Page last updated: 2024-08-16

spiperone and ergoline

spiperone has been researched along with ergoline in 104 studies

Research

Studies (104)

TimeframeStudies, this research(%)All Research%
pre-199054 (51.92)18.7374
1990's49 (47.12)18.2507
2000's1 (0.96)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Battista, AF; Fuxe, K; Goldstein, M; Lew, JY; Lieberman, A; Nakamura, S1
Cote, T; Kebabian, J; Munemura, M1
Battista, AF; Goldstein, M; Lew, JY; Nakamura, S1
Fuller, RW; Snoddy, HD3
Fujita, N; Saito, K; Yonehara, N; Yoshida, H1
Jenner, P; Marsden, CD; Rose, S; Thomas, KL1
Esterle, TM; Sanders-Bush, E1
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD1
Lucki, I; McGonigle, P; Subramaniam, S1
DeSouza, EB; Grigoriadis, DE; Levant, B2
LaHoste, GJ; Marshall, JF1
Kozlowski, MR; Neve, KA; Rosser, MP1
Pawlikowski, M; Pisarek, H; Stepien, H1
Aulakh, CS; Hill, JL; Murphy, DL1
Choudhary, MS; Craigo, S; Roth, BL1
Todd, RD1
Boroni, F; Castelletti, L; Memo, M; Missale, C; Spano, P1
Gong, L; Kostrzewa, RM1
Michel, AD; Nunes, JL; Sharif, NA; Whiting, RL1
Schaus, JM; Seeman, P1
Brus, R; Kalbfleisch, J; Kostrzewa, RM1
Bourque, CW; Renaud, LP; Yang, CR1
Aghajanian, GK; Sheldon, PW1
Courtney, ND; Howlett, AC; Westfall, TC1
Bancroft, C; Dong, KW; McChesney, R; Roberts, JL; Sealfon, SC; Tsutsumi, M1
Hashimoto, T; Katsura, M; Kuriyama, K1
Linseman, MA1
Nowak, JZ; Schorderet, M1
Axel, R; Huang, KN; Jessell, TM; Julius, D; Livelli, TJ1
Gessa, GL; Olianas, MC; Onali, P1
Iuvone, PM1
Beaulieu, M; Felder, R; Kebabian, JW1
Cohen, ML; Kurz, KD; Schenck, KW1
Brazell, C; Dourish, CT; King, BH; Middlemiss, DN1
Doty, RL; Risser, JM1
Segawa, T; Zhang, X1
Allin, R; Reyneke, L; Russell, VA; Taljaard, JJ1
Klimek, V; Maj, J1
Dlabac, A; Dobrovský, K; Krejcí, I; Valchár, M1
Chojnacka-Wójcik, E; Jaros, T; Kłodzińska, A; Maj, J1
Fuller, RW; Hemrick-Luecke, SK; Perry, KW; Toomey, RE1
Arnt, J; Hyttel, J1
Crocker, AD; Faunt, JE2
Battaglia, G; Creese, I; Hess, EJ; Norman, AB1
Kidric, M; Petrović, J; Soskić, V; Trajković, D1
Beart, PM; Bridge, S; Christie, MJ1
Amedro, J; Brown, L; Smith, D; Williams, G1
Ares, J; Chang, YA; Farooqui, T; Miller, D; Uretsky, N; Wallace, L; Wallace, RA1
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW1
Arnt, J; Hyttel, J; Nowak, G1
Burchill, SA; Thody, AJ1
Bondy, SC; Breese, GR; Duncan, GE; Iorio, LC; Mueller, RA; Napier, TC1
Nakagawa, K; Sekihara, S; Somei, M; Watanabe, H; Yamada, F1
Fuller, RW; Hemrick-Luecke, SK1
Dlabac, A; Krejcí, I; Valchár, M; Vrsecká, M1
Anderson, D; Gordon, J; Herbster, G; Koller, W; Wack, R1
Brunello, N; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC1
Bymaster, FP; Kornfeld, EC; Nichols, CL; Reid, LR; Wong, DT1
Arnt, J1
Liskowsky, DR; Potter, LT1
Cohen, ML; Fuller, RW; Garbrecht, WL; Kurz, KD; Marzoni, GP; Mason, NR1
Dow, RC; Hill, AG; McQueen, JK1
Hruska, RE; Silbergeld, EK1
Filburn, CR; Joseph, JA; Roth, GS1
Fuller, RW; Hemrick-Luecke, SK; Perry, KW1
Beart, PM; McDonald, D1
Ferrer, JM; Mora, F; Sanguinetti, AM; Vives, F1
Creese, I; De Lean, A; Sibley, DR1
Beart, PM; Gundlach, AL; Krstich, M1
Koller, WC1
Hruska, RE; Silbergeld, EK; Weir, RL1
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K1
Asano, T; Goldstein, M; Lew, JY; Lieberman, A; Makman, MH; Rosenfeld, MR1
Reynolds, GP; Riederer, P1
Battaglia, G; Titeler, M1
Senogles, SE1
Bancroft, C; Fischberg, DJ1
Barrett, RJ; Caul, WF; Huffman, EM; Jones, JR; Strand, EJ1
Erol, DD; Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD; Smith, LA1
Abarca, J; Bustos, G; Gysling, K; Roth, RH1
Chaouche-Teyara, K; Dabiré, H; Fournier, B; Safar, M1
Katz, JL; Witkin, JM1
Contestabile, A; Dall'Olio, R; Facchinetti, F; Gandolfi, O1
Guo, J; Kostrzewa, FP; Kostrzewa, RM1
Bernard, A; Cavegn, C; Chabert, C; Mills, A1
Dall'Olio, R; Gandolfi, O; Rimondini, R1
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD1
Bole-Vunduk, B; Budihna, MV; Krisch, I; Lavric, B; Ocvirk, A; Pepelnak, M; Sket, D1
Nowak, JZ; Zawilska, JB1
Burnham, P; Louis, JC; Magal, E; Varon, S1
Dall'Olio, R; Gandolfi, O1
Aloyo, VJ; Chen, JF; Weiss, B1
Ball, S; Boyfield, I; Coldwell, MC; Cook, T; Gloger, IS; Herrity, N; McHale, M; Robinson, JH; Winn, FM1
Craig, DA; Martin, GR1
Allard, S; Falardeau, P; Lapointe, S1
Allet, B; Bernard, A; Brandt, E; Cavegn, C; Chabert, C; Chollet, A; Kawashima, E; Mills, A1
Felder, RA; Jose, PA; Walk, SF; Yamaguchi, I1
Cheng, CC; Leonard, NL; Levant, B; Moehlenkamp, JD; Morgan, KA1
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Clifton, PG; Dourish, CT; Kennett, GA; Lee, MD; Somerville, EM1

