spiperone has been researched along with bromocriptine in 59 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 42 (71.19) | 18.7374 |
1990's | 15 (25.42) | 18.2507 |
2000's | 2 (3.39) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH | 1 |
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P | 1 |
Battista, AF; Fuxe, K; Goldstein, M; Lew, JY; Lieberman, A; Nakamura, S | 1 |
Iversen, LL; Quik, M | 1 |
List, SJ; Seeman, P | 1 |
Agnati, L; Fuxe, K; Köhler, C; Ogren, SO | 1 |
Creese, I; Sibley, DR | 1 |
Agnati, LF; Fuxe, K; Gustafsson, JA; Schwarcz, R | 1 |
Seeman, P; Titeler, M | 1 |
Choi, AL; Gallo, F; Martínez de la Escalera, G; Weiner, RI | 1 |
Pawlikowski, M; Pisarek, H; Stepien, H | 1 |
Ahlskog, JE; Carmichael, SW; Kelly, PJ; Nelson, A; Okazaki, H; Richelson, E; Stoddard, SL; Tyce, GM; van Heerden, JA | 1 |
Bédard, PJ; Di Paolo, T; Gagnon, C | 1 |
Amlaiky, N; Bausero, P; Borrelli, E; Hen, R; Maroteaux, L; Montmayeur, JP | 1 |
Amenta, F; Ianni, L; Lanzillotti, R; Mannelli, M; Pupilli, C; Ricci, A; Serio, M | 1 |
Bédard, PJ; Di Paolo, T; Rouillard, C | 1 |
Gessa, GL; Olianas, MC; Onali, P | 1 |
Beaulieu, M; Felder, R; Kebabian, JW | 1 |
Bertrand, P; Delivet, S; Enjalbert, A; Gunz, G; Jaquet, P; Jedynak, CP; Kordon, C; Peillon, F; Pellegrini, I; Rasolonjanahary, R | 1 |
Fregly, MJ; Rowland, NE | 1 |
Battaglia, G; Creese, I; Hess, EJ; Norman, AB | 1 |
Jin, GZ; Le, WD; Zhou, XD | 1 |
Govoni, S; Lucchi, L; Memo, M; Missale, C; Spano, PF; Trabucchi, M | 1 |
Burchill, SA; Thody, AJ | 1 |
Day, RN; Hinkle, PM | 1 |
Bhatnagar, RK; Chatterjee, TK; Scott, CE; Vazquez, DM | 1 |
Bédard, PJ; Dipaolo, T; Falardeau, P; Rouillard, C | 1 |
Bédard, PJ; Boucher, R; Di Paolo, T; Falardeau, P | 1 |
Bazan, E; de Yebenes, JG; Gervas, JJ; Mena, MA; Muradas, V | 1 |
Arao, M; Kishimoto, S; Koga, M; Mori, S; Morimoto, Y; Nakao, H; Noma, K; Sato, B; Uozumi, T | 1 |
Ozaki, L; Stern, N; Tuck, ML | 1 |
Fahn, S; Hassan, M; Jackson-Lewis, V; Traub, M; Wagner, HR | 1 |
Affolter, HU; Cote, TE; Felder, R; Kebabian, JW; Reisine, T; Sekura, RD | 1 |
Israel, JM; Jaquet, P; Vincent, JD | 1 |
Bannon, MJ; Bunney, BS; Grace, AA; Roth, RH | 1 |
Hruska, RE; Silbergeld, EK | 1 |
Costall, B; Lim, SK; Naylor, RJ | 1 |
Briley, M; Langer, SZ; Lehmann, J | 1 |
Ferrer, JM; Mora, F; Sanguinetti, AM; Vives, F | 1 |
Cronin, MJ; Thorner, MO | 1 |
Beaulieu, M; Cote, TE; Eskay, RL; Frey, EA; Goldman, ME; Kebabian, JW; Miyazaki, K | 1 |
Deupree, JD; Murrin, LC; Pfeiffer, RF; Schneider, MB | 1 |
Di Paolo, T; Falardeau, P | 1 |
Cronin, MJ; Hellmann, P; Rogol, AD; Thorner, MO | 1 |
Cronin, MJ; Evans, WS; Thorner, MO | 1 |
Hruska, RE; Silbergeld, EK; Weir, RL | 1 |
Bannet, J; Belmaker, RH; Globus, M; Lerer, B | 1 |
Gee, KW; Hollinger, MA; Killam, EK | 1 |
Finch, CE; Randall, PK; Severson, JA | 1 |
Reynolds, GP; Riederer, P | 1 |
Cocchi, D; Gil-Ad, I; Locatelli, V; Müller, EE; Parenti, M; Stefanini, E | 1 |
Atrens, DM; Hunt, GE; Jackson, DM | 1 |
Alberici, A; Memo, M; Spano, P; Tinti, C; Valerio, A | 1 |
Bhargava, HN; Reddy, PL | 1 |
Bhargava, HN; Reddy, PL; Thorat, SN | 1 |
Braghiroli, L; De Feo, G; Giacomelli, S; Koppenaal, DW; Ponzianelli, A | 1 |
Haida, M; Kozuma, R; Shinohara, Y; Takagi, S; Takahashi, W; Yoshii, F | 1 |
Gu, Q; Kwong, E | 1 |
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J | 1 |
59 other study(ies) available for spiperone and bromocriptine
Article | Year |
---|---|
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection | 1991 |
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution | 1990 |
Dopaminephilic properties of ergot alkaloids.
