Page last updated: 2024-08-16

spiperone and amphetamine

spiperone has been researched along with amphetamine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199023 (63.89)18.7374
1990's9 (25.00)18.2507
2000's3 (8.33)29.6817
2010's1 (2.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Andrews, PR; Craik, DJ; Martin, JL1
Colpaert, FC; Janssen, PA; Niemegeers, CJ1
Mogenson, GJ; Robertson, A1
Mogenson, GJ; Robertson, A; Takigawa, M1
Howlett, DR; Nahorski, SR1
Cadet, JL; Zhu, SM1
Belknap, JK; de Paulis, T; Janowsky, A; Kinzie, JM; Neve, KA; Taylor, B1
Angrist, B; Brodie, JD; Dewey, SL; Fowler, JS; Gatley, SJ; Logan, J; Volkow, ND; Wolf, AP1
Chen, C; Goldman, S; Matsumura, K; Minkin, E; Scheffel, U; Wagner, HN; Wong, DF; Young, LT1
Bédard, PJ; Di Paolo, T; Gagnon, C; Gaudin, D; Martinoli, MG; Pelletier, G; Rioux, L1
Linseman, MA1
Fung, YK; Lau, YS1
Pan, ZZ; Williams, JT1
Lum, JT; Piercey, MF1
Agrawal, AK; Goel, SK; Pandya, KP; Seth, PK1
Speiser, Z; Weinstock, M1
Dow, RC; Hill, AG; McQueen, JK1
Harbert, CA; Koe, BK; Plattner, JJ; Weissman, A; Welch, WM1
Costall, B; Dannenburg, WN; Johnson, DN; Naylor, RJ1
Arnt, J; Hyttel, J; Larsen, JJ1
Braestrup, C; Nielsen, EB; Nielsen, M1
Eison, MS; Riblet, LA; Taylor, DP; Temple, DL1
Robertson, HA1
Hruska, RE; Silbergeld, EK1
Bentall, AC; Herberg, LJ1
Bischoff, S; Bittiger, H; Delini-Stula, A; Ortmann, R1
Heffner, TG; Stricker, EM; Zigmond, MJ1
Braestrup, C; Ellison, G; Nielsen, EB; Nielsen, M1
Atrens, DM; Hunt, GE; Jackson, DM1
Albin, RL; Becker, JB; Curran, EJ1
Bjurling, P; Fasth, KJ; Hartvig, P; Långström, B; Tedroff, J; Torstenson, R; Watanabe, Y1
Joksimović, J; Tomić, M1
Ginovart, N; Kapur, S; Ko, F; Seeman, P; Sun, W1
Atack, JR; Bromidge, FA; Dawson, GR; Newman, RJ; O'Meara, GF; Reynolds, DS; Rosahl, TW; Whiting, PJ1
Ahnert-Hilger, G; Bilbao, A; Blex, C; Brunk, I; Perreau-Lenz, S; Sanchis-Segura, C; Spanagel, R1

Reviews

1 review(s) available for spiperone and amphetamine

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Other Studies

35 other study(ies) available for spiperone and amphetamine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Neuroleptic interference with the cocaine cue: internal stimulus control of behavior and psychosis.
    Psychopharmacology, 1978, Jul-19, Volume: 58, Issue:3

    Topics: Amphetamine; Animals; Antipsychotic Agents; Behavior; Cocaine; Cues; Drug Interactions; Haloperidol; Humans; Male; Pimozide; Psychotic Disorders; Rats; Spiperone

1978
Facilitation of self-stimulation of the prefrontal cortex in rats following chronic administration of spiroperidol or amphetamine.
    Psychopharmacology, 1979, Volume: 65, Issue:2

    Topics: Amphetamine; Animals; Butyrophenones; Cerebral Cortex; Dopamine; Male; Rats; Self Stimulation; Spiperone; Stimulation, Chemical; Time Factors

1979
Brain-stimulation reward associated with stimulation of the supracallosal bundle.
    Experimental neurology, 1978, Jan-01, Volume: 58, Issue:1

    Topics: Amphetamine; Animals; Colchicine; Corpus Callosum; Dextroamphetamine; Electric Stimulation; Locus Coeruleus; Male; Neurons; Rats; Self Stimulation; Spiperone; Sympathetic Nervous System