Reviews

1 review(s) available for spiperone and ergoline

ArticleYear
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates

1990

Other Studies

103 other study(ies) available for spiperone and ergoline

ArticleYear
Dopaminephilic properties of ergot alkaloids.
    Federation proceedings, 1978, Volume: 37, Issue:8

    Topics: Acetonitriles; Animals; Bromocriptine; Corpus Striatum; Ergolines; Ergot Alkaloids; Haplorhini; Humans; Levodopa; Parkinson Disease; Receptors, Dopamine; Spiperone; Substantia Nigra; Synaptosomes; Tremor; Tyrosine 3-Monooxygenase

1978
Lisuride hydrogen maleate: an ergoline with beta-adrenergic antagonist activity.
    European journal of pharmacology, 1979, Nov-16, Volume: 59, Issue:3-4

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding Sites; Cerebellum; Dihydroalprenolol; Ergolines; Isoproterenol; Lisuride; Rabbits; Spiperone

1979
Dopamine agonist potencies of ergolines.
    Communications in psychopharmacology, 1979, Volume: 3, Issue:3

    Topics: Animals; Cattle; Corpus Striatum; Dopamine; Ergolines; Haplorhini; Humans; Neural Pathways; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra; Tegmentum Mesencephali; Tremor

1979
The effects of metergoline and other serotonin receptor antagonists on serum corticosterone in rats.
    Endocrinology, 1979, Volume: 105, Issue:4

    Topics: Animals; Corticosterone; Cyproheptadine; Ergolines; Male; Metergoline; Methysergide; Rats; Serotonin Antagonists; Spiperone; Structure-Activity Relationship

1979
Lisuride inhibits 3H-spiroperidol binding to membranes isolated from striatum.
    Neuropharmacology, 1978, Volume: 17, Issue:12

    Topics: Animals; Butyrophenones; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Ergolines; In Vitro Techniques; Lisuride; Male; Membranes; Rats; Spiperone

1978
Dissociation of the striatal D-2 dopamine receptor from adenylyl cyclase following 6-hydroxydopamine-induced denervation.
    Biochemical pharmacology, 1992, Jul-07, Volume: 44, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Denervation; Dopamine; Ergolines; Female; Homovanillic Acid; Oxidopamine; Prosencephalon; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1992
Serotonin agonists increase transferrin levels via activation of 5-HT1C receptors in choroid plexus epithelium.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: Amino Acid Isomerases; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Choroid Plexus; Cyclosporins; Epithelium; Ergolines; Fibroblasts; Kinetics; Male; Mianserin; Peptidylprolyl Isomerase; Phosphatidylinositols; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA Probes; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Thymidine; Time Factors; Transferrin

