Page last updated: 2024-08-16

spiperone and clonidine

spiperone has been researched along with clonidine in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-199026 (70.27)18.7374
1990's9 (24.32)18.2507
2000's2 (5.41)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Carmichael, R; Di Paolo, T; Labrie, F; Raynaud, JP1
Giachetti, A; Hefco, E; Jameson, HE; Krulich, L; Marchlewska-Koj, A1
Maj, J; Palider, W; Rawłów, A1
Kojima, C; Satoh, M; Takayanagi, I1
Harris, LT; King, KA; McCall, RB1
Ramage, AG1
Iuvone, PM; Zawilska, J1
Costa, LG; Murphy, SD; Olibet, G1
Gallager, D; Goldman-Rakic, PS; Rakic, P1
Hyttel, J; Skarsfeldt, T1
Baldwin, JJ; Clineschmidt, BV; Huff, JR; Lotti, VJ; Pettibone, DJ; Randall, WC; Vacca, J; Young, SD1
Carlson, KR; Cooper, DO1
Audiau, F; Benavides, J; Guérémy, C; Le Fur, G; Renault, C; Uzan, A1
Arbilla, S; Bartholini, G; Claustre, Y; Dedek, J; Dennis, T; Langer, SZ; Lloyd, KG; Scatton, B; Zivkovic, B1
Garattini, S; Mennini, T; Mocaer, E1
Bymaster, FP; Kornfeld, EC; Nichols, CL; Reid, LR; Wong, DT1
Carlson, KR; Cooper, DO; McKearney, JW1
Bischoff, S; Ortmann, R; Waldmeier, PC1
Barbaz, B; Bernard, P; Braunwalder, A; Kim, HS; Liebman, JM; Lovell, RA; Robson, RD; Stone, G; Wasley, JW; Welch, J1
Hartley, EJ; Seeman, P1
Brenner, M; Dandridge, PA; Davis, LD; Foley, JJ; Gaitanopoulos, D; Kaiser, C; Sarau, HM; Webb, RL1
Berry-Kravis, E; Dawson, G; Freedman, SB1
Ackerman, DM; Hieble, JP; Jain, TC; Sarau, HM1
Bhatnagar, RK; Cannon, JG; Chatterjee, TK; Long, JP1
Iwamoto, ET1
Kwan, S; Seeman, P; Tang, SW1
Connor, TM; Fregly, MJ; Kikta, DC; Threatte, RM1
Clincke, G; Fransen, J; Wauquier, A1
Guarneri, L; Leonardi, A; Poggesi, E; Simonazzi, I; Taddei, C; Testa, R1
Lidow, MS; Rakic, P1
Klimek, V; Nikulina, EM1
Docherty, JR; Kearns, S; O'Rourke, M1
Blier, P; de Montigny, C; Mongeau, R; Weiss, M1
Amobi, N; Coker, C; Guillebaud, J; Mulvin, D; Smith, IC1
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K1
Avellar, MC; Caricati-Neto, A; Jurkiewicz, A; Jurkiewicz, NH; Reuter, HR; Verde, LF1

Other Studies

37 other study(ies) available for spiperone and clonidine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Effects of estrogens on the characteristics of [3H]spiroperidol and [3H]RU24213 binding in rat anterior pituitary gland and brain.
    Molecular and cellular endocrinology, 1979, Volume: 16, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Brain; Butyrophenones; Castration; Clonidine; Dihydroergotoxine; Estradiol; Female; Phenethylamines; Phentolamine; Pituitary Gland, Anterior; Rats; Receptors, Dopamine; Spiperone

1979
On the role of the central noradrenergic and dopaminergic systems in the regulation of TSH secretion in the rat.
    Endocrinology, 1977, Volume: 100, Issue:2

    Topics: Animals; Apomorphine; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Clonidine; Ditiocarb; Dopamine; Kinetics; Male; Methyltyrosines; Norepinephrine; Phenoxybenzamine; Phentolamine; Pituitary Gland; Propranolol; Rats; Spiperone; Stress, Physiological; Thyrotropin; Thyrotropin-Releasing Hormone

1977
The effect of haloperidol, spiperone and pimozide on the flexor reflex of the hind limb of the spinal rat.
    Journal of neural transmission, 1978, Volume: 43, Issue:2

