spiperone has been researched along with eedq in 20 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (50.00) | 18.7374 |
1990's | 9 (45.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (5.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Black, LE; Creese, I; Hatada, Y; Sibley, DR; Xu, SX | 1 |
Di Paolo, T; Lévesque, D | 1 |
Ekman, A; Eriksson, E | 1 |
Bolaños, FJ; Gozlan, H; Hamon, M; Laporte, AM; Schechter, LE | 1 |
Agnati, LF; Cimino, M; Farabegoli, C; Fuxe, K; Merlo Pich, E | 1 |
Battaglia, G; Creese, I; Norman, AB | 1 |
Henry, JM; Joseph, JA; Kochman, K; Roth, GS | 1 |
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW | 1 |
Cameron, DL; Crocker, AD | 1 |
Arnt, J; Hyttel, J; Nowak, G | 1 |
Loeschen, S; Marshall, JF; Neve, KA | 1 |
Agnati, LF; Benfenati, F; Fuxe, K; Goldstein, M; Meller, E | 1 |
Creese, I; Hamblin, MW | 1 |
Henry, JM; Roth, GS | 1 |
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD | 1 |
Bardo, MT; Crawford, CA; McDougall, SA; Rowlett, JK | 1 |
Burger, LY; Martin-Iverson, MT | 1 |
Baldessarini, RJ; Kula, NS; Neumeyer, JL; Tarazi, FI; Zhang, K | 1 |
Baldessarini, RJ; Kula, NS; Tarazi, FI; Weiss, NT; Zhang, K | 1 |
20 other study(ies) available for spiperone and eedq
Article | Year |
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Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
N-(p-isothiocyanatophenethyl)spiperone, a selective and irreversible antagonist of D2 dopamine receptors in brain.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Cells, Cultured; Dopamine Antagonists; Injections, Subcutaneous; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1991 |
Dopamine receptor reappearance after irreversible receptor blockade: effect of chronic estradiol treatment of ovariectomized rats.
Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Dopamine Antagonists; Drug Administration Schedule; Estradiol; Female; Ovariectomy; Pituitary Gland, Anterior; Prolactin; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1991 |
Pituitary and brain D2 receptor density measured in vitro and in vivo in EEDQ treated male rats.
Topics: 4-Butyrolactone; Animals; Brain; Cell Membrane; Corpus Striatum; Kinetics; Limbic System; Male; Pituitary Gland; Quinolines; Raclopride; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Tritium | 1991 |
Recovery of 5-HT 1A receptors after irreversible blockade by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alkylating Agents; Animals; Autoradiography; Brain; Hippocampus; Quinolines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1991 |
Chronic uridine treatment reduces the level of [3H]spiperone-labelled dopamine receptors and enhances their turnover rate in striatum of young rats: relationship to dopamine-dependent behaviours.
Topics: Adrenergic alpha-Antagonists; Age Factors; Animals; Catalepsy; Corpus Striatum; Male; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Uridine | 1988 |
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone | 1987 |
Effect of aging on striatal dopamine receptor subtype recovery following N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline blockade and relation to motor function in Wistar rats.
Topics: Aging; Animals; Corpus Striatum; Male; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Thioxanthenes | 1987 |
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior | 1988 |
Alkylation of striatal dopamine receptors abolishes stereotyped behavior but has no effect on dopamine stimulated adenylate cyclase activity.
Topics: Adenylyl Cyclases; Alkylating Agents; Animals; Apomorphine; Benzazepines; Corpus Striatum; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1988 |
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone | 1988 |
Denervation accelerates the reappearance of neostriatal D-2 receptors after irreversible receptor blockade.
Topics: Animals; Corpus Striatum; Dopamine; Hydroxydopamines; Male; Oxidopamine; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Analysis of [3H]spiperone binding sites in the rat striatum and frontoparietal cortex by means of quantitative receptor autoradiography after inactivation of dopamine receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo: selective protectio
Topics: Animals; Autoradiography; Butyrophenones; Cerebral Cortex; Corpus Striatum; Male; Quinolines; Rats; Receptors, Dopamine; Spiperone; Sulpiride | 1986 |
Behavioral and radioligand binding evidence for irreversible dopamine receptor blockade by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline.
Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Catalepsy; Dose-Response Relationship, Drug; Humans; Injections, Intraperitoneal; Male; Quinolines; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors | 1983 |
Effect of aging on recovery of striatal dopamine receptors following N-ethoxycarbonyl-2-ethoxy-1, 2-dihydroquinoline (EEDQ) blockade.
Topics: Aging; Animals; Corpus Striatum; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1984 |
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1994 |
Age-dependent differences in the rate of recovery of striatal dopamine D1 and D2 receptors after inactivation with EEDQ.
Topics: Aging; Animals; Behavior, Animal; Benzazepines; Dopamine D2 Receptor Antagonists; Female; Injections, Intraperitoneal; Male; Neostriatum; Nerve Tissue Proteins; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1994 |
Increased occupation of D1 and D2 dopamine receptors accompanies cocaine-induced behavioral sensitization.
Topics: Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine D2 Receptor Antagonists; Male; Motor Activity; Neostriatum; Nimodipine; Nucleus Accumbens; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1994 |
Selective alkylatation of dopamine D2 and D4 receptors in rat brain by N-(p-isothiocyanatophenethyl)spiperone.
Topics: Alkylation; Animals; Autoradiography; Brain Chemistry; Dopamine Antagonists; Male; Neostriatum; Nucleus Accumbens; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Serotonin; Spiperone | 1999 |
Effects of alkylating agents on dopamine D(3) receptors in rat brain: selective protection by dopamine.
Topics: Alkylating Agents; Animals; Brain; Dopamine; Dopamine Antagonists; Male; Neuroprotective Agents; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone | 1999 |