1992
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Dec-15, Volume: 89, Issue:24

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone

1992
Effects of chronic treatment with selective agonists on the subtypes of dopamine receptors.
    Brain research, 1992, Feb-07, Volume: 571, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Body Temperature Regulation; Brain; Caudate Nucleus; Dopamine Agents; Drug Interactions; Ergolines; Kinetics; Male; Nucleus Accumbens; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reference Values; Spiperone; Substantia Nigra

1992
Characterization of [3H]quinpirole binding to D2-like dopamine receptors in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Binding Sites; Brain; Culture Techniques; Dopamine Agents; Dopamine Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone

1992
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
    Synapse (New York, N.Y.), 1992, Volume: 12, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium

1992
Dopamine D2 receptor stimulation of Na+/H+ exchange assessed by quantification of extracellular acidification.
    The Journal of biological chemistry, 1992, Dec-25, Volume: 267, Issue:36

    Topics: Amiloride; Animals; Carrier Proteins; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Glioma; Hydrogen-Ion Concentration; Kinetics; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Sodium-Hydrogen Exchangers; Spiperone; Tumor Cells, Cultured

1992
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.
    Endocrine regulations, 1992, Volume: 26, Issue:1

    Topics: Animals; Antiparkinson Agents; Bromocriptine; Diethylstilbestrol; Dose-Response Relationship, Drug; Ergolines; Female; Hyperplasia; Hyperprolactinemia; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Time Factors; Tritium

1992
Effects of various serotonin receptor subtype-selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Corticosterone; Ergolines; Male; Metergoline; Mianserin; Neurosecretory Systems; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1992
Identification of receptor domains that modify ligand binding to 5-hydroxytryptamine2 and 5-hydroxytryptamine1c serotonin receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Base Sequence; Binding, Competitive; Ergolines; Haloperidol; In Vitro Techniques; Ketanserin; Molecular Sequence Data; Oligodeoxyribonucleotides; Receptors, Serotonin; Recombinant Fusion Proteins; Spiperone; Structure-Activity Relationship; Transfection

1992
Neural development is regulated by classical neurotransmitters: dopamine D2 receptor stimulation enhances neurite outgrowth.
    Biological psychiatry, 1992, Apr-15, Volume: 31, Issue:8

    Topics: Animals; Base Sequence; Brain; Cells, Cultured; Cerebral Cortex; Ergolines; Female; Male; Mental Disorders; Models, Biological; Molecular Sequence Data; Nerve Growth Factors; Neurites; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; RNA, Messenger; Salicylamides; Spiperone

1992
Epidermal growth factor induces the functional expression of dopamine receptors in the GH3 cell line.
    Endocrinology, 1991, Volume: 128, Issue:1

    Topics: Animals; Binding, Competitive; Cell Line; Cells, Cultured; Dopamine Agents; Epidermal Growth Factor; Ergolines; Kinetics; Pituitary Gland, Anterior; Pituitary Neoplasms; Potassium; Prolactin; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1991
Supersensitized D1 receptors mediate enhanced oral activity after neonatal 6-OHDA.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Mouth; Movement; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1991
Dopamine D2-receptors mediate hypothermia in mice: ICV and IP effects of agonists and antagonists.
    Neurochemical research, 1991, Volume: 16, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Body Temperature Regulation; Cerebral Ventricles; Domperidone; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1991
Dopamine receptors labelled by [3H]quinpirole.
    European journal of pharmacology, 1991, Oct-02, Volume: 203, Issue:1

    Topics: Animals; Corpus Striatum; Dogs; Dopamine Agents; Dopamine Antagonists; Ergolines; Guanine Nucleotides; Haloperidol; In Vitro Techniques; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1991
Ontogenetic homologous sensitization to the antinociceptive action of quinpirole in rats.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Aging; Analgesics; Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Female; Pain Measurement; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1991
Dopamine D2 receptor activation depolarizes rat supraoptic neurones in hypothalamic explants.
    The Journal of physiology, 1991, Volume: 443

    Topics: Animals; Calcium; Dopamine; Dopamine Agents; Ergolines; Membrane Potentials; Neurons; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Sulpiride; Supraoptic Nucleus