1978
Acute and chronic amphetamine treatments modulate striatal dopamine receptor binding sites.
    Brain research, 1979, Jan-26, Volume: 161, Issue:1

    Topics: Adenylyl Cyclases; Amphetamine; Animals; Binding Sites; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Rats; Receptors, Dopamine; Spiperone

1979
The intrastriatal 6-hydroxydopamine model of hemiparkinsonism: quantitative receptor autoradiographic evidence of correlation between circling behavior and presynaptic as well as postsynaptic nigrostriatal markers in the rat.
    Brain research, 1992, Nov-13, Volume: 595, Issue:2

    Topics: Amphetamine; Animals; Apomorphine; Autoradiography; Biomarkers; Corpus Striatum; Immunohistochemistry; Injections; Male; Mazindol; Oxidopamine; Parkinson Disease, Secondary; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substantia Nigra; Synapses

1992
Extrastriatal dopamine D2 receptors: distribution, pharmacological characterization and region-specific regulation by clozapine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Amphetamine; Animals; Autoradiography; Benzamides; Brain; Clozapine; Haloperidol; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1992
Effects of endogenous dopamine on measures of [18F]N-methylspiroperidol binding in the basal ganglia: comparison of simulations and experimental results from PET studies in baboons.
    Synapse (New York, N.Y.), 1991, Volume: 9, Issue:3

    Topics: Amphetamine; Animals; Basal Ganglia; Computer Simulation; Dopamine; Dopamine Agents; Fluorine Radioisotopes; Ligands; Models, Biological; Papio; Pulsatile Flow; Spiperone; Tomography, Emission-Computed

1991
Effects of endogenous dopamine on kinetics of [3H]N-methylspiperone and [3H]raclopride binding in the rat brain.
    Synapse (New York, N.Y.), 1991, Volume: 9, Issue:3

    Topics: Amphetamine; Animals; Brain; Dopamine; Dopamine Antagonists; Kinetics; Male; Raclopride; Rats; Reserpine; Salicylamides; Spiperone; Tomography, Emission-Computed; Tritium

1991
Regional changes of striatal dopamine receptors following denervation by 6-hydroxydopamine and fetal mesencephalic grafts in the rat.
    Brain research, 1991, Sep-06, Volume: 558, Issue:2

    Topics: Amphetamine; Animals; Benzazepines; Brain Tissue Transplantation; Corpus Striatum; Female; Fetal Tissue Transplantation; Mesencephalon; Oxidopamine; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical

1991
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
    Psychopharmacology, 1990, Volume: 100, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1990
Effect of nicotine pretreatment on striatal dopaminergic system in rats.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:1

    Topics: Amphetamine; Animals; Corpus Striatum; Cotinine; Dopamine; Infusion Pumps; Locomotion; Male; Nicotine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tyrosine

1989
Differential actions of cocaine and amphetamine on dorsal raphe neurons in vitro.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:1

    Topics: Amphetamine; Animals; Cocaine; In Vitro Techniques; Membrane Potentials; Neurons; Prazosin; Raphe Nuclei; Rats; Serotonin; Spiperone

1989
Electrophysiological evidence that spiperone is an antagonist of 5-HT1A receptors in the dorsal raphe nucleus.
    European journal of pharmacology, 1988, Apr-27, Volume: 149, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Buspirone; Dopamine; Electrodes; Electrophysiology; Male; Neurons; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Spiperone; Tetrahydronaphthalenes

1988
Central nervous system effect of 2,5-hexane diol.
    Neurotoxicology, 1985,Fall, Volume: 6, Issue:3

    Topics: Amphetamine; Animals; Apomorphine; Binding Sites; Corpus Striatum; Glycols; Kinetics; Male; Membranes; Mice; Motor Activity; Spiperone; Stereotyped Behavior

1985
Modification by propranolol and related compounds of motor activity and stereotype behaviour induced in the rat by amphetamine.
    European journal of pharmacology, 1974, Volume: 25, Issue:1

    Topics: Amphetamine; Animals; Behavior; Chlorpromazine; Dose-Response Relationship, Drug; Humans; Male; Motor Activity; Moxisylyte; Norepinephrine; Oxprenolol; Practolol; Propranolol; Rats; Spiperone; Stereotyped Behavior; Stimulation, Chemical

1974
Proceedings: Effects of some dopamine receptor stimulants on cobalt-induced epilepsy in the rat.
    British journal of pharmacology, 1974, Volume: 52, Issue:1

    Topics: Amphetamine; Animals; Apomorphine; Cobalt; Dopamine; Electroencephalography; Epilepsy; Ergolines; Male; Rats; Receptors, Adrenergic; Spiperone; Stimulation, Chemical

1974
Neuroleptic activity of the 5-aryltetrahydro-gamma-carboline series. Conformational requirements for interaction with central dopamine receptors.
    Molecular pharmacology, 1980, Volume: 17, Issue:1

    Topics: Amphetamine; Animals; Antipsychotic Agents; Binding Sites; Carbolines; Humans; In Vitro Techniques; Indoles; Male; Molecular Conformation; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Structure-Activity Relationship

1980
Aminoalkylindoles: atypical dopamine antagonists.
    The Journal of pharmacy and pharmacology, 1983, Volume: 35, Issue:4

    Topics: Amphetamine; Animals; Antipsychotic Agents; Catalepsy; Corpus Striatum; Dopamine Antagonists; Haloperidol; Humans; Indoles; Male; Mice; Prolactin; Rats; Rats, Inbred Strains; Spiperone

1983
The citalopram/5-HTP-induced head shake syndrome is correlated to 5-HT2 receptor affinity and also influenced by other transmitters.
    Acta pharmacologica et toxicologica, 1984, Volume: 55, Issue:5

    Topics: 5-Hydroxytryptophan; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Brain; Citalopram; Female; Guinea Pigs; Histamine Antagonists; Humans; Hydroxydopamines; In Vitro Techniques; Male; Neurotransmitter Agents; Oxidopamine; Prazosin; Propylamines; Propylbenzilylcholine Mustard; Rats; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Stereotyped Behavior

1984
Reduction of 3H-spiroperidol binding in rat striatum and frontal cortex by chronic amphetamine: dose response, time course and role of sustained dopamine release.
    Psychopharmacology, 1983, Volume: 81, Issue:1

    Topics: alpha-Methyltyrosine; Amphetamine; Animals; Binding, Competitive; Butyrophenones; Cerebral Cortex; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Hydroxydopamines; Male; Methyltyrosines; Oxidopamine; Rats; Rats, Inbred Strains; Spiperone; Time Factors

1983
Determination of functionally-relevant serum levels of MJ 13859-1 in the dog: relationship to blockade of amphetamine stereotypy.
    Methods and findings in experimental and clinical pharmacology, 1984, Volume: 6, Issue:5

    Topics: Amphetamine; Animals; Behavior, Animal; Binding, Competitive; Corpus Striatum; Dogs; Humans; In Vitro Techniques; Male; Psychotropic Drugs; Radioligand Assay; Rats; Spiperone; Spiro Compounds; Stereotyped Behavior

1984
Chronic phencyclidine, like amphetamine, produces a decrease in [3H]spiroperidol binding in rat striatum.
    European journal of pharmacology, 1982, Mar-12, Volume: 78, Issue:3

    Topics: Amphetamine; Animals; Butyrophenones; Corpus Striatum; Depression, Chemical; In Vitro Techniques; Kinetics; Male; Phencyclidine; Rats; Rats, Inbred Strains; Spiperone

1982
Estrogen treatment enhances dopamine receptor sensitivity in the rat striatum.
    European journal of pharmacology, 1980, Volume: 61, Issue:4

    Topics: Amphetamine; Animals; Apomorphine; Corpus Striatum; Estrogens; Humans; Kinetics; Male; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors

1980
Blockade of amphetamine-induced locomotor activity and stereotypy in rats by spiroperidol but not by an atypical neuroleptic, thioridazine.
    Neuropharmacology, 1980, Volume: 19, Issue:8

    Topics: Amphetamine; Animals; Butyrophenones; Humans; Male; Motor Activity; Rats; Spiperone; Stereotyped Behavior; Thioridazine

1980
Septo-hippocampal system: target for substituted benzamides.
    European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4

    Topics: Adenylyl Cyclases; Amphetamine; Animals; Apomorphine; Benzamides; Binding, Competitive; Brain; Corpus Striatum; Hippocampus; Humans; Male; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1982
The effect of altered dopaminergic activity on food intake in the rat: evidence for an optimal level of dopaminergic activity for behavior.
    Progress in neuro-psychopharmacology, 1980, Volume: 4, Issue:4-5

    Topics: Amphetamine; Amphetamines; Animals; Apomorphine; Brain; Cocaine; Dextroamphetamine; Dopamine; Feeding Behavior; Haloperidol; Levodopa; Methylphenidate; Rats; Spiperone

1980
Decreased spiroperidol and LSD binding in rat brain after continuous amphetamine.
    European journal of pharmacology, 1980, Aug-29, Volume: 66, Issue:2-3

    Topics: Amphetamine; Animals; Brain; Butyrophenones; Corpus Striatum; Frontal Lobe; In Vitro Techniques; Lysergic Acid Diethylamide; Male; Rats; Receptors, Dopamine; Receptors, Serotonin; Spiperone

1980
Reward summation and the effects of dopamine D1 and D2 agonists and antagonists on fixed-interval responding for brain stimulation.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Brain; Bromocriptine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Drug Interactions; Electric Stimulation; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Self Stimulation; Spiperone

1994
Adrenal medulla grafts in the hemiparkinsonian rat: profile of behavioral recovery predicts restoration of the symmetry between the two striata in measures of pre- and postsynaptic dopamine function.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:9

    Topics: Adrenal Medulla; Amphetamine; Animals; Apomorphine; Benzazepines; Cerebral Ventricles; Corpus Striatum; Denervation; Female; Functional Laterality; In Situ Hybridization; Motor Activity; Oxidopamine; Parkinson Disease, Secondary; Rats; Receptors, Dopamine D2; RNA, Messenger; Rotation; Spiperone; Substantia Nigra; Transplantation, Heterotopic; Tyrosine 3-Monooxygenase

1993
Amphetamine effects on dopamine release and synthesis rate studied in the Rhesus monkey brain by positron emission tomography.
    Journal of neural transmission (Vienna, Austria : 1996), 1997, Volume: 104, Issue:4-5

    Topics: Amphetamine; Animals; Brain; Cerebrovascular Circulation; Decarboxylation; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Female; Levodopa; Macaca mulatta; Raclopride; Salicylamides; Spiperone; Tomography, Emission-Computed

1997
Psychotomimetics moderately affect dopamine receptor binding in the rat brain.
    Neurochemistry international, 2000, Volume: 36, Issue:2

    Topics: Amphetamine; Animals; Benzazepines; Brain; Central Nervous System Stimulants; Corpus Striatum; Dextroamphetamine; Hallucinogens; Lysergic Acid Diethylamide; Male; Nucleus Accumbens; Phencyclidine; Rats; Receptors, Dopamine; Spiperone; Tritium

2000
In vivo evidence for dopamine-mediated internalization of D2-receptors after amphetamine: differential findings with [3H]raclopride versus [3H]spiperone.
    Molecular pharmacology, 2003, Volume: 63, Issue:2

    Topics: Amphetamine; Animals; Binding Sites; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Endocytosis; Guanylyl Imidodiphosphate; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Subcellular Fractions; Time Factors; Tritium

2003
GABA(A) alpha 1 subunit knock-out mice do not show a hyperlocomotor response following amphetamine or cocaine treatment.
    Neuropharmacology, 2003, Volume: 44, Issue:2

    Topics: Amphetamine; Animals; Benzazepines; Binding, Competitive; Central Nervous System Stimulants; Cocaine; Diazepam; Dizocilpine Maleate; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Modulators; Habituation, Psychophysiologic; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Protein Subunits; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Spiperone

2003
Amphetamine regulates NR2B expression in Go2α knockout mice and thereby sustains behavioral sensitization.
    Journal of neurochemistry, 2010, Volume: 115, Issue:1

    Topics: Amphetamine; Animals; Behavior, Animal; Blotting, Western; Central Nervous System Stimulants; Conditioning, Operant; Dopamine; Dopamine Antagonists; Gene Deletion; GTP-Binding Protein alpha Subunit, Gi2; Immunoprecipitation; Mice; Mice, Knockout; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Spiperone; Synaptosomes

2010