Page last updated: 2024-09-05

sorafenib and tanespimycin

sorafenib has been researched along with tanespimycin in 4 studies

Compound Research Comparison

Studies
(sorafenib)
Trials
(sorafenib)
Recent Studies (post-2010)
(sorafenib)
Studies
(tanespimycin)
Trials
(tanespimycin)
Recent Studies (post-2010) (tanespimycin)
6,5207305,25192139496

Protein Interaction Comparison

ProteinTaxonomysorafenib (IC50)tanespimycin (IC50)
Corticotropin releasing hormone receptor 2Sus scrofa (pig)0.004
Lysine-specific demethylase 6BHomo sapiens (human)0.4
Lysine-specific demethylase 4BHomo sapiens (human)0.7
Tyrosine-protein kinase ABL1Homo sapiens (human)3
ATP-dependent molecular chaperone HSP82Saccharomyces cerevisiae S288C7.65
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.031
Heat shock protein HSP 90-alphaHomo sapiens (human)0.9391
Heat shock protein HSP 90-betaHomo sapiens (human)0.5124
Breakpoint cluster region proteinHomo sapiens (human)3
Lysine-specific demethylase 5AHomo sapiens (human)0.13
EndoplasminCanis lupus familiaris (dog)0.031
Heat shock protein 75 kDa, mitochondrialHomo sapiens (human)1.496
Putative heat shock protein HSP 90-alpha A4Homo sapiens (human)0.78
Lysine-specific demethylase 4CHomo sapiens (human)0.7

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blanke, C1
Burger, AM; Egorin, MJ; Heilbrun, LK; Horiba, MN; Ivy, P; Li, J; Lorusso, PM; Pacey, S; Sausville, EA; Vaishampayan, UN1
Arango, BA; Cohen, EE; Perez, CA; Raez, LE; Santos, ES1
Chen, R; Curley, SA; Liu, H; McConkey, DJ; Ward, JF; Zhang, T1

Reviews

1 review(s) available for sorafenib and tanespimycin

ArticleYear
Novel molecular targeted therapies for refractory thyroid cancer.
    Head & neck, 2012, Volume: 34, Issue:5

    Topics: Angiogenesis Inhibitors; Anilides; Antineoplastic Agents; Axitinib; Benzamides; Benzenesulfonates; Benzoquinones; Bibenzyls; Boronic Acids; Bortezomib; Depsipeptides; ErbB Receptors; Gefitinib; Histone Deacetylase Inhibitors; HSP90 Heat-Shock Proteins; Humans; Hydroxamic Acids; Imatinib Mesylate; Imidazoles; Indazoles; Indoles; Lactams, Macrocyclic; Lenalidomide; Niacinamide; Oligonucleotides; Phenylurea Compounds; Piperazines; Piperidines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrazines; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Quinolines; Receptor Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Sorafenib; Sulfonamides; Sunitinib; Thalidomide; Thyroid Neoplasms; Valproic Acid; Vorinostat

2012

Trials

1 trial(s) available for sorafenib and tanespimycin

ArticleYear
Safety, efficacy, pharmacokinetics, and pharmacodynamics of the combination of sorafenib and tanespimycin.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2010, Jul-15, Volume: 16, Issue:14

    Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzenesulfonates; Benzoquinones; Clinical Trials, Phase II as Topic; Cohort Studies; Colorectal Neoplasms; Drug Administration Schedule; Drug-Related Side Effects and Adverse Reactions; Female; Follow-Up Studies; Humans; Kidney Neoplasms; Lactams, Macrocyclic; Male; Melanoma; Middle Aged; Niacinamide; Phenylurea Compounds; Pyridines; Sorafenib; Survival Analysis

2010

Other Studies

2 other study(ies) available for sorafenib and tanespimycin

ArticleYear
Current and future management of GIST.
    Clinical advances in hematology & oncology : H&O, 2006, Volume: 4, Issue:8

    Topics: Antineoplastic Agents; Benzamides; Benzenesulfonates; Benzoquinones; Disease Progression; Dose-Response Relationship, Drug; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Indoles; Lactams, Macrocyclic; Niacinamide; Phenylurea Compounds; Piperazines; Pyridines; Pyrimidines; Pyrroles; Sorafenib; Sunitinib; Treatment Outcome

2006
Multiple kinase pathways involved in the different de novo sensitivity of pancreatic cancer cell lines to 17-AAG.
    The Journal of surgical research, 2012, Volume: 176, Issue:1

    Topics: Antineoplastic Agents; Benzenesulfonates; Benzoquinones; Cell Line, Tumor; Cell Survival; Drug Resistance, Neoplasm; HSP90 Heat-Shock Proteins; Humans; Lactams, Macrocyclic; Mutation; Niacinamide; Pancreatic Neoplasms; Phenylurea Compounds; Protein Kinase Inhibitors; Protein Kinases; Pyridines; RNA, Small Interfering; Signal Transduction; Sorafenib; Tumor Suppressor Protein p53

2012