1991
Excitatory responses to serotonin (5-HT) in neurons of the rat piriform cortex: evidence for mediation by 5-HT1C receptors in pyramidal cells and 5-HT2 receptors in interneurons.
    Synapse (New York, N.Y.), 1991, Volume: 9, Issue:3

    Topics: Animals; Electrophysiology; Ergolines; Interneurons; Limbic System; Male; Neurons; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone

1991
Dopaminergic regulation of dopamine release from PC12 cells via a pertussis toxin-sensitive G protein.
    Neuroscience letters, 1991, Jan-28, Volume: 122, Issue:2

    Topics: Adrenal Gland Neoplasms; Animals; Apomorphine; Cell Line; Dopamine; Dopamine Antagonists; Ergolines; GTP-Binding Proteins; Haloperidol; Nicotine; Pertussis Toxin; Pheochromocytoma; Potassium; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Virulence Factors, Bordetella

1991
Either isoform of the dopamine D2 receptor can mediate dopaminergic repression of the rat prolactin promoter.
    Molecular and cellular endocrinology, 1991, Volume: 79, Issue:1-3

    Topics: Animals; Cell Line; Ergolines; Female; Hysterectomy; Ovariectomy; Pituitary Neoplasms; Plasmids; Prolactin; Prolactinoma; Promoter Regions, Genetic; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D1; RNA, Messenger; Signal Transduction; Spiperone; Transcription, Genetic

1991
On the mechanism of mergocryptine-induced suppression of dopamine turnover in the rat striatum.
    European journal of pharmacology, 1991, Jun-06, Volume: 198, Issue:2-3

    Topics: Animals; Apomorphine; Benzazepines; Corpus Striatum; Dopamine; Ergolines; Half-Life; Male; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1991
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
    Psychopharmacology, 1990, Volume: 100, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1990
The 5HT2 receptor defines a family of structurally distinct but functionally conserved serotonin receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1990, Volume: 87, Issue:3

    Topics: Amino Acid Sequence; Animals; Antiparkinson Agents; Brain; DNA; Ergolines; Fibroblasts; Gene Library; Genes; Mice; Molecular Sequence Data; Organ Specificity; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Nucleic Acid; Spiperone; Transfection; Type C Phospholipases

1990
Characterization of dopamine receptors mediating inhibition of adenylate cyclase activity in rat striatum.
    Molecular pharmacology, 1985, Volume: 28, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butaclamol; Corpus Striatum; Dopamine; Enzyme Activation; Ergolines; Guanine Nucleotides; Norepinephrine; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Sulpiride

1985
Evidence for a D2 dopamine receptor in frog retina that decreases cyclic AMP accumulation and serotonin N-acetyltransferase activity.
    Life sciences, 1986, Jan-27, Volume: 38, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Bucladesine; Calcium; Circadian Rhythm; Cyclic AMP; Dopamine; Ergolines; Light; Metoclopramide; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Retina; Spiperone; Xenopus laevis

1986
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1988
MK-212 increases rat plasma ACTH concentration by activation of the 5-HT1C receptor subtype.
    Neuroscience letters, 1989, Oct-23, Volume: 105, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Antiparkinson Agents; Ergolines; Ketanserin; Male; Metergoline; Pindolol; Piperazines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1989
Influence of the D-2 dopamine receptor agonist quinpirole on the odor detection performance of rats before and after spiperone administration.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Acetates; Animals; Behavior, Animal; Conditioning, Operant; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Smell; Spiperone

1989
Selective blockade of dopamine D-1 receptor by SCH 23390 affects dopamine agonist binding to 3H-spiperone labeled D-2 receptors in rat striatum.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Guanosine Triphosphate; In Vitro Techniques; Male; Pertussis Toxin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Virulence Factors, Bordetella

1989
Lack of effect of chronic desipramine treatment on dopaminergic activity in the nucleus accumbens of the rat.
    Neurochemical research, 1989, Volume: 14, Issue:7

    Topics: Acetylcholine; Animals; Benzazepines; Desipramine; Dopamine; Dopamine Agents; Dopamine Antagonists; Electric Stimulation; Ergolines; Male; Nomifensine; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Septal Nuclei; Spiperone

1989
Repeated administration of antidepressants enhances agonist affinity for mesolimbic D2-receptors.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:8

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Binding, Competitive; Ergolines; Imipramine; Limbic System; Male; Mianserin; Motor Activity; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spiperone

1989
Comparison of (3H)-terguride and (3H)-spiperone binding to dopamine receptors in the rat striatum.
    Activitas nervosa superior, 1989, Volume: 31, Issue:1

    Topics: Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Ergolines; Ergotamines; Lisuride; Male; Rats; Receptors, Dopamine; Spiperone