Topics: Acetonitriles; Animals; Bromocriptine; Corpus Striatum; Ergolines; Ergot Alkaloids; Haplorhini; Humans; Levodopa; Parkinson Disease; Receptors, Dopamine; Spiperone; Substantia Nigra; Synaptosomes; Tremor; Tyrosine 3-Monooxygenase | 1978 |
Subsensitivity of the rat striatal dopaminergic system after treatment with bromocriptine: effects on [3H]spiperone binding and dopamine-stimulated cyclic AMP formation.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Corpus Striatum; Cyclic AMP; Dopamine; Male; Rats; Spiperone; Time Factors | 1978 |
Dopamine agonists reverse the elevated 3H-neuroleptic binding in neuroleptic-pretreated rats.
Topics: Animals; Apomorphine; Bromocriptine; Carbidopa; Corpus Striatum; Dyskinesia, Drug-Induced; Haloperidol; Levodopa; Male; Radioligand Assay; Rats; Receptors, Dopamine; Receptors, Drug; Spiperone | 1979 |
Evidence for in vivo binding of apomorphine and bromocriptine to receptor sites not labelled by 3H-spiperone.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Brain; Bromocriptine; Butyrophenones; In Vitro Techniques; Male; Rats; Spiperone | 1979 |
Radioligand binding studies: evidence for multiple dopamine receptors.
Topics: Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Cattle; Guanine Nucleotides; In Vitro Techniques; Pituitary Gland; Pituitary Gland, Anterior; Radioligand Assay; Receptors, Dopamine; Retina; Spiperone | 1979 |
Effects of bromocriptine on 3H-spiroperidol binding sites in rat striatum. Evidence for actions of dopamine receptors not linked to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Bromocriptine; Butyrophenones; Caudate Nucleus; Cerebral Cortex; Kainic Acid; Male; Putamen; Rats; Receptors, Dopamine; Spiperone | 1978 |
Antiparkinsonian drug doses and neuroleptic receptors.
Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Cattle; Caudate Nucleus; Haloperidol; In Vitro Techniques; Receptors, Dopamine; Spiperone; Tritium | 1978 |
Dopaminergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via D1-receptors positively coupled to adenylate cyclase.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Benzazepines; Bromocriptine; Cell Line; Cyclic AMP; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Gonadotropin-Releasing Hormone; Kinetics; Nerve Tissue Proteins; Neurons; Norepinephrine; Phosphoproteins; Receptors, Dopamine D1; RNA, Messenger; Spiperone | 1992 |
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.
Topics: Animals; Antiparkinson Agents; Bromocriptine; Diethylstilbestrol; Dose-Response Relationship, Drug; Ergolines; Female; Hyperplasia; Hyperprolactinemia; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Time Factors; Tritium | 1992 |
Reduced D2 dopamine and muscarinic cholinergic receptor densities in caudate specimens from fluctuating parkinsonian patients.
Topics: Adult; Brain Tissue Transplantation; Bromocriptine; Caudate Nucleus; Down-Regulation; Humans; Levodopa; Middle Aged; Parkinson Disease; Pergolide; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, Neurotransmitter; Spiperone | 1991 |
Effect of chronic treatment of MPTP monkeys with dopamine D-1 and/or D-2 receptor agonists.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Brain; Bromocriptine; Carbidopa; Catecholamines; Dopamine Agents; Female; Levodopa; Macaca fascicularis; Receptors, Dopamine; Spiperone | 1990 |
Differential expression of the mouse D2 dopamine receptor isoforms.
Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Southern; Brain; Brain Mapping; Bromocriptine; Cloning, Molecular; DNA; Mice; Molecular Sequence Data; Receptors, Dopamine; Recombinant Proteins; RNA, Messenger; Spiperone | 1991 |
Dopamine modulation of pathological human chromaffin tissue.
Topics: Adrenal Gland Neoplasms; Autoradiography; Binding Sites; Bromocriptine; Catecholamines; Chromaffin System; Dopamine; Female; Humans; Male; Pheochromocytoma; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1990 |
Effects of chronic treatment of MPTP monkeys with bromocriptine alone or in combination with SKF 38393.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Brain; Brain Chemistry; Bromocriptine; Dopamine; Female; Homovanillic Acid; Kinetics; Levodopa; Macaca fascicularis; Motor Activity; MPTP Poisoning; Parkinson Disease, Secondary; Receptors, Dopamine; Spiperone | 1990 |
Characterization of dopamine receptors mediating inhibition of adenylate cyclase activity in rat striatum.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butaclamol; Corpus Striatum; Dopamine; Enzyme Activation; Ergolines; Guanine Nucleotides; Norepinephrine; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Sulpiride | 1985 |
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone | 1986 |
Resistance to bromocriptine in prolactinomas.
Topics: 17-Hydroxycorticosteroids; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adolescent; Adult; Bromocriptine; Cell Membrane; Dopamine; Drug Resistance; Female; Growth Hormone; Humans; Kinetics; Luteinizing Hormone; Male; Middle Aged; Pituitary Neoplasms; Prolactin; Prolactinoma; Receptors, Dopamine; Spiperone; Thyrotropin; Thyroxine; Tumor Cells, Cultured | 1989 |
Augmentation of isoproterenol-induced drinking by acute treatment with certain dopaminergic agonists.
Topics: Animals; Brain; Bromocriptine; Dopamine Agents; Dose-Response Relationship, Drug; Drinking; Female; Isoproterenol; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Thirst; Water-Electrolyte Balance | 1988 |
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Enhanced stereotypic behavior by chronic treatment with bromocriptine accompanies increase of D-1 receptor binding.
Topics: Animals; Apomorphine; Benzazepines; Bromocriptine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior | 1988 |
Chronic lead exposure alters dopaminergic mechanisms in rat pituitary.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Bromocriptine; Cyclic AMP; Dopamine; Female; Lead; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride | 1986 |
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride | 1986 |
Transient dopaminergic inhibition of prolactin release from hybrid cells derived by fusion of normal rat pituitary and GH4C1 tumor cells.
Topics: Animals; Bromocriptine; Cell Fusion; Cell Line; Cells, Cultured; Dopamine; Female; Growth Hormone; Hybrid Cells; Pituitary Gland; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred WF; Spiperone; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide | 1988 |
Interaction of [3H]spiperone with rat striatal dopamine D-2 receptors: kinetic evidence for antagonist-induced formation of ternary complex.
Topics: Algorithms; Animals; Bromocriptine; Corpus Striatum; Guanylyl Imidodiphosphate; Kinetics; Male; Pertussis Toxin; Polymers; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Virulence Factors, Bordetella | 1988 |
Behavioral and biochemical evidence for a different effect of repeated administration of L-dopa and bromocriptine on denervated versus non-denervated striatal dopamine receptors.
Topics: Animals; Behavior, Animal; Benserazide; Bromocriptine; Corpus Striatum; Denervation; Female; In Vitro Techniques; Levodopa; Rats; Receptors, Dopamine; Spiperone | 1987 |
Chronic treatment with L-DOPA, but not bromocriptine induces dyskinesia in MPTP-parkinsonian monkeys. Correlation with [3H]spiperone binding.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Binding Sites; Bromocriptine; Butyrophenones; Female; Kinetics; Levodopa; Macaca fascicularis; Movement Disorders; Parkinson Disease, Secondary; Pyridines; Spiperone; Time Factors | 1986 |
The effect of single and repeated administration of bromocriptine on monoamine metabolism in rat brain and [3H]spiroperidol binding to striatal membranes.
Topics: Animals; Biogenic Monoamines; Brain; Bromocriptine; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Synaptic Membranes; Tritium | 1986 |
Demonstration of specific dopamine receptors on human pituitary adenomas.
Topics: Adenoma; Adult; Bromocriptine; Female; Growth Hormone; Humans; Male; Middle Aged; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Spiperone | 1987 |
Evidence for dopaminergic binding sites in the human adrenal cortex.
Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors | 1986 |
The effects of chronic bromocriptine treatment on behaviour and dopamine receptor binding in the rat striatum.
Topics: Animals; Apomorphine; Bromocriptine; Corpus Striatum; Hydroxydopamines; Kainic Acid; Male; Motor Activity; Muscle Denervation; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra | 1985 |
D-2 dopamine receptor-mediated inhibition of pro-opiomelanocortin synthesis in rat intermediate lobe. Abolition by pertussis toxin or activators of adenylate cyclase.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bromocriptine; Butyrophenones; Cholera Toxin; Colforsin; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; In Vitro Techniques; Male; Molecular Weight; Pertussis Toxin; Pituitary Gland; Pro-Opiomelanocortin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Virulence Factors, Bordetella | 1986 |
The electrical properties of isolated human prolactin-secreting adenoma cells and their modification by dopamine.
Topics: Adenoma; Bromocriptine; Domperidone; Dopamine; Dose-Response Relationship, Drug; Electrophysiology; Flupenthixol; Haloperidol; Humans; In Vitro Techniques; Membrane Potentials; Phenethylamines; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Spiperone; Time Factors | 1985 |
Evidence for an irreversible interaction of bromocryptine with central dopamine receptors.
Topics: 4-Butyrolactone; Animals; Brain; Bromocriptine; Corpus Striatum; Dopa Decarboxylase; Electrophysiology; Kinetics; Male; Olfactory Bulb; Rats; Receptors, Dopamine; Spiperone; Tyrosine 3-Monooxygenase | 1980 |
Inhibition of neurotransmitter receptor binding by ergot derivatives.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Bromocriptine; Dioxanes; Ergolines; Ergot Alkaloids; gamma-Aminobutyric Acid; Lysergic Acid Diethylamide; Male; Metergoline; Organ Specificity; Quinuclidinyl Benzilate; Rats; Receptors, Neurotransmitter; Serotonin; Spiperone; Structure-Activity Relationship; Synapses | 1981 |
Characterisation of the mechanisms by which purported dopamine agonists reduce spontaneous locomotor activity of mice.
Topics: Animals; Antipsychotic Agents; Apomorphine; Bromocriptine; Catecholamines; Dopamine; Dose-Response Relationship, Drug; Imidazolines; Male; Mice; Motor Activity; Prazosin; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes; Yohimbine | 1981 |
Characterization of dopamine autoreceptor and [3H]spiperone binding sites in vitro with classical and novel dopamine receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Apomorphine; Benzazepines; Binding Sites; Bromocriptine; Butyrophenones; Cats; Caudate Nucleus; Dopamine; Electric Stimulation; Female; In Vitro Techniques; Male; Phentolamine; Receptors, Dopamine; Spiperone; Sulpiride; Tritium | 1983 |
Effects of agonists and antagonists of D1 and D2 dopamine receptors on self-stimulation of the medial prefrontal cortex in the rat.
Topics: Animals; Apomorphine; Bromocriptine; Cerebral Cortex; Dose-Response Relationship, Drug; Ergolines; Functional Laterality; Male; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Self Stimulation; Spiperone; Sulpiride; Synaptic Transmission | 1983 |
Dopamine and bromocriptine inhibit cyclic AMP accumulation in the anterior pituitary: the effect of cholera toxin.
Topics: Animals; Bromocriptine; Cholera Toxin; Cyclic AMP; Dopamine; Female; Growth Hormone; In Vitro Techniques; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Spiperone; Time Factors | 1982 |
Bromocriptine-induced changes in the biochemistry, physiology, and histology of the intermediate lobe of the rat pituitary gland.
Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Male; Melanocyte-Stimulating Hormones; Peptide Fragments; Pituitary Gland; Pituitary Hormones, Anterior; Pro-Opiomelanocortin; Protein Precursors; Rats; Rats, Inbred Strains; RNA, Messenger; Spiperone | 1984 |
Dopamine receptors: effects of chronic L-dopa and bromocriptine treatment in an animal model of Parkinson's disease.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Bromocriptine; Corpus Striatum; Disease Models, Animal; Dopamine; Humans; Hydroxydopamines; Kinetics; Levodopa; Male; Membranes; Oxidopamine; Parkinson Disease; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra | 1984 |
Dopamine receptors in rat pituitary and estradiol-induced pituitary tumor: effect of chronic treatment with bromocriptine.
