Page last updated: 2024-08-16

spiperone and cocaine

spiperone has been researched along with cocaine in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-199015 (32.61)18.7374
1990's22 (47.83)18.2507
2000's7 (15.22)29.6817
2010's2 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Brouillette, WJ; Brown, GB; Zha, C1
Dismukes, K; Mulder, AH1
Colpaert, FC; Janssen, PA; Niemegeers, CJ1
Fagan, JD; Ho, BT; Taylor, DL1
Heffner, TG; Stricker, EM; Zigmond, MJ2
Farfel, GM; Kleven, MS; Perry, BD; Seiden, LS; Woolverton, WL1
Byrd, LD; Howell, LL1
Coleman-Hardee, M; Millard, WJ; Peris, J1
Coen, KM; Corrigall, WA2
Hubner, CB; Moreton, JE1
Gessa, GL; Kuzmin, A; Pani, L; Rossetti, ZL; Stefanini, E1
Ali, SF; Frambes, NA; Scalzo, FM; Spear, LP1
George, FR; Ritz, MC1
Alpert, R; Bendriem, B; Christman, D; Dewey, SL; Fowler, JS; Logan, J; Schlyer, D; Shiue, CY; Volkow, ND; Wolf, AP1
Frenken, M1
Fung, YK; Lau, YS; Reed, JA1
Pan, ZZ; Williams, JT1
Langer, SZ; Pimoule, C; Reynolds, GP; Schoemaker, H1
Creese, I; Koob, GF; Le, HT1
Dwoskin, LP; Peris, J; Philpott, K; Yasuda, RP; Zahniser, NR1
Lajtha, A; Reith, ME; Sershen, H1
Hashim, A; Lajtha, A; Reith, ME; Sershen, H1
Hanbauer, I; Memo, M; Pradhan, S1
Pecins-Thompson, M; Peris, J1
Cooper, DC; Graybiel, AM; Hu, XT; Moratalla, R; Tonegawa, S; White, FJ; Xu, M1
De Souza, EB; Griffiths, JW; Katz, JL; Sharpe, LG; Witkin, JM1
Dewey, SL; Fowler, JS; Hitzemann, R; Logan, J; Schlyer, DJ; Volkow, ND; Wang, GJ; Wolf, AP1
Burger, LY; Martin-Iverson, MT1
Gatley, SJ1
Futatsubashi, M; Kakiuchi, T; Kreek, MJ; Kreuter, J; Maggos, CE; Nishiyama, S; Tsukada, H; Unterwald, EM1
Ali, SF; Benson, KA; Wilson, MC1
Fujita, M; Ito, Y; Kusuoka, H; Nishimura, T; Okada, T; Watanabe, Y1
Ho, A; Kakiuchi, T; Kreek, MJ; Kreuter, J; Maggos, CE; Myers, JE; Nishiyama, S; Schlussman, SD; Tsukada, H; Unterwald, EM1
Gee, A; Hosoi, R; Inoue, O; Kobayashi, K1
Chang, YH; Liao, RM; Wang, SH1
Huber, J; Kolta, MG; Park, K; Samaan, SS; Soliman, KF; Stino, FK1
Araujo, DM; Cherry, SR; Kornblum, HI; Tatsukawa, KJ; Toyokuni, T1
Atack, JR; Bromidge, FA; Dawson, GR; Newman, RJ; O'Meara, GF; Reynolds, DS; Rosahl, TW; Whiting, PJ1
Aguiar, LM; Correia, EE; Macêdo, DS; Sousa, FC; Vasconcelos, SM; Viana, GS1
Childers, SR; Davies, HM; Gregg, TC; O'Connor, KA1
Arias-Montaño, JA; Díaz-Romero, M; Eguibar, JR; Flores, G1
Andrade-Neto, M; Barros Viana, GS; Florençode Sousa, FC; França Fonteles, MM; Mendes Vasconcelos, SM; Silveira Macêdo, D; Vasconcelos Aguiar, LM1
Ananth, M; Hadjiargyrou, M; Komatsu, DE; Robison, LS; Thanos, PK1