1989
Exploratory hypoactivity induced by m-trifluoromethylphenylpiperazine (TFMPP) and m-chlorophenylpiperazine (m-CPP).
    Journal of neural transmission. Parkinson's disease and dementia section, 1989, Volume: 1, Issue:3

    Topics: Animals; Ergolines; Exploratory Behavior; Male; Metergoline; Mianserin; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1989
Pergolide elevation of MHPG sulphate concentration in rat hypothalamus blocked by spiperone and mimicked by other dopamine agonists.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Butyrophenones; Dopamine; Ergolines; Glycols; Homovanillic Acid; Hypothalamus; Male; Methoxyhydroxyphenylglycol; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
Differential involvement of dopamine D-1 and D-2 receptors in the circling behaviour induced by apomorphine, SK & F 38393, pergolide and LY 171555 in 6-hydroxydopamine-lesioned rats.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Appetite Depressants; Benzazepines; Electric Stimulation; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical; Time Factors

1985
Adrenocortical hormone status affects responses to dopamine receptor agonists.
    European journal of pharmacology, 1988, Aug-02, Volume: 152, Issue:3

    Topics: Adrenal Cortex Hormones; Adrenalectomy; Animals; Apomorphine; Behavior, Animal; Benzazepines; Body Temperature; Corticosterone; Dopamine Agents; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1988
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
    Neuroscience letters, 1985, Aug-30, Volume: 59, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Dopaminergic activity of some ergot alkaloid derivatives: relationship to their chemical structure.
    Pharmacology, 1986, Volume: 32, Issue:3

    Topics: Animals; Cattle; Caudate Nucleus; Dopamine; Ergolines; Ergot Alkaloids; Guanosine Triphosphate; In Vitro Techniques; Molecular Conformation; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Tritium

1986
No change in neostriatal D-2 dopamine receptors after NMDA lesions of rat prefrontal cortex.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:6

    Topics: Animals; Aspartic Acid; Corpus Striatum; Ergolines; Female; Frontal Lobe; Male; N-Methylaspartate; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tritium

1986
The effects of selective dopamine receptor agonists and antagonists on body temperature in rats.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Temperature; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1987
A pharmacological analysis of the rat spinal cord serotonin (5-HT) autoreceptor.
    European journal of pharmacology, 1988, Jan-12, Volume: 145, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Male; Piperazines; Potassium; Quipazine; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Spiperone; Tetrahydronaphthalenes; Tritium

1988
Interaction of permanently uncharged dopamine analogs with the D-2 dopaminergic receptor.
    Biochemical pharmacology, 1988, May-15, Volume: 37, Issue:10

    Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Ergolines; In Vitro Techniques; Male; Mice; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sodium Chloride; Spiperone; Sulfides

1988
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
    Advances in experimental medicine and biology, 1988, Volume: 235

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
    European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone

1988
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
    The Journal of endocrinology, 1986, Volume: 111, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride

1986
6-hydroxydopamine treatments enhance behavioral responses to intracerebral microinjection of D1- and D2-dopamine agonists into nucleus accumbens and striatum without changing dopamine antagonist binding.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Ergolines; Female; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Microinjections; Motor Activity; Nucleus Accumbens; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone

1987
Dopamine receptor stimulating effects of chanoclavine analogues, tricyclic ergot alkaloids, in the brain.
    Japanese journal of pharmacology, 1987, Volume: 45, Issue:4

    Topics: 4-Butyrolactone; Animals; Binding, Competitive; Brain; Catechols; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Ergot Alkaloids; In Vitro Techniques; Male; Mice; Rats; Rats, Inbred Strains; Receptors, Dopamine; Rotation; Spiperone; Stereotyped Behavior; Time Factors

1987
Decrease in hypothalamic epinephrine concentration and other neurochemical changes produced by quinpirole, a dopamine agonist, in rats.
    Journal of neural transmission, 1985, Volume: 61, Issue:3-4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Epinephrine; Ergolines; Homovanillic Acid; Hypothalamus; Male; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Binding characteristics of the dopamine agonist/antagonist [3H]terguride (transdihydrolisuride) in the rat striatum.
    European journal of pharmacology, 1987, Apr-07, Volume: 136, Issue:1

    Topics: Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Kinetics; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1987
Quinpirole hydrochloride, a potential anti-parkinsonism drug.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: Animals; Benzazepines; Corpus Striatum; Dogs; Dose-Response Relationship, Drug; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride

1987
Absence of [3H]SCH 23390 specific binding sites in anterior pituitary: dissociation from effects on prolactin secretion.
    European journal of pharmacology, 1987, Mar-17, Volume: 135, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Corpus Striatum; Cyproheptadine; Ergolines; Kinetics; Male; Metergoline; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1987
Elevation of acetylcholine levels in striatum of rat brain by LY163502, trans-(-)-5,5a,6,7,8,9a,10-octahydro-6-propylpyrimido less than 4,5-g greater than quinolin-2-amine dihydrochloride, a potent and stereospecific dopamine (D2) agonist.
    Life sciences, 1986, Jan-27, Volume: 38, Issue:4

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Apomorphine; Clonidine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Ergolines; Pergolide; Quinolines; Rats; Receptors, Dopamine; Spiperone

1986
Hyperactivity induced by stimulation of separate dopamine D-1 and D-2 receptors in rats with bilateral 6-OHDA lesions.
    Life sciences, 1985, Aug-26, Volume: 37, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Benzazepines; Clopenthixol; Dopamine; Dose-Response Relationship, Drug; Ergolines; Flupenthixol; Hydroxydopamines; Hypothalamus; Male; Motor Activity; Oxidopamine; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
D-2 dopamine receptors in the frontal cortex of rat and human.
    Life sciences, 1985, Apr-22, Volume: 36, Issue:16

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Cinanserin; Dopamine; Ergolines; Humans; Kinetics; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
Pharmacological activity of the isomers of LY53857, potent and selective 5-HT2 receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Blood Pressure; Cerebral Cortex; Corticosterone; Decerebrate State; Ergolines; Isomerism; Male; Mathematics; Quipazine; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Time Factors

1985
Proceedings: Effects of some dopamine receptor stimulants on cobalt-induced epilepsy in the rat.
    British journal of pharmacology, 1974, Volume: 52, Issue:1

    Topics: Amphetamine; Animals; Apomorphine; Cobalt; Dopamine; Electroencephalography; Epilepsy; Ergolines; Male; Rats; Receptors, Adrenergic; Spiperone; Stimulation, Chemical

1974
Inhibition of neurotransmitter receptor binding by ergot derivatives.
    Journal of neuroscience research, 1981, Volume: 6, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Bromocriptine; Dioxanes; Ergolines; Ergot Alkaloids; gamma-Aminobutyric Acid; Lysergic Acid Diethylamide; Male; Metergoline; Organ Specificity; Quinuclidinyl Benzilate; Rats; Receptors, Neurotransmitter; Serotonin; Spiperone; Structure-Activity Relationship; Synapses

1981
Development of dopamine receptor denervation supersensitivity in the neostriatum of the senescent rat.
    Life sciences, 1981, Aug-10, Volume: 29, Issue:6

    Topics: Adenylyl Cyclases; Aging; Animals; Corpus Striatum; Dextroamphetamine; Ergolines; Female; Male; Motor Activity; Rats; Receptors, Dopamine; Rotation; Sex Factors; Spiperone

1981
Elevation of serum corticosterone concentrations in rats by pergolide and other dopamine agonists.
    Endocrinology, 1981, Volume: 109, Issue:4

    Topics: Animals; Antiparkinson Agents; Corticosterone; Domperidone; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Metergoline; Mianserin; Pergolide; Rats; Rats, Inbred Strains; Spiperone

1981
Depletion of epinephrine in rat hypothalamus by a dopamine agonist, pergolide.
    Neurochemical research, 1982, Volume: 7, Issue:4

    Topics: Animals; Antiparkinson Agents; Dopamine Antagonists; Epinephrine; Ergolines; Haloperidol; Hypothalamus; Kinetics; Male; Pergolide; Rats; Rats, Inbred Strains; Spiperone

1982
Neurochemical studies of the mesolimbic dopaminergic pathway: [3H]spiperone labels two bindings sites in homogenates of the nucleus accumbens of rat brain.
    Journal of neurochemistry, 1982, Volume: 39, Issue:5

    Topics: Animals; Antipsychotic Agents; Apomorphine; Butyrophenones; Dopamine; Ergolines; Kinetics; Nucleus Accumbens; Rats; Receptors, Dopamine; Septal Nuclei; Spiperone

1982
Serum corticosterone elevation by pergolide in rats: prevention of tolerance development by spiperone.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:9

    Topics: Animals; Butyrophenones; Corticosterone; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Ergolines; Male; Pergolide; Rats; Rats, Inbred Strains; Spiperone

