Page last updated: 2024-08-16

spiperone and diazepam

spiperone has been researched along with diazepam in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-199013 (72.22)18.7374
1990's1 (5.56)18.2507
2000's2 (11.11)29.6817
2010's2 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Artursson, P; Mateus, A; Matsson, P1
Enna, SJ; Möhler, H; Okada, T1
Carlson, KR; Eibergen, RD2
Engel, JA; Hulthe, P; Johannessen, K; Söderpalm, B; Svensson, L1
Alleva, FR; Balazs, T; Seth, PK; Takagi, S; Yen-Koo, HC1
Laduron, PM; Luabeya, MK; Maloteaux, JM1
Biggio, G; Concas, A; Corda, MG; Corongiu, FP; Guarneri, P; Rossetti, Z1
Braestrup, C; Divac, I; Nielsen, M1
Britton, DR1
Gardner, CR; Huot-Olivier, S; Klein, J; Mallorga, P; Palfreyman, MG1
Flohé, L; Hennies, HH; Hess, V1
Anderson, D; Deering, J; Henn, FA1
Atack, JR; Bromidge, FA; Dawson, GR; Newman, RJ; O'Meara, GF; Reynolds, DS; Rosahl, TW; Whiting, PJ1
Avakyan, GN; Borlikova, GG; Burd, SG; Garibova, TL; Petrichenko, OB; Proskuryakova, TV; Voronina, TA1

Other Studies

18 other study(ies) available for spiperone and diazepam

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
Benzodiasepine and neurotransmitter receptor binding in rat brain after chronic administration of diazepam or phenobarbital.
    Brain research, 1978, Nov-10, Volume: 156, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Dopamine; gamma-Aminobutyric Acid; Neurotransmitter Agents; Phenobarbital; Quinuclidines; Rats; Receptors, Dopamine; Receptors, Drug; Receptors, Neurotransmitter; Spiperone

1978
Dyskinesias in monkeys: interaction of methamphetamine with prior methadone treatment.
    Pharmacology, biochemistry, and behavior, 1976, Volume: 5, Issue:2

    Topics: Animals; Chlorpromazine; Clozapine; Diazepam; Dyskinesia, Drug-Induced; Haloperidol; Haplorhini; Humans; Macaca mulatta; Male; Methadone; Methamphetamine; Naloxone; Phenobarbital; Phentolamine; Physostigmine; Spiperone; Stereotyped Behavior

1976
Susceptibility to amphetamine-elicited dyskinesias following chronic methadone treatment in monkeys.
    Annals of the New York Academy of Sciences, 1976, Volume: 281

    Topics: Animals; Chlorpromazine; Clozapine; Diazepam; Drug Interactions; Dyskinesia, Drug-Induced; Haloperidol; Haplorhini; Macaca mulatta; Male; Methadone; Methamphetamine; Phenobarbital; Phentolamine; Physostigmine; Spiperone; Time Factors

1976
Evidence for a role for dopamine in the diazepam locomotor stimulating effect.
    Psychopharmacology, 1991, Volume: 104, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Benzazepines; Diazepam; Dopamine; Flumazenil; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Spiperone; Stimulation, Chemical; Tyrosine 3-Monooxygenase

1991
Brain neurotransmitter receptor alterations in offspring of rats exposed to phenobarbital, phenytoin or their combination during pregnancy.
    Neurotoxicology, 1987,Spring, Volume: 8, Issue:1

    Topics: Animals; Brain; Cerebral Cortex; Corpus Striatum; Diazepam; Female; Fetus; Kinetics; Male; Phenobarbital; Phenytoin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Serotonin; Spiperone

1987
Regional and cortical laminar distributions of serotonin S2, benzodiazepine, muscarinic, and dopamine D2 receptors in human brain.
    Journal of neurochemistry, 1984, Volume: 43, Issue:4

    Topics: Adult; Aged; Brain; Cerebral Cortex; Diazepam; Humans; Ketanserin; Male; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Serotonin; Spiperone; Tissue Distribution

1984
Methyl mercury enhances [3H]diazepam binding in different areas of the rat brain.
    Brain research, 1981, Dec-14, Volume: 229, Issue:1

    Topics: Animals; Brain; Diazepam; gamma-Aminobutyric Acid; Male; Methylmercury Compounds; Muscimol; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Retina; Spiperone

1981
Spiroperidol, naloxone, diazepam and QNB binding in the monkey cerebral cortex.
    Brain research bulletin, 1981, Volume: 7, Issue:5

    Topics: Animals; Butyrophenones; Cerebral Cortex; Chlorocebus aethiops; Diazepam; Female; Male; Naloxone; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Dopamine; Receptors, Drug; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Spiperone

1981
A convergent approach to the pharmacology of tetrahydroisoquinolines.
    Progress in clinical and biological research, 1982, Volume: 90

    Topics: Animals; Diazepam; Hypothalamus; Isoquinolines; Kinetics; Naloxone; Receptors, Dopamine; Receptors, Opioid; Salsoline Alkaloids; Spiperone; Tetrahydroisoquinolines; Tetrahydropapaveroline

1982
Chronic elevation of brain GABA by gamma-vinyl GABA treatment does not alter the sensitivity of GABAergic or dopaminergic receptors in rat CNS.
    Psychopharmacology, 1983, Volume: 79, Issue:2-3

    Topics: Adenylyl Cyclases; Aminocaproates; Animals; Brain Chemistry; Diazepam; gamma-Aminobutyric Acid; Male; Motor Activity; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Spiperone; Vigabatrin

1983
Antagonism by supidimide of haloperidol-induced augmentation of [3H]-spiperone binding in rat striatum.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:11

    Topics: Animals; Butyrophenones; Corpus Striatum; Diazepam; Haloperidol; Kinetics; Male; Membranes; Phenobarbital; Rats; Rats, Inbred Strains; Spiperone; Thalidomide

1984
Receptor studies on isolated astroglial cell fractions prepared with and without trypsin.
    Neurochemical research, 1980, Volume: 5, Issue:4

    Topics: Animals; Astrocytes; Brain; Brain Chemistry; Cell Separation; Diazepam; Methods; Rats; Receptors, Dopamine; Receptors, Drug; Spiperone; Subcellular Fractions; Trypsin

1980
GABA(A) alpha 1 subunit knock-out mice do not show a hyperlocomotor response following amphetamine or cocaine treatment.
    Neuropharmacology, 2003, Volume: 44, Issue:2

    Topics: Amphetamine; Animals; Benzazepines; Binding, Competitive; Central Nervous System Stimulants; Cocaine; Diazepam; Dizocilpine Maleate; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Modulators; Habituation, Psychophysiologic; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Protein Subunits; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Spiperone

2003
Effect of nooglutil on benzodiazepine withdrawal syndrome and binding of 3H-spiperone with D2 receptors in rat striatum.
    Bulletin of experimental biology and medicine, 2002, Volume: 134, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Corpus Striatum; Diazepam; Glutamates; In Vitro Techniques; Kinetics; Male; Nicotinic Acids; Nootropic Agents; Rats; Receptors, AMPA; Receptors, Dopamine D2; Spiperone; Substance Withdrawal Syndrome

2002