Page last updated: 2024-08-16

spiperone and bromocriptine

spiperone has been researched along with bromocriptine in 59 studies

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-199042 (71.19)18.7374
1990's15 (25.42)18.2507
2000's2 (3.39)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P1
Battista, AF; Fuxe, K; Goldstein, M; Lew, JY; Lieberman, A; Nakamura, S1
Iversen, LL; Quik, M1
List, SJ; Seeman, P1
Agnati, L; Fuxe, K; Köhler, C; Ogren, SO1
Creese, I; Sibley, DR1
Agnati, LF; Fuxe, K; Gustafsson, JA; Schwarcz, R1
Seeman, P; Titeler, M1
Choi, AL; Gallo, F; Martínez de la Escalera, G; Weiner, RI1
Pawlikowski, M; Pisarek, H; Stepien, H1
Ahlskog, JE; Carmichael, SW; Kelly, PJ; Nelson, A; Okazaki, H; Richelson, E; Stoddard, SL; Tyce, GM; van Heerden, JA1
Bédard, PJ; Di Paolo, T; Gagnon, C1
Amlaiky, N; Bausero, P; Borrelli, E; Hen, R; Maroteaux, L; Montmayeur, JP1
Amenta, F; Ianni, L; Lanzillotti, R; Mannelli, M; Pupilli, C; Ricci, A; Serio, M1
Bédard, PJ; Di Paolo, T; Rouillard, C1
Gessa, GL; Olianas, MC; Onali, P1
Beaulieu, M; Felder, R; Kebabian, JW1
Bertrand, P; Delivet, S; Enjalbert, A; Gunz, G; Jaquet, P; Jedynak, CP; Kordon, C; Peillon, F; Pellegrini, I; Rasolonjanahary, R1
Fregly, MJ; Rowland, NE1
Battaglia, G; Creese, I; Hess, EJ; Norman, AB1
Jin, GZ; Le, WD; Zhou, XD1
Govoni, S; Lucchi, L; Memo, M; Missale, C; Spano, PF; Trabucchi, M1
Burchill, SA; Thody, AJ1
Day, RN; Hinkle, PM1
Bhatnagar, RK; Chatterjee, TK; Scott, CE; Vazquez, DM1
Bédard, PJ; Dipaolo, T; Falardeau, P; Rouillard, C1
Bédard, PJ; Boucher, R; Di Paolo, T; Falardeau, P1
Bazan, E; de Yebenes, JG; Gervas, JJ; Mena, MA; Muradas, V1
Arao, M; Kishimoto, S; Koga, M; Mori, S; Morimoto, Y; Nakao, H; Noma, K; Sato, B; Uozumi, T1
Ozaki, L; Stern, N; Tuck, ML1
Fahn, S; Hassan, M; Jackson-Lewis, V; Traub, M; Wagner, HR1
Affolter, HU; Cote, TE; Felder, R; Kebabian, JW; Reisine, T; Sekura, RD1
Israel, JM; Jaquet, P; Vincent, JD1
Bannon, MJ; Bunney, BS; Grace, AA; Roth, RH1
Hruska, RE; Silbergeld, EK1
Costall, B; Lim, SK; Naylor, RJ1
Briley, M; Langer, SZ; Lehmann, J1
Ferrer, JM; Mora, F; Sanguinetti, AM; Vives, F1
Cronin, MJ; Thorner, MO1
Beaulieu, M; Cote, TE; Eskay, RL; Frey, EA; Goldman, ME; Kebabian, JW; Miyazaki, K1
Deupree, JD; Murrin, LC; Pfeiffer, RF; Schneider, MB1
Di Paolo, T; Falardeau, P1
Cronin, MJ; Hellmann, P; Rogol, AD; Thorner, MO1
Cronin, MJ; Evans, WS; Thorner, MO1
Hruska, RE; Silbergeld, EK; Weir, RL1
Bannet, J; Belmaker, RH; Globus, M; Lerer, B1
Gee, KW; Hollinger, MA; Killam, EK1
Finch, CE; Randall, PK; Severson, JA1
Reynolds, GP; Riederer, P1
Cocchi, D; Gil-Ad, I; Locatelli, V; Müller, EE; Parenti, M; Stefanini, E1
Atrens, DM; Hunt, GE; Jackson, DM1
Alberici, A; Memo, M; Spano, P; Tinti, C; Valerio, A1
Bhargava, HN; Reddy, PL1
Bhargava, HN; Reddy, PL; Thorat, SN1
Braghiroli, L; De Feo, G; Giacomelli, S; Koppenaal, DW; Ponzianelli, A1
Haida, M; Kozuma, R; Shinohara, Y; Takagi, S; Takahashi, W; Yoshii, F1
Gu, Q; Kwong, E1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1