1982
Effects of agonists and antagonists of D1 and D2 dopamine receptors on self-stimulation of the medial prefrontal cortex in the rat.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Animals; Apomorphine; Bromocriptine; Cerebral Cortex; Dose-Response Relationship, Drug; Ergolines; Functional Laterality; Male; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Self Stimulation; Spiperone; Sulpiride; Synaptic Transmission

1983
Anterior pituitary dopamine receptors. Demonstration of interconvertible high and low affinity states of the D-2 dopamine receptor.
    The Journal of biological chemistry, 1982, Jun-10, Volume: 257, Issue:11

    Topics: Animals; Binding, Competitive; Butaclamol; Cattle; Cell Membrane; Computers; Ergolines; Guanylyl Imidodiphosphate; Kinetics; Pergolide; Pituitary Gland, Anterior; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1982
Guanine nucleotides reveal differential actions of ergot derivatives at D-2 receptors labelled by [3H]spiperone in striatal homogenates.
    Brain research, 1983, Nov-14, Volume: 278, Issue:1-2

    Topics: Animals; Binding, Competitive; Butyrophenones; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Guanine Nucleotides; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Tritium

1983
Attenuation by pergolide of haloperidol-induced striatal dopamine receptor density.
    Journal of clinical psychopharmacology, 1984, Volume: 4, Issue:6

    Topics: Animals; Corpus Striatum; Ergolines; Guinea Pigs; Haloperidol; Male; Membranes; Pergolide; Receptors, Dopamine; Spiperone

1984
Binding of antiparkinsonian ergot derivatives to the dopamine receptor.
    Psychopharmacology, 1981, Volume: 75, Issue:2

    Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Caudate Nucleus; Ergolines; Lisuride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1981
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
    Acta physiologica Scandinavica, 1983, Volume: 117, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
Interaction of pergolide with central dopaminergic receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:6

    Topics: Adenylyl Cyclases; Animals; Behavior, Animal; Binding, Competitive; Cattle; Cerebral Decortication; Chlorocebus aethiops; Corpus Striatum; Ergolines; Guanosine Triphosphate; Hot Temperature; Male; Pergolide; Rats; Receptors, Dopamine; Spiperone; Tegmentum Mesencephali; Tremor

1980
The effects of lisuride and some other dopaminergic agonists on receptor binding in human brain.
    Journal of neural transmission, 1981, Volume: 51, Issue:1-2

    Topics: Brain; Bromocriptine; Ergolines; Humans; Kinetics; Lisuride; Receptors, Dopamine; Spiperone

1981
Direct binding of 3H-lisuride to adrenergic and serotonergic receptors.
    Life sciences, 1981, Aug-31, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Ergolines; Haloperidol; In Vitro Techniques; Kinetics; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Spiperone

1981
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
    Endocrinology, 1994, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1994
The D2 receptor: blocked transcription in GH3 cells and cellular pathways employed by D2A to regulate prolactin promoter activity.
    Molecular and cellular endocrinology, 1995, Volume: 111, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Cell Line; Chloramphenicol O-Acetyltransferase; DNA-Binding Proteins; Ergolines; Gene Expression Regulation; Pertussis Toxin; Pituitary Gland; Prolactin; Promoter Regions, Genetic; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Spiperone; Thyrotropin-Releasing Hormone; Transcription Factor Pit-1; Transcription Factors; Transcription, Genetic; Transfection; Virulence Factors, Bordetella

1995
D2-specific discriminative stimuli: parameters, blocking, and rebound.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 51, Issue:1

    Topics: Animals; Cues; Discrimination, Psychological; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Food Deprivation; Haloperidol; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Spiperone

1995
Differential anti-parkinsonian effects of benzazepine D1 dopamine agonists with varying efficacies in the MPTP-treated common marmoset.
    Psychopharmacology, 1995, Volume: 117, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antiparkinson Agents; Behavior, Animal; Benzazepines; Binding, Competitive; Callithrix; Dopamine Agonists; Ergolines; In Vitro Techniques; Male; Parkinson Disease, Secondary; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1995
Changes in extracellular levels of glutamate and aspartate in rat substantia nigra induced by dopamine receptor ligands: in vivo microdialysis studies.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aspartic Acid; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Extracellular Space; Glutamic Acid; Kinetics; Ligands; Male; Microdialysis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Substantia Nigra; Tetrodotoxin; Time Factors

1995
Systemic and regional haemodynamic effects of 1-(2,5-dimethoxy-4-iodo-phenyl)-2-aminopropane (DOI) and alpha-methyl-5-HT, in the anaesthetised rat.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 1994, Volume: 16, Issue:6

    Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Ergolines; Hemodynamics; Injections, Intravenous; Injections, Intraventricular; Male; Rats; Rats, Wistar; Regional Blood Flow; Renal Circulation; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Splanchnic Circulation

