spiperone has been researched along with 4-iodo-2,5-dimethoxyphenylisopropylamine in 24 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (4.17) | 18.7374 |
1990's | 20 (83.33) | 18.2507 |
2000's | 3 (12.50) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Adham, N; Branchek, T; Hartig, PR; Kao, HT; Macchi, M | 1 |
Glennon, RA; Herrick-Davis, K; Lyon, RA; Seggel, MR; Soine, WH; Titeler, M | 1 |
Baez, M; Kursar, JD; Nelson, DL; Wainscott, DB | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Mutel, V; Sleight, AJ; Stam, NJ; Vanderheyden, PM | 1 |
Kristiansen, K; Kroeze, WK; Roth, BL; Shapiro, DA | 1 |
Glennon, RA | 1 |
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R | 1 |
Jeffrey, JJ; Rydelek-Fitzgerald, L; Wilcox, BD | 1 |
Done, CJ; Sharp, T | 1 |
Beck, SG | 1 |
Ashby, CR; Wang, RY | 1 |
Darmani, NA; Glennon, RA; Martin, BR; Pandey, U | 1 |
Chaouche-Teyara, K; Dabiré, H; Fournier, B; Safar, M | 1 |
Bobker, DH | 1 |
Jeffrey, JJ; Rydelek-Fitzgerald, L; Teitler, M; Wilcox, BD | 2 |
Coulson, A; Grahame-Smith, DG; Leslie, RA; Moorman, JM | 1 |
Kagaya, A; Mikuni, M; Muraoka, S; Saitoh, K; Takahashi, K | 1 |
Grignaschi, G; Samanin, R; Sironi, F | 1 |
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL | 1 |
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP | 1 |
Knowles, ID; Ramage, AG | 1 |
Currie, PJ; Saxena, N; Tu, AY | 1 |
1 review(s) available for spiperone and 4-iodo-2,5-dimethoxyphenylisopropylamine
Article | Year |
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Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 2003 |
23 other study(ies) available for spiperone and 4-iodo-2,5-dimethoxyphenylisopropylamine
Article | Year |
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[3H]-DOB(4-bromo-2,5-dimethoxyphenylisopropylamine) and [3H] ketanserin label two affinity states of the cloned human 5-hydroxytryptamine2 receptor.
Topics: Affinity Labels; Animals; Binding Sites; Binding, Competitive; Cell Line; Chlorocebus aethiops; Cloning, Molecular; DOM 2,5-Dimethoxy-4-Methylamphetamine; Genetic Vectors; Guanylyl Imidodiphosphate; Ketanserin; Mice; Receptors, Serotonin; Transfection; Tritium | 1990 |
[125I]-1-(2,5-dimethoxy-4-iodophenyl)-2-amino-propane: an iodinated radioligand that specifically labels the agonist high-affinity state of 5-HT2 serotonin receptors.
Topics: Amphetamines; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Radioligand Assay; Receptors, Serotonin | 1988 |
Molecular cloning, functional expression, and mRNA tissue distribution of the human 5-hydroxytryptamine2B receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; DNA, Complementary; Humans; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution | 1994 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Radiolabelling of the human 5-HT2A receptor with an agonist, a partial agonist and an antagonist: effects on apparent agonist affinities.
Topics: 3T3 Cells; Animals; Binding, Competitive; Cell Membrane; DOM 2,5-Dimethoxy-4-Methylamphetamine; Humans; Ketanserin; Mice; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1996 |
Differential modes of agonist binding to 5-hydroxytryptamine(2A) serotonin receptors revealed by mutation and molecular modeling of conserved residues in transmembrane region 5.
Topics: Amino Acid Substitution; Animals; Binding, Competitive; Conserved Sequence; COS Cells; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hydrolysis; Membrane Proteins; Models, Molecular; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Folding; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tryptamines | 2000 |
Physical binding pocket induction for affinity prediction.
Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A | 2009 |
Regulation of collagenase gene expression by serotonin and progesterone in rat uterine smooth muscle cells.
Topics: Amphetamines; Animals; Cell Nucleus; Cells, Cultured; Collagenases; DNA Probes; Female; Gene Expression Regulation, Enzymologic; Ketanserin; Kinetics; Muscle, Smooth; Myometrium; Progesterone; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Spiperone; Tetradecanoylphorbol Acetate; Transcription, Genetic; Uterus | 1992 |
Evidence that 5-HT2 receptor activation decreases noradrenaline release in rat hippocampus in vivo.
Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electrophysiology; Hippocampus; Male; Neurons; Norepinephrine; p-Chloroamphetamine; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Receptor Agonists; Spiperone; Sulpiride | 1992 |
5-Hydroxytryptamine increases excitability of CA1 hippocampal pyramidal cells.
Topics: Action Potentials; Amphetamines; Animals; Electric Stimulation; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neurons; Pyramidal Tracts; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Synapses | 1992 |
Effects of antipsychotic drugs on 5-HT2 receptors in the medial prefrontal cortex: microiontophoretic studies.
Topics: Amphetamines; Animals; Antipsychotic Agents; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Evoked Potentials; Frontal Lobe; Haloperidol; Iontophoresis; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone | 1990 |
Do functional relationships exist between 5-HT1A and 5-HT2 receptors?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Injections, Intravenous; Ketanserin; Male; Methoxydimethyltryptamines; Mice; Mice, Inbred ICR; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Stereoisomerism; Tetrahydronaphthalenes | 1990 |
Systemic and regional haemodynamic effects of 1-(2,5-dimethoxy-4-iodo-phenyl)-2-aminopropane (DOI) and alpha-methyl-5-HT, in the anaesthetised rat.
Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Ergolines; Hemodynamics; Injections, Intravenous; Injections, Intraventricular; Male; Rats; Rats, Wistar; Regional Blood Flow; Renal Circulation; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Splanchnic Circulation | 1994 |
A slow excitatory postsynaptic potential mediated by 5-HT2 receptors in nucleus prepositus hypoglossi.
Topics: Amphetamines; Animals; Brain Stem; Cyclohexane Monoterpenes; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Medulla Oblongata; Membrane Potentials; Neurons; Pindolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Synaptic Transmission | 1994 |
Serotonin-mediated 5-HT2 receptor gene regulation in rat myometrial smooth muscle cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Biguanides; Cells, Cultured; Cycloheximide; Female; Gene Expression Regulation; Ketanserin; Medroxyprogesterone Acetate; Myometrium; Piperazines; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sulpiride; Transcription, Genetic; Up-Regulation | 1993 |
Serotonin-dependent collagenase induction in rat myometrial smooth muscle cells: mediation by the 5-HT2 receptor.
Topics: Amphetamines; Animals; Base Sequence; Blotting, Northern; Collagenases; Female; Iodine Radioisotopes; Ketanserin; Molecular Sequence Data; Myometrium; Polymerase Chain Reaction; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Receptor Agonists; Spiperone | 1993 |
Serotonin2/1C receptor activation causes a localized expression of the immediate-early gene c-fos in rat brain: evidence for involvement of dorsal raphe nucleus projection fibres.
Topics: Amphetamines; Animals; Behavior, Animal; Brain Chemistry; Deoxyglucose; Gene Expression; Genes, fos; Immunohistochemistry; Male; Nerve Fibers; Neural Pathways; Proto-Oncogene Proteins c-fos; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Receptor Agonists; Spiperone | 1993 |
Dexamethasone potentiates serotonin-2 receptor-mediated intracellular Ca2+ mobilization in C6 glioma cells.
Topics: Amphetamines; Animals; Calcium; Dexamethasone; Glioma; Ketanserin; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tumor Cells, Cultured | 1993 |
Stimulation of 5-HT2A receptors in the paraventricular hypothalamus attenuates neuropeptide Y-induced hyperphagia through activation of corticotropin releasing factor.
Topics: Amphetamines; Animals; Corticotropin-Releasing Hormone; Feeding Behavior; Hyperphagia; Indoles; Male; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Receptor Agonists; Spiperone | 1996 |
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1998 |
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1999 |
Evidence for a role for central 5-HT2B as well as 5-HT2A receptors in cardiovascular regulation in anaesthetized rats.
Topics: Amidines; Amphetamines; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine Derivatives; Blood Pressure; Cardiovascular Physiological Phenomena; Cinanserin; Injections, Intraventricular; Male; Polyethylene Glycols; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Spiperone | 1999 |
5-HT(2A/2C) receptor antagonists in the paraventricular nucleus attenuate the action of DOI on NPY-stimulated eating.
Topics: Amphetamines; Animals; Appetite Stimulants; Eating; Male; Mianserin; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Ventromedial Hypothalamic Nucleus | 1999 |