Other Studies

59 other study(ies) available for spiperone and bromocriptine

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
    Nature, 1990, Sep-13, Volume: 347, Issue:6289

    Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution

1990
Dopaminephilic properties of ergot alkaloids.
    Federation proceedings, 1978, Volume: 37, Issue:8

    Topics: Acetonitriles; Animals; Bromocriptine; Corpus Striatum; Ergolines; Ergot Alkaloids; Haplorhini; Humans; Levodopa; Parkinson Disease; Receptors, Dopamine; Spiperone; Substantia Nigra; Synaptosomes; Tremor; Tyrosine 3-Monooxygenase

1978
Subsensitivity of the rat striatal dopaminergic system after treatment with bromocriptine: effects on [3H]spiperone binding and dopamine-stimulated cyclic AMP formation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 304, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Corpus Striatum; Cyclic AMP; Dopamine; Male; Rats; Spiperone; Time Factors

1978
Dopamine agonists reverse the elevated 3H-neuroleptic binding in neuroleptic-pretreated rats.
    Life sciences, 1979, Apr-16, Volume: 24, Issue:16

    Topics: Animals; Apomorphine; Bromocriptine; Carbidopa; Corpus Striatum; Dyskinesia, Drug-Induced; Haloperidol; Levodopa; Male; Radioligand Assay; Rats; Receptors, Dopamine; Receptors, Drug; Spiperone

1979
Evidence for in vivo binding of apomorphine and bromocriptine to receptor sites not labelled by 3H-spiperone.
    European journal of pharmacology, 1979, Oct-01, Volume: 58, Issue:3

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Brain; Bromocriptine; Butyrophenones; In Vitro Techniques; Male; Rats; Spiperone

1979
Radioligand binding studies: evidence for multiple dopamine receptors.
    Communications in psychopharmacology, 1979, Volume: 3, Issue:6

    Topics: Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Cattle; Guanine Nucleotides; In Vitro Techniques; Pituitary Gland; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Retina; Spiperone

1979
Effects of bromocriptine on 3H-spiroperidol binding sites in rat striatum. Evidence for actions of dopamine receptors not linked to adenylate cyclase.
    Life sciences, 1978, Aug-07, Volume: 23, Issue:5

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Bromocriptine; Butyrophenones; Caudate Nucleus; Cerebral Cortex; Kainic Acid; Male; Putamen; Rats; Receptors, Dopamine; Spiperone

1978
Antiparkinsonian drug doses and neuroleptic receptors.
    Experientia, 1978, Nov-15, Volume: 34, Issue:11

    Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Cattle; Caudate Nucleus; Haloperidol; In Vitro Techniques; Receptors, Dopamine; Spiperone; Tritium

1978
Dopaminergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via D1-receptors positively coupled to adenylate cyclase.
    Endocrinology, 1992, Volume: 131, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Benzazepines; Bromocriptine; Cell Line; Cyclic AMP; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Gonadotropin-Releasing Hormone; Kinetics; Nerve Tissue Proteins; Neurons; Norepinephrine; Phosphoproteins; Receptors, Dopamine D1; RNA, Messenger; Spiperone

1992
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.
    Endocrine regulations, 1992, Volume: 26, Issue:1

    Topics: Animals; Antiparkinson Agents; Bromocriptine; Diethylstilbestrol; Dose-Response Relationship, Drug; Ergolines; Female; Hyperplasia; Hyperprolactinemia; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Time Factors; Tritium