Other Studies

46 other study(ies) available for spiperone and cocaine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
Effects of neuroleptics on release of 3H-dopamine from slices of rat corpus striatum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 297, Issue:1

    Topics: Animals; Antipsychotic Agents; Apomorphine; Chlorpromazine; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; Fluphenazine; Haloperidol; Male; Rats; Spiperone

1977
Neuroleptic interference with the cocaine cue: internal stimulus control of behavior and psychosis.
    Psychopharmacology, 1978, Jul-19, Volume: 58, Issue:3

    Topics: Amphetamine; Animals; Antipsychotic Agents; Behavior; Cocaine; Cues; Drug Interactions; Haloperidol; Humans; Male; Pimozide; Psychotic Disorders; Rats; Spiperone

1978
Increased dopamine receptor binding in rat brain by repeated cocaine injections.
    Communications in psychopharmacology, 1979, Volume: 3, Issue:3

    Topics: Animals; Apomorphine; Butyrophenones; Cocaine; Dose-Response Relationship, Drug; Male; Motor Activity; Rats; Receptors, Dopamine; Spiperone

1979
Effects of dopaminergic agonists and antagonists of feeding in intact and 6-hydroxydopamine-treated rats.
    The Journal of pharmacology and experimental therapeutics, 1977, Volume: 201, Issue:2

    Topics: Animals; Apomorphine; Benztropine; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Brain; Catecholamines; Cocaine; Dextroamphetamine; Dopamine; Dopamine Antagonists; Eating; Hydroxydopamines; Levodopa; Male; Methylphenidate; Methyltyrosines; Motor Activity; Rats; Spiperone; Telencephalon

1977
Effects of repeated injections of cocaine on catecholamine receptor binding sites, dopamine transporter binding sites and behavior in rhesus monkey.
    Brain research, 1992, Apr-24, Volume: 578, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Benzazepines; Brain; Carrier Proteins; Caudate Nucleus; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Administration Schedule; Grooming; Homovanillic Acid; Hydroxyindoleacetic Acid; Iodocyanopindolol; Macaca mulatta; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Organ Specificity; Pindolol; Piperazines; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin; Spiperone; Stereotyped Behavior; Time Factors

1992
Enhanced sensitivity to the behavioral effects of cocaine after chronic administration of D2-selective dopamine antagonists in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Fluoxetine; Infusion Pumps; Male; Quipazine; Receptors, Dopamine; Receptors, Dopamine D2; Saimiri; Spiperone

1992
Cocaine in utero enhances the behavioral response to cocaine in adult rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 42, Issue:3

    Topics: Animals; Body Weight; Cocaine; Corpus Striatum; Female; Male; Motor Activity; Nucleus Accumbens; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1992
Cocaine self-administration is increased by both D1 and D2 dopamine antagonists.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: Animals; Benzazepines; Cocaine; Conditioning, Operant; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement, Psychology; Self Administration; Spiperone

1991
Effects of selective D1 and D2 dopamine antagonists on cocaine self-administration in the rat.
    Psychopharmacology, 1991, Volume: 105, Issue:2

    Topics: Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Self Administration; Spiperone

1991
Flunarizine potentiates cocaine-induced dopamine release and motor stimulation in rats.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: Animals; Brain Chemistry; Cocaine; Corpus Striatum; Dopamine; Drug Synergism; Flunarizine; Male; Membranes; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride

1990
Weanling rats exposed prenatally to cocaine exhibit an increase in striatal D2 dopamine binding associated with an increase in ligand affinity.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:2

    Topics: Animals; Benzazepines; Cocaine; Corpus Striatum; Female; Nucleus Accumbens; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Weaning

1990
Cocaine produces locomotor stimulation in SS but not LS mice: relationship to dopaminergic function.
    Psychopharmacology, 1990, Volume: 101, Issue:1

    Topics: Animals; Benzazepines; Brain Chemistry; Cocaine; Dopamine; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred Strains; Motor Activity; Receptors, Dopamine; Species Specificity; Spiperone

1990
Effects of chronic cocaine abuse on postsynaptic dopamine receptors.
    The American journal of psychiatry, 1990, Volume: 147, Issue:6