    Topics: Animals; Butyrophenones; Clonidine; Denervation; Fenfluramine; Haloperidol; Hindlimb; Lysergic Acid Diethylamide; Male; Muscle Contraction; Norepinephrine; Pimozide; Rats; Receptors, Adrenergic; Receptors, Serotonin; Reflex; Serotonin; Spinal Cord; Spiperone

1978
Characterization of alpha 1-adrenoceptor subtypes labeled by [3H]prazosin in single cells prepared from rabbit thoracic aorta.
    European journal of pharmacology, 1992, Oct-06, Volume: 221, Issue:1

    Topics: Animals; Aorta, Thoracic; Binding Sites; Calcium; Clonidine; Dioxanes; In Vitro Techniques; Methoxamine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Spiperone

1992
Sympatholytic action of yohimbine mediated by 5-HT1A receptors.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Heart Rate; Injections, Intravenous; Receptors, Serotonin; Spiperone; Sympathetic Nervous System; Tetrahydronaphthalenes; Yohimbine

1991
The mechanism of the sympathoinhibitory action of urapidil: role of 5-HT1A receptors.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: Anesthesia; Animals; Blood Pressure; Cats; Clonidine; Heart; Heart Rate; Kidney; Male; Piperazines; Prazosin; Receptors, Serotonin; Regional Blood Flow; Spiperone; Splanchnic Nerves; Sympatholytics

1991
Catecholamine receptors regulating serotonin N-acetyltransferase activity and melatonin content of chicken retina and pineal gland: D2-dopamine receptors in retina and alpha-2 adrenergic receptors in pineal gland.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: Acetyltransferases; Adrenergic beta-Antagonists; Animals; Apomorphine; Arylamine N-Acetyltransferase; Chickens; Clonidine; Darkness; Dopamine Antagonists; Light; Male; Melatonin; Pineal Gland; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Reference Values; Retina; Spiperone; Yohimbine

1989
Alpha 2-adrenoceptors as a target for formamidine pesticides: in vitro and in vivo studies in mice.
    Toxicology and applied pharmacology, 1988, Volume: 93, Issue:2

    Topics: Amidines; Animals; Chlorphenamidine; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Insecticides; Male; Mice; Receptors, Adrenergic, alpha; Spiperone; Toluidines

1988
Quantitative autoradiography of major neurotransmitter receptors in the monkey striate and extrastriate cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:10

    Topics: Animals; Autoradiography; Cerebral Cortex; Clonidine; Female; Flunitrazepam; Ketanserin; Macaca mulatta; Male; Muscimol; Pindolol; Prazosin; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Neurotransmitter; Serotonin; Spiperone; Visual Cortex

1988
The St 587-induced flexor reflex in pithed rats: a model to evaluate central alpha 1-receptor blocking properties.
    European journal of pharmacology, 1986, Jun-24, Volume: 125, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Binding, Competitive; Clonidine; Decerebrate State; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reflex; Spiperone

1986
Pharmacological profile of a new potent and specific alpha 2-adrenoceptor antagonist, L-657,743.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Blood Platelets; Cattle; Cerebral Cortex; Clonidine; Humans; In Vitro Techniques; Ketanserin; Male; Prazosin; Quinolizines; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Vas Deferens

1987
Morphine dependence and protracted abstinence: regional alterations in CNS radioligand binding.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:6

    Topics: Animals; Brain Chemistry; Clonidine; Dihydroalprenolol; Male; Morphine Dependence; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Spiperone; Substance Withdrawal Syndrome; Time Factors

1985
4-Amino-6-chloro-2-piperazinopyrimidines with selective affinity for alpha 2-adrenoceptors.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:8

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Clonidine; Corpus Striatum; Dioxanes; Idazoxan; Piperazines; Pyrimidines; Rats; Receptors, Adrenergic, alpha; Spiperone; Structure-Activity Relationship

1986
Fengabine, a novel antidepressant GABAergic agent. II. Effect on cerebral noradrenergic, serotonergic and GABAergic transmission in the rat.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Animals; Antidepressive Agents; Brain; Chlorophenols; Clonidine; Dihydroalprenolol; gamma-Aminobutyric Acid; Imipramine; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Spiperone; Synaptic Transmission