1992
Reduced D2 dopamine and muscarinic cholinergic receptor densities in caudate specimens from fluctuating parkinsonian patients.
    Annals of neurology, 1991, Volume: 30, Issue:2

    Topics: Adult; Brain Tissue Transplantation; Bromocriptine; Caudate Nucleus; Down-Regulation; Humans; Levodopa; Middle Aged; Parkinson Disease; Pergolide; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, Neurotransmitter; Spiperone

1991
Effect of chronic treatment of MPTP monkeys with dopamine D-1 and/or D-2 receptor agonists.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Brain; Bromocriptine; Carbidopa; Catecholamines; Dopamine Agents; Female; Levodopa; Macaca fascicularis; Receptors, Dopamine; Spiperone

1990
Differential expression of the mouse D2 dopamine receptor isoforms.
    FEBS letters, 1991, Jan-28, Volume: 278, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Southern; Brain; Brain Mapping; Bromocriptine; Cloning, Molecular; DNA; Mice; Molecular Sequence Data; Receptors, Dopamine; Recombinant Proteins; RNA, Messenger; Spiperone

1991
Dopamine modulation of pathological human chromaffin tissue.
    American journal of hypertension, 1990, Volume: 3, Issue:6 Pt 2

    Topics: Adrenal Gland Neoplasms; Autoradiography; Binding Sites; Bromocriptine; Catecholamines; Chromaffin System; Dopamine; Female; Humans; Male; Pheochromocytoma; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1990
Effects of chronic treatment of MPTP monkeys with bromocriptine alone or in combination with SKF 38393.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Brain; Brain Chemistry; Bromocriptine; Dopamine; Female; Homovanillic Acid; Kinetics; Levodopa; Macaca fascicularis; Motor Activity; MPTP Poisoning; Parkinson Disease, Secondary; Receptors, Dopamine; Spiperone

1990
Characterization of dopamine receptors mediating inhibition of adenylate cyclase activity in rat striatum.
    Molecular pharmacology, 1985, Volume: 28, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butaclamol; Corpus Striatum; Dopamine; Enzyme Activation; Ergolines; Guanine Nucleotides; Norepinephrine; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Sulpiride

1985
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
Resistance to bromocriptine in prolactinomas.
    The Journal of clinical endocrinology and metabolism, 1989, Volume: 69, Issue:3

    Topics: 17-Hydroxycorticosteroids; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adolescent; Adult; Bromocriptine; Cell Membrane; Dopamine; Drug Resistance; Female; Growth Hormone; Humans; Kinetics; Luteinizing Hormone; Male; Middle Aged; Pituitary Neoplasms; Prolactin; Prolactinoma; Receptors, Dopamine; Spiperone; Thyrotropin; Thyroxine; Tumor Cells, Cultured

1989
Augmentation of isoproterenol-induced drinking by acute treatment with certain dopaminergic agonists.
    Physiology & behavior, 1988, Volume: 44, Issue:4-5

    Topics: Animals; Brain; Bromocriptine; Dopamine Agents; Dose-Response Relationship, Drug; Drinking; Female; Isoproterenol; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Thirst; Water-Electrolyte Balance

1988
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
    Neuroscience letters, 1985, Aug-30, Volume: 59, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Enhanced stereotypic behavior by chronic treatment with bromocriptine accompanies increase of D-1 receptor binding.
    Life sciences, 1988, Volume: 42, Issue:19

    Topics: Animals; Apomorphine; Benzazepines; Bromocriptine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
Chronic lead exposure alters dopaminergic mechanisms in rat pituitary.
    Toxicology letters, 1986, Volume: 32, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Bromocriptine; Cyclic AMP; Dopamine; Female; Lead; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride

1986
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
    The Journal of endocrinology, 1986, Volume: 111, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride

1986
Transient dopaminergic inhibition of prolactin release from hybrid cells derived by fusion of normal rat pituitary and GH4C1 tumor cells.
    Endocrinology, 1988, Volume: 122, Issue:5

    Topics: Animals; Bromocriptine; Cell Fusion; Cell Line; Cells, Cultured; Dopamine; Female; Growth Hormone; Hybrid Cells; Pituitary Gland; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred WF; Spiperone; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide

1988
Interaction of [3H]spiperone with rat striatal dopamine D-2 receptors: kinetic evidence for antagonist-induced formation of ternary complex.
    Molecular pharmacology, 1988, Volume: 33, Issue:4

    Topics: Algorithms; Animals; Bromocriptine; Corpus Striatum; Guanylyl Imidodiphosphate; Kinetics; Male; Pertussis Toxin; Polymers; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Virulence Factors, Bordetella

1988
Behavioral and biochemical evidence for a different effect of repeated administration of L-dopa and bromocriptine on denervated versus non-denervated striatal dopamine receptors.
    Neuropharmacology, 1987, Volume: 26, Issue:11

    Topics: Animals; Behavior, Animal; Benserazide; Bromocriptine; Corpus Striatum; Denervation; Female; In Vitro Techniques; Levodopa; Rats; Receptors, Dopamine; Spiperone

1987
Chronic treatment with L-DOPA, but not bromocriptine induces dyskinesia in MPTP-parkinsonian monkeys. Correlation with [3H]spiperone binding.
    Brain research, 1986, Aug-06, Volume: 379, Issue:2

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Binding Sites; Bromocriptine; Butyrophenones; Female; Kinetics; Levodopa; Macaca fascicularis; Movement Disorders; Parkinson Disease, Secondary; Pyridines; Spiperone; Time Factors

1986
The effect of single and repeated administration of bromocriptine on monoamine metabolism in rat brain and [3H]spiroperidol binding to striatal membranes.
    Movement disorders : official journal of the Movement Disorder Society, 1986, Volume: 1, Issue:2

    Topics: Animals; Biogenic Monoamines; Brain; Bromocriptine; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Synaptic Membranes; Tritium

1986
Demonstration of specific dopamine receptors on human pituitary adenomas.
    Acta endocrinologica, 1987, Volume: 114, Issue:4

    Topics: Adenoma; Adult; Bromocriptine; Female; Growth Hormone; Humans; Male; Middle Aged; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Spiperone

1987
Evidence for dopaminergic binding sites in the human adrenal cortex.
    Metabolism: clinical and experimental, 1986, Volume: 35, Issue:12

    Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors

1986
The effects of chronic bromocriptine treatment on behaviour and dopamine receptor binding in the rat striatum.
    European journal of pharmacology, 1985, Nov-26, Volume: 118, Issue:1-2

    Topics: Animals; Apomorphine; Bromocriptine; Corpus Striatum; Hydroxydopamines; Kainic Acid; Male; Motor Activity; Muscle Denervation; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra

1985
D-2 dopamine receptor-mediated inhibition of pro-opiomelanocortin synthesis in rat intermediate lobe. Abolition by pertussis toxin or activators of adenylate cyclase.
    The Journal of biological chemistry, 1986, Apr-05, Volume: 261, Issue:10

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Cholera Toxin; Colforsin; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; In Vitro Techniques; Male; Molecular Weight; Pertussis Toxin; Pituitary Gland; Pro-Opiomelanocortin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Virulence Factors, Bordetella

1986
The electrical properties of isolated human prolactin-secreting adenoma cells and their modification by dopamine.
    Endocrinology, 1985, Volume: 117, Issue:4

    Topics: Adenoma; Bromocriptine; Domperidone; Dopamine; Dose-Response Relationship, Drug; Electrophysiology; Flupenthixol; Haloperidol; Humans; In Vitro Techniques; Membrane Potentials; Phenethylamines; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Spiperone; Time Factors

1985
Evidence for an irreversible interaction of bromocryptine with central dopamine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1980, Volume: 312, Issue:1

    Topics: 4-Butyrolactone; Animals; Brain; Bromocriptine; Corpus Striatum; Dopa Decarboxylase; Electrophysiology; Kinetics; Male; Olfactory Bulb; Rats; Receptors, Dopamine; Spiperone; Tyrosine 3-Monooxygenase