    Topics: Adult; Basal Ganglia; Cocaine; Corpus Striatum; Down-Regulation; Fluorine Radioisotopes; Humans; Receptors, Dopamine; Spiperone; Substance-Related Disorders; Tomography, Emission-Computed; Up-Regulation

1990
Evidence for two populations of 5-hydroxytryptamine receptors in dog basilar artery.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: Animals; Basilar Artery; Cocaine; Dogs; In Vitro Techniques; Indomethacin; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Potassium; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Spiperone; Vasoconstriction

1989
Prenatal cocaine exposure fails to modify neurobehavioral responses and the striatal dopaminergic system in newborn rats.
    General pharmacology, 1989, Volume: 20, Issue:5

    Topics: Animals; Animals, Newborn; Behavior, Animal; Body Weight; Cocaine; Corpus Striatum; Dopamine; Drinking; Eating; Female; Male; Motor Activity; Nervous System; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Sexual Behavior, Animal; Spiperone

1989
Differential actions of cocaine and amphetamine on dorsal raphe neurons in vitro.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:1

    Topics: Amphetamine; Animals; Cocaine; In Vitro Techniques; Membrane Potentials; Neurons; Prazosin; Raphe Nuclei; Rats; Serotonin; Spiperone

1989
[3H]SCH 23390 labeled D1 dopamine receptors are unchanged in schizophrenia and Parkinson's disease.
    European journal of pharmacology, 1985, Aug-15, Volume: 114, Issue:2

    Topics: Aged; Antipsychotic Agents; Benzazepines; Cocaine; Humans; In Vitro Techniques; Middle Aged; Parkinson Disease; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Schizophrenia; Spiperone

1985
The D1 dopamine receptor antagonist SCH 23390 increases cocaine self-administration in the rat.
    Neuroscience letters, 1987, Aug-31, Volume: 79, Issue:3

    Topics: Animals; Benzazepines; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Self Administration; Spiperone

1987
Repeated cocaine administration results in supersensitivity of striatal D-2 dopamine autoreceptors to pergolide.
    Life sciences, 1988, Volume: 42, Issue:3

    Topics: Animals; Benzazepines; Binding, Competitive; Cocaine; Corpus Striatum; Dopamine Antagonists; Male; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1988
Endogenous peptide(s) inhibiting [3H]cocaine binding in mouse brain.
    Neurochemical research, 1980, Volume: 5, Issue:12

    Topics: Animals; Binding Sites; Cell Membrane; Cerebral Cortex; Cocaine; Cyclazocine; Dihydromorphine; Dioxanes; Ethylketocyclazocine; Mice; Molecular Weight; Naloxone; Peptides; Receptors, Opioid; Spiperone

1980
Reduction of dopamine uptake and cocaine binding in mouse striatum by N-methyl-4-phenyl-1,2,3,6-tetrahydropyridine.
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Cocaine; Corpus Striatum; Depression, Chemical; Dopamine; Hydroxydopamines; In Vitro Techniques; Kinetics; Mice; Mice, Inbred BALB C; Pyridines; Spiperone; Synaptosomes

1984
The effect of altered dopaminergic activity on food intake in the rat: evidence for an optimal level of dopaminergic activity for behavior.
    Progress in neuro-psychopharmacology, 1980, Volume: 4, Issue:4-5

    Topics: Amphetamine; Amphetamines; Animals; Apomorphine; Brain; Cocaine; Dextroamphetamine; Dopamine; Feeding Behavior; Haloperidol; Levodopa; Methylphenidate; Rats; Spiperone

1980
Cocaine-induced supersensitivity of striatal dopamine receptors: role of endogenous calmodulin.
    Neuropharmacology, 1981, Volume: 20, Issue:12A

    Topics: Animals; Apomorphine; Calcium-Binding Proteins; Calmodulin; Cocaine; Corpus Striatum; Dopamine; Enzyme-Linked Immunosorbent Assay; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1981
Behavioral and neurochemical changes caused by repeated ethanol and cocaine administration.
    Psychopharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Autoradiography; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Convulsants; Dopamine; Ethanol; gamma-Aminobutyric Acid; Limbic System; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Substantia Nigra