1994
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
    Psychopharmacology, 1993, Volume: 113, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone

1993
Chronic neonatal blockade of N-methyl-D-aspartate receptor by CGP 39551 increases dopaminergic function in adult rat.
    Neuroscience, 1994, Volume: 63, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Apomorphine; Behavior, Animal; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Motor Activity; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; Spiperone; Stereotyped Behavior; Time Factors

1994
Ontogenetic quinpirole treatment induces vertical jumping activity in rats.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Injections, Intraperitoneal; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1993
Characterization of the functional activity of dopamine ligands at human recombinant dopamine D4 receptors.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: Animals; Cell Line; Clozapine; DNA; Dopamine; Dopamine Agents; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Ligands; Moths; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Sulfur Radioisotopes; Tritium

1994
D-cycloserine decreases both D1 and D2 dopamine receptors number and their function in rat brain.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Cell Membrane; Cycloserine; Dizocilpine Maleate; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; In Vitro Techniques; Kinetics; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1994
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
    Neuropharmacology, 1994, Volume: 33, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Pharmacological studies with two new ergoline derivatives, the potential antipsychotics LEK-8829 and LEK-8841.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Antipsychotic Agents; Benzazepines; Blood Pressure; Catalepsy; Clozapine; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Lysergic Acid; Male; Mice; Muscarinic Antagonists; Rats; Serotonin Antagonists; Spiperone

1994
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
    Neuroscience, 1993, Volume: 52, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase

1993
Chronic treatment with MK-801 decreases D2 dopamine receptor function in rat striatum.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Grooming; In Vitro Techniques; Kinetics; Ligands; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone

1993
Continuous treatment with the D2 dopamine receptor agonist quinpirole decreases D2 dopamine receptors, D2 dopamine receptor messenger RNA and proenkephalin messenger RNA, and increases mu opioid receptors in mouse striatum.
    Neuroscience, 1993, Volume: 54, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Behavior, Animal; Blotting, Northern; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Down-Regulation; Enkephalins; Ergolines; Image Processing, Computer-Assisted; Male; Mice; Nucleic Acid Hybridization; Oligonucleotide Probes; Protein Precursors; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Spiperone; Up-Regulation

1993
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone

1993
Expression and functional characterisation of a synthetic version of the human D4 dopamine receptor in a stable human cell line.
    FEBS letters, 1994, May-30, Volume: 345, Issue:2-3

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Binding, Competitive; Cell Line; Chlorocebus aethiops; Colforsin; DNA; Ergolines; Genes, Synthetic; Humans; Kidney; Kinetics; Molecular Sequence Data; Plasmids; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; Spiperone; Transfection

1994
5-HT1B receptors mediate potent contractile responses to 5-HT in rat caudal artery.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arteries; Ergolines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Vasoconstrictor Agents

1993
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
    Biochemical and biophysical research communications, 1993, Jun-15, Volume: 193, Issue:2

    Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1993
Expression and characterization of human D4 dopamine receptors in baculovirus-infected insect cells.
    FEBS letters, 1993, Apr-05, Volume: 320, Issue:2

    Topics: Animals; Baculoviridae; Base Sequence; Cell Line; Ergolines; Genetic Vectors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Introns; Molecular Sequence Data; Moths; Occlusion Body Matrix Proteins; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Fusion Proteins; Spiperone; Viral Proteins; Viral Structural Proteins

1993
Dopamine D2L receptors stimulate Na+/K(+)-ATPase activity in murine LTK- cells.
    Molecular pharmacology, 1996, Volume: 49, Issue:2

    Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dideoxyadenosine; Dopamine Agonists; Ergolines; Kinetics; L Cells; Mice; Ouabain; Pertussis Toxin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Rubidium; Sodium-Potassium-Exchanging ATPase; Spiperone; Transfection; Virulence Factors, Bordetella

1996
Modulation of [3H]quinpirole binding in brain by monoamine oxidase inhibitors: evidence for a potential novel binding site.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone

1996
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice.
    Psychopharmacology, 2004, Volume: 176, Issue:1

    Topics: Animals; Binding Sites; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Evaluation, Preclinical; Eating; Ergolines; Fenfluramine; Genotype; Injections, Intraperitoneal; Injections, Subcutaneous; Isomerism; Mianserin; Mice; Mice, Knockout; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Satiation; Satiety Response; Serotonin 5-HT2 Receptor Agonists; Species Specificity; Spiperone; Spiro Compounds; Time Factors; Tritium; United Kingdom

2004