1980
Inhibition of neurotransmitter receptor binding by ergot derivatives.
    Journal of neuroscience research, 1981, Volume: 6, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Bromocriptine; Dioxanes; Ergolines; Ergot Alkaloids; gamma-Aminobutyric Acid; Lysergic Acid Diethylamide; Male; Metergoline; Organ Specificity; Quinuclidinyl Benzilate; Rats; Receptors, Neurotransmitter; Serotonin; Spiperone; Structure-Activity Relationship; Synapses

1981
Characterisation of the mechanisms by which purported dopamine agonists reduce spontaneous locomotor activity of mice.
    European journal of pharmacology, 1981, Jul-17, Volume: 73, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Bromocriptine; Catecholamines; Dopamine; Dose-Response Relationship, Drug; Imidazolines; Male; Mice; Motor Activity; Prazosin; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine

1981
Characterization of dopamine autoreceptor and [3H]spiperone binding sites in vitro with classical and novel dopamine receptor agonists.
    European journal of pharmacology, 1983, Mar-18, Volume: 88, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Apomorphine; Benzazepines; Binding Sites; Bromocriptine; Butyrophenones; Cats; Caudate Nucleus; Dopamine; Electric Stimulation; Female; In Vitro Techniques; Male; Phentolamine; Receptors, Dopamine; Spiperone; Sulpiride; Tritium

1983
Effects of agonists and antagonists of D1 and D2 dopamine receptors on self-stimulation of the medial prefrontal cortex in the rat.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Animals; Apomorphine; Bromocriptine; Cerebral Cortex; Dose-Response Relationship, Drug; Ergolines; Functional Laterality; Male; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Self Stimulation; Spiperone; Sulpiride; Synaptic Transmission

1983
Dopamine and bromocriptine inhibit cyclic AMP accumulation in the anterior pituitary: the effect of cholera toxin.
    Journal of cyclic nucleotide research, 1982, Volume: 8, Issue:4

    Topics: Animals; Bromocriptine; Cholera Toxin; Cyclic AMP; Dopamine; Female; Growth Hormone; In Vitro Techniques; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Spiperone; Time Factors

1982
Bromocriptine-induced changes in the biochemistry, physiology, and histology of the intermediate lobe of the rat pituitary gland.
    Endocrinology, 1984, Volume: 114, Issue:5

    Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Male; Melanocyte-Stimulating Hormones; Peptide Fragments; Pituitary Gland; Pituitary Hormones, Anterior; Pro-Opiomelanocortin; Protein Precursors; Rats; Rats, Inbred Strains; RNA, Messenger; Spiperone

1984
Dopamine receptors: effects of chronic L-dopa and bromocriptine treatment in an animal model of Parkinson's disease.
    Clinical neuropharmacology, 1984, Volume: 7, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Bromocriptine; Corpus Striatum; Disease Models, Animal; Dopamine; Humans; Hydroxydopamines; Kinetics; Levodopa; Male; Membranes; Oxidopamine; Parkinson Disease; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra

1984
Dopamine receptors in rat pituitary and estradiol-induced pituitary tumor: effect of chronic treatment with bromocriptine.
    Biochemical and biophysical research communications, 1984, Aug-30, Volume: 123, Issue:1

    Topics: Adenoma; Animals; Bromocriptine; Estradiol; Female; Kinetics; Organ Size; Pituitary Gland, Anterior; Pituitary Neoplasms; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1984
Bromocriptine inhibits growth hormone release from rat pituitary cells in primary culture.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1984, Volume: 175, Issue:2

    Topics: Animals; Bromocriptine; Cells, Cultured; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Spiperone

1984
One minute of bromocriptine irreversibly inhibits prolactin release for hours.
    European journal of pharmacology, 1984, Mar-16, Volume: 99, Issue:1

    Topics: Animals; Bromocriptine; Dopamine; Dopamine Antagonists; Female; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1984
Binding of antiparkinsonian ergot derivatives to the dopamine receptor.
    Psychopharmacology, 1981, Volume: 75, Issue:2

    Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Caudate Nucleus; Ergolines; Lisuride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1981
The effect of chronic bromocriptine and L-dopa on spiperone binding and apomorphine-induced stereotypy.
    Psychopharmacology, 1982, Volume: 78, Issue:1

