Page last updated: 2024-08-16

spiperone and eedq

spiperone has been researched along with eedq in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-199010 (50.00)18.7374
1990's9 (45.00)18.2507
2000's0 (0.00)29.6817
2010's1 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Black, LE; Creese, I; Hatada, Y; Sibley, DR; Xu, SX1
Di Paolo, T; Lévesque, D1
Ekman, A; Eriksson, E1
Bolaños, FJ; Gozlan, H; Hamon, M; Laporte, AM; Schechter, LE1
Agnati, LF; Cimino, M; Farabegoli, C; Fuxe, K; Merlo Pich, E1
Battaglia, G; Creese, I; Norman, AB1
Henry, JM; Joseph, JA; Kochman, K; Roth, GS1
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW1
Cameron, DL; Crocker, AD1
Arnt, J; Hyttel, J; Nowak, G1
Loeschen, S; Marshall, JF; Neve, KA1
Agnati, LF; Benfenati, F; Fuxe, K; Goldstein, M; Meller, E1
Creese, I; Hamblin, MW1
Henry, JM; Roth, GS1
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD1
Bardo, MT; Crawford, CA; McDougall, SA; Rowlett, JK1
Burger, LY; Martin-Iverson, MT1
Baldessarini, RJ; Kula, NS; Neumeyer, JL; Tarazi, FI; Zhang, K1
Baldessarini, RJ; Kula, NS; Tarazi, FI; Weiss, NT; Zhang, K1

Other Studies

20 other study(ies) available for spiperone and eedq

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
N-(p-isothiocyanatophenethyl)spiperone, a selective and irreversible antagonist of D2 dopamine receptors in brain.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Cells, Cultured; Dopamine Antagonists; Injections, Subcutaneous; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1991
Dopamine receptor reappearance after irreversible receptor blockade: effect of chronic estradiol treatment of ovariectomized rats.
    Molecular pharmacology, 1991, Volume: 39, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Dopamine Antagonists; Drug Administration Schedule; Estradiol; Female; Ovariectomy; Pituitary Gland, Anterior; Prolactin; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1991
Pituitary and brain D2 receptor density measured in vitro and in vivo in EEDQ treated male rats.
    Life sciences, 1991, Volume: 48, Issue:4

    Topics: 4-Butyrolactone; Animals; Brain; Cell Membrane; Corpus Striatum; Kinetics; Limbic System; Male; Pituitary Gland; Quinolines; Raclopride; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Tritium

1991
Recovery of 5-HT 1A receptors after irreversible blockade by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
    Proceedings of the Western Pharmacology Society, 1991, Volume: 34

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alkylating Agents; Animals; Autoradiography; Brain; Hippocampus; Quinolines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1991
Chronic uridine treatment reduces the level of [3H]spiperone-labelled dopamine receptors and enhances their turnover rate in striatum of young rats: relationship to dopamine-dependent behaviours.
    Acta physiologica Scandinavica, 1988, Volume: 132, Issue:2

    Topics: Adrenergic alpha-Antagonists; Age Factors; Animals; Catalepsy; Corpus Striatum; Male; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Uridine

1988
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:5

    Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone

1987
Effect of aging on striatal dopamine receptor subtype recovery following N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline blockade and relation to motor function in Wistar rats.
    Brain research, 1987, Aug-25, Volume: 418, Issue:2

    Topics: Aging; Animals; Corpus Striatum; Male; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Thioxanthenes

1987
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
    Advances in experimental medicine and biology, 1988, Volume: 235

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
Alkylation of striatal dopamine receptors abolishes stereotyped behavior but has no effect on dopamine stimulated adenylate cyclase activity.
    Neuroscience letters, 1988, Jul-19, Volume: 90, Issue:1-2

    Topics: Adenylyl Cyclases; Alkylating Agents; Animals; Apomorphine; Benzazepines; Corpus Striatum; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1988
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
    European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone

1988
Denervation accelerates the reappearance of neostriatal D-2 receptors after irreversible receptor blockade.
    Brain research, 1985, Mar-11, Volume: 329, Issue:1-2

    Topics: Animals; Corpus Striatum; Dopamine; Hydroxydopamines; Male; Oxidopamine; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Analysis of [3H]spiperone binding sites in the rat striatum and frontoparietal cortex by means of quantitative receptor autoradiography after inactivation of dopamine receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo: selective protectio
    Neuroscience letters, 1986, Feb-28, Volume: 64, Issue:2

    Topics: Animals; Autoradiography; Butyrophenones; Cerebral Cortex; Corpus Striatum; Male; Quinolines; Rats; Receptors, Dopamine; Spiperone; Sulpiride

1986
Behavioral and radioligand binding evidence for irreversible dopamine receptor blockade by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline.
    Life sciences, 1983, May-09, Volume: 32, Issue:19

    Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Catalepsy; Dose-Response Relationship, Drug; Humans; Injections, Intraperitoneal; Male; Quinolines; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors

1983
Effect of aging on recovery of striatal dopamine receptors following N-ethoxycarbonyl-2-ethoxy-1, 2-dihydroquinoline (EEDQ) blockade.
    Life sciences, 1984, Aug-20, Volume: 35, Issue:8

    Topics: Aging; Animals; Corpus Striatum; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1984
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
    Neuropharmacology, 1994, Volume: 33, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Age-dependent differences in the rate of recovery of striatal dopamine D1 and D2 receptors after inactivation with EEDQ.
    European journal of pharmacology, 1994, Feb-03, Volume: 252, Issue:2

    Topics: Aging; Animals; Behavior, Animal; Benzazepines; Dopamine D2 Receptor Antagonists; Female; Injections, Intraperitoneal; Male; Neostriatum; Nerve Tissue Proteins; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Increased occupation of D1 and D2 dopamine receptors accompanies cocaine-induced behavioral sensitization.
    Brain research, 1994, Mar-14, Volume: 639, Issue:2

    Topics: Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine D2 Receptor Antagonists; Male; Motor Activity; Neostriatum; Nimodipine; Nucleus Accumbens; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Selective alkylatation of dopamine D2 and D4 receptors in rat brain by N-(p-isothiocyanatophenethyl)spiperone.
    Neuroscience letters, 1999, Oct-29, Volume: 274, Issue:3

    Topics: Alkylation; Animals; Autoradiography; Brain Chemistry; Dopamine Antagonists; Male; Neostriatum; Nucleus Accumbens; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Serotonin; Spiperone

1999
Effects of alkylating agents on dopamine D(3) receptors in rat brain: selective protection by dopamine.
    Brain research, 1999, Nov-13, Volume: 847, Issue:1

    Topics: Alkylating Agents; Animals; Brain; Dopamine; Dopamine Antagonists; Male; Neuroprotective Agents; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone

1999