Topics: Adenoma; Animals; Bromocriptine; Estradiol; Female; Kinetics; Organ Size; Pituitary Gland, Anterior; Pituitary Neoplasms; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1984 |
Bromocriptine inhibits growth hormone release from rat pituitary cells in primary culture.
Topics: Animals; Bromocriptine; Cells, Cultured; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Spiperone | 1984 |
One minute of bromocriptine irreversibly inhibits prolactin release for hours.
Topics: Animals; Bromocriptine; Dopamine; Dopamine Antagonists; Female; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1984 |
Binding of antiparkinsonian ergot derivatives to the dopamine receptor.
Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Caudate Nucleus; Ergolines; Lisuride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1981 |
The effect of chronic bromocriptine and L-dopa on spiperone binding and apomorphine-induced stereotypy.
Topics: Animals; Apomorphine; Bromocriptine; Butyrophenones; Corpus Striatum; Dose-Response Relationship, Drug; Haloperidol; Humans; Levodopa; Male; Muridae; Receptors, Dopamine; Spiperone; Stereotyped Behavior | 1982 |
Effects of haloperidol-induced dopamine receptor supersensitivity on kindled seizure development.
Topics: Amygdala; Animals; Bromocriptine; Dose-Response Relationship, Drug; Haloperidol; Kindling, Neurologic; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Seizures; Spiperone; Time Factors | 1983 |
Aging and the regulation of striatal dopaminergic mechanisms in mice.
Topics: Aging; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Haloperidol; Humans; Male; Mice; Mice, Inbred C57BL; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors | 1981 |
The effects of lisuride and some other dopaminergic agonists on receptor binding in human brain.
Topics: Brain; Bromocriptine; Ergolines; Humans; Kinetics; Lisuride; Receptors, Dopamine; Spiperone | 1981 |
Prolactin-releasing effect of a novel anti-dopaminergic drug, domperidone, in the rat.
Topics: Animals; Benzimidazoles; Bromocriptine; Caudate Nucleus; Corpus Striatum; Dopamine Antagonists; Haloperidol; Male; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Spiperone | 1980 |
Reward summation and the effects of dopamine D1 and D2 agonists and antagonists on fixed-interval responding for brain stimulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Brain; Bromocriptine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Drug Interactions; Electric Stimulation; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Self Stimulation; Spiperone | 1994 |
Antisense strategy unravels a dopamine receptor distinct from the D2 subtype, uncoupled with adenylyl cyclase, inhibiting prolactin release from rat pituitary cells.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Base Sequence; Bromocriptine; Cells, Cultured; Cyclic AMP; Female; Molecular Sequence Data; Oligonucleotides, Antisense; Pituitary Gland, Anterior; Polymerase Chain Reaction; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Vasoactive Intestinal Peptide | 1994 |
Effect of chronic administration of U-50,488H, a kappa-opioid receptor agonist, on central dopamine D2 receptors of the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Binding Sites; Brain; Bromocriptine; Drug Tolerance; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Opioid, kappa; Spinal Cord; Spiperone; Up-Regulation | 1993 |
Evidence for the behavioral supersensitivity of dopamine D2 receptors without receptor up-regulation in morphine-abstinent rats.
Topics: Animals; Behavior, Animal; Body Temperature; Brain Chemistry; Bromocriptine; Drug Tolerance; Kinetics; Male; Morphine Dependence; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spinal Cord; Spiperone; Substance Withdrawal Syndrome; Up-Regulation | 1993 |
A sensitive assay for studying dopaminergic activity in cultures of rat pituitary cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cell Count; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation, Preclinical; Female; Haloperidol; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Spiperone | 1997 |
Magnetic resonance imaging and 11C-N-methylspiperone/positron emission tomography studies in a patient with the interval form of carbon monoxide poisoning.
Topics: Basal Ganglia; Bromocriptine; Carbon Monoxide Poisoning; Carbon Radioisotopes; Caudate Nucleus; Cerebral Hemorrhage; Combined Modality Therapy; Convalescence; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Globus Pallidus; Humans; Hyperbaric Oxygenation; Levodopa; Magnetic Resonance Imaging; Male; Middle Aged; Necrosis; Nerve Tissue Proteins; Parkinson Disease, Secondary; Psychomotor Performance; Putamen; Receptors, Dopamine D2; Spiperone; Tomography, Emission-Computed | 1998 |
Activity-dependent and use-dependent regulation of dopamine-receptor clustering.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Microscopy, Confocal; Rats; Rats, Long-Evans; Receptor Aggregation; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 2000 |
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine | 2001 |