    Topics: Animals; Apomorphine; Bromocriptine; Butyrophenones; Corpus Striatum; Dose-Response Relationship, Drug; Haloperidol; Humans; Levodopa; Male; Muridae; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1982
Effects of haloperidol-induced dopamine receptor supersensitivity on kindled seizure development.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:1

    Topics: Amygdala; Animals; Bromocriptine; Dose-Response Relationship, Drug; Haloperidol; Kindling, Neurologic; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Seizures; Spiperone; Time Factors

1983
Aging and the regulation of striatal dopaminergic mechanisms in mice.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 219, Issue:3

    Topics: Aging; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Haloperidol; Humans; Male; Mice; Mice, Inbred C57BL; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors

1981
The effects of lisuride and some other dopaminergic agonists on receptor binding in human brain.
    Journal of neural transmission, 1981, Volume: 51, Issue:1-2

    Topics: Brain; Bromocriptine; Ergolines; Humans; Kinetics; Lisuride; Receptors, Dopamine; Spiperone

1981
Prolactin-releasing effect of a novel anti-dopaminergic drug, domperidone, in the rat.
    Neuroendocrinology, 1980, Volume: 30, Issue:2

    Topics: Animals; Benzimidazoles; Bromocriptine; Caudate Nucleus; Corpus Striatum; Dopamine Antagonists; Haloperidol; Male; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Spiperone

1980
Reward summation and the effects of dopamine D1 and D2 agonists and antagonists on fixed-interval responding for brain stimulation.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Brain; Bromocriptine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Drug Interactions; Electric Stimulation; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Self Stimulation; Spiperone

1994
Antisense strategy unravels a dopamine receptor distinct from the D2 subtype, uncoupled with adenylyl cyclase, inhibiting prolactin release from rat pituitary cells.
    Journal of neurochemistry, 1994, Volume: 62, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Base Sequence; Bromocriptine; Cells, Cultured; Cyclic AMP; Female; Molecular Sequence Data; Oligonucleotides, Antisense; Pituitary Gland, Anterior; Polymerase Chain Reaction; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Vasoactive Intestinal Peptide

1994
Effect of chronic administration of U-50,488H, a kappa-opioid receptor agonist, on central dopamine D2 receptors of the rat.
    European journal of pharmacology, 1993, Apr-22, Volume: 235, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Binding Sites; Brain; Bromocriptine; Drug Tolerance; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Opioid, kappa; Spinal Cord; Spiperone; Up-Regulation

1993
Evidence for the behavioral supersensitivity of dopamine D2 receptors without receptor up-regulation in morphine-abstinent rats.
    Brain research, 1993, Apr-02, Volume: 607, Issue:1-2

    Topics: Animals; Behavior, Animal; Body Temperature; Brain Chemistry; Bromocriptine; Drug Tolerance; Kinetics; Male; Morphine Dependence; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spinal Cord; Spiperone; Substance Withdrawal Syndrome; Up-Regulation

1993
A sensitive assay for studying dopaminergic activity in cultures of rat pituitary cells.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cell Count; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation, Preclinical; Female; Haloperidol; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Spiperone

1997
Magnetic resonance imaging and 11C-N-methylspiperone/positron emission tomography studies in a patient with the interval form of carbon monoxide poisoning.
    Journal of the neurological sciences, 1998, Sep-18, Volume: 160, Issue:1

    Topics: Basal Ganglia; Bromocriptine; Carbon Monoxide Poisoning; Carbon Radioisotopes; Caudate Nucleus; Cerebral Hemorrhage; Combined Modality Therapy; Convalescence; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Globus Pallidus; Humans; Hyperbaric Oxygenation; Levodopa; Magnetic Resonance Imaging; Male; Middle Aged; Necrosis; Nerve Tissue Proteins; Parkinson Disease, Secondary; Psychomotor Performance; Putamen; Receptors, Dopamine D2; Spiperone; Tomography, Emission-Computed

1998
Activity-dependent and use-dependent regulation of dopamine-receptor clustering.
    Neuroreport, 2000, Aug-21, Volume: 11, Issue:12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Microscopy, Confocal; Rats; Rats, Long-Evans; Receptor Aggregation; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

2000
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001