1987
Tianeptine, a selective enhancer of serotonin uptake in rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:5

    Topics: Animals; Brain; Cerebral Cortex; Clonidine; Dihydroalprenolol; Dopamine; Hippocampus; Imipramine; In Vitro Techniques; Male; Mesencephalon; Norepinephrine; Rats; Serotonin; Spiperone; Synaptosomes; Thiazepines

1987
Elevation of acetylcholine levels in striatum of rat brain by LY163502, trans-(-)-5,5a,6,7,8,9a,10-octahydro-6-propylpyrimido less than 4,5-g greater than quinolin-2-amine dihydrochloride, a potent and stereospecific dopamine (D2) agonist.
    Life sciences, 1986, Jan-27, Volume: 38, Issue:4

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Apomorphine; Clonidine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Ergolines; Pergolide; Quinolines; Rats; Receptors, Dopamine; Spiperone

1986
Comparison of regional CNS ligand binding in two inbred rat strains: effects of chronic morphine.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:3

    Topics: Animals; Brain; Clonidine; Dihydroalprenolol; Ligands; Male; Morphine; Rats; Rats, Inbred BUF; Rats, Inbred F344; Species Specificity; Spiperone

1985
Modulation of dopaminergic transmission by alpha-noradrenergic agonists and antagonists: evidence for antidopaminergic properties of some alpha antagonists.
    Experientia, 1982, Oct-15, Volume: 38, Issue:10

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Clonidine; Dopamine; Female; Haloperidol; Homovanillic Acid; Male; Prazosin; Rats; Spiperone; Synaptic Transmission; Yohimbine

1982
CGS 7525A, a new, centrally active alpha 2 adrenoceptor antagonist.
    Life sciences, 1983, Jan-24, Volume: 32, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Benzodiazepines; Chemical Phenomena; Chemistry; Clonidine; Male; Mesencephalon; Mianserin; Norepinephrine; Prazosin; Quinones; Rats; Rats, Inbred Strains; Spiperone; Yohimbine

1983
Development of receptors for dopamine and noradrenaline in rat brain.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Animals; Brain; Clonidine; Dioxanes; Female; Limbic System; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Spiperone

1983
Synthesis, resolution, absolute stereochemistry, and enantioselectivity of 3',4'-dihydroxynomifensine.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:1

    Topics: Adenylyl Cyclases; Animals; Biological Assay; Caudate Nucleus; Cerebral Cortex; Circular Dichroism; Clonidine; Imidazoline Receptors; Indicators and Reagents; Isoquinolines; Kinetics; Models, Molecular; Molecular Conformation; Nomifensine; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-2; Receptors, Dopamine; Spiperone; Stereoisomerism; Structure-Activity Relationship

1984
Specific receptor-mediated inhibition of cyclic AMP synthesis by dopamine in a neuroblastoma X brain hybrid cell line NCB-20.
    Journal of neurochemistry, 1984, Volume: 43, Issue:2

    Topics: Alprostadil; Animals; Apomorphine; Brain; Cell Line; Cell Membrane; Clonidine; Cricetinae; Cricetulus; Cyclic AMP; Dopamine; Hybrid Cells; Mice; Neuroblastoma; Prostaglandins E; Receptors, Dopamine; Serotonin; Spiperone

1984
Pharmacological characterization of dopamine-4-O-sulfate.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 267, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Anesthesia; Animals; Clonidine; Dioxanes; Dogs; Dopamine; Ear; Female; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Rabbits; Regional Blood Flow; Renal Circulation; Spiperone

1984
Interaction of dihydroxy-2-aminotetralin derivatives at sites labelled with [3H]clonidine, [3H]prazosin and [3H]spiperone in rat brain membranes.
    European journal of pharmacology, 1984, Feb-17, Volume: 98, Issue:2

    Topics: Animals; Binding Sites; Brain; Butyrophenones; Cell Membrane; Cerebral Cortex; Clonidine; Drug Interactions; Male; Naphthalenes; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Spiperone; Tetrahydronaphthalenes

