spermine has been researched along with piperidines in 46 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (8.70) | 18.7374 |
1990's | 25 (54.35) | 18.2507 |
2000's | 12 (26.09) | 29.6817 |
2010's | 5 (10.87) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Alexander, SP; Hill, SJ; Kendall, DA | 1 |
Abe, K; Chida, N; Saito, H | 1 |
Cler, JA; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL | 1 |
Canton, H; Colpaert, F; Lehmann, J | 1 |
Ransom, RW | 1 |
Carter, CJ; Lloyd, KG; Scatton, B; Zivkovic, B | 1 |
Maki, Y; Nagaya, H; Satoh, H | 1 |
Richter, S; Stüttgen, G; Wildberger, D | 1 |
Creveling, CR; Daly, JW; Kondo, K | 1 |
Bagga, L; Derks, M; Doyle, KM; Purcell, WM | 1 |
Williams, K | 1 |
Baxter, K; Church, J; Fletcher, EJ; MacDonald, JF | 1 |
Oblin, A; Schoemaker, H | 1 |
Baudry, M; Marvizón, JC | 1 |
Carter, C; Nicolas, C | 1 |
Carter, C; Fage, D; Voltz, C | 1 |
Abe, K; Chida, N; Nishiyama, N; Saito, H | 1 |
Atterwill, CK; Doyle, KM; Purcell, WM; Westgate, C | 1 |
Chao, J; Fukuchi, J; Igarashi, K; Kashiwagi, K; Williams, K | 1 |
Doyle, KM; Shaw, GG | 1 |
Johnson, SW; Wu, YN | 1 |
Abe, K; Chu, P; Saito, H; Samejima, K; Shirahata, A | 1 |
Ciani, E; Contestabile, A; Dall'Olio, R; Gandolfi, O; Sparapani, M | 1 |
Segal, JA; Skolnick, P | 1 |
Kemp, JA; Kew, JN | 1 |
Berger, ML; Rebernik, P | 1 |
Fukuchi, J; Igarashi, K; Kashiwagi, K; Kuno, T; Masuko, T; Nguyen, ND; Pahk, AJ; Williams, K | 1 |
Rumbaugh, G; Vicini, S | 1 |
Bunney, BS; Shi, WX; Zhang, XX | 1 |
Mo, LL; Sundström, E | 1 |
Arai, T; Haradahira, T; Hojo, J; Kida, T; Maeda, J; Maeda, M; Okauchi, T; Sasaki, S; Suhara, T; Suzuki, K; Yamamoto, F; Zhang, MR | 1 |
D'Hooge, R; De Deyn, PP; Marescau, B; Van Bogaert, PP; Van de Vijver, G; Vanholder, R | 1 |
FOULKS, JG; HANSEN, S; LING, GM; PERRY, TL | 1 |
Haradahira, T; Kurosaki, F; Maeda, J; Maeda, M; Okauchi, T; Sasaki, S; Suhara, T; Suzuki, K; Yamamoto, F | 1 |
Kirby, BP; Shaw, GG | 1 |
Dodd, PR; Lewis, RJ; Tsai, VW | 1 |
Grant, GH; Huggins, DJ | 1 |
Kamei, C; Masuoka, T; Saito, S | 1 |
Hirose, T; Igarashi, K; Jin, L; Kashiwagi, K; Miyazaki, M; Mizuno, S; Nishimura, K; Takigawa, M; Toida, T; Williams, K | 1 |
Fukiwake, T; Füll, C; Han, X; Higashi, K; Igarashi, K; Kashiwagi, K; Leewanich, P; Mizuno, S; Nishimura, K; Terui, Y; Toida, T; Tomitori, H; Williams, K | 1 |
Gavazzo, P; Guida, P; Marchetti, C; Zanardi, I | 1 |
Armand, V; Arrang, JM; Bayard, C; Burban, A; Faucard, R; Vorobjev, V | 1 |
Igarashi, K; Kashiwagi, K; Masuko, T; Mizuno, S; Nishimura, K; Saiki, R; Suganami, A; Tamura, Y; Toida, T; Tomitori, H; Williams, K; Yoshizawa, Y | 1 |
Nowak, G; Poleszak, E; Serefko, A; Socała, K; Szewczyk, B; Wlaź, P; Wośko, S; Wróbel, A | 1 |
Duarte, T; Frühauf, PK; Ineu, RP; Mello, CF; Rubin, MA; Tomazi, L | 1 |
Cheng, X; Lian, Y; Wang, C; Wu, C; Xie, N; Zhang, H; Zhang, L | 1 |
46 other study(ies) available for spermine and piperidines
Article | Year |
---|---|
Excitatory amino acid-induced phosphoinositide turnover in guinea pig cerebral cortical slices: selective enhancement by spermine of the response to DL-1-aminocyclopentane-trans-1,3-dicarboxylate.
Topics: Adrenergic alpha-Antagonists; Alkaloids; Amino Acids; Animals; Calcium; Cerebral Cortex; Cycloleucine; Dose-Response Relationship, Drug; Female; Glutamates; Guinea Pigs; Hydrolysis; Male; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Piperidines; Polyamines; Protein Kinase C; Receptors, Amino Acid; Receptors, Cell Surface; Spermine; Staurosporine | 1992 |
Spermine facilitates the generation of long-term potentiation of evoked potential in the dentate gyrus of anesthetized rats.
Topics: Adrenergic alpha-Antagonists; Anesthesia, General; Animals; Cerebral Ventricles; Electric Stimulation; Evoked Potentials; Hippocampus; Injections, Intraventricular; Male; Piperidines; Putrescine; Rats; Rats, Wistar; Spermidine; Spermine; Time Factors | 1992 |
Polyamines modulate events mediated by the N-methyl-D-aspartate (NMDA) receptor complex through an ifenprodil-insensitive pathway: in vivo measurements of cyclic GMP in the cerebellum.
Topics: Animals; Biogenic Polyamines; Cerebellum; Cyclic GMP; Dizocilpine Maleate; Injections, Intraventricular; Male; Methamphetamine; Mice; Neural Pathways; Ornithine; Pentylenetetrazole; Piperidines; Putrescine; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine | 1991 |
Glutamate and glycine co-activate while polyamines merely modulate the NMDA receptor complex.
Topics: 2-Amino-5-phosphonovalerate; Adrenergic alpha-Antagonists; Animals; Biguanides; Binding, Competitive; Biogenic Polyamines; Biotransformation; Brain; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; In Vitro Techniques; Kynurenic Acid; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine | 1991 |
Polyamine and ifenprodil interactions with the NMDA receptor's glycine site.
Topics: Animals; Binding Sites; Drug Interactions; Glutamates; Glutamic Acid; Glycine; Male; Piperidines; Polyamines; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine; Statistics as Topic | 1991 |
Ifenprodil and SL 82.0715 as cerebral antiischemic agents. III. Evidence for antagonistic effects at the polyamine modulatory site within the N-methyl-D-aspartate receptor complex.
Topics: Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Binding Sites; Binding, Competitive; Brain; Cells, Cultured; Drug Interactions; Female; Glycine; Male; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spermidine; Spermine; Spinal Cord | 1990 |
Actions of antisecretory agents on proton transport in hog gastric microsomes.
Topics: Adenosine Triphosphatases; Animals; Diffusion; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Magnesium; Microscopy, Electron; Microsomes; Piperidines; Potassium; Sodium Cyanide; Spermine; Swine; Valinomycin | 1987 |
[On the demonstration of biogenic amines in animal as well as in human skin and its tumors by thin layer chromatographic methods (according to Seiler). I. Alkylamines, colamine, piperidine, histamine, spermine and spermidine].
Topics: Amines; Animals; Chromatography, Thin Layer; Fluorometry; Guinea Pigs; Histamine; Humans; Indicators and Reagents; Mice; Piperidines; Rats; Skin; Skin Neoplasms; Spectrophotometry; Spermine; Sweat; Ultraviolet Rays | 1967 |
Use of dansyl derivatives and mass spectrometry for identification of biogenic amines.
Topics: Amines; Amino Acids; Animals; Chromatography, Thin Layer; Fluorescence; Fluorometry; Mice; Myocardium; Phenethylamines; Piperidines; Spectrum Analysis; Spermine; Tissue Extracts; Tyramine | 1968 |
Histamine release from mast cells by polyamines: an NMDA receptor-mediated event?
Topics: Animals; Biguanides; Dizocilpine Maleate; Histamine Release; In Vitro Techniques; Kinetics; Mast Cells; p-Methoxy-N-methylphenethylamine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermine | 1994 |
Pharmacological properties of recombinant N-methyl-D-aspartate (NMDA) receptors containing the epsilon 4 (NR2D) subunit.
Topics: Animals; Glutamic Acid; Glycine; Histamine; Oocytes; Piperidines; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Spermine; Xenopus laevis | 1995 |
Blockade by ifenprodil of high voltage-activated Ca2+ channels in rat and mouse cultured hippocampal pyramidal neurones: comparison with N-methyl-D-aspartate receptor antagonist actions.
Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Electrophysiology; Excitatory Amino Acids; Fluorescent Dyes; Hippocampus; Mice; Patch-Clamp Techniques; Piperidines; Potassium; Pyramidal Cells; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermine | 1994 |
Complex allosteric modulation of the binding of the NMDA receptor antagonist [3H]CGP39653.
Topics: 2-Amino-5-phosphonovalerate; Allosteric Regulation; Animals; Biguanides; Binding Sites; Glycine; In Vitro Techniques; Kynurenic Acid; Male; Piperidines; Prosencephalon; Putrescine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine | 1994 |
[3H]dizocilpine association kinetics distinguish stimulatory and inhibitory polyamine sites of N-methyl-D-aspartate receptors.
Topics: Animals; Biguanides; Binding Sites; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; Kinetics; Male; Piperidines; Polyamines; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Tritium | 1994 |
Autoradiographic distribution and characteristics of high- and low-affinity polyamine-sensitive [3H]ifenprodil sites in the rat brain: possible relationship to NMDAR2B receptors and calmodulin.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Calmodulin; Hippocampus; Imidazoles; Male; Piperidines; Polyamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Sepharose; Spermidine; Spermine; Sulfonamides; Tissue Distribution; Trifluoperazine; Tritium | 1994 |
Synergism between the NMDA receptor antagonistic effects of ifenprodil and the glycine antagonist, 7-chlorokynurenate, in vivo.
Topics: Animals; Chromatography, High Pressure Liquid; Drug Synergism; Glycine; Injections; Kynurenic Acid; Male; N-Methylaspartate; Neostriatum; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine | 1994 |
Spermine promotes the survival of primary cultured brain neurons.
Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Hippocampus; Neurons; Piperidines; Putrescine; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine | 1993 |
Characterisation of a functional polyamine site on rat mast cells: association with a NMDA receptor macrocomplex.
Topics: Animals; Binding Sites; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Histamine Release; Mast Cells; p-Methoxy-N-methylphenethylamine; Peritoneum; Piperidines; Polyamines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermine; Thalamus | 1996 |
An aspartate residue in the extracellular loop of the N-methyl-D-aspartate receptor controls sensitivity to spermine and protons.
Topics: Amino Acid Sequence; Animals; Female; Hydrogen-Ion Concentration; Magnesium; Molecular Sequence Data; Mutagenesis, Site-Directed; Piperidines; Receptors, N-Methyl-D-Aspartate; Spermine; Structure-Activity Relationship; Xenopus | 1996 |
Investigation of the involvement of the N-methyl-D-aspartate receptor macrocomplex in the development of spermine-induced CNS excitation in vivo.
Topics: Animals; Brain; Cerebral Ventricles; Dizocilpine Maleate; Female; Kynurenic Acid; Mice; Neuroprotective Agents; Piperazines; Piperidines; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Seizures; Spermine; Tremor | 1996 |
Pharmacological characterization of inward current evoked by N-methyl-D-aspartate in dopamine neurons in the rat brain slice.
Topics: Animals; Dizocilpine Maleate; Excitatory Amino Acid Agonists; In Vitro Techniques; Kynurenic Acid; Magnesium; Male; Membrane Potentials; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Sodium; Spermine; Substantia Nigra; Ventral Tegmental Area | 1996 |
Structural requirement for axonal regeneration-promoting effect of polyamines in cultured rat hippocampal neurons.
Topics: Animals; Axons; Axotomy; Cadaverine; Cells, Cultured; Diamines; Hippocampus; Nerve Regeneration; Neurons; Piperidines; Polyamines; Putrescine; Rats; Rats, Wistar; Spermine | 1997 |
Neurotoxicity of polyamines and pharmacological neuroprotection in cultures of rat cerebellar granule cells.
Topics: 2-Amino-5-phosphonovalerate; Animals; Apoptosis; Aspartic Acid; Butylated Hydroxytoluene; Cells, Cultured; Cerebellar Cortex; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Female; Free Radical Scavengers; Glutamic Acid; L-Lactate Dehydrogenase; Male; Nerve Tissue Proteins; Neurons; Neuroprotective Agents; Nitric Oxide Synthase; Nitroarginine; Piperidines; Putrescine; Quinoxalines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine; Vitamin E | 1997 |
Polyamine-like actions of aminoglycosides and aminoglycoside derivatives at NMDA receptors.
Topics: Adrenergic alpha-Antagonists; Animals; Anti-Bacterial Agents; Carbohydrate Sequence; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kanamycin; Male; Molecular Sequence Data; Neomycin; Piperidines; Polyamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine | 1998 |
An allosteric interaction between the NMDA receptor polyamine and ifenprodil sites in rat cultured cortical neurones.
Topics: Allosteric Regulation; Allosteric Site; Animals; Benzamides; Binding Sites; Cells, Cultured; Cerebral Cortex; Embryo, Mammalian; Evoked Potentials; Excitatory Amino Acid Antagonists; Magnesium; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Piperidines; Pyridines; Rats; Receptors, N-Methyl-D-Aspartate; Spermine | 1998 |
Zinc and ifenprodil allosterically inhibit two separate polyamine-sensitive sites at N-methyl-D-aspartate receptor complex.
Topics: Allosteric Regulation; Animals; Binding, Competitive; Brain; Cell Membrane; Dentate Gyrus; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Hippocampus; Kinetics; Male; Neurons; Organ Specificity; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermine; Tritium; Zinc | 1999 |
A regulatory domain (R1-R2) in the amino terminus of the N-methyl-D-aspartate receptor: effects of spermine, protons, and ifenprodil, and structural similarity to bacterial leucine/isoleucine/valine binding protein.
Topics: Amino Acid Sequence; Animals; Bacterial Proteins; Binding Sites; Carrier Proteins; Excitatory Amino Acid Antagonists; Exons; Hydrogen-Ion Concentration; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Piperidines; Protein Conformation; Protons; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; RNA Splicing; Sequence Homology, Amino Acid; Spermine; Xenopus laevis | 1999 |
Distinct synaptic and extrasynaptic NMDA receptors in developing cerebellar granule neurons.
Topics: Aging; Animals; Animals, Newborn; Cerebellum; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Kinetics; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Synapses | 1999 |
Enhancement of NMDA-induced current by the putative NR2B selective antagonist ifenprodil.
Topics: 2-Amino-5-phosphonovalerate; Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Kynurenic Acid; Male; Membrane Potentials; N-Methylaspartate; Organ Culture Techniques; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine | 2000 |
Polyamine and redox modulation of [3H]MK-801 binding to N-methyl-D-aspartate receptors in the spinal cord and cerebral cortex.
Topics: Animals; Biguanides; Cerebral Cortex; Dizocilpine Maleate; Hydrogen-Ion Concentration; Male; Neuroprotective Agents; Oxidation-Reduction; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Spinal Cord; Tritium | 2001 |
Synthesis, in vitro and in vivo pharmacology of a C-11 labeled analog of CP-101,606, (+/-)threo-1-(4-hydroxyphenyl)-2-[4-hydroxy-4-(p-[11C]methoxyphenyl)piperidino]-1-propanol, as a PET tracer for NR2B subunit-containing NMDA receptors.
Topics: Animals; Brain; Carbon Radioisotopes; Isotope Labeling; Macaca; Male; Metals; Mice; Piperidines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reproducibility of Results; Sensitivity and Specificity; Spermine; Tissue Distribution; Tomography, Emission-Computed; Whole-Body Counting | 2002 |
Involvement of voltage- and ligand-gated Ca2+ channels in the neuroexcitatory and synergistic effects of putative uremic neurotoxins.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Calcium Channels; Cells, Cultured; Drug Synergism; Excitatory Amino Acid Antagonists; GABA Antagonists; Guanidines; Membrane Potentials; Mice; Neurons; Nickel; Piperidines; Potassium Channel Blockers; Seizures; Spermine; Spinal Cord; Succinates; Synapses; Tetraethylammonium; Tetrodotoxin; Uremia | 2003 |
ALIPHATIC AND AROMATIC AMINES OF CAT BRAIN.
Topics: Amines; Amino Alcohols; Brain; Brain Chemistry; Cats; Chromatography; Ion Exchange Resins; Organic Chemicals; Piperidines; Research; Serotonin; Spermine | 1965 |
Synthesis of 11C-labelled bis(phenylalkyl)amines and their in vitro and in vivo binding properties in rodent and monkey brains.
Topics: Amines; Animals; Binding Sites; Brain; Butylamines; Carbon Radioisotopes; In Vitro Techniques; Injections, Intravenous; Isotope Labeling; Macaca mulatta; Male; Mice; Piperidines; Propylamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Tissue Distribution | 2004 |
The neuroprotective effects of N1-dansyl-spermine in the gerbil model of cerebral ischaemia.
Topics: Analysis of Variance; Animals; Behavior, Animal; Body Temperature; Brain Ischemia; Cell Count; Dansyl Compounds; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Gerbillinae; Hippocampus; Male; Motor Activity; Neurons; Neuroprotective Agents; Piperidines; Polyamines; Spermine; Time Factors | 2004 |
The effects of alanine-substituted conantokin-G and ifenprodil on the human spermine-activated N-methyl-D-aspartate receptor.
Topics: Alanine; Binding, Competitive; Cell Membrane; Cerebral Cortex; Conotoxins; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Humans; Neurons; Neurotoxins; Piperidines; Radioligand Assay; Receptors, N-Methyl-D-Aspartate; Spermine | 2005 |
The function of the amino terminal domain in NMDA receptor modulation.
Topics: Amino Acid Sequence; Binding Sites; Dimerization; Humans; Models, Molecular; Molecular Sequence Data; Piperidines; Protein Structure, Tertiary; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Sequence Homology, Amino Acid; Spermine; Zinc | 2005 |
Participation of hippocampal ionotropic glutamate receptors in histamine H(1) antagonist-induced memory deficit in rats.
Topics: Animals; Concanavalin A; Cycloserine; Dioxoles; Dose-Response Relationship, Drug; Electroencephalography; Fourier Analysis; GluK2 Kainate Receptor; Hippocampus; Histamine H1 Antagonists; Injections; Male; Maze Learning; Mental Recall; Orientation; Piperidines; Pyrilamine; Pyrrolidinones; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Histamine H1; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Signal Processing, Computer-Assisted; Spermidine; Spermine; Theta Rhythm | 2008 |
The pore region of N-methyl-D-aspartate receptors differentially influences stimulation and block by spermine.
Topics: Animals; Dose-Response Relationship, Drug; Mice; Mutagenesis, Site-Directed; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermine; Structure-Activity Relationship | 2008 |
Binding of spermine and ifenprodil to a purified, soluble regulatory domain of the N-methyl-D-aspartate receptor.
Topics: Aminoglycosides; Animals; Binding Sites; Biophysical Phenomena; Carbon Isotopes; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Piperidines; Protein Conformation; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Spermine; Time Factors; Tritium; Xenopus laevis | 2008 |
Molecular determinants of multiple effects of nickel on NMDA receptor channels.
Topics: Animals; Binding Sites; Biophysical Phenomena; Cell Line, Transformed; Dose-Response Relationship, Drug; Electric Stimulation; Glutamic Acid; Humans; Membrane Potentials; Models, Molecular; Nickel; Oocytes; Patch-Clamp Techniques; Piperidines; Point Mutation; Protein Structure, Tertiary; Receptors, N-Methyl-D-Aspartate; Spermine; Trace Elements; Transfection; Xenopus; Zinc | 2009 |
Histamine potentiates N-methyl-D-aspartate receptors by interacting with an allosteric site distinct from the polyamine binding site.
Topics: 2-Amino-5-phosphonovalerate; Allosteric Site; Animals; Binding Sites; Calcium; Dizocilpine Maleate; Drug Synergism; Hippocampus; Histamine; In Vitro Techniques; Intracellular Space; Male; Methylhistamines; N-Methylaspartate; Neurons; Norepinephrine; Piperidines; Polyamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermine; Synaptosomes | 2010 |
Structural changes of regulatory domain heterodimer of N-methyl-D-aspartate receptor subunits GluN1 and GluN2B through the binding of spermine and ifenprodil.
Topics: Amino Acid Sequence; Animals; Female; Molecular Sequence Data; Piperidines; Protein Binding; Protein Multimerization; Protein Structure, Secondary; Protein Structure, Tertiary; Protein Subunits; Rats; Receptors, N-Methyl-D-Aspartate; Spermine; Xenopus laevis | 2012 |
An anti-immobility effect of spermine in the forced swim test in mice.
Topics: Animals; Antidepressive Agents; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Mice; Motor Activity; Piperidines; Receptors, N-Methyl-D-Aspartate; Spermine; Swimming | 2014 |
Spermine reverses lipopolysaccharide-induced memory deficit in mice.
Topics: Analysis of Variance; Animals; Cytokines; Discrimination, Psychological; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Excitatory Amino Acid Antagonists; Exploratory Behavior; Lipopolysaccharides; Male; Memory Disorders; Mice; Piperidines; Recognition, Psychology; Spermine | 2015 |
Inhibition of the mitochondrial calcium uniporter inhibits Aβ-induced apoptosis by reducing reactive oxygen species-mediated endoplasmic reticulum stress in cultured microglia.
Topics: Amyloid beta-Peptides; Animals; Antioxidants; Apoptosis; Calcium; Calcium Channels; Cell Survival; Cells, Cultured; Endoplasmic Reticulum Chaperone BiP; Endoplasmic Reticulum Stress; Mice; Microglia; Mitochondria; Neuroprotection; Neuroprotective Agents; Organophosphorus Compounds; Peptide Fragments; Piperidines; Reactive Oxygen Species; Ruthenium Compounds; Spermine | 2017 |