Promoter Regions, Genetic; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Thyrotropin-Releasing Hormone; Transcription Factor Pit-1; Transcription Factors; Transcription, Genetic; Transfection; Virulence Factors, Bordetella | 1995 |
D2-specific discriminative stimuli: parameters, blocking, and rebound.
Topics: Animals; Cues; Discrimination, Psychological; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Food Deprivation; Haloperidol; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Spiperone | 1995 |
Differential anti-parkinsonian effects of benzazepine D1 dopamine agonists with varying efficacies in the MPTP-treated common marmoset.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antiparkinson Agents; Behavior, Animal; Benzazepines; Binding, Competitive; Callithrix; Dopamine Agonists; Ergolines; In Vitro Techniques; Male; Parkinson Disease, Secondary; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1995 |
Changes in extracellular levels of glutamate and aspartate in rat substantia nigra induced by dopamine receptor ligands: in vivo microdialysis studies.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aspartic Acid; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Extracellular Space; Glutamic Acid; Kinetics; Ligands; Male; Microdialysis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Substantia Nigra; Tetrodotoxin; Time Factors | 1995 |
Systemic and regional haemodynamic effects of 1-(2,5-dimethoxy-4-iodo-phenyl)-2-aminopropane (DOI) and alpha-methyl-5-HT, in the anaesthetised rat.
Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Ergolines; Hemodynamics; Injections, Intravenous; Injections, Intraventricular; Male; Rats; Rats, Wistar; Regional Blood Flow; Renal Circulation; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Splanchnic Circulation | 1994 |
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone | 1993 |
Chronic neonatal blockade of N-methyl-D-aspartate receptor by CGP 39551 increases dopaminergic function in adult rat.
Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Apomorphine; Behavior, Animal; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Motor Activity; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; Spiperone; Stereotyped Behavior; Time Factors | 1994 |
Ontogenetic quinpirole treatment induces vertical jumping activity in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Injections, Intraperitoneal; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1993 |
Characterization of the functional activity of dopamine ligands at human recombinant dopamine D4 receptors.
Topics: Animals; Cell Line; Clozapine; DNA; Dopamine; Dopamine Agents; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Ligands; Moths; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Sulfur Radioisotopes; Tritium | 1994 |
D-cycloserine decreases both D1 and D2 dopamine receptors number and their function in rat brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Cell Membrane; Cycloserine; Dizocilpine Maleate; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; In Vitro Techniques; Kinetics; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone | 1994 |
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1994 |
Pharmacological studies with two new ergoline derivatives, the potential antipsychotics LEK-8829 and LEK-8841.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Antipsychotic Agents; Benzazepines; Blood Pressure; Catalepsy; Clozapine; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Lysergic Acid; Male; Mice; Muscarinic Antagonists; Rats; Serotonin Antagonists; Spiperone | 1994 |
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride | 1994 |
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase | 1993 |
Chronic treatment with MK-801 decreases D2 dopamine receptor function in rat striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Grooming; In Vitro Techniques; Kinetics; Ligands; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone | 1993 |
Continuous treatment with the D2 dopamine receptor agonist quinpirole decreases D2 dopamine receptors, D2 dopamine receptor messenger RNA and proenkephalin messenger RNA, and increases mu opioid receptors in mouse striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Behavior, Animal; Blotting, Northern; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Down-Regulation; Enkephalins; Ergolines; Image Processing, Computer-Assisted; Male; Mice; Nucleic Acid Hybridization; Oligonucleotide Probes; Protein Precursors; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Spiperone; Up-Regulation | 1993 |
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone | 1993 |
Expression and functional characterisation of a synthetic version of the human D4 dopamine receptor in a stable human cell line.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Binding, Competitive; Cell Line; Chlorocebus aethiops; Colforsin; DNA; Ergolines; Genes, Synthetic; Humans; Kidney; Kinetics; Molecular Sequence Data; Plasmids; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; Spiperone; Transfection | 1994 |
5-HT1B receptors mediate potent contractile responses to 5-HT in rat caudal artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arteries; Ergolines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Vasoconstrictor Agents | 1993 |
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide | 1993 |
Expression and characterization of human D4 dopamine receptors in baculovirus-infected insect cells.
Topics: Animals; Baculoviridae; Base Sequence; Cell Line; Ergolines; Genetic Vectors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Introns; Molecular Sequence Data; Moths; Occlusion Body Matrix Proteins; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Fusion Proteins; Spiperone; Viral Proteins; Viral Structural Proteins | 1993 |
Dopamine D2L receptors stimulate Na+/K(+)-ATPase activity in murine LTK- cells.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dideoxyadenosine; Dopamine Agonists; Ergolines; Kinetics; L Cells; Mice; Ouabain; Pertussis Toxin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Rubidium; Sodium-Potassium-Exchanging ATPase; Spiperone; Transfection; Virulence Factors, Bordetella | 1996 |
Modulation of [3H]quinpirole binding in brain by monoamine oxidase inhibitors: evidence for a potential novel binding site.
Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone | 1996 |
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1999 |
Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice.
Topics: Animals; Binding Sites; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Evaluation, Preclinical; Eating; Ergolines; Fenfluramine; Genotype; Injections, Intraperitoneal; Injections, Subcutaneous; Isomerism; Mianserin; Mice; Mice, Knockout; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Satiation; Satiety Response; Serotonin 5-HT2 Receptor Agonists; Species Specificity; Spiperone; Spiro Compounds; Time Factors; Tritium; United Kingdom | 2004 |