1984
Pharmacologic effects of N-allylnormetazocine (SKF-10047).
    NIDA research monograph, 1981, Volume: 34

    Topics: Analgesics; Animals; Behavior, Animal; Clonidine; Cyclazocine; Ethylketocyclazocine; Male; Morphine; Motor Activity; Phenazocine; Rats; Receptors, Dopamine; Spiperone

1981
Differential effect of chronic desipramine and amitriptyline treatment on rat brain adrenergic and serotonergic receptors.
    Psychiatry research, 1981, Volume: 4, Issue:2

    Topics: Amitriptyline; Animals; Brain; Cerebral Cortex; Clonidine; Desipramine; Dihydroalprenolol; Dioxanes; Male; Radioligand Assay; Rats; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Spiperone

1981
L-5-Hydroxytryptophan-induced drinking in rats: possible mechanisms for induction.
    Pharmacology, biochemistry, and behavior, 1981, Volume: 14, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Captopril; Clonidine; Drinking; Drug Interactions; Female; Haloperidol; Propranolol; Rats; Spiperone; Stimulation, Chemical

1981
Brain reinforcement mechanisms: alpha-adrenergic and dopaminergic agonists and antagonists.
    Progress in clinical and biological research, 1981, Volume: 71

    Topics: Animals; Apomorphine; Brain; Clonidine; Electric Stimulation; Hypothalamus; Locus Coeruleus; Neurons; Phenoxybenzamine; Rats; Receptors, Adrenergic; Receptors, Dopamine; Reinforcement, Psychology; Saimiri; Self Stimulation; Spiperone; Substantia Nigra

1981
Mediation of noradrenaline-induced contractions of rat aorta by the alpha 1B-adrenoceptor subtype.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Computer Simulation; Hippocampus; In Vitro Techniques; Liver; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Regression Analysis; Spiperone; Stereoisomerism; Sulfonamides

1995
Distribution and density of monoamine receptors in the primate visual cortex devoid of retinal input from early embryonic stages.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:3 Pt 2

    Topics: Animals; Anophthalmos; Benzazepines; Clonidine; Eye Enucleation; Gene Expression Regulation, Developmental; Gestational Age; Ketanserin; Macaca mulatta; Pindolol; Prazosin; Radioligand Assay; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Spiperone; Visual Cortex; Visual Pathways

1995
Strain differences in clonidine-induced aggressiveness in mice and its interaction with the dopamine system.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Aggression; Animals; Benzazepines; Binding, Competitive; Brain; Clonidine; Dopamine; Dopamine Agents; Dopamine Antagonists; Male; Mice; Mice, Inbred A; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred CBA; Mice, Inbred DBA; Mice, Inbred Strains; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity; Spiperone

1993
Investigation of the actions of chloroethylclonidine in rat aorta.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine

1995
Effect of acute, short- and long-term milnacipran administration on rat locus coeruleus noradrenergic and dorsal raphe serotonergic neurons.
    Neuropharmacology, 1998, Volume: 37, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic Uptake Inhibitors; Animals; Biological Transport; Brimonidine Tartrate; Clonidine; Cyclopropanes; Desipramine; Drug Administration Schedule; gamma-Aminobutyric Acid; Hippocampus; Hypothalamus; Injections, Subcutaneous; Kinetics; Locus Coeruleus; Lysergic Acid Diethylamide; Male; Mesencephalon; Milnacipran; Neurons; Norepinephrine; Quinoxalines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Spiperone; Time Factors

1998
Functional characterization of alpha1-adrenoceptor subtypes in longitudinal and circular muscle of human vas deferens.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Alkylating Agents; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Piperazines; Prazosin; Receptors, Adrenergic; Spiperone; Vas Deferens

1999
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
    European journal of pharmacology, 2000, Jan-03, Volume: 387, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine

2000
Sympathetic neurotransmission in the rat testicular capsule: functional characterization and identification of mRNA encoding alpha1-adrenoceptor subtypes.
    European journal of pharmacology, 2006, Aug-14, Volume: 543, Issue:1-3

    Topics: Acetyl-CoA C-Acyltransferase; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Calcium Channel Blockers; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Male; Muscle Contraction; Nifedipine; Norepinephrine; Prazosin; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Purinergic P2; Reserpine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spiperone; Suramin; Sympathetic Nervous System; Synaptic Transmission; Testis

2006