1993
Dopamine mechanisms play at best a small role in the nicotine discriminative stimulus.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:3

    Topics: Animals; Benzazepines; Cocaine; Cues; Discrimination Learning; Discrimination, Psychological; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Neurotransmitter Uptake Inhibitors; Nicotine; Piperazines; Rats; Receptors, Dopamine D1; Reinforcement Schedule; Spiperone

1994
Elimination of cocaine-induced hyperactivity and dopamine-mediated neurophysiological effects in dopamine D1 receptor mutant mice.
    Cell, 1994, Dec-16, Volume: 79, Issue:6

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine; Electric Conductivity; Hyperkinesis; Male; Mice; Mice, Mutant Strains; Neurons; Nucleus Accumbens; Receptors, Dopamine D1; Receptors, Dopamine D2; Signal Transduction; Spiperone

1994
Cocaine tolerance and cross-tolerance.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:1

    Topics: Animals; Behavior, Animal; Benzazepines; Binding Sites; Cocaine; Corpus Striatum; Dopamine Agents; Drug Tolerance; Male; Neurotransmitter Uptake Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tritium

1993
Decreased dopamine D2 receptor availability is associated with reduced frontal metabolism in cocaine abusers.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:2

    Topics: Adult; Brain; Cocaine; Deoxyglucose; Dopamine Agents; Fluorodeoxyglucose F18; Frontal Lobe; Glucose; Humans; Male; Receptors, Dopamine D2; Reference Values; Spiperone; Substance-Related Disorders; Tomography, Emission-Computed

1993
Increased occupation of D1 and D2 dopamine receptors accompanies cocaine-induced behavioral sensitization.
    Brain research, 1994, Mar-14, Volume: 639, Issue:2

    Topics: Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine D2 Receptor Antagonists; Male; Motor Activity; Neostriatum; Nimodipine; Nucleus Accumbens; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Estimation of upper limits on human radiation absorbed doses from carbon-11-labeled compounds.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1993, Volume: 34, Issue:12

    Topics: Animals; Benztropine; Carbon Radioisotopes; Cocaine; Deoxyglucose; Dogs; Humans; Mice; Models, Biological; Papio; Putrescine; Radiation Dosage; Selegiline; Spiperone; Tissue Distribution

1993
Effects of binge pattern cocaine administration on dopamine D1 and D2 receptors in the rat brain: an in vivo study using positron emission tomography.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Dec-01, Volume: 16, Issue:23

    Topics: Animals; Benzazepines; Brain; Cocaine; Dopamine Agonists; Dopamine Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tomography, Emission-Computed

1996
The effects of prenatal cocaine exposure on dopaminergic challenge and receptor binding in Wistar rats.
    Annals of the New York Academy of Sciences, 1996, Oct-31, Volume: 801

    Topics: Animals; Avoidance Learning; Benzazepines; Cocaine; Dopamine; Dopamine Agonists; Female; Male; Motor Activity; Pregnancy; Prenatal Exposure Delayed Effects; Protein Binding; Rats; Rats, Wistar; Receptors, Dopamine; Spiperone; Tritium

1996
Brain dopamine transporter in spontaneously hypertensive rats.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1997, Volume: 38, Issue:3

    Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Brain Chemistry; Carrier Proteins; Caudate Nucleus; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Hypertension; Image Enhancement; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Putamen; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Dopamine; Spiperone

1997
Sustained withdrawal allows normalization of in vivo [11C]N-methylspiperone dopamine D2 receptor binding after chronic binge cocaine: a positron emission tomography study in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1998, Volume: 19, Issue:2

    Topics: Analysis of Variance; Animals; Benzazepines; Brain; Carbon Radioisotopes; Cocaine; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors; Tomography, Emission-Computed

1998
Opposing effects of clomipramine on [125I]RTI-55 and [3H]N-methylspiperone binding in mouse striatum: important role of other factors than endogenous dopamine?
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:3

    Topics: Animals; Brain; Carrier Proteins; Clomipramine; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Organ Specificity; Radioligand Assay; Serotonin; Serotonin Plasma Membrane Transport Proteins; Spiperone; Tritium

1998
Influence of SCH23390 and spiperone on the expression of conditioned place preference induced by d-amphetamine or cocaine in the rat.
    The Chinese journal of physiology, 1998, Jun-30, Volume: 41, Issue:2

    Topics: Animals; Benzazepines; Cocaine; Conditioning, Operant; Dextroamphetamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1998
Behavioral responses to repeated cocaine exposure in mice selectively bred for differential sensitivity to pentobarbital.
    Annals of the New York Academy of Sciences, 2000, Volume: 914

    Topics: Analysis of Variance; Animals; Behavior, Animal; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Hypnotics and Sedatives; Male; Mice; Motor Activity; Nucleus Accumbens; Pentobarbital; Protein Binding; Receptors, Dopamine D2; Spiperone; Tritium

2000
Deficits in striatal dopamine D(2) receptors and energy metabolism detected by in vivo microPET imaging in a rat model of Huntington's disease.
    Experimental neurology, 2000, Volume: 166, Issue:2

    Topics: Animals; Autoradiography; Benzazepines; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Energy Metabolism; Female; Fluorodeoxyglucose F18; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Huntington Disease; In Situ Hybridization; Nerve Degeneration; Neurotoxins; Quinolinic Acid; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Substantia Nigra; Tomography, Emission-Computed; Tritium

2000
GABA(A) alpha 1 subunit knock-out mice do not show a hyperlocomotor response following amphetamine or cocaine treatment.
    Neuropharmacology, 2003, Volume: 44, Issue:2

    Topics: Amphetamine; Animals; Benzazepines; Binding, Competitive; Central Nervous System Stimulants; Cocaine; Diazepam; Dizocilpine Maleate; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Modulators; Habituation, Psychophysiologic; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Protein Subunits; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Spiperone

2003
Cocaine treatment causes early and long-lasting changes in muscarinic and dopaminergic receptors.
    Cellular and molecular neurobiology, 2004, Volume: 24, Issue:1

    Topics: Animals; Benzazepines; Binding, Competitive; Brain; Cocaine; Cocaine-Related Disorders; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Down-Regulation; Male; N-Methylscopolamine; Neuronal Plasticity; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Muscarinic; Spiperone; Synaptic Transmission

2004
Effects of long-term biogenic amine transporter blockade on receptor/G-protein coupling in rat brain.
    Neuropharmacology, 2005, Volume: 48, Issue:1

    Topics: Animals; Apomorphine; Biogenic Monoamines; Brain; Cocaine; Dopamine Antagonists; Drug Administration Schedule; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guanosine 5'-O-(3-Thiotriphosphate); Isotopes; Male; Membrane Transport Modulators; Membrane Transport Proteins; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Spiperone; Time

2005
Enhanced binding of dopamine D1 receptors in caudate-putamen subregions in High-Yawning Sprague-Dawley rats.
    Synapse (New York, N.Y.), 2005, Volume: 56, Issue:2

    Topics: Animals; Benzazepines; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Male; Neostriatum; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tritium; Yawning

2005
Differential effects of cocaine-induced seizures and lethality on M(1)-like muscarinic and dopaminergic D (1)- and D (2)-like binding receptors in mice brain.
    Cellular and molecular neurobiology, 2006, Volume: 26, Issue:1

    Topics: Acetylcholinesterase; Animals; Benzazepines; Binding Sites; Brain; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Humans; Male; Mice; N-Methylscopolamine; Parasympatholytics; Receptor, Muscarinic M1; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Status Epilepticus

2006
Chronic oral methylphenidate treatment reversibly increases striatal dopamine transporter and dopamine type 1 receptor binding in rats.
    Journal of neural transmission (Vienna, Austria : 1996), 2017, Volume: 124, Issue:5

    Topics: Administration, Oral; Animals; Autoradiography; Benzazepines; Central Nervous System Stimulants; Cocaine; Corpus Striatum; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Male; Methylphenidate; Radiopharmaceuticals; Rats, Inbred SHR; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tritium

2017