Page last updated: 2024-08-16

spiperone and 1,3-ditolylguanidine

spiperone has been researched along with 1,3-ditolylguanidine in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (75.00)18.2507
2000's1 (12.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brasili, L; Costantino, L; Franchini, S; Gandolfi, F; Leonardi, A; Poggesi, E; Prezzavento, O; Ronsisvalle, G; Sorbi, C; Vittorio, F1
Kitamura, Y; Kozaka, T; Miwa, D; Ogawa, K; Shiba, K; Uno, I1
Blier, P; de Montigny, C; Debonnel, G; Monnet, FP1
de Montigny, C; Debonnel, G; Fournier, A; Monnet, FP1
De Montigny, C; Debonnel, G; Junien, JL; Monnet, FP1
Barfknecht, CF; Cheng, B; Ignace, CC; Iwai, Y; Newton, RE; Schoenwald, RD; Shirolkar, S; Vidvauns, S; Xia, E1
Barfknecht, CF; Newton, RE; Schoenwald, RD; Xia, E1
Bergeron, R; de Montigny, C; Debonnel, G1

Other Studies

8 other study(ies) available for spiperone and 1,3-ditolylguanidine

ArticleYear
Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.
    Journal of medicinal chemistry, 2005, Jan-13, Volume: 48, Issue:1

    Topics: Animals; Binding Sites; Biochemistry; Cells, Cultured; Drug Evaluation, Preclinical; Guinea Pigs; Humans; Inhibitory Concentration 50; Ligands; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Serotonin 5-HT1 Receptor Agonists; Sigma-1 Receptor; Structure-Activity Relationship

2005
Syntheses and in vitro evaluation of decalinvesamicol analogues as potential imaging probes for vesicular acetylcholine transporter (VAChT).
    Bioorganic & medicinal chemistry, 2012, Aug-15, Volume: 20, Issue:16

    Topics: Animals; Male; Molecular Structure; Piperidines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, sigma; Vesicular Acetylcholine Transport Proteins

2012
Modulation by sigma ligands of N-methyl-D-aspartate-induced [3H]noradrenaline release in the rat hippocampus: G-protein dependency.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:1

    Topics: Animals; Calcium; Cinnamates; Cyclopropanes; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanidines; Haloperidol; Hippocampus; In Vitro Techniques; Magnesium; Male; N-Methylaspartate; Norepinephrine; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Tritium; Virulence Factors, Bordetella

1992
Neuropeptide Y potentiates the N-methyl-D-aspartate response in the CA3 dorsal hippocampus. II. Involvement of a subtype of sigma receptor.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:3

    Topics: Animals; Cinnamates; Cyclopropanes; Drug Synergism; Guanidines; Haloperidol; Hippocampus; Male; N-Methylaspartate; Neuropeptide Y; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Neuropeptide Y; Receptors, sigma; Spiperone

1992
N-methyl-D-aspartate-induced neuronal activation is selectively modulated by sigma receptors.
    European journal of pharmacology, 1990, Apr-25, Volume: 179, Issue:3

    Topics: Animals; Aspartic Acid; Guanidines; Haloperidol; In Vitro Techniques; Iontophoresis; Kainic Acid; Male; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Spiperone

1990
Lacrimal secretion stimulants: sigma receptors and drug implications.
    Journal of ocular pharmacology, 1993,Fall, Volume: 9, Issue:3

    Topics: Animals; Bromhexine; Dose-Response Relationship, Drug; Eye Proteins; Female; Guanidines; Haloperidol; In Vitro Techniques; Lacrimal Apparatus; Male; Rabbits; Receptors, sigma; Secretory Rate; Spiperone; Tears

1993
The presence of sigma-receptors in the lacrimal gland.
    Journal of ocular pharmacology, 1993,Summer, Volume: 9, Issue:2

    Topics: Animals; Binding, Competitive; Cell Membrane; Female; Guanidines; Haloperidol; Lacrimal Apparatus; Male; Rabbits; Radioligand Assay; Receptors, sigma; Spiperone

1993
Potentiation of neuronal NMDA response induced by dehydroepiandrosterone and its suppression by progesterone: effects mediated via sigma receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Feb-01, Volume: 16, Issue:3

    Topics: Animals; Anisoles; Dehydroepiandrosterone; Drug Synergism; Female; Guanidines; Haloperidol; Hippocampus; Iontophoresis; Ligands; Male; N-Methylaspartate; Pertussis Toxin; Pregnenolone; Progesterone; Propylamines; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Spiperone; Virulence Factors